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    N-ACYLIMINO HETEROCYCLIC COMPOUNDS
    21.
    发明申请
    N-ACYLIMINO HETEROCYCLIC COMPOUNDS 审中-公开
    N-乙酰氨基杂环化合物

    公开(公告)号：WO2016062680A1

    公开(公告)日：2016-04-28

    申请号：PCT/EP2015/074199

    申请日：2015-10-20

    Applicant: BASF SE

    Inventor： KÖRBER, Karsten ,  MCLAUGHLIN, Martin John ,  GOCKEL, Birgit ,  VON DEYN, Wolfgang

    IPC: C07D401/14 ,  C07D405/14 ,  C07D413/14 ,  A01N43/50 ,  C07D401/06 ,  C07D409/14 ,  C07D417/14 ,  A01N43/78 ,  C07D413/06 ,  C07D417/06

    CPC classification number: C07D401/06 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N43/88 ,  C07D401/14 ,  C07D405/14 ,  C07D409/14 ,  C07D413/06 ,  C07D413/14 ,  C07D417/06 ,  C07D417/14

    Abstract: The present invention relates to N-acylimino compound of formula (I): wherein X is O or S, in particular O; Y indicates a single bond between N and R 4 or Y is O, S, S(=O), S(=O) 2 , CHR 5a or N-R 5 ; Het is a 5 or 6 membered carbon-bound or nitrogen-bound heterocyclic ring, W 1 represents O, S or NR w1 ; W 2 -W 3 -W 4 represents a bivalent radical selected from -C(R v2 R w2 )-C(R v3 R w3 )-, -C(R v4 )=C(R v5 )- and -C(R v2 R w2 )-O-C(R v3 R w3 )-; R 1 , R 2 may be hydrogen, halogen, etc.; R 3 may be hydrogen, CN, C 1 -C 6 -alkyl, etc.; R 4 may be of hydrogen, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkinyl, C 3 -C 8 -cycloalkyl, Q- phenyl, Q'-O-phenyl, Q'-S-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R 10 , and the moieties Q-Het#, Q'-O-Het# and Q'-S-Het# where Het# represents a heterocyclic radical and where Q and Q' are C 1 -C 6 -alkandiyl, C 2 -C 6 -alkendiyl, or C 2 -C 6 -alkyndiyl, and where Q may also be a single bond; R 3 and R 4 together may also a bivalent radical, selected from the group consisting of C 2 -C 5 -alkandiyl, C 2 -C 5 -alkendiyl, Q"-C 1 -C 4 -alkandiyl and Q"-C 2 -C 4 -alkendiyl, where Q" is O or S. The invention also relates to the use of the N-acylimino heterocyclic compounds, their ste-reoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明涉及式（I）的N-酰基亚胺基化合物：其中X是O或S，特别是O; Y表示N和R4之间的单键，或Y表示O，S，S（= O），S（= O）2，CHR5a或N-R5; Het是5或6元碳键或氮键的杂环，W1表示O，S或NRw1; W2-W3-W4表示选自-C（Rv2Rw2）-C（Rv3Rw3） - ， - C（Rv4）= C（Rv5） - 和-C（Rv2Rw2）-O-C（Rv3Rw3） - 的二价基团。 R1，R2可以是氢，卤素等; R3可以是氢，CN，C1-C6-烷基等; R4可以是氢，C1-C6-烷基，C2-C6-烯基，C2-C6-炔基，C3-C8-环烷基，Q-苯基，Q'-O-苯基，Q'-S-苯基，其中 苯环任选被一个或多个，例如， 1,2,3或4或5个相同或不同的取代基R10，以及Q-Het＃，Q'-O-Het和Q'-S-Het的部分，其中Het＃表示杂环基团，其中Q和Q '是C 1 -C 6 - 烷二基，C 2 -C 6 - 烷基或C 2 -C 6 - 炔二基，其中Q也可以是单键; R 3和R 4一起也可以是选自C 2 -C 5 - 烷二基，C 2 -C 5 - 烷基，Q“-C 1 -C 4 - 烷二基和Q”-C 2 -C 4 - 烷二基的二价基团，其中Q“ 本发明还涉及N-酰基亚氨基杂环化合物及其互变异构体及其互变异构体及其盐对抗无脊椎动物害虫的用途，本发明还涉及无脊椎动物害虫的防治方法，其包括施用 这样的化合物。

