公开(公告)号：WO2007063028A3

公开(公告)日：2007-08-23

申请号：PCT/EP2006068832

申请日：2006-11-23

Applicant: BASF AG ,  SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  RACK MICHAEL ,  MAYER GUIDO ,  PLESCHKE AXEL

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  RACK MICHAEL ,  MAYER GUIDO ,  PLESCHKE AXEL

IPC: C07C303/38 ,  C07C201/12 ,  C07C205/58 ,  C07C303/40 ,  C07C311/51

CPC classification number: C07C303/38 ,  C07C201/12 ,  C07C303/40 ,  C07C311/51 ,  C07C205/58

Abstract: The invention relates to methods for producing sulfonamides of formula I, wherein the variables have the designations cited in the description, by reacting m-nitro-benzoic acid chlorides of formula II with aminosulfons of formula III, under the influence of B equivalents of base IV. Said method is characterised in that, during step a) the aminosulfon of formula III is reacted with B1 equivalents of base IV, and during step b), the reaction mixture resulting from step a) is reacted with m-nitro-benzoic acid chlorides of formula II and B2 equivalents of base IV; B, B1 and B2 having the designations cited in the description.

Abstract translation: 一种用于磺酰胺的制备（I）其中各变量具有说明书中给出的含义，由间硝基 - 苯甲酰氯II与aminosulfones III的反应中，碱IV的乙等同物的影响下，其特征在于在步骤a工艺）包括一 氨基砜III用碱IV的B1当量反应，和在步骤b），其从步骤a）的反应混合物结果与间 - 硝基 - 苯甲酰氯Ⅱ和的碱IV发生反应B2当量; 其中B，B1和B2具有说明书中给出的含义。

公开(公告)号：WO2008043835A2

公开(公告)日：2008-04-17

申请号：PCT/EP2007060879

申请日：2007-10-12

Applicant: BASF AG ,  SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  ERK PETER ,  SAXELL HEIDI EMILIA ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  MAYER GUIDO ,  WOLF BERND ,  COX GERHARD ,  MICHEL ALFRED ,  ZAGAR CYRILL ,  REINHARD ROBERT ,  SIEVERNICH BERND

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  ERK PETER ,  SAXELL HEIDI EMILIA ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  MAYER GUIDO ,  WOLF BERND ,  COX GERHARD ,  MICHEL ALFRED ,  ZAGAR CYRILL ,  REINHARD ROBERT ,  SIEVERNICH BERND

CPC classification number: C07D239/54

Abstract: The present invention relates to a crystalline form of 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethyl)-1-(2H)-pyrimidinyl]-4-fluoro-N-[[methyl-(1-methylethyl)amino]sulphonyl]benzamide. The invention also relates to a method for preparing this crystalline form and to formulations for crop protection which comprise this crystalline form of the phenyluracil.

Abstract translation: 本发明涉及2-氯-5- [3,6-二氢-3-甲基-2,6-二氧-4-（三氟甲基）-1（2H） - 嘧啶基] -4-氟的结晶形式 N - [[甲基 - （1-甲基乙基）氨基]磺酰基]苯甲酰胺。 本发明还涉及一种用于该结晶形式的制备以及制剂，其包含苯基尿嘧啶的该晶形的作物保护的方法。

公开(公告)号：CA2574406C

公开(公告)日：2013-02-19

申请号：CA2574406

申请日：2005-07-13

Applicant: BASF AG

Inventor： LOEHR SANDRA ,  GEBHARDT JOACHIM ,  MAYER GUIDO ,  KEIL MICHAEL ,  SCHMIDT THOMAS ,  WOLF BERND

IPC: C07D239/54 ,  C07C307/06

Abstract: The invention relates to a method for the production of 3-phenyl(thio)uracils and dithiouracils of formula I, wherein the variables have the meanings cited in the description, characterized in that carbamates of formula II, wherein variables X1, X3, Ar and A have the above-mentioned meanings and L1 represents a nucleophilically displaceable nucleofuge, can be reacted with enamines of formula III, wherein variables X2, R1, R2 and R3 have the above-mentioned meanings and L2 represents a nucleophilically displaceable nucleofuge. The invention also relates to intermediate products for the production thereof.

