公开(公告)号：EP0775124B1

公开(公告)日：2001-09-19

申请号：EP95928489.4

申请日：1995-07-29

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： PLATH, Peter ,  RANG, Harald ,  WESTPHALEN, Karl-Otto ,  GERBER, Matthias ,  WALTER, Helmut

IPC: C07D275/06 ,  A01N43/80 ,  C07B41/08

CPC classification number: C07D275/06 ,  A01N43/80

Abstract: The invention pertains to novel herbicidally effective saccharin carboxylic acids or carboxylic acid esters of formula (Ia), in which the substituents are as follows: L, M are hydrogen, C1-C4 alkyl, C1-C4 alkoxy C1-C4 alkylthio, chlorine, cyano, methyl sulfonyl, nitro or trifluoromethyl; Z is hydrogen, C1-C4 alkyl, C3-C8 cycloalkyl, benzyl or phenyl, where the penyl rings can in each case be substituted by C1-C4 alkyl, and R is H, C1-C6 alkyl, with the proviso that if L and M are hydrogen, Z is not methyl, phenyl hydrogen or an alkali metal cation or silver cation, and also excepting 5-carboxy-7-methyl saccharin and 5-carboxy-4-chlorosaccharin.

公开(公告)号：EP0888343A1

公开(公告)日：1999-01-07

申请号：EP97903334.0

申请日：1997-02-20

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： OTTEN, Martina ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  VOSSEN, Marcus ,  PLATH, Peter ,  GÖTZ, Norbert ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut ,  MISSLITZ, Ulf

IPC: A01N43 ,  C07D409 ,  C07D411

CPC classification number: C07D409/06 ,  A01N43/56 ,  C07D411/06

Abstract: The invention concerns pyrazolylhetaroyl derivatives of formula (I) in which the substituents have the following meanings: L, M are hydrogen, C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkinyl, C1-C4 alkoxy, wherein these groups can optionally be substituted by between one and five halogen atoms or C1-C4 alkoxy; halogen, cyano, nitro; X is oxygen or sulphur which can be substituted by one or two oxygens; n is zero, one, two; and Q, R?1, R2, R3, R4¿ have the meanings given in claim 1. The invention further concerns a process for preparing the pyrazole-4-yl-hetaroyl derivatives, agents containing the latter, and the use of these derivatives or agents containing them for weed control.

公开(公告)号：EP0888334A1

公开(公告)日：1999-01-07

申请号：EP97906099.0

申请日：1997-02-20

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： OTTEN, Martina ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  VOSSEN, Marcus ,  PLATH, Peter ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: A01N43 ,  C07D327 ,  C07D339 ,  C07D407 ,  C07D411

CPC classification number: A01N43/32 ,  C07D327/06 ,  C07D339/08

Abstract: The invention concerns hetaroyl derivatives of formula (I) in which the substituents have the following meanings: L, M are hydrogen, C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkinyl, C1-C4 alkoxy, wherein these groups can optionally be substituted by between one and five halogen atoms or C1-C4 alkoxy; halogen, cyano, nitro; X is oxygen or sulphur which can be substituted by one or two oxygens; n is zero, one, two; and Q, R?1, R2, R3, R4¿ have the meanings given in claim 1. The invention further concerns a process for preparing the hetaroyl derivatives, agents containing the latter, and the use of these derivatives or agents containing them for weed control.

Abstract translation: 本发明涉及式（I）的丁二酰衍生物，其中取代基具有以下含义：L，M为氢，C 1 -C 6烷基，C 2 -C 6烯基，C 2 -C 6炔基，C 1 -C 4烷氧基，其中这些基团可任选地 被一个和五个卤素原子或C1-C4烷氧基取代; 卤素，氰基，硝基; X是可被一个或两个氧原子取代的氧或硫; n是零，一，二; 和Q，R 1，R 2，R 3，R 4具有权利要求1中给出的含义。本发明进一步涉及制备杂芳酰基衍生物的方法，含有后者的药剂，以及这些衍生物或含有它们的药剂用于杂草 控制。

公开(公告)号：EP0788479A1

公开(公告)日：1997-08-13

申请号：EP95936508.0

申请日：1995-10-17

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： HEISTRACHER, Elisabeth ,  PLATH, Peter ,  VON DEM BUSSCHE-HÜNNEFELD, Christoph-Sweder ,  HAMPRECHT, Gerhard ,  KLINTZ, Ralf ,  SCHÄFER, Peter ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut ,  GERBER, Matthias ,  MISSLITZ, Ulf

