-
公开(公告)号:ZA991738B
公开(公告)日:2000-10-11
申请号:ZA991738
申请日:1999-03-04
Applicant: BASF AG
Inventor: AMBERG WILHELM , KLINGE ROLF JANSEN DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: C07D251/22 , A61K31/192 , A61K31/216 , A61K31/505 , A61K31/506 , A61K31/519 , A61K31/53 , A61P9/04 , A61P9/06 , A61P9/10 , A61P9/12 , A61P11/06 , A61P13/08 , A61P13/12 , A61P35/00 , A61P43/00 , C07C59/66 , C07C59/68 , C07C69/734 , C07D213/63 , C07D239/34 , C07D239/52 , C07D239/60 , C07D405/12 , C07D491/048 , C07D , A61K
Abstract: The invention relates to carboxylic acid derivatives of formula (I), wherein R -R , Q, W, X, Y and Z have the meanings given in the description. The novel compounds are suitable for combating diseases.
-
公开(公告)号:CZ20001582A3
公开(公告)日:2000-10-11
申请号:CZ20001582
申请日:1998-10-16
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: A61K31/495 , A61P9/00 , C07D239/00
-
公开(公告)号:BR9814951A
公开(公告)日:2000-10-03
申请号:BR9814951
申请日:1998-10-16
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: A61K31/505 , A61K31/506 , A61K31/517 , A61K31/519 , A61K31/5377 , A61P9/02 , A61P9/10 , A61P9/12 , A61P13/08 , A61P13/12 , A61P35/00 , A61P43/00 , C07D239/34 , C07D239/36 , C07D239/52 , C07D239/60 , C07D239/70 , C07D401/12 , C07D403/12 , C07D491/048 , C07D239/00
Abstract: The invention relates to carboxylic acid derivatives of formula (I), wherein the substituents have the meaning as commented in the description. It also relates to the production and use of same as endothelin receptor antagonists.
-
公开(公告)号:TR200001365T2
公开(公告)日:2000-09-21
申请号:TR200001365
申请日:1998-11-04
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , HILLEN HEINZ , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: C07D249/12 , A61K31/41 , A61K31/415 , A61K31/4164 , A61K31/42 , A61K31/421 , A61K31/422 , A61K31/4245 , A61K31/425 , A61K31/426 , A61K31/427 , A61K31/428 , A61K31/433 , A61P9/04 , A61P9/08 , A61P9/10 , A61P9/12 , A61P11/06 , A61P13/08 , A61P13/12 , A61P35/00 , A61P43/00 , C07D231/20 , C07D233/70 , C07D261/12 , C07D263/38 , C07D271/06 , C07D271/10 , C07D273/01 , C07D275/02 , C07D275/03 , C07D277/20 , C07D277/32 , C07D277/34 , C07D277/60 , C07D277/68 , C07D285/00 , C07D285/08 , C07D285/12 , C07D291/04 , C07D413/12 , C07D417/12
Abstract: The present invention relates to carboxylic acid derivatives of the formula Ithe substituents having the meanings explained in the description, preparation and use as endothelin receptor antagonists.
-
135.
公开(公告)号:ZA9901214B
公开(公告)日:2000-08-16
申请号:ZA9901214
申请日:1999-02-16
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , KLING ANDREAS , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASHACK MANFRED , UNGER LILIAN
IPC: A61K31/505 , A61K31/506 , A61P5/14 , A61P9/02 , A61P9/10 , A61P9/12 , A61P11/06 , A61P13/12 , A61P35/00 , A61P43/00 , C07D239/34 , C07D239/46 , C07D239/52 , C07D239/60 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D417/12 , C07D , A62K
CPC classification number: C07D239/47 , C07D239/60 , C07D403/12
-
136.
公开(公告)号:CZ20001788A3
公开(公告)日:2000-08-16
申请号:CZ20001788
申请日:1998-11-04
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , HILLEN HEINZ , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: A61K31/42 , A61K31/425 , A61P9/00 , A61P11/06 , A61P13/00 , C07D261/12 , C07D263/38 , C07D275/03 , C07D277/34 , C07D413/12 , C07D417/12
-
公开(公告)号:CZ20001326A3
公开(公告)日:2000-08-16
申请号:CZ20001326
申请日:1998-09-18
Applicant: BASF AG
Inventor: PUHL MICHAEL , ZECHEL JOHANN-CHRISTIAN , DITRICH KLAUS , HILLEN HEINZ , KOHL TANJA , ERHARDT MELANIE , HERGENROEDER STEFAN , MARKERT CLAUS OTTO
IPC: A61K31/381 , A61K31/47 , A61K31/498 , A61P9/00 , A61P9/12 , C07C271/22 , C07C321/06 , C07D215/48 , C07D241/44 , C07D333/24
-
公开(公告)号:NO20004075A
公开(公告)日:2000-08-15
申请号:NO20004075
申请日:2000-08-15
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , KLING ANDREAS , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: A61K31/505 , A61K31/506 , A61P5/14 , A61P9/02 , A61P9/10 , A61P9/12 , A61P11/06 , A61P13/12 , A61P35/00 , A61P43/00 , C07D239/34 , C07D239/46 , C07D239/52 , C07D239/60 , C07D401/12 , C07D403/12 , C07D405/12 , C07D409/12 , C07D417/12
CPC classification number: C07D239/47 , C07D239/60 , C07D403/12
-
公开(公告)号:TR199903159T2
公开(公告)日:2000-07-21
申请号:TR9903159
申请日:1998-06-05
Applicant: BASF AG
Inventor: AMBERG WILHELM , KLING ANDREAS , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: C07D251/16 , A61K31/4965 , A61K31/50 , A61K31/505 , A61K31/517 , A61K31/519 , A61K31/53 , A61P7/02 , A61P9/02 , A61P9/04 , A61P9/10 , A61P9/12 , A61P11/06 , A61P13/08 , A61P13/12 , A61P25/06 , A61P35/00 , A61P35/04 , A61P43/00 , C07C247/12 , C07D213/68 , C07D237/14 , C07D237/16 , C07D239/34 , C07D239/52 , C07D239/56 , C07D239/60 , C07D239/70 , C07D239/80 , C07D239/95 , C07D241/18 , C07D251/22 , C07D251/34 , C07D251/52 , C07D253/06 , C07D403/12 , C07D491/048
Abstract: The invention relates to carboxylic acid derivatives of formula (I) wherein the constituents have the meaning given in the description. The invention also relates to the production of said derivatives, and to their use as endothelin receptor antagonists.
-
公开(公告)号:CZ2000743A3
公开(公告)日:2000-06-14
申请号:CZ2000743
申请日:1998-08-24
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: A61K31/505 , A61P9/10 , A61P9/12 , C07D239/04 , C07D263/38 , C07D277/34
-
-
-
-
-
-
-
-
-