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公开(公告)号:CA2917183A1
公开(公告)日:2015-01-29
申请号:CA2917183
申请日:2014-07-22
Applicant: BASF SE
Inventor: HAFNER ANDREAS , BLATTER FRITZ , SZELAGIEWICZ MARTIN , SIEBENHAAR BERND , CHIODO TIZIANA , HINTERMANN TOBIAS , SALVADOR BEATE , VOSSEN MARCUS
IPC: A61K31/506 , A61K31/191 , A61K31/428 , A61K31/455
Abstract: The present invention primarily relates to molecular crystalline substances, preferably salts of Dasatinib in crystalline form, comprising a compound of formula 1, preferably a cation of a compound of formula 1, and a second compound selected from the group consisting of glutaric acid, nicotinic acid and saccharin, preferably an anion thereof. The invention is further related to pharmaceutical compositions comprising such a substance. Furthermore, the invention relates to processes for preparing said substances. The invention also relates to several aspects of using said substances or pharmaceutical compositions to treat a disease.
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公开(公告)号:AU2013265471A1
公开(公告)日:2014-12-04
申请号:AU2013265471
申请日:2013-05-15
Applicant: BASF SE
Inventor: REINHARD ROBERT , CHIODO TIZIANA , WOLF BERND , SCHERER STEFAN , BRATZ MATTHIAS , WITSCHEL MATTHIAS , NEWTON TREVOR WILLIAM , SEITZ THOMAS
IPC: C07D413/04 , A01N43/84 , A01P13/00
Abstract: The present invention relates to a novel crystalline form A of 1,5-dimethyl-6-thioxo-3-(2,2,7-trifluoro-3-oxo-4-(prop-2-ynyl)-3,4- dihydro-2H-benzo[b][1,4]oxazin-6-yl)-1,3,5-triazinane-2,4-dione. The invention also relates to a process for the production of this crystalline form and formulations for plant protection which contains the novel crystalline form of 1,5-dimethyl-6-thioxo-3-(2,2,7-trifluoro-3- oxo-4-(prop-2-ynyl)-3,4-dihydro-2H-benzo[b][1,4]oxazin-6-yl)-1,3,5- triazinane-2,4-dione.
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公开(公告)号:PE20141533A1
公开(公告)日:2014-11-14
申请号:PE2014000267
申请日:2012-08-30
Applicant: BASF SE
Inventor: SOWA CHRISTIAN , GOLD RANDALL EVAN , CHIODO TIZIANA , VOGEL RALF
IPC: C07D239/42 , A01N43/32 , A01N43/54 , A01P3/00 , C07D339/08
Abstract: SE REFIERE A COCRISTALES QUE COMPRENDEN CYPRODINIL Y DITHIANON, QUE EN UN DIFRACTOGRAMA DE RAYOS X EN POLVO A 20�C, MUESTRAN HASTA TRES DE LOS SIGUIENTES VALORES 2TETHA[�]: 7,47�0,2�; 9,86�0,2�; 12,34�0,2�; 12,88�0,2�; 13,92�0,2�; 14,88�0,2�; 15,34�0,2�; 16,20�0,2�; 17,85�0,2�; 18,97�0,2�; ENTRE OTROS. SE REFIERE TAMBIEN A UN PROCESO PARA LA PREPARACION DE DICHOS COCRISTALES Y A UNA COMPOSICION QUE COMPRENDEN COCRISTALES. DICHOS COCRISTALES SON UTILES PARA COMBATIR HONGOS FITOPATOGENOS
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公开(公告)号:AU2013242103A1
公开(公告)日:2014-10-16
申请号:AU2013242103
申请日:2013-03-20
Applicant: BASF SE
Inventor: CHIODO TIZIANA , KLIMOV EVGUENI , SCHAFER ANSGAR , HOFFKEN HANS WOLFGANG , HELLMANN ROLF , KABAT ANDRE , ISRAELS RAFEL , SCHNABEL GERHARD , BRATZ MATTHIAS , KIBAT CHRISTINE , HOUY WOLFGANG
IPC: A01N37/40 , A01N25/12 , A01P13/00 , C07C63/06 , C07D239/42 , C07D239/47 , C07D277/40 , C07D473/12
Abstract: Co-crystals comprising a) a herbicide compound A, which is 3,6-dichloro-2-methoxybenzoic acid (dicamba), and b) a co-crystal former B, which is selected from the group of aromatic, N- containing heterocycles; and their use in agrochemical compositions.
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公开(公告)号:CA2879792A1
公开(公告)日:2014-02-13
申请号:CA2879792
申请日:2013-08-05
Applicant: BASF SE
Inventor: HAFNER ANDREAS , BLATTER FRITZ , RODEL EVA , SZELAGIEWICZ MARTIN , CHIODO TIZIANA , HINTERMANN TOBIAS , SALVADOR BEATE , VOSSEN MARCUS
IPC: C07D249/08 , A61K31/4196 , A61P7/00
Abstract: The present invention refers to a multicomponent crystalline system (co-crystal) comprising a compound of formula (1) (4-[3,5-Bis(2-hydroxyphenyl)-1H-1,2,4-triazol-1-yl]benzoic acid; INN:Deferasirox) formula (1) and a compound of formula (2) (Isonicotinamide; pyridine-4-carboxamide) formula (2), as well as to a process for obtaining the same.