IPC: C07D403 ,  A01N37 ,  A01N43 ,  C07C205 ,  C07C229 ,  C07D209 ,  C07D417 ,  C07F7

CPC classification number: C07D209/48 ,  A01N37/46 ,  C07C205/56 ,  C07C229/44 ,  C07F7/0812

Abstract: Disclosed are substituted phthalimido-cinnamic acid derivatives of formula (I), wherein R1 is H, C¿1?-C4-alkyl; R?2¿ is H, halogen; R3 is CN, NO¿2?, halogen, C1-C6-alkyl, C1-C6-alkyl halide, C1-C6-alkoxy, C1-C6-alkoxy halide; R?4¿ is H, CN, NO¿2?, halogen, C1-C6-alkyl; R?5¿ is H, C¿1?-C6-alkyl, C2-C6-alkenyl, C2-C6-alkinyl, substituted C1-C6-alkyl; R?6¿ is one of the radicals indicated under R5 or CN, NO¿2?, C1-C6-alkoxy, C1-C6-alkoxy halide, C1-C6-alkyl thio, C1-C6 alkyl thio halide, C3-C6-cycloalkyl, sustituted alkyl, C3-C6-alkenyl halide, (C1-C6-alkoxy)-carbonyl, COOH, (C1-C6-alkyl amino)carbonyl, di-(C1-C6-alkyl)amino carbonyl, (C1-C6-alkyl) carbonyl, (C1-C6-alkyl halide) carbonyl, optionally substituted aryl, hetaryl, aryl C1-C6 alkyl or hetaryl C1-C6 alkyl; or R?5 and R6¿ together are an alkylene chain, in which a methylene unit can be substituted a C¿1?-C4-alkyl imino group; R?7¿ is H, C¿1?-C6-alkyl, C3-C6-alkenyl, C3-C6 alkinyl, C2-C6 alkyl halide, C1-C6 cyanoalkyl, C1-C6 alkoxy C2-C6 alkyl, C1-C6-alkyl thio C2-C6 alkyl, (C1-C6-alkoxy)carbonyl-C1-C6-alkyl, optionally substituted phenyl or benzyl; X is O, S or N(R?8¿), as well as the salts of formula (I). Disclose also is their use as herbicides and for desication/defoliation of plants.

公开(公告)号：EP0775136A1

公开(公告)日：1997-05-28

申请号：EP95927734.0

申请日：1995-07-27

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： PLATH, Peter ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  KARDORFF, Uwe ,  KÖNIG, Hartmann ,  RANG, Harald ,  GERBER, Matthias ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto

IPC: A01N43 ,  A01P13 ,  C07D417

CPC classification number: C07D417/06 ,  A01N43/80

Abstract: The disclosure is of 5-hydroxypyrazol-4-yl-carbonyl-substituted saccharin derivatives of formula (I), in which the substituents have the following meanings: L,M stand for hydrogen, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 alkylthio, chlorine, cyano, methylsulphonyl, nitro or trifluoromethyl; Z stands for hydrogen, C1-C4 alkyl, C3-C8 cycloalkyl, C3-C6-alkenyl, C3-C5-alkinyl, C1-C4 acyl, benzyl or phenyl (the phenyl rings optionally being each substituted by a halogen or C1-C4 alkyl); Q stands for a CO-J group; J stands for a 5-hydroxypyrazol ring linked at position 4 and of formula (II), in which R1 represents C¿1?-C4 alkyl, and R?2¿ represents hydrogen or methyl. Also disclosed are the salts of formula (I) compounds commonly used in agriculture.

公开(公告)号：EP0775125A1

公开(公告)日：1997-05-28

申请号：EP95929016.0

申请日：1995-07-27

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： PLATH, Peter ,  VON DEYN, Wolfgang ,  ENGEL, Stefan ,  KARDORFF, Uwe ,  NÜBLING, Christoph ,  KÖNIG, Hartmann ,  RANG, Harald ,  GERBER, Matthias ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto

IPC: C07D275 ,  A01N43

CPC classification number: C07D275/06 ,  A01N43/80

Abstract: The invention concerns saccharine derivatives of the formula (I) in which the substituents are defined as follows: L, M hydrogen, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 alkylthio, chlorine, cyano, methylsulphonyl, nitro or trifluoromethyl; Z hydrogen, C1-C4 alkyl, C3-C8 cycloalkyl, C3-C6 alkenyl, C3-C5 alkinyl, C1-C4 acyl, benzyl or phenyl, wherein any of the phenyl rings may be substituted by halogen or C1-C4 alkyl; R1 cyclopropyl, 1-methylcyclopropyl, 1-methylthiocyclopropyl or tert.-butyl. The invention also concerns salts of such compounds usually used in agriculture.

