Abstract:
Disclosed are herbicides containing at least one 3-aminobenzo[b]thiophene (I) with an antagonistic action (in which R1 = -COX or -COOX; X = H, halogen, optionally substituted amino, optionally substituted C¿1?-C10 alkyl, optionally sustituted C1-C8 alkenyl, optionally substituted C3-C10 cycloalkyl, optionally substituted C3-C10 cycloalkenyl, a 5/6-membered heterocyclic aromatic, optionally substituted phenyl or optionally substituted naphthyl; R?2 and R3¿ = H, CN, NO¿2?, SH, halogen, optionally substituted amino, optionally substituted C1-C10 alkyl, optionally substituted C1-C6 alkoxy, optionally substituted C2-C8 alkenyl, optionally substituted C3-C10 cycloalkyl, optionally substituted C3-C10 cycloalkenyl, optionally substituted phenyl, optionally substituted naphthyl or a 5/6-membered heterocyclic aromatic; R?4 to R7¿ = H, optionally substituted C¿1?-C10 alkyl, optionally substituted C2-C8 alkenyl, optionally substituted C3-C10 cycloalkyl, optionally substituted C3-C10 cycloalkenyl, an optionally substituted 5/6-membered heterocyclic aromatic, optionally substituted phenyl or optionally substituted naphthyl or R?4 + R5¿ and/or R6 + R7 form, together with the N-atom to which they are bound, a 5- to 7-membered ring), plus the basic salts of those compounds of formula (I) which carry at least one carboxyl, hydroxythiocarbonyl or sulphonic acid group and the acid salts of those compounds of formula (I) which contain a basic nitrogen atom, and at least one herbicidal substance selected (A) from the group comprising the cyclohexenone derivatives or (B) from the group comprising the 4-(hetero)aryloxyphenoxyacetic acid derivatives.
Abstract:
The invention relates to a method for producing isoxazolene of the formula (1), where the substituents have the following meanings: R1 is hydrogen, C1-C6 alkyl, R2 is C1-C6 alkyl, R3, R4, R5 are hydrogen, C1-C6 alkyl or R4 and R5 together form a linkage, R6 is a heterocyclic ring, and n is 0, 1 or 2. Said method comprises the production of an intermediate compound of the formula (VI) where R1, R3, R4 and R5 have the meanings given above. This step is followed by halogenation, thiomethylation, oxidation and acylation to yield compounds of formula (I). The invention also relates to new intermediate products for producing compounds of formula (I) and new methods for producing the intermediate products.
Abstract:
Изобретениеотноситсяк способуполучениясоединенийформулы XVгдеостаткиимеютследующеезначение: X - NO, S(O)Ry; Rx, Ry независимодруготдругаозначаютгалоген, карбоксил, карбоксамид, N-алкилкарбоксамид, N,N-диалкилкарбоксамид, фенил, C-Cалкил, C-Cалкокси, C-Cалкилтио; m равно 0, 1, 2, 3 или 4; n равно 0, 1 или 2. Изобретениеотноситсятакжек новомусоединениюформулы XV ик применениюспособаполучениясоединенияформулы XV.
Abstract:
The present invention describes a process for preparing isoxazoles of the formula Iwhere:R is hydrogen, C1-C6-alkyl,R is hydrogen, C1-C6-alkyl,R , R , R are each hydrogen, C1-C6-alkyl or R and R together form a bond,R is a heterocyclic ring,n is 0, 1 or 2;which comprises preparing an intermediate of the formula VIwhere R , R , R and R are each as defined above, followed by halogenation, thiomethylation, oxidation and acylation to give compounds of the formula I.Furthermore, the invention describes novel intermediates for preparing the compounds of the formula I and novel processes for preparing the intermediates.
Abstract:
The invention relates to a method for producing isoxazolene of the formula (I): (See formula I) where the substituents have the following meanings: R1 is hydrogen, C1-C6 alkyl, R2 is C1-C6 alkyl, R3, R4, R5 are hydrogen, C1-C6 alkyl or R4 and R5 togethe r form a linkage, R6 is a heterocyclic ring, and n is 0, 1 or 2. Said method comprises the production of an intermediate compound of the formula (VI): (See formula VI) where R1, R3, R4 and R5 have the meanings given above. This step is followed by halogenation, thiomethylation, oxidation and acylation to yield compounds of formula (I). The invention also relates to new intermediate products for producing compounds of formula (I) and new methods for producing the intermediate products.