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公开(公告)号:CA2867504A1
公开(公告)日:2013-10-03
申请号:CA2867504
申请日:2013-03-20
Applicant: BASF SE
Inventor: CHIODO TIZIANA , KLIMOV EVGUENI , SCHAFER ANSGAR , HOFFKEN HANS WOLFGANG , HELLMANN ROLF , KABAT ANDRE , ISRAELS RAFEL , SCHNABEL GERHARD , BRATZ MATTHIAS , KIBAT CHRISTINE , HOUY WOLFGANG
IPC: A01N37/40 , A01N25/12 , A01P13/00 , C07C63/06 , C07D239/42 , C07D239/47 , C07D277/40 , C07D473/12
Abstract: Co-crystals comprising a) a herbicide compound A, which is 3,6-dichloro-2-methoxybenzoic acid (dicamba), and b) a co-crystal former B, which is selected from the group of aromatic, N- containing heterocycles; and their use in agrochemical compositions.
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公开(公告)号:CA2844014A1
公开(公告)日:2013-03-07
申请号:CA2844014
申请日:2012-08-30
Applicant: BASF SE
Inventor: SOWA CHRISTIAN , GOLD RANDALL EVAN , CHIODO TIZIANA , VOGEL RALF
IPC: C07D239/42 , A01N43/32 , A01N43/54 , A01P3/00 , C07D339/08
Abstract: The present invention relates to co-crystals of cyprodinil and dithianon as defined in the description, processes for preparing these co-crystals and also to compositions comprising at least such co-crystals. The invention also relates to the use of such co- crystals or compositions for combating harmful fungi.
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18.
公开(公告)号:CL2021001826A1
公开(公告)日:2022-01-14
申请号:CL2021001826
申请日:2021-07-08
Applicant: BASF SE
Inventor: GOCKEL BIRGIT , KLAUBER ERIC GEORGE , RACK MICHAEL , SOERGEL SEBASTIAN , GOETZ ROLAND , VOGT FLORIAN , GEBHARDT JOACHIM , VIERTELHAUS MARTIN , CHIODO TIZIANA , XU WEN
IPC: C07D403/12
Abstract: La invención describe a una forma cristalina de 1-(1,2-dimetilpropil)-N-etil-5-metil-N-piridazin-4-il-pirazol-4-carboxamida a la que recientemente se le asignó el nombre común dimpropyridaz y al uso de dicha forma cristalina B para combatir plagas de invertebrados y a formulaciones para la protección de plantas.
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公开(公告)号:UA116887C2
公开(公告)日:2018-05-25
申请号:UAA201413770
申请日:2013-05-15
Applicant: BASF SE
Inventor: REINHARD ROBERT , CHIODO TIZIANA , WOLF BERND , SCHERER STEFAN , BRATZ MATTHIAS , WITSCHEL MATTIAS , NEWTON TREVOR WILLIAM , SEITZ THOMAS
IPC: C07D413/04 , A01N43/90
Abstract: ВинахідстосуєтьсяновоїкристалічноїформиВ 1,5-диметил-6-тіоксо-3-(2,2,7-трифтор-3-оксо-4-(проп-2-ініл)-3,4-дигідро-2Н-бензо[b][1,4]оксазин-6-іл)-1,3,5-триазинан-2,4-діону. Винахідтакожстосуєтьсяспособуотриманняцієїкристалічноїформитарецептурдлязахистурослин, якімістятьновукристалічнуформу 1,5-диметил-6-тіоксо-3-(2,2,7-трифтор-3-оксо-4-(проп-2-ініл)-3,4-дигідро-2Н-бензо[b][1,4]оксазин-6-іл)-1,3,5-триазинан-2,4-діону.
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公开(公告)号:EA027898B1
公开(公告)日:2017-09-29
申请号:EA201401310
申请日:2013-05-15
Applicant: BASF SE
Inventor: REINHARD ROBERT , CHIODO TIZIANA , WOLF BERND , SCHERER STEFAN , BRATZ MATTHIAS , WITSCHEL MATTHIAS , NEWTON TREVOR WILLIAM , SEITZ THOMAS
IPC: C07D413/04 , A01N43/84 , A01P13/00
Abstract: Изобретениеотноситсяк новойкристаллическойформеА 1,5-диметил-6-тиоксо-3-(2,2,7-трифтор-3-оксо-4-(проп-2-инил)-3,4-дигидро-2Н-бензо[b][1,4]оксазин-6-ил)-1,3,5-триазинан-2,4-диона. Изобретениетакжеотноситсяк способуполученияэтойкристаллическойформыи рецептурдлязащитырастений, которыесодержатновуюкристаллическуюформу 1,5-диметил-6-тиоксо-3-(2,2,7-трифтор-3-оксо-4-(проп-2-инил)-3,4-дигидро-2Н-бензо[b][1,4]оксазин-6-ил)-1,3,5-триазинан-2,4-диона.
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