公开(公告)号：CA2652071C

公开(公告)日：2012-01-17

申请号：CA2652071

申请日：1999-05-04

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  VON DEYN WOLFGANG ,  GEBHARDT JOACHIM ,  RACK MICHAEL ,  LOCHTMAN RENE ,  GOETZ NORBERT ,  KEIL MICHAEL ,  WITSCHEL MATTHIAS ,  HAGEN HELMUT ,  MISSLITZ ULF ,  BAUMANN ERNST

IPC: C07C251/48 ,  C07C20060101 ,  C07C201/12 ,  C07C205/44 ,  C07C249/06 ,  C07C251/52 ,  C07C253/00 ,  C07C255/50 ,  C07C315/04 ,  C07C317/32 ,  C07C317/36 ,  C07C319/14 ,  C07C319/20 ,  C07C321/28 ,  C07C323/09 ,  C07D20060101 ,  C07D261/02 ,  C07D261/04 ,  C07D261/08 ,  C07D413/02 ,  C07D413/10

Abstract: The invention relates to a compound of the formula III: (see formula III) where R1 is C1-C6-alkyl. It also relates to a process for preparing compounds of the formula XV: (see formula XV) wherein: X is S(O)n Ry, R1 is C1-C6-alkyl, halogen, C1-C6-alkoxy or C1-C6-alkylthio, R X is halogen, carboxamide, N-alkyl-carboxamide, N,Ndialkylcarboxamide, phenyl, C1-C6-alkyl, C1-C6 alkoxy or C1-C6-alkylthio, R y is C1-C6-alkyl, m is 1, and n is 0, 1 or 2.

公开(公告)号：PL209931B1

公开(公告)日：2011-11-30

申请号：PL34433299

申请日：1999-05-04

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  VON DEYN WOLFGANG ,  GEBHARDT JOACHIM ,  RACK MICHAEL ,  LOCHTMAN RENE ,  GOETZ NORBERT ,  KEIL MICHAEL ,  WITSCHEL MATTHIAS ,  HAGEN HELMUT ,  MISSLITZ ULF ,  BAUMANN ERNST

IPC: C07D261/04 ,  C07C20060101 ,  C07C201/12 ,  C07C205/44 ,  C07C249/06 ,  C07C251/48 ,  C07C251/52 ,  C07C253/00 ,  C07C255/50 ,  C07C317/32 ,  C07C319/14 ,  C07C323/09 ,  C07D20060101 ,  C07D261/02 ,  C07D261/08 ,  C07D413/02 ,  C07D413/10

公开(公告)号：NO327975B1

公开(公告)日：2009-11-02

申请号：NO20030212

申请日：2003-01-16

Applicant: BASF AG

Inventor： KEIL MICHAEL ,  RACK MICHAEL ,  GEBHARDT JOACHIM ,  LOCHTMAN RENE ,  DEYN WOLFGANG VON

IPC: C07B61/00 ,  C07C319/14 ,  C07C323/62 ,  C07D261/04 ,  C07D413/04

Abstract: A process for preparing 4-thioalkylbromobenzene derivatives of the formula I where: R 1 is C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, C 1 -C 6 -alkoxy, C 1 -C 6 -haloalkoxy, C 3 -C 8 -cycloalkyl, halogen, R 2 is C 1 -C 6 -alkyl, C 1 -C 6 -alkoxy, C 3 -C 8 -cycloalkyl, C 2 -C 6 -alkenyl, cyano or a heterocyclic radical, R 3 is C 1 -C 6 -alkyl, which comprises reacting a compound of the formula II, in which R 1 and R 2 are as defined above, with a dialkyl disulfide of the formula III R 3 -S-S-R 3 III in the presence of a nitrite and a catalyst in a suitable solvent is described.

