公开(公告)号：WO2016062814A1

公开(公告)日：2016-04-28

申请号：PCT/EP2015/074507

申请日：2015-10-22

Applicant: BASF SE

Inventor： BESONG, Gilbert ,  WITSCHEL, Matthias ,  SEITZ, Thomas ,  PARRA RAPADO, Liliana ,  EVANS, Richard ,  HANZLIK, Kristin ,  KRAEMER, Gerd ,  RACK, Michael

IPC: C07D495/04 ,  A01N43/90

CPC classification number: C07D495/04 ,  A01N43/90 ,  A01N47/20 ,  A01N53/00

Abstract: The present invention provides a substituted pyridine compound of the formula I or an agriculturally suitable salt or N-oxide thereof, wherein the variables in the formula I defined as in the description. Substituted pyridine compounds of formula I are useful as herbicides.

Abstract translation: 本发明提供式I的取代的吡啶化合物或其农业上合适的盐或N-氧化物，其中式I中的变量如说明书所述定义。 式I的取代的吡啶化合物可用作除草剂。

公开(公告)号：WO2015158565A1

公开(公告)日：2015-10-22

申请号：PCT/EP2015/057458

申请日：2015-04-07

Applicant: BASF SE

Inventor： BESONG, Gilbert ,  WITSCHEL, Matthias ,  REINGRUBER, Rüdiger ,  KRAUS, Helmut ,  SEITZ, Thomas ,  PARRA RAPADO, Liliana ,  NEWTON, Trevor William ,  KRÄMER, Gerd ,  EVANS, Richard Roger ,  RACK, Michael

IPC: C07D495/04 ,  A01N43/90

CPC classification number: C07D495/04 ,  A01N43/90

Abstract: The present invention provides a substituted pyridine compound of the formula (I) or an agriculturally suitable salt or N-oxide thereof, wherein the variables in the formula (I) are defined as in the description. Substituted pyridine compounds of formula I are useful as herbicides.

Abstract translation: 本发明提供式（I）的取代的吡啶化合物或其农业上合适的盐或N-氧化物，其中式（I）中的变量如描述中所定义。 式I的取代的吡啶化合物可用作除草剂。

公开(公告)号：WO2015158518A1

公开(公告)日：2015-10-22

申请号：PCT/EP2015/056541

申请日：2015-03-26

Applicant: BASF SE

Inventor： WOLF, Bernd ,  RACK, Michael ,  MAYWALD, Volker ,  GÖTZ, Roland ,  FRASSETTO, Timo

IPC: C07D265/36

CPC classification number: C07D265/36

Abstract: The present invention relates to for manufacturing benzoxazinones of formula (I), characterized in that amino compounds of formula (II) are added to an acid; wherein the substituents are defined according to the specification.

Abstract translation: 本发明涉及制备式（I）的苯并恶嗪酮，其特征在于将式（II）的氨基化合物加入酸中; 其中取代基根据说明书定义。

公开(公告)号：WO2015049360A1

公开(公告)日：2015-04-09

申请号：PCT/EP2014/071210

申请日：2014-10-02

Applicant: BASF SE

Inventor： KLAUBER, Eric George ,  RACK, Michael ,  ZIERKE, Thomas ,  HOLUB, Nicole ,  CORTES, David ,  SCHMELEBECK, Gerald ,  JI, Junmin

IPC: C07C37/02 ,  C07C41/16

CPC classification number: C07C51/377 ,  C07C37/02 ,  C07C41/16 ,  C07C67/297 ,  C07F1/005 ,  C07F1/04 ,  C07C39/30 ,  C07C43/225

Abstract: The present invention relates to a process for providing a compound of formula (I):, wherein R is hydrogen or R', wherein R' is –(C 1 -C 4 )alkyl, and Hal is a halogen, the process comprising the step of: reacting a compound of formula (II) wherein Hal is defined as above, with an alkali metal alkoxide of the formula XOR', wherein X is an alkali metal, and R' is defined as above.

