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公开(公告)号:PL2663550T4
公开(公告)日:2017-07-31
申请号:PL12734770
申请日:2012-01-12
Applicant: VENTIRX PHARMACEUTICALS INC , ARRAY BIOPHARMA INC
Inventor: HOWBERT JAMES JEFFRY , HERSHBERG ROBERT , BURGESS LAURENCE E , YANG HONG WOON
IPC: C07D223/16 , A61K31/55 , A61P29/00 , A61P35/00 , C07D401/04 , C07D403/10 , C07D413/10 , C07D487/04
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公开(公告)号:HRP20170404T1
公开(公告)日:2017-05-19
申请号:HRP20170404
申请日:2017-03-10
Applicant: VENTIRX PHARMACEUTICALS INC , ARRAY BIOPHARMA INC
Inventor: HOWBERT JAMES JEFFRY , DIETSCH GREGORY , HERSHBERG ROBERT , BURGESS LAURENCE E , LYSSIKATOS JOSEPH P , NEWHOUSE BRAD , YANG HONG WOON
IPC: C07D401/14 , A61K31/4025 , A61K31/454 , A61K31/55 , A61P31/00 , A61P35/00 , C07D223/14 , C07D403/10
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公开(公告)号:HRP20170401T1
公开(公告)日:2017-05-19
申请号:HRP20170401
申请日:2017-03-10
Applicant: VENTIRX PHARMACEUTICALS INC , ARRAY BIOPHARMA INC
Inventor: HOWBERT JAMES JEFFRY , HERSHBERG ROBERT , BURGESS LAURENCE E , YANG HONG WOON
IPC: C07D223/16 , A61K31/55 , A61P29/00 , A61P35/00 , C07D401/04 , C07D403/10 , C07D413/10 , C07D487/04
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公开(公告)号:DK2663555T3
公开(公告)日:2017-03-27
申请号:DK12733896
申请日:2012-01-12
Applicant: VENTIRX PHARMACEUTICALS INC , ARRAY BIOPHARMA INC
Inventor: DOHERTY GEORGE A , LYSSIKATOS JOSEPH P , YANG HONG WOON , HOWBERT JAMES JEFFRY , HERSHBERG ROBERT , EARY CHARLES TODD , GRONEBERG ROBERT D , JONES ZACHARY , BURGESS LAURENCE E
IPC: A61K31/55 , A61P37/00 , C07D223/16 , C07D243/14 , C07D401/12 , C07D487/04
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公开(公告)号:DK2467380T3
公开(公告)日:2017-03-13
申请号:DK10810564
申请日:2010-08-18
Applicant: VENTIRX PHARMACEUTICALS INC , ARRAY BIOPHARMA INC
Inventor: HOWBERT JAMES JEFFRY , DIETSCH GREGORY , HERSHBERG ROBERT , BURGESS LAURENCE E , DOHERTY GEORGE A , EARY C TODD , GRONEBERG ROBERT D , JONES ZACHARY
IPC: C07D403/10 , A61K31/4025 , A61K31/55 , A61P31/00 , A61P35/00 , C07D223/14 , C07D401/14 , C07D403/14
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公开(公告)号:AU2010284240B2
公开(公告)日:2016-11-10
申请号:AU2010284240
申请日:2010-08-18
Applicant: ARRAY BIOPHARMA INC , VENTIRX PHARMACEUTICALS INC
Inventor: HOWBERT JAMES JEFFRY , DIETSCH GREGORY , HERSHBERG ROBERT , BURGESS LAURENCE E , LYSSIKATOS JOSEPH P , NEWHOUSE BRAD , YANG HONG WOON
IPC: C07D223/14 , A61K31/4025 , A61K31/454 , A61K31/55 , A61P31/00 , A61P35/00 , C07D401/14 , C07D403/10
Abstract: Provided are compositions and methods useful for modulation of signaling through the Toll-like receptors TLR7 and/or TLR8. The compositions and methods have use in treating or preventing disease, including cancer, autoimmune disease, infectious disease, inflammatory disorder, graft rejection, and graft-verses-host disease.
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公开(公告)号:CA2729217C
公开(公告)日:2016-09-06
申请号:CA2729217
申请日:2009-06-24
Applicant: ARRAY BIOPHARMA INC
Inventor: BURGESS LAURENCE E , CLARK CHRISTOPHER T , COOK ADAM , CORRETTE CHRISTOPHER P , DELISLE ROBERT KIRK , DOHERTY GEORGE A , HUNT KEVIN W , ROMOFF TODD , KIM GANGHYEOK
IPC: C07D311/04 , A61K31/353 , A61P29/00 , C07D405/12 , C07D407/12
Abstract: Compounds of Formula (I): in which A1, A2, W, L, G, R7a, R7b, R8, R9 and R10 have the meanings given in the specification, are DP2 receptor modulators useful in the treatment of immunologic diseases.
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公开(公告)号:UA109131C2
公开(公告)日:2015-07-27
申请号:UAA201212901
申请日:2011-04-11
Applicant: ARRAY BIOPHARMA INC
Inventor: BOYS MARK LAURENCE , BURGESS LAURENCE E , GRONEBERG ROBERT D , HARVEY DARREN M , HUANG LILY , KERCHER TIMOTHY , KRASER CHRISTOPHER F , LAIRD ELLEN , TARLTON EUGENE , ZHAO QIAN
IPC: C07D487/04 , A61K31/519 , A61P29/00 , A61P37/00
Abstract: СоединенияФормулы I: EMBED ISISServer , I иихстереоизомерыи фармацевтическиприемлемыесоли, исольваты, где R1, R2, R3, R4, R5, R6, R7, X1 и X2 имеютзначения, приведенныев описании, являетсяингибиторамиоднойилибольше JAK-кинази пригодныедлялеченияаутоиммунныхзаболеваний, воспалительныхзаболеваний, отторженияпересаженныхорганов, тканейи клеток, атакжегематологическихрасстройстви злокачественныхновообразований, исопутствующихзаболеваний.
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公开(公告)号:AU2015201991A1
公开(公告)日:2015-05-07
申请号:AU2015201991
申请日:2015-04-21
Applicant: ARRAY BIOPHARMA INC
Inventor: BOYS MARK LAURENCE , BURGESS LAURENCE E , GRONEBERG ROBERT D , HARVEY DARREN M , HUANG LILY , KERCHER TIMOTHY , KRASER CHRISTOPHER F , LAIRD ELLEN , TARLTON EUGENE , ZHAO QIAN
IPC: C07D487/04 , A61K31/519 , A61P29/00 , A61P37/00
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公开(公告)号:PH12014500079B1
公开(公告)日:2015-02-09
申请号:PH12014500079
申请日:2014-01-08
Applicant: ARRAY BIOPHARMA INC
Inventor: BURGESS LAURENCE E , CLARK CHRISTOPHER T , ADAM COOK , CORRETTE CHRISTOPHER P , KIRK DELISLE ROBERT , DOHERTY GEORGE A , HUNT KEVIN W , TODD ROMOFF , GANGHYEOK KIM
IPC: A61K31/353 , A61P29/00 , C07D311/04 , C07D405/12 , C07D407/12
Abstract: Compounds of Formula (I): in which A1, A2, W, L, G, R7a, R7b, R8, R9 and R10 have the meanings given in the specification, are DP2 receptor modulators useful in the treatment of immunologic diseases.
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