公开(公告)号：EP0680481A1

公开(公告)日：1995-11-08

申请号：EP94905039.0

申请日：1994-01-12

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： PLATH, Peter ,  RENTZEA, Costin ,  MEYER, Norbert ,  KAST, Juergen ,  KARDORFF, Uwe ,  GERBER, Matthias ,  WALTER, Helmut ,  LANDES, Andreas ,  WESTPHALEN, Karl-Otto

IPC: A01N43 ,  C07D221 ,  C07D491

CPC classification number: C07D491/04 ,  A01N43/42 ,  A01N43/90 ,  C07D221/08

Abstract: A process is disclosed for controlling undesirable plant growth and for regulating plant growth, by applying to the plants derivatives of azaanthraquinones and/or azaxanthones having formula (I), in which X, Y, Z and the residues R1 to R5 have the following meanings: R1 is hydrogen, methyl; R2-R5 are (a) hydrogen, (b) halogen, (c) nitro, (d) COOR6, in which R6 stands for C¿1?-C4-alkyl, (e) CONH2 and CONR?6R7¿, in which R?6 and R7¿ stand for C¿1?-C4-alkyl, (f) C1-C8-alkyl, which may bear one to three of the following substituents: halogen, hydroxy, C1-C6-alkoxy, (g) C3-C6-alkenyl, (h) C1-C4-alkoxy, (i) hydroxy, (j) amino or NR?6R7¿, (k) phenyl, which may bear one to five halogen atoms or one to three of the following substituents: nitro, C¿1?-C4-alkoxy, C1-C4-alkyl or C1-C4alkyl halide; X, Y are N, N?+-O-¿ or CH, with the proviso that only a nitrogen atom or a N-oxide group be contained in the ring; Z is oxygen, sulphur or a C = O group; A is oxygen or sulphur. Also disclosed are new azaanthraquinones and azaxanthones and herbicidal and bioregulatory agents containing the same.

公开(公告)号：EP1716120A1

公开(公告)日：2006-11-02

申请号：EP04803998.6

申请日：2004-12-17

Applicant: BASF Aktiengesellschaft

Inventor： WITSCHEL, Matthias ,  PUHL, Michael ,  RACK, Michael ,  PARRA RAPADO, Liliana ,  MISSLITZ, Ulf ,  ZAGAR, Cyrill ,  PLATH, Peter ,  REINHARD, Robert ,  SIEVERNICH, Bernd ,  LIEBL, Rex

IPC: C07D231/14 ,  C07D333/38 ,  C07D307/68 ,  C07D277/56 ,  C07D213/81 ,  C07D213/82 ,  C07D207/34 ,  A01N43/56 ,  A01N43/08 ,  A01N43/10 ,  A01N43/78 ,  A01N43/36 ,  A01N43/40

CPC classification number: C07D213/81 ,  A01N43/08 ,  A01N43/10 ,  A01N43/36 ,  A01N43/40 ,  A01N43/56 ,  A01N43/78 ,  A01N47/12 ,  A01N47/20 ,  A01N47/28 ,  A01N47/30 ,  C07D207/34 ,  C07D213/82 ,  C07D231/14 ,  C07D277/56 ,  C07D307/68 ,  C07D333/38

Abstract: The invention relates to heteroaroyl-substituted phenylalanine amides of formula (I), in which A represents a C-bonded heteroaryl, in addition to their salts that can be used for agricultural applications. The invention also relates to methods and intermediate products for the production of said compounds and to the use of said compounds or agents containing said compounds for controlling undesirable plants.

