PIRIDIN-4-ILMETILAMIDAS
    31.
    发明专利

    公开(公告)号:PE20080107A1

    公开(公告)日:2008-04-18

    申请号:PE2007000160

    申请日:2007-02-14

    Applicant: BASF AG

    Abstract: SE REFIERE A UN COMPUESTO DE FORMULA I, DONDE R1 ES H, ALQUILO C1-C6, ALCOXI C1-C6, CIANO-ALQUILO C1-C4, HALOALQUILO C1-C4, ENTRE OTROS; R2, R3, R4 Y R5 SON CADA UNO H, HALOGENO, ALQUILO C1-C4, ALQUENILO C2-C4, HALOALCOXI C2-C4, ENTRE OTROS; R6 ES HALOGENO, CIANO, NITRO, ALQUILO C1-C10, ALQUENILO C2-C10, ENTRE OTROS; n ES 0-2. TAMBIEN SE REFIERE A COMPOSICIONES FARMACEUTICAS EN FORMA DE SOLUCIONES, EMULSIONES DIRECTAMENTE ROCIABLES, PASTAS, DISPERSIONES EN ACEITE. DICHOS COMPUESTOS SON UTILES PARA COMBATIR HONGOS FITOPATOGENOS, PLAGAS DE ARTROPODOS, EN PARTICULAR INSECTOS, ARACNIDOS, ENTRE OTROS

    3-(PYRIDIN-2-YL)-[1,2,4]-TRIAZINES FOR USE AS FUNGICIDES

    公开(公告)号:CA2648496A1

    公开(公告)日:2007-10-18

    申请号:CA2648496

    申请日:2007-04-11

    Applicant: BASF AG

    Abstract: The invention relates to 3-(pyridin-2-yl)-[1,2,4]-triazines of formula (I) a nd their use in the control of parasitic fungi and to herbicides that contain said compounds as an effective ingredient thereof. In formula (I), R1, R2 independently represent OH, halogen, NO2, NH2, C1-C8 alkyl, C1-C8 alkoxy, C1 - C8 halogenalkyl, C1-C8 halogenalkoxy, C1-C8 alkylamino or di(C1-C8 alkyl)amino, or they form, together with the C atoms to which they are bound , a saturated five-, six- or seven-membered carbocycle or heterocycle, which, in addition to the carbon ring members, has one or two heteroatoms selected fro m oxygen or sulfur as the ring members, the carbocycle and the heterocycle bei ng unsubstituted or having 1, 2, 3 or 4 C1-C4 alkyl groups as the substituents; R3 represents hydrogen, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy, C3-C6 cycloalkyl, C3-C6 cycloalkylmethyl, or halogen; R4 represents hydrogen, C1-C4 alkyl, C1-C4 alkoxy, C1-C4 halogenalkyl, C1-C4 halogenalkoxy or halogen; R5 represents C1-C8 alkyl, C1-C8 halogenalkyl, C1- C8 alkoxy, C1-C8 halogenalkoxy, C3-C8 cycloalkyl, C3-C8 cycloalkyloxy, five- or six-membered heteroaryl, phenyl, phenoxy, benzyl, benzyloxy, five- or six- membered heteroarylmethyl or five- or six-membered heteroaryloxy, said cycli c groups being unsubstituted or having 1, 2, 3, 4 or 5 groups Ra.

    Use of new or known imidazopyrimidine derivatives control phytopathogenic fungi

    公开(公告)号:DE102007012627A1

    公开(公告)日:2007-10-04

    申请号:DE102007012627

    申请日:2007-03-16

    Applicant: BASF AG

    Abstract: Imidazopyrimidine derivatives (I) are used to control phytopathogenic fungi. Imidazopyrimidine derivatives of formula (I) are used to control phytopathogenic fungi. R1>, R2>H, CN, NO2, 1-8C (halo)alkyl, 1-8C hydroxyalkyl, (1-4C)alkoxy(1-8C)alkyl, 2-8C (halo)alkenyl, 2-8C (halo)alkynyl, 1-8C (halo)alkoxy, 3-8C (halo)cycloalkyl, SR, SOR, SO2R, CHO, CSNH2, 1-8C alkylcarbonyl, 1-8C alkoxycarbonyl, 1-8C alkylcarbamoyl, 1-8C alkoximinocarbonyl, (1-8C)alkoximino(1-8C)alkyl, hydroximino(1-8C)alkyl, CRcRdORe or C(Rf)=NRg, optionally substituted; Rc, Rd, Re : H, R, 3-8C cycloalkyl, (1-8C)alkoxy(1-8C)alkyl, 2-8C alkenyl, 2-8C alkynyl, benzyl; Rd+Re : 1-5C alkylenedioxy optionally substituted with 1-2 of Me, Et, OH, OMe, OEt, CH2OH, CH2OMe, CH2OEt; Rf : H or R; Rg : R, 3-8C cycloalkyl, or optionally substituted phenyl or phenylamino; R : 1-8C alkyl; X : H, halo, OH, CN, NAA', 1-8C (halo)alkoxy,SR, SOR, SO2R, 1-8C (halo)alkyl, 2-8C (halo)alkenyl, 2-8C (halo)alkynyl, cyano(1-4C)alkyl or (1-4C)alkoxy(1-4C)alkyl; Y' : optionally substituted 5- to 10-membered heterocyclyl or optionally substituted phenyl; Z' : 1-10C (halo)alkyl, 2-10C (halo)alkenyl, 2-10C (halo)alkynyl, 3-10C (halo)cycloalkyl, 3-10C (halo)cycloalkenyl, (halo)phenyl, (halo)napthyl or 5- to