Abstract translation: 本发明涉及提供式（I）化合物的方法：其中R是氢或R'，其中R'是 - （C 1 -C 4）烷基，而Hal是卤素，该方法包括以下步骤： ：将其中Hal如上定义的式（II）化合物与式XOR'的碱金属醇盐反应，其中X为碱金属，R'如上定义。

公开(公告)号：WO2014202589A1

公开(公告)日：2014-12-24

申请号：PCT/EP2014/062695

申请日：2014-06-17

Applicant: BASF SE

Inventor： FRASSETTO, Timo ,  DOCHNAHL, Maximilian ,  RACK, Michael ,  MAYWALD, Volker ,  WOLF, Bernd ,  GÖTZ, Roland ,  MÜLHEIMS, Philip ,  HÄBERLE, Rudolf

IPC: C07D265/36 ,  C07C17/16

CPC classification number: C07D265/36 ,  C07C17/16 ,  C07D413/04 ,  C07C21/22

Abstract: The present invention relates to a process for manufacturing 4-propargylated amino- benzoxazinones of formula (I), comprising the following steps: step a) preparing propargyl chloride by reacting propargyl alcohol with thionyl chloride optionally in the presence of a catalyst; and step b) reacting the propargyl chloride prepared in step (a) with a NH-benzoxazinone of formula (II); wherein the variables are defined according to the description.

Abstract translation: 本发明涉及一种制备式（I）的4-炔丙基化 - 苯并恶嗪酮的方法，包括以下步骤：步骤a）任选地在催化剂存在下，将炔丙醇与亚硫酰氯反应制备炔丙基氯; 和步骤b）使步骤（a）中制备的炔丙基氯与式（II）的NH-苯并嗪酮反应; 其中根据描述定义变量。

公开(公告)号：WO2014108286A1

公开(公告)日：2014-07-17

申请号：PCT/EP2013/077083

申请日：2013-12-18

Applicant: BASF SE

Inventor： ZIERKE, Thomas ,  GEBHARDT, Joachim ,  SCHÄFER, Peter ,  VOGELBACHER, Uwe Josef ,  RACK, Michael ,  LOHMANN, Jan Klaas

IPC: C07D301/02

CPC classification number: C07D301/02 ,  A01N43/653 ,  C07B2200/13 ,  C07D249/08

Abstract: The present invention relates to a process for the preparation of the compounds (II) from the respective oxo compounds. Furthermore, he invention relates to a process for the preparation of triazole compounds from oxiranes II.

Abstract translation: 本发明涉及由各种氧化合物制备化合物（II）的方法。 此外，本发明涉及从环氧乙烷II制备三唑化合物的方法。

公开(公告)号：WO2012168241A1

公开(公告)日：2012-12-13

申请号：PCT/EP2012/060600

申请日：2012-06-05

Applicant: BASF SE ,  WITSCHEL, Matthias ,  KRAUS, Helmut ,  HUTZLER, Johannes ,  NEWTON, Trevor, William ,  LERCHL, Jens ,  KREUZ, Klaus ,  GROßMANN, Klaus ,  EVANS, Richard, Roger ,  REINGRUBER, Rüdiger ,  PARRA RAPADO, Liliana ,  BESONG, Gilbert ,  RACK, Michael ,  KLOET, Andree van der ,  SEITZ, Thomas

Inventor： WITSCHEL, Matthias ,  KRAUS, Helmut ,  HUTZLER, Johannes ,  NEWTON, Trevor, William ,  LERCHL, Jens ,  KREUZ, Klaus ,  GROßMANN, Klaus ,  EVANS, Richard, Roger ,  REINGRUBER, Rüdiger ,  PARRA RAPADO, Liliana ,  BESONG, Gilbert ,  RACK, Michael ,  KLOET, Andree van der ,  SEITZ, Thomas

IPC: C07D497/04 ,  A01N43/60

CPC classification number: C07D497/04 ,  A01N43/90

Abstract: The present invention provides substituted pyrazine compounds of the formula (I) or N-oxides or agriculturally suitable salts thereof, wherein the variables in the formula (I) are defined as in the description. Substituted pyrazines of formula I are useful as herbicides.

Abstract translation: 本发明提供式（I）的取代的吡嗪化合物或其N-氧化物或农业上合适的盐，其中式（I）中的变量如描述中所定义。 式I的取代的吡嗪可用作除草剂。

公开(公告)号：WO2012146598A1

公开(公告)日：2012-11-01

申请号：PCT/EP2012/057517

申请日：2012-04-25

Applicant: BASF SE ,  DOCHNAHL, Maximilian ,  GEBHARDT, Joachim ,  KEIL, Michael ,  RACK, Michael ,  VOGELBACHER, Uwe Josef ,  GÖTZ, Roland ,  NOACK, Rainer

Inventor： DOCHNAHL, Maximilian ,  GEBHARDT, Joachim ,  KEIL, Michael ,  RACK, Michael ,  VOGELBACHER, Uwe Josef ,  GÖTZ, Roland ,  NOACK, Rainer

IPC: C07D405/06 ,  C07D249/12

CPC classification number: C07D405/06

Abstract: Preparation of 2-substituted 4-amino-2,4-dihydro-[1,2,4]triazole 3-thiones of the formula (I), by reacting 1-substituted 4-amino-4H-[1,2,4]-triazolium salts with sulfur in water or in a protic organic solvent or mixtures of such solvents in the presence of a base.