    N-ACYLIMINO HETEROCYCLIC COMPOUNDS
    22.
    发明申请
    N-ACYLIMINO HETEROCYCLIC COMPOUNDS 审中-公开
    N-乙酰氨基杂环化合物

    公开(公告)号：WO2016062678A1

    公开(公告)日：2016-04-28

    申请号：PCT/EP2015/074196

    申请日：2015-10-20

    Applicant: BASF SE

    Inventor： KÖRBER, Karsten ,  MCLAUGHLIN, Martin John ,  GOCKEL, Birgit ,  VON DEYN, Wolfgang ,  KOJIMA, Kenichi

    IPC: C07D401/06 ,  C07D405/06 ,  C07D413/06 ,  C07D417/06 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78

    CPC classification number: C07D401/06 ,  A01N43/50 ,  A01N43/76 ,  A01N43/78 ,  A01N43/88 ,  A01N53/00 ,  C07D405/06 ,  C07D413/06 ,  C07D417/06

    Abstract: The present invention relates to N-acylimino compound of formula (I): (I) wherein X 1 is O or S, in particular O; X 2 is CN or NO 2 ; m is an integer selected from 0, 1, 2, 3, 4, 5 and 6; Het is a 5- or 6- membered carbon-bound or nitrogen-bound heterocyclic or heteroaromatic ring, W 1 is O, S or NR w1 ; W 2 -W 3 -W 4 isa bivalent radical selected from -C(R v2 R w2 )-C(R v3 R w3 )-, -C(R v4 )=C(R v5 )- and - C(R v2 R w2 )-O-C(R v3 R w3 )-; R 1 , R 2 may be hydrogen, halogen, etc. R 3 may be hydrogen, halogen, CN, C 1 -C 6 -alkyl, etc. R 4a , R 4b if present, may be hydrogen, halogen, C 1 -C 6 -alkyl, etc. R 5 may be hydrogen, halogen, C 1 -C 6 -alkyl, C 1 -C 6 -alkenyl, C 1 -C 6 -alkynyl, C 3 -C 8 - cycloalkyl, S(O) n NR 9a R 9b , NR 9a R 9b , C(=O)OR 8 , C(=O)NR 9a R 9b , C(=S)NR 9a R 9b , C(=O)R 7a , C(=S)R 7a , NR 9a -C(=O)R 7a , NR 9a -C(=S)R 7a , NR 9a -S(O) n R 8a , a moitey Q-phenyl, where the phenyl ring is optionally substituted with one or more, e.g. 1, 2, 3, 4 or 5 identical or different substituents R 10 , or a moiety Q-Het # , or R 3 and R 5 together may also form with the carbon atom they are bound to, a 3-, 4-, 5- or 6- membered saturated partially unsaturated carbocycle or heterocycle, wherein R w1 , R w2 , R w3 , R v2 , R v3 , R v5 , R 7a , R 8 , R 8a , R 9a , R 9b , Q, Het # are as defomed in the claims. The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: 本发明涉及式（I）的N-酰基亚氨基化合物：（I）其中X1是O或S，特别是O; X2为CN或NO2; m是选自0,1,2,3,4,5和6的整数; Het是5-或6-元碳键或氮键合的杂环或杂芳环，W1是O，S或NRw1; W2-W3-W4是选自-C（Rv2Rw2）-C（Rv3Rw3） - ， - C（Rv4）= C（Rv5） - 和-C（Rv2Rw2）-O-C（Rv3Rw3） - 的二价基团。 R 1，R 2可以是氢，卤素等。R 3可以是氢，卤素，CN，C 1 -C 6烷基等。如果存在，R 4a，R 4b可以是氢，卤素，C 1 -C 6烷基等。 C 1 -C 6 - 烷基，C 1 -C 6 - 烯基，C 1 -C 6 - 炔基，C 3 -C 8环烷基，S（O）n NR 9 a R 9 b，NR 9 a R 9 b，C（= O）OR 8，C（= O）NR 9a R 9b ，C（= S）NR9aR9b，C（= O）R7a，C（= S）R7a，NR9a-C（= O）R7a，NR9a-C（= S）R7a，NR9a-S（O）nR8a， Q-苯基，其中苯环任选被一个或多个例如， 1,2,3或4或5个相同或不同的取代基R10或部分Q-Het＃，或R3和R5一起也可以与它们所键合的碳原子形成，3-，4-，5-或 6-元饱和部分不饱和碳环或杂环，其中Rw1，Rw2，Rw3，Rv2，Rv3，Rv5，R7a，R8，R8a，R9a，R9b，Q，Het＃如权利要求中所述。 本发明还涉及N-酰基亚氨基杂环化合物，其立体异构体，其互变异构体及其盐的用途，用于防治无脊椎动物害虫。 此外，本发明还涉及防治无脊椎害虫的方法，其包括施用这样的化合物。