公开(公告)号：EP0811007B1

公开(公告)日：2005-11-23

申请号：EP96902274.8

申请日：1996-02-14

Applicant: BASF Aktiengesellschaft

Inventor： VON DEYN, Wolfgang ,  HILL, Regina, Luise ,  KARDORFF, Uwe ,  ENGEL, Stefan ,  OTTEN, Martina ,  VOSSEN, Marcus ,  PLATH, Peter ,  RANG, Harald ,  HARREUS, Albrecht ,  KÖNIG, Hartmann ,  WALTER, Helmut ,  WESTPHALEN, Karl-Otto ,  MISSLITZ, Ulf

IPC: C07D409/10 ,  C07D413/10 ,  C07D417/10 ,  A01N43/56

CPC classification number: C07D401/10 ,  A01N43/56 ,  A01N43/74 ,  A01N43/80 ,  C07D231/24 ,  C07D403/10 ,  C07D405/10 ,  C07D409/10 ,  C07D411/10 ,  C07D413/10 ,  C07D417/10

Abstract: Pyrazol-4-yl-benzoyl derivatives have the formula (I), in which the substituents have the following meanings: L, M are hydrogen, C1-C6 alkyl, C2-C6 alkenyl, C2-C6 alkinyl, C1-C4 alkoxy, these groups being optionally substituted by 1 to 5 halogen atoms or C1-C4 alkoxy, halogen, cyano, nitro, a group -(Y)n-S(O)mR7 or a group -(Y)¿n-CO-R?8; Z is a 5 or 6-membered saturated or unsaturated heterocyclic rest, that contains 1 to 3 heteroatoms selected from the group that includes oxygen, sulphur or nitrogen, optionally substituted by halogen, cyano, nitro, a group -CO-R8, C1-C4 alkyl, C1-C4 halogen alkyl, C3-C8 cycloalkyl, C1-C4 alkoxy, C1-C4 halogen alkoxy, C1-C4 alkylthio, C1-C4 halogen alkylthio, di-C1-C4-alkylamino, a phenyl optionally substituted by halogen, cyano, nitro C1-C4 alkyl or C1-C4 halogen alkyl or a twice bound oxygen that optionally in the tautomer form may also be a hydroxy group, or that forms a bicyclic system together with a condensed phenyl ring optionally substituted by halogen, cyano, nitro, C1-C4 alkyl or C1-C4 halogen alkyl, with a condensed carbon cycle or with a second condensed heterocycle optionally substituted by halogen, cyano, nitro, C1-C4 alkyl, di-C1-C4-alkylamino, C1-C4 alkoxy, C1-C4 halogen alkoxy or C1-C4 halogen alkyl; Y is O, NR9; n equals 0 or 1; m equals 0, 1 or 2; R7 is C1-C4 alkyl, C1-C4 halogen alkyl or NR?9R10; R8 is C¿1-C4 alkyl, C1-C4 halogen alkyl, C1-C4 alkoxy or NR?9R10; R9¿ is hydrogen or C¿1?-C4 alkyl; R?10 is C¿1-C4 alkyl; Q is a pyrazol ring linked at position 4 having the formula (II) in which R1 is C1-C4 alkyl; R2 is hydrogen or C¿1?-C4 alkyl; and R?3¿ is hydrogen, C¿1?-C4 alkyl sulphonyl, phenyl sulphonyl or alkyl phenyl sulphonyl. Also disclosed are the salts of compounds (I) usually utilized in agriculture.

公开(公告)号：EP1163232A1

公开(公告)日：2001-12-19

申请号：EP00906364.5

申请日：2000-02-21

Applicant: BASF AKTIENGESELLSCHAFT

Inventor： MISSLITZ, Ulf ,  BAUMANN, Ernst ,  VON DEYN, Wolfgang ,  KUDIS, Steffen ,  LANGEMANN, Klaus ,  MAYER, Guido ,  NEIDLEIN, Ulf ,  WITSCHEL, Matthias ,  GÖTZ, Roland ,  RACK, Michael ,  PLATH, Peter ,  OTTEN, Martina ,  WESTPHALEN, Karl-Otto ,  WALTER, Helmut

IPC: C07D275/06 ,  A01N43/80

CPC classification number: C07D275/06 ,  A01N43/80

Abstract: The invention relates to saccharin 5 carbonyl derivatives of formula (I), wherein the substituents have the following meaning: L represents C1-C6-alkyl, C1-C6-alkoxy; Z represents C1-C6-alkyl, C3-C8-cycloalkyl, C3-C6-alkenyl, C3-C5-alkinyl, phenyl-C1-C6-alkyl or phenyl, wherein the phenyl rings are optionally substituted once or several times by C1-C6-alkyl, C1-C6-alkoxy or halogen; M represents hydrogen, C1-C6-alkyl, C1-C6-alkoxy, halogen, cyano, nitro or halogen-C1-C6-alkyl; R?1, R2, R3, R4, R5, R6, R7, R8¿ represent hydrogen, C¿1?-C6-alkyl. The invention also relates to the agriculturally usable salts of compound (I).