公开(公告)号：UY32286A

公开(公告)日：2010-06-30

申请号：UY32286

申请日：2009-12-02

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： MICHEL MUEHLEBACH ,  JEANGUENAT ANDRE ,  OLIVIER LOISELEUR ,  THOMAS PITTERNA ,  PETER MAIENFISCH ,  QACEMI MYRIEM EL ,  CASSAYRE JEROME YVES ,  HALL ROGER GRAHAM ,  ANDREW EDMUNDS ,  CAMILLA CORSI ,  STOLLER ANDRE DENIS ,  GODFREY CHRISTOPHER RICHARD AYLES ,  SCHAETZER JUERGEN HARRY

IPC: C07D471/20 ,  A01N43/40

Abstract: Nuevos derivados de pirrolidindiona espiroheterocíclica N-oxiamida sustituidas de fórmula I donde los sustituyentes son tales como se definene en la reivindicación 1; composiciones que los contienen y sus usos como insecticidas, acaricidas, nematicidas o molusquicidas.

公开(公告)号：GB2520098A

公开(公告)日：2015-05-13

申请号：GB201410899

申请日：2014-06-19

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： PITTERNA THOMAS ,  GODFREY CHRISTOPHER RICHARD AYLES ,  HUETER OTTMAR FRANZ ,  STOLLER ANDRE DENIS ,  JUNG PIERRE JOSEPH MARCEL ,  EDMUNDS ANDREW

IPC: C07D335/02 ,  A01N43/18 ,  A01N43/20 ,  A01N43/26 ,  A01P5/00 ,  A01P7/00 ,  A01P9/00 ,  C07D331/04 ,  C07D339/04 ,  C07D409/04

Abstract: The present invention relates to bis-amide derivatives of formula (I): wherein Q1 is a saturated 4-6-membered heterocyclic ring comprising 1-2 sulfur atoms in addition to the carbon atoms, preferably a thietan-3-yl, dithiolan-4-yl or tetrahydrothiopyran-4-yl group, which may be unsubstituted or substituted on a sulphur atom with one or more substituents selected from =O, =N-Z and =NCZ1Z2; Z is H or cyano; Z1 and Z2 are cyano or together form a C(O)-O-CH2-C(O)- or C(O)-S-CH2-C(O)- bridge; Y1 and Y5 are Cl, Br, I, C1-4alkyl, C1-4alkoxy, C1-4haloalkyl, C1-4haloalkoxy, C1-4alkylthio, C1-4alkylsulfinyl, C1-4alkylsulfonyl or C1-4alkoxy- C1-4alkyl; Y3 is C1-4haloalkyl; Xa is H, methoxy or halogen; Xb is H, halogen or cyano; R1 and R2 are H or substituents; or an agronomically acceptable salt thereof may be useful as an insecticide, in particular insecticidal, acaricidal, nematicidal or molluscicidal activity. Methods of preparing these compounds, including intermediates, and insecticidal, acaricidal, nematicidal or molluscicidal compositions comprising them are also disclosed.

公开(公告)号：UA102676C2

公开(公告)日：2013-08-12

申请号：UAA201005712

申请日：2008-10-13

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： STOLLER ANDRE DENIS ,  JUNG PIERRE JOSEPH MARCEL ,  GODFREY CHRISTOPHER RICHARD AYLES ,  LUTZ WILLIAM ,  MAIENFISCH PETER ,  ZAMBACH WERNER

IPC: A01N37/46 ,  A01N41/10 ,  A01P7/04 ,  C07C317/40 ,  C07C323/60 ,  C07D213/64

Abstract: Соединениеформулы (I), вкоторой A, A, A, A, R, R, R, G, G, Q, Q, Y, Y, Yи Yявляютсятакими, какопределенов пункте 1 формулыизобретения, илиихсолями, или N-оксидами. Крометого, описаныпромежуточноесоединениеи инсектицидная, акарицидная, нематоциднаяилимоллюскоциднаякомпозиция, содержащаясоединениеформулы (I), испособборьбыс насекомыми, клещами, нематодамиилимоллюсками, илиихуничтожение.

公开(公告)号：UY32324A

公开(公告)日：2010-07-30

申请号：UY32324

申请日：2009-12-14

Applicant: SYNGENTA LTD ,  SYNGENTA PARTICIPATIONS AG

Inventor： MICHEL MUEHLEBACH ,  JEANGUENAT ANDRE ,  OLIVIER LOISELEUR ,  THOMAS PITTERNA ,  PETER MAIENFISCH ,  QACEMI MYRIEM EL ,  CASSAYRE JEROME YVES ,  CAMILLA CORSI ,  STOLLER ANDRE DENIS ,  SCHAETZER JUERGEN HARRY ,  ANDREW EDMUNDS ,  HALL ROGER GRAHAM ,  AYLES GODFREY CRISTOPHER RICHARD ,  CARTER NEIL BRIAN

IPC: A01N43/34 ,  A01N43/90 ,  C07D471/10

Abstract: Nuevos derivados de pirrolidinidona espiroheterocíclica N-alquilmida sustituidas de fórmula donde los sustituyentes son tales como se definen en la reivindicación 1; composiciones que los contienen y sus usos como pesticidas.

公开(公告)号：GB2463736A

公开(公告)日：2010-03-31

申请号：GB0817909

申请日：2008-09-30

Applicant: SYNGENTA PARTICIPATIONS AG

Inventor： HALL ROGER GRAHAM ,  EDMUNDS ANDREW ,  JEANGUENAT ANDRE ,  LOISELEUR OLIVIER ,  STOLLER ANDRE DENIS

IPC: C07D231/56

Abstract: The invention relates to the preparation of an insecticide of formula (I), wherein X is a bivalent group selected from X1-X8; R1is C1-C4alkyl or halogen; and R2and R3are hydrogen, C1-C4alkyl, C1-C4alkoxy, cyano, nitro or halogen. The process is depicted below and comprises (a) reacting a pyrroline dione of formula (II) with a source of hydroxylamine, preferably hydroxylamine hydrochloride, to give a compound of formula (III); (b) converting the intermediate (III) into the ortho amino-substituted aromatic cyano compound of formula (IV) by heating; and (c) hydrolysing the nitrile group of precursor (IV) to obtain the product of formula (I). A particular example is the synthesis of 6-amino-5-methyl-1H-indazole-7-carboxylic acid. The preparation of 6-amino-5-methyl-1H-indazole-7-carboxamide is also outlined. Compounds of formula (IV) are claimed separately.