    C3-C4-CYCLOALKENYL-COMPRISING PYRAZOLES FOR CONTROLLING INVERTEBRATE PESTS
    23.
    发明申请
    C3-C4-CYCLOALKENYL-COMPRISING PYRAZOLES FOR CONTROLLING INVERTEBRATE PESTS 审中-公开
    用于控制反相胶束的C3-C4-环烯基包含吡咯

    公开(公告)号：WO2015162133A1

    公开(公告)日：2015-10-29

    申请号：PCT/EP2015/058608

    申请日：2015-04-21

    Applicant: BASF SE

    Inventor： SAELINGER, Daniel ,  GOCKEL, Birgit ,  SOERGEL, Sebastian

    IPC: C07D403/12 ,  C07D401/12 ,  A01N43/56 ,  A01N43/58

    CPC classification number: C07D401/12 ,  A01N43/56 ,  A01N43/58 ,  C07D403/12

    Abstract: The present invention relates to novel pyrazoles of formula (I). Moreover, the invention relates to processes and intermediates for preparing the pyrazoles of formula (I), and also to active compound combinations comprising them, to compositions comprising them, and to their use for protecting growing plants from attack or infestation by invertebrate pests. Furthermore, the invention relates to methods of applying such compounds. The present invention also relates to seed comprising such compounds.

    Abstract translation: 本发明涉及式（I）的新型吡唑。 此外，本发明涉及用于制备式（I）的吡唑的方法和中间体，还涉及包含它们的活性化合物组合物，包含它们的组合物以及用于保护生长植物免受无脊椎害虫侵袭或侵袭的用途。 此外，本发明涉及应用这些化合物的方法。 本发明还涉及包含这种化合物的种子。

    N-ACYLIMINO HETEROCYCLIC COMPOUNDS AND THEIR USE AS PESTICIDES
    24.
    发明申请
    N-ACYLIMINO HETEROCYCLIC COMPOUNDS AND THEIR USE AS PESTICIDES 审中-公开
    N-乙酰氨基杂环化合物及其作为农药的用途

    公开(公告)号：WO2015086790A1

    公开(公告)日：2015-06-18

    申请号：PCT/EP2014/077488

    申请日：2014-12-12

    Applicant: BASF SE

    Inventor： MCLAUGHLIN, Martin, John ,  GOCKEL, Birgit ,  KÖRBER, Karsten ,  DIETZ, Jochen ,  VON DEYN, Wolfgang ,  POHLMAN, Matthias