Abstract translation: 式（I）的2-取代的4-氨基-2,4-二氢 - [1,2,4]三唑-3-硫酮的制备，通过1-取代的4-氨基-4H- [1,2,4 ] - 三唑鎓盐与硫在水中或质子有机溶剂或这些溶剂的混合物在碱的存在下反应。

公开(公告)号：WO2012146535A1

公开(公告)日：2012-11-01

申请号：PCT/EP2012/057230

申请日：2012-04-20

Applicant: BASF SE ,  DOCHNAHL, Maximilian ,  GEBHARDT, Joachim ,  KEIL, Michael ,  RACK, Michael ,  VOGELBACHER, Uwe Josef ,  GÖTZ, Roland ,  NOACK, Rainer

Inventor： DOCHNAHL, Maximilian ,  GEBHARDT, Joachim ,  KEIL, Michael ,  RACK, Michael ,  VOGELBACHER, Uwe Josef ,  GÖTZ, Roland ,  NOACK, Rainer

IPC: C07D405/06 ,  C07D249/12

CPC classification number: C07D405/06 ,  C07D405/14

Abstract: Preparation of 2-substituted 2,4-dihydro-[1,2,4]triazole-3-thiones of the formula (III), comprising the steps i), diazotation of 2-substituted 4-amino-2,4-dihydro-[1,2,4]triazole- 3-thiones by treatment with inorganic nitrites and an acid or in the presence of organic nitrites in an organic solvent or water or mixtures thereof, giving the corresponding 4- diazo-2,4-dihydro-[1,2,4]triazole-3-thiones, and ii), reduction of the diazo intermediate to provide mixtures of compounds of the formula (III) and compounds of the formula (VII), by means of a reducing agent, followed by, iii), treating the reaction mixture with a reducing reagent suitable to cleave disulfide groups.

Abstract translation: 制备式（III）的2-取代的2,4-二氢 - [1,2,4]三唑-3-硫酮，包括步骤i），2-取代的4-氨基-2,4-二氢 - [1,2,4]三唑-3-硫酮通过用无机亚硝酸盐和酸或有机亚硝酸盐在有机溶剂或水或其混合物中的存在下处理，得到相应的4-重氮基-2,4-二氢 - [1,2,4]三唑-3-硫酮，和ii），通过还原剂还原重氮中间体以提供式（III）化合物和式（VII）化合物的混合物， 随后，iii）用适合于裂解二硫基的还原剂处理反应混合物。

公开(公告)号：WO2011161612A1

公开(公告)日：2011-12-29

申请号：PCT/IB2011/052681

申请日：2011-06-20

Applicant: BASF SE ,  MAYWALD, Volker ,  MENGES, Frederik ,  VOGELBACHER, Uwe Josef ,  RACK, Michael ,  KEIL, Michael ,  GRAMMENOS, Wassilios ,  VRETTOU-SCHULTES, Marianna ,  LOHMANN, Jan Klaas ,  MÜLLER, Bernd ,  JABS, Thorsten ,  BASF (CHINA) COMPANY LIMITED

Inventor： MAYWALD, Volker ,  MENGES, Frederik ,  VOGELBACHER, Uwe Josef ,  RACK, Michael ,  KEIL, Michael ,  GRAMMENOS, Wassilios ,  VRETTOU-SCHULTES, Marianna ,  LOHMANN, Jan Klaas ,  MÜLLER, Bernd ,  JABS, Thorsten

IPC: C07D213/68 ,  C07D213/61

CPC classification number: C07D213/68 ,  C07D213/08 ,  C07D213/61

Abstract: A process for preparing 4-hydroxypyridines of formula I, wherein R 1 , R 2 , R 3 and R 4 have the meaning defined in the description.

Abstract translation: 制备式I的4-羟基吡啶的方法，其中R1，R2，R3和R4具有说明书中定义的含义。