公开(公告)号：US20230271929A1

公开(公告)日：2023-08-31

申请号：US18040365

申请日：2021-08-06

Applicant: Kureha Corporation

Inventor： Ryo HARIGAE ,  Chiemi KOJIMA ,  Shingo KONNO ,  Toru YAMAZAKI

IPC: C07D301/02 ,  C07D303/48 ,  C07C67/42 ,  C07D249/08

CPC classification number: C07D301/02 ,  C07D303/48 ,  C07C67/42 ,  C07D249/08

Abstract: A method by which an intermediate product of an azole derivative can be produced at a lower cost than known production methods is provided. A method for producing a compound represented by General Formula (IV) includes converting a compound represented by General Formula (II) into the compound represented by General Formula (IV) using (a) dimethyl sulfide and/or dimethyl sulfoxide, and (b) a methyl-LG (an LG is a nucleophilically substitutable leaving group and is selected from the group consisting of a halogen group, an alkoxysulfonyloxy group, an aryloxysulfonyloxy group, an alkylsulfonyloxy group, a haloalkylsulfonyloxy group, and an arylsulfonyloxy group) in the presence of an inorganic base.

公开(公告)号：US20200288714A1

公开(公告)日：2020-09-17

申请号：US16636502

申请日：2018-11-13

Applicant: Kureha Corporation

Inventor： Ryo HARIGAE ,  Atsushi ITO ,  Taiji MIYAKE ,  Toru YAMAZAKI

IPC: A01N43/653 ,  C07D249/08

Abstract: It is provided a plant disease controlling agent having low toxicity to human and animals and excellent handling safety, and showing excellent controlling effects on various plant diseases and high antibiotic action to plant disease germs.A compound represented by the following the general formula (I), or an N-oxide or agrochemically acceptable salt thereof.

公开(公告)号：US20140213794A1

公开(公告)日：2014-07-31

申请号：US14213240

申请日：2014-03-14

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki ARAKI ,  Toru YAMAZAKI ,  Nobuyuki KUSANO ,  Eiyu IMAI ,  Hisashi KANNO ,  Masaru MORI ,  Taiji MIYAKE

IPC: C07D405/06 ,  C07C201/12 ,  C07C67/31

CPC classification number: C07C67/31 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12 ,  C07C2601/08 ,  C07D405/06

Abstract: An azole derivative according to the invention is represented by Formula (I), wherein each of Ra and Rb denotes a hydrogen atom, or a C1-C6 alkyl group, a C2-C6 alkenyl group or a C2-C6 alkynyl group; Ra and Rb may be substituted with Xa or Xb which is a halogen atom; each of na and nb denotes 0 or the number of Xa- or Xb-substituted hydrogen atoms among the hydrogen atoms in Ra or Rb; each Y denotes a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a C1-C4 alkoxy group, a C1-C4 haloalkoxy group, a phenyl group, a cyano group or a nitro group; m denotes 0 to 5; and A denotes a nitrogen atom or a methyne group. As a result, an azole derivative contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases can be provided.

Abstract translation: 根据本发明的唑衍​​生物由式（I）表示，其中R a和R b各自表示氢原子或C 1 -C 6烷基，C 2 -C 6烯基或C 2 -C 6炔基; Ra和Rb可以被Xa或Xb取代，Xb或Xb是卤素原子; na和nb中的每一个表示0或Ra或Rb中的氢原子中的X a或X b取代的氢原子的数目; 每个Y表示卤素原子，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基，C1-C4卤代烷氧基，苯基，氰基或硝基; m表示0〜5; A表示氮原子或甲炔基。 结果，可以提供在对疾病具有优异控制作用的农业园艺剂中作为活性成分含有的唑衍生物。

公开(公告)号：US20140200352A1

公开(公告)日：2014-07-17

申请号：US14213043

申请日：2014-03-14

Applicant: KUREHA CORPORATION

Inventor： Nobuyuki ARAKI ,  Toru YAMAZAKI ,  Nobuyuki KUSANO ,  Eiyu IMAI ,  Hisashi KANNO ,  Masaru MORI ,  Taiji MIYAKE

IPC: A01N43/50 ,  A01N43/653 ,  A01N37/10

CPC classification number: C07C67/31 ,  A01N37/10 ,  A01N43/50 ,  A01N43/653 ,  C07C201/12 ,  C07C2601/08 ,  C07D405/06

Abstract: An azole derivative according to the invention is represented by Formula (I), wherein each of Ra and Rb denotes a hydrogen atom, or a C1-C6 alkyl group, a C2-C6 alkenyl group or a C2-C6 alkynyl group; Ra and Rb may be substituted with Xa or Xb which is a halogen atom; each of na and nb denotes 0 or the number of Xa- or Xb-substituted hydrogen atoms among the hydrogen atoms in Ra or Rb; each Y denotes a halogen atom, a C1-C4 alkyl group, a C1-C4 haloalkyl group, a C1-C4 alkoxy group, a C1-C4 haloalkoxy group, a phenyl group, a cyano group or a nitro group; m denotes 0 to 5; and A denotes a nitrogen atom or a methyne group.As a result, an azole derivative contained as an active ingredient in an agro-horticultural agent having an excellent controlling effect on diseases can be provided.