    IPC: C07D213/75 ,  C07D409/14 ,  A01N43/14 ,  A01P5/00 ,  A01P7/00

    CPC classification number: C07D213/75 ,  C07D409/14

    Abstract: N-acylimino heterocyclic compounds The present invention relates to N-acylimino compound of formula (I): wherein X is 0 or S, in particular 0; Y is 0, S or NR 5 ; D is a bivalent radical such as optionally substituted C 1 -C 6 - alkandiyl, Het is a 5- or 6-membered carbon-bound or nitrogen-bound heterocyclic ring, W 1 -W 2 -W 3 -W Represents a carbon chain group connected to N and C=N, and thus forming a saturated, unsaturated, or partially unsaturated 5 or 6 membered nitrogen containing heterocycle, wherein W 1, , W 2 , W 3 and W 4 each individually represent CR vR W; R', R 2 may be hydrogen, halogen, C 1 -C 6 -alkyl etc.; R 3 hydrogen, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 8 - cycloalkyl, C 3 -C 8 -cycloalkyl-Ci-C 4 -alkyl, etc.; R 4 hydrogen, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 -C 8 - cycloalkyl, C 3 -C 8 -cycloalkyl-Ci-C 4 -alkyl, etc.; R 3 and R 4 together may also form a bivalent radical, selected from the group consisting of C 3 -C 6 -alkandiyl, C 3 -C e-alkendiyl, Q'-C 2 -C 5 -alkandiyl, Q'-C 2 -C 5 -alkendiyl, Q '"C 2 -C 4 -alkandiyl-Q 2 and Q i- C 2 - C 4 -alkendiyl-Q 2 , where Q 1 , Q 2 are 0, S or NR 7d ; R 5 hydrogen, CN, C 1 -C 6 -alkyl, C 2 -C 6 -alkenyl, C 2 -C 6 -alkynyl, C 3 - C 8 -cycloalkyl, C 3 -C 8 -cycloalkyl-Ci-C 4 -alkyl, C 1 -C 6 -alkylcarbonyl, C 1 -C 6 -alkylsulfonyl, etc.; The invention also relates to the use of the N-acylimino heterocyclic compounds, their stereoisomers, their tautomers and their salts, for combating invertebrate pests. Furthermore the invention relates also to methods of combating invertebrate pests, which comprises applying such compounds.

    Abstract translation: N-酰基亚氨基杂环化合物本发明涉及式（I）的N-酰基亚氨基化合物：其中X为0或S，特别是0; Y为0，S或NR 5; D是二价基团，例如任选取代的C 1 -C 6 - 烷二基，Het是5-或6-元碳结合或氮键合的杂环，W 1 -W 2 -W 3 -W表示碳链 连接到N和C = N的基团，从而形成饱和的，不饱和的或部分不饱和的5或6元含氮杂环，其中W 1，W 2，W 3和W 4各自独立地表示CR vRW; R'，R 2可以是氢，卤素，C 1 -C 6 - 烷基等; R 3氢，C 1 -C 6烷基，C 2 -C 6链烯基，C 2 -C 6炔基，C 3 -C 8环烷基，C 3 -C 8 - 环烷基-C 1 -C 4烷基， 等等。; R 4氢，C 1 -C 6烷基，C 2 -C 6链烯基，C 2 -C 6炔基，C 3 -C 8环烷基，C 3 -C 8 - 环烷基-C 1 -C 4 - 烷基， 等等。; R 3和R 4一起也可以形成二价基团，其选自C 3 -C 6 - 烷二基，C 3 -C e - 烷二基，Q'-C 2 -C 5 - 烷二基，Q'-C 2- C 5 - 烷基，Q'“C 2 -C 4 - 二烷基-Q 2和Q iC 2 -C 4 - 烷基-Q 2，其中Q 1，Q 2为0，S或NR 7d; R 5氢，CN，C 1 C 1-6烷基，C 2 -C 6链烯基，C 2 -C 6炔基，C 3 -C 8环烷基，C 3 -C 8 - 环烷基-C 1 -C 4 - 烷基，C 1 -C 6 - 烷基羰基，C 1 -C 6 - 烷基磺酰基等;本发明还涉及N-酰基亚氨基杂环化合物，其立体异构体，其互变异构体及其盐的用途，用于防治无脊椎动物害虫。此外，本发明还涉及方法 防治无脊椎动物害虫，其中包括施用这些化合物。