公开(公告)号：UA88377C2

公开(公告)日：2009-10-12

申请号：UAA200713919

申请日：2006-05-18

Applicant: BASF AG

Inventor： GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  SCHMIDT THOMAS ,  WEVERS JAN HENDRIK ,  ZECH HELMUT ,  HAEBERLE RUDOLF

IPC: C07D239/54

Abstract: Данноеизобретениекасаетсяспособаполучения 1-алкил-3-фенилурациловформулыІ, Iгдепеременныеот Rдо Rимеютзначения, приведенныев описании, прикоторых 3-фенилурацилыформулы IIIIиалкилировочныйагентформулы IIIR-LIIIподвергаютвзаимодействиюдругс другом, причемнапротяженииобщеговзаимодействиярН-значенияблагодаряпорционномудобавлениюосновысохраняютв пределахот 1 до 6.

公开(公告)号：SK286986B6

公开(公告)日：2009-08-06

申请号：SK462003

申请日：2001-07-17

Applicant: BASF AG

Inventor： LOCHTMAN RENE ,  KEIL MICHAEL ,  GEBHARDT JOACHIM ,  RACK MICHAEL ,  VON DEYN WOLFGANG

IPC: C07C251/00 ,  C07B61/00 ,  C07C319/00 ,  C07C319/14 ,  C07C323/62 ,  C07D261/00 ,  C07D261/04 ,  C07D413/00 ,  C07D413/04

Abstract: The invention relates a process for preparing 4-thioalkylbromobenzene derivtaes of the formula (I) where R1 is C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6haloalkoxy, C3-C8-cykloalkyl, halogen, R2 is C1-C6-alkyl, C1-C6-alkoxy, C3-C8-cykloalkyl, C2-C6-alkenyl, cyano or a heterocyclic radical, R3is C1-C6 alkyl, which comprises reacting a compound of the formula (II), in which R1 and R2 are as defined above, with dialkyl disulfide of the formula (III), in the presence of a nitrite and catalyst in a suitable solvent and molar ratio of catalyst and compound of the formula (II) is 0.005 : 1 to 0.05 : 1.

公开(公告)号：EA012035B1

公开(公告)日：2009-06-30

申请号：EA200700289

申请日：2005-07-13

Applicant: BASF AG

Inventor： LOHR SANDRA ,  GEBHARDT JOACHIM ,  MAYER GUIDO ,  KEIL MICHAEL ,  SCHMIDT THOMAS ,  WOLF BERND

IPC: C07D239/54 ,  C07C307/06

Abstract: Настоящееизобретениекасаетсяспособаполучения 3-фенилурациловформулы Iгдезначениякаждогоиззаместителейприведеныв описании, итакжепромежуточныхпродуктовдляихполучения.

公开(公告)号：ES2288021T3

公开(公告)日：2007-12-16

申请号：ES99922160

申请日：1999-05-04

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  VON DEYN WOLFGANG ,  GEBHARDT JOACHIM ,  RACK MICHAEL ,  LOCHTMAN RENE ,  GOTZ NORBERT

IPC: C07D261/04 ,  C07C20060101 ,  C07C201/12 ,  C07C205/44 ,  C07C249/06 ,  C07C251/40 ,  C07C251/48 ,  C07C251/52 ,  C07C253/00 ,  C07C255/50 ,  C07C317/32 ,  C07C319/14 ,  C07C323/09 ,  C07D20060101 ,  C07D261/02 ,  C07D261/08 ,  C07D413/02 ,  C07D413/10

Abstract: Un proceso de preparación de los isoxazoles de la fórmula I donde los sustituyentes son como se definen abajo: R1 es un hidrógeno, alquilo C1-C6, R2 es un alquilo C1-C6, R3, R4, R5 son hidrógeno, alquilo C1-C6, o R4 y R5 juntos forman un enlace, R6 es un anillo heterocíclico, n es 0, 1 o 2; que comprende la preparación de un intermediario de la fórmula VI donde R1, R3, R4 y R5 son como se definieron arriba.