AMIDRAZONE COMPOUNDS FOR COMBATING ANIMAL PESTS
    3.
    发明申请
    AMIDRAZONE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    用于组合动物疫苗的咪唑啉酮化合物

    公开(公告)号:WO2006097279A8

    公开(公告)日:2007-05-18

    申请号:PCT/EP2006002331

    申请日:2006-03-14

    CPC classification number: C07C259/20 A01N37/52 C07C2601/02

    Abstract: The present invention relates to new amidrazone compounds which are useful for combating animal pests, in particular insects, arachnids and nematodes. The invention also relates to a method for combating insects, nematodes and arachnids. The amidrazone compounds are of the general formula (I) including the tautomers of I and the salts thereof; wherein X and Y are hydrogen or together form a chemical bond; Ar is an aromatic radical selected from phenyl and a 5- or 6-membered heteroaryl having 1 , 2, 3 or 4 heteroatoms as ring members, which are selected, independently of one another, from O, N and S, and where the aromatic radical may have 1 , 2, 3, 4 or 5 substituents R a ; R 1 is selected from the group consisiting of C 1 -C 1O -alkyl, C 1 -C 4 -alkoxy-C 1 -C 4 -alkyl, cyano-C 1 -C 4 -alkyl, hydroxy-C 1- C 4 -alkyl, C 1 -C 10 -haloalkyl, tri-(C 1 -C 4 -alkyl)-silyl-C 1 - C 4 -alkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, C 2 -C 10 -alkynyl, C 2 -C 10 -haloalkynyl, C 3 -C 10 -cycloalkyl, phenyl, heteroaryl, C 3 -C 10 -cycloalkyl-C 1 C 4 -alkyl, phenyl-C 1 -C 4 - alkyl and heteroaryl-C 1 C 4 alkyl, wherein C 3 -C 10 -cycloalkyl, heteroaryl and phenyl in the last six mentioned radicals may be unsubstituted or carry 1 , 2, 3, 4 or 5 substituents R b as defined above; R 2 is selected from the group consisiting of C 1- C 1 0-alkyl, c 1- c 4 -alkoxy- C 1- C 4 -alkyl, C 1- C 10 -haloalkyl, C 2 -C 10 -alkenyl, C 2 -C 10 -haloalkenyl, C 2 -C 10 -alkynyl, C 2 -C 10 - haloalkynyl,c 3 -C 10 -cycloalkyl, phenyl, heteroaryl, C 3 -C 10 -cycloalkyl-C 1- C 4 -alkyl, phenyl-C 1 -C 4 -alkyl and heteroaryI-C 1- C 4 -alkyl, wherein C 3 -C 10 -cycloalkyl, heteroaryl and phenyl in the last six mentioned radicals may be unsubstituted or carry 1 , 2, 3, 4 or 5 substituents R b as defined above.

    Abstract translation: 本发明涉及可用于对抗动物害虫,特别是昆虫,蜘蛛和线虫的新的氨基腙化合物。 本发明还涉及一种防治昆虫,线虫和蜘蛛的方法。 氨基腙化合物具有通式(I),其包括I的互变异构体及其盐; 其中X和Y是氢或一起形成化学键; Ar是选自苯基和具有1,2,3或4个杂原子作为环成员的5-或6-元杂芳基的芳族基团,其彼此独立地选自O,N和S,并且其中芳族 基团可以具有1,2,3,4或5个取代基R a, R 1选自C 1 -C 10 - 烷基,C 1 -C 1 - 烷基, C 1 -C 4烷基,C 1 -C 4烷基,C 1 -C 4烷基,氰基-C 1 -C 4烷基, C 1 -C 6烷基,羟基-C 1 -C 4 - 亚烷基,C 1 -C 10 - 烷基, 卤代烷基,三 - (C 1 -C 4 - 烷基) - 甲硅烷基-C 1 -C 4 - 烷基,C 2 -C 10 - 烯基,C 2 -C 10 - 卤代烯基,C 1 -C 10 - C 2 -C 10 - 炔基,C 2 -C 10 - 卤代炔基,C 3 - C 10 - 环烷基,苯基,杂芳基,C 3 -C 10 - 环烷基-C 1 -C C 1-4烷基,苯基-C 1 -C 4 - 烷基和杂芳基-C 1 -C 4烷基, 其中C 3 -C 10 - 环烷基,杂芳基和苯基在后面六个提及的基团中可以是未取代的或携带1,2,3,4或4个 5个取代基R b如上所定义; R 2选自C 1 -C 1-4烷基,C 1 -C 4烷基, C 1-4烷基,C 1 -C 10烷基,C 1 -C 4烷基,C 1〜 亚烷基,C 2 -C 10 - 烯基,C 2 -C 10 - 卤代烯基,C C 2 -C 10 - 炔基,C 2 -C 10 - 卤代炔基,C 3 - C 1 -C 10 - 环烷基,苯基,杂芳基,C 3 -C 10 - 环烷基-C 1 - C 1 -C 4 - 烷基,苯基-C 1 -C 4 - 烷基和杂芳基C 1 -C 其中C 3 -C 10 - 环烷基,最后六个所述基团中的杂芳基和苯基可以是未取代的或携带1, 2,3,4或5个如上定义的取代基R b。

    PROCESS FOR PREPARING AMIDRAZONES
    4.
    发明申请
    PROCESS FOR PREPARING AMIDRAZONES 审中-公开
    制备AMIDRAZONES的方法

    公开(公告)号:WO2008015133A3

    公开(公告)日:2008-03-20

    申请号:PCT/EP2007057645

    申请日:2007-07-25

    CPC classification number: C07C257/22 C07C233/58 C07C257/02 C07C2601/02

    Abstract: The present invention relates to a novel process for preparing amidrazones of the formula (I) wherein R, R 1 , R 2 , A, B, W, Y and n have the meanings as indicated in the description. Further, the invention relates to novel compounds used as intermediates in this process and to processes for their preparation.

    Abstract translation: 本发明涉及一种制备式(I)的氨基腙的新方法,其中R 1,R 2,R 2,A,B,W,Y和n具有 说明中指出的含义。 此外,本发明涉及在该方法中用作中间体的新化合物及其制备方法。

    NOVEL 2-CYANO-3-(HALO)ALKOXY-BENZENESULFONAMIDE COMPOUNDS FOR COMBATING ANIMAL PESTS
    6.
    发明申请
    NOVEL 2-CYANO-3-(HALO)ALKOXY-BENZENESULFONAMIDE COMPOUNDS FOR COMBATING ANIMAL PESTS 审中-公开
    新型2-氰基-3-(卤代)烷氧基苯磺酰胺化合物用于防治动物病虫害

    公开(公告)号:WO2006056433A2

    公开(公告)日:2006-06-01

    申请号:PCT/EP2005012561

    申请日:2005-11-24

    CPC classification number: C07C319/20 A01N41/06 C07C311/29 C07C323/62

    Abstract: The invention relates to 2-cyano-3-(halo)alkoxy-benzenesulfonamide compounds (I), where the variables Alk and R1 to R5 are as defined in claim 1, and/or to their agriculturally useful salts. Moreover, the present invention relates to: the use of compounds (I) and/or their salts for combating animal pests; agricultural compositions comprising such an amount of at least one compound of the general formula (I) and/or at least one agriculturally useful salt of (I) and at least one inert liquid and/or solid agronomically acceptable carrier that it has a pesticidal action and, if desired, at least one surfactant; and a method of combating animal pests which comprises contacting the animal pests, their habit, breeding ground, food supply, plant, seed, soil, area, material or environment in which the animal pests are growing or may grow, or the materials, plants, seeds, soils, surfaces or spaces to be protected from animal attack or infestation with a pesticidally effective amount of at least one2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the formula (I) and/or at least one agriculturally acceptable salt thereof; a method for the for the protection of seeds from soil insects and of the resulting plant's roots and shoots from soil and foliar insects comprising contacting the seeds before sowing and/or after pregermination with a 2-cyano-3-(halo)alkoxy-benzenesulfonamide compound of the general formula (I).

    Abstract translation: 本发明涉及2-氰基-3-(卤代)烷氧基 - 苯磺酰胺化合物(I),其中变量Alk和R1-R5如权利要求1中所定义,和/或其可农用盐。 此外,本发明涉及:化合物(I)和/或其盐用于对抗动物害虫的用途; 包含这种量的至少一种通式(I)的化合物和/或至少一种(I)的农业上有用的盐和至少一种惰性液体和/或固体农艺上可接受的载体的农业组合物,其具有杀虫作用 和如果需要的话,至少一种表面活性剂; 以及防治动物害虫的方法,其包括使动物害虫,其习性,繁殖场,食物供应,植物,种子,土壤,面积,动物害虫正在生长或可能生长的材料或环境,或材料,植物 (I)的至少一种2-氰基-3-(卤代)烷氧基 - 苯磺酰胺化合物和/或至少一种农业上受到保护的种子,土壤,表面或空间免于动物攻击或侵染 其可接受的盐; 一种用于保护种子免受土壤昆虫以及所得植物的根和茎由土壤和叶面昆虫引起的方法,包括在播种之前和/或在萌芽后使种子与2-氰基-3-(卤代)烷氧基 - 苯磺酰胺 通式(I)的化合物。

    THE USE OF N-ARYLHYDRAZINE DERIVATIVES FOR COMBATING PESTS IN AND ON ANIMALS
    9.
    发明申请
    THE USE OF N-ARYLHYDRAZINE DERIVATIVES FOR COMBATING PESTS IN AND ON ANIMALS 审中-公开
    使用N-芳基衍生物在动物体内和动物体内

    公开(公告)号:WO2005053402A3

    公开(公告)日:2005-08-04

    申请号:PCT/EP2004013685

    申请日:2004-12-02

    CPC classification number: A01N37/52

    Abstract: Use of compounds of formula (I) wherein Q is (II), (III), or (IV) ; X is chlorine, bromine, or fluorine; R , R are each independently H, alkyl, alkenyl, alkynyl, or cycloalkyl, alkylamino, dialkylamino, alkylcarbonylamino, alkylsulfonyl, or alkylsulfinyl, wherein the carbon atoms in these groups may be substituted, or R and R may be taken together to form a ring represented by the structure (V); p,m are 1, 2 or 3; X' is oxygen, sulfur, amino, alkylamino, phenylamino, or methylene; Z is alkyl or phenyl; R is H, alkyl, alkenyl, alkynyl, cycloalkyl, wherein the carbon atoms in these groups may be substituted; R, R are H or alkyl, alkoxycarbonyl, alkylaminocarbonyl, or dialkylaminocarbonyl, wherein the carbon atoms in the these groups may be substituted; A is C-R or N; B is C-R or N; W is C-R or N; with the proviso that one of A, B and W is other than N; R , R , R are H, halogen, nitro, cyano, amino, mercapto, hydroxy, alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkylamino, dialkylamino, alkylthio, alkylsulfonyl, or alkylsulfinyl, wherein the carbon atoms in these groups may be substituted, a 5- to 6-membered aromatic ringsystem which may contain 1 to 4 heteroatoms selected from oxygen, sulfur and nitrogen and which may be substituted; Y is hydrogen, halogen, cyano, nitro, amino, hydroxy, mercapto, alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkylamino, dialkylamino, alkylthio, alkylsulfonyl, or alkylsulfinyl, wherein the carbon atoms in these groups may be substituted; n is 0, 1, or 2; for combating parasites in and on animals.

    Abstract translation: 其中Q为(II),(III)或(IV)的式(I)化合物; X 1是氯,溴或氟; R 1,R 2各自独立地为H,烷基,烯基,炔基或环烷基,烷基氨基,二烷基氨基,烷基羰基氨基,烷基磺酰基或烷基亚磺酰基,其中这些基团中的碳原子可以被取代,或R 1, 和R 2可以一起形成由结构(Ⅴ)表示的环; p,m为1,2或3; X'是氧,硫,氨基,烷基氨基,苯基氨基或亚甲基; Z是烷基或苯基; R 3是H,烷基,烯基,炔基,环烷基,其中这些基团中的碳原子可以被取代; R 4是H或烷基,烷氧基羰基,烷基氨基羰基或二烷基氨基羰基,其中这些基团中的碳原子可以被取代; A为C-R 5或N; B是C-R 6或N; W是C-R 7或N; 条件是A,B和W之一不是N; R 5,R 6,R 7是H,卤素,硝基,氰基,氨基,巯基,羟基,烷基,烯基,炔基,环烷基,烷氧基,烷基氨基,二烷基氨基,烷硫基,烷基磺酰基或烷基亚磺酰基, 其中这些基团中的碳原子可以被取代,可以含有1至4个选自氧,硫和氮并且可以被取代的杂原子的5至6元芳族环系统; Y是氢,卤素,氰基,硝基,氨基,羟基,巯基,烷基,烯基,炔基,环烷基,烷氧基,烷基氨基,二烷基氨基,烷硫基,烷基磺酰基或烷基亚磺酰基,其中这些基团中的碳原子可以被取代; n为0,1或2; 用于对抗动物体内及其上的寄生虫。

    THE USE OF N-ARYLHYDRAZINE DERIVATIVES FOR COMBATING PESTS
    10.
    发明申请
    THE USE OF N-ARYLHYDRAZINE DERIVATIVES FOR COMBATING PESTS 审中-公开
    使用N-芳基衍生物来制备PES

    公开(公告)号:WO2005053403A2

    公开(公告)日:2005-06-16

    申请号:PCT/EP2004013687

    申请日:2004-12-02

    CPC classification number: A01N37/52

    Abstract: Use of hydrazine derivatives of formula (I) wherein W is chlorine or trifluoromethyl; X and Y are each independently chlorine or bromine; R is alkyl, alkenyl, alkynyl, or cycloalkyl which may be substituted with 1 to 3 halogen atoms, or alkyl which is substituted by alkoxy; R and R are alkyl or may be taken together to form cycloalkyl which may be unsubstituted or substituted by 1 to 3 halogen atoms; R is hydrogen or alkyl, or the enantiomers or salts thereof, for combating non-crop pests. Use of compounds of formula (I) for the protection of non-living organic materials and for the protection of animals against non-crop pests.

    Abstract translation: 式(I)的肼衍生物的用途,其中W是氯或三氟甲基; X和Y各自独立地为氯或溴; R 1是可以被1至3个卤素原子取代的烷基,烯基,炔基或环烷基,或被烷氧基取代的烷基; R 2和R 3是烷基或可以一起形成可被未取代或被1至3个卤素原子取代的环烷基; R 4是氢或烷基,或其对映异构体或盐,用于防治非作物害虫。 使用式(I)化合物用于保护非生物有机物质和保护动物免受非作物害虫的侵害。

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