    CRYSTALLINE FORMS OF 1-(1,2-DIMETHYLPROPYL)-N-ETHYL-5-METHYL-N-PYRIDAZIN-4-YL-PYRAZOLE-4-CARBOXAMIDE
    27.
    发明申请
    CRYSTALLINE FORMS OF 1-(1,2-DIMETHYLPROPYL)-N-ETHYL-5-METHYL-N-PYRIDAZIN-4-YL-PYRAZOLE-4-CARBOXAMIDE 审中-公开

    公开(公告)号：WO2020144308A1

    公开(公告)日：2020-07-16

    申请号：PCT/EP2020/050493

    申请日：2020-01-10

    Applicant: BASF SE

    Inventor： GEBHARDT, Joachim ,  VIERTELHAUS, Martin ,  CHIODO, Tiziana ,  RACK, Michael ,  KLAUBER, Eric George ,  XU, Wen ,  GOETZ, Roland ,  VOGT, Florian ,  GOCKEL, Birgit ,  SOERGEL, Sebastian

    IPC: C07D403/12

    Abstract: The present invention relates to a novel crystalline form of 1-(1,2-dimethylpropyl)- N-ethyl-5-methyl-N-pyridazin-4-yl-pyrazole-4-carboxamide recently assigned the common name dimpropyridaz. The invention also relates to the use of the crystalline form B for combating invertebrate pests and to formulations for plant protection which contain the crystalline form B of 1-(1,2-dimethylpropyl)-N-ethyl-5-methyl-N-pyridazin-4- yl-pyrazole-4-carboxamide. The crystalline form B according to the present invention can be identified by powder X-ray diffractometry on the basis of its powder X-ray diffraction diagram, hereinafter also termed powder X-ray diffraction pattern or PXRD pattern,of the polymorph form B recorded using Cu-Kα radiation (1.54178 Å) at 25°C displays the 3 following reflections, quoted as 2θ values: 20.69±0.10°, 24.15±0.10°and 30.52± 0.10°.In addition to these 3 reflections, the polymorph B of the present invention may display in such a PXRD pattern one or more, in particular at least 2, often at least 4, in particular at least 6 or at least 8 reflections and especially all of the reflections quoted hereinafter as 2θ values:7.99±0.10°, 10.07±0.10°, 12.38±0.10°,15.31±0.10°, 15.97±0.10°, 16.50±0.10°, 18.03±0.10°,19.29±0.10°, 20.22±.0.10°, 20.96± 0.10°, 23.40±0.10°, 23.70±0.10°,26.09±0.10°, 27.26±0.10°and 32.91±0.10°.

    PROCESS FOR PREPARATION OF BENZYLIC AMIDES
    30.
    发明申请
    PROCESS FOR PREPARATION OF BENZYLIC AMIDES 审中-公开

    公开(公告)号：WO2018137959A1

    公开(公告)日：2018-08-02

    申请号：PCT/EP2018/050937

    申请日：2018-01-16

    Applicant: BASF SE

    Inventor： MCLAUGHLIN, Martin John ,  KOERBER, Karsten ,  GOCKEL, Birgit ,  VYAS, Devendra ,  NARINE, Arun

    IPC: C07D413/04 ,  C07D307/79

    Abstract: The present invention relates to a process for preparing benzylic amides of formula (I) wherein the variables have the meaning as defined in the description, by reductive amidation of a nitrile of formula (II) wherein the variables have the meanings given for formula I, with an activated carbonyl compound of formula (III), and which nitrile is obtained by reaction of a compound of formula (IV) with a halogen compound of formula (V), wherein X is a halogen atom, preferably bromo, which halogen compound V in turn is obtained by Sandmeyer reaction of an aniline derivative of formula (VI) novel compounds of formula (I), and processes for preparing compounds of formula (XII) wherein the variables have the meaning as defined in the description by condensing compounds of formula I with compounds of formula (X) and subjecting the resulting α,β-unsaturated ketone of formula (XI) to a reaction with hydroxylamine to yield compounds of formula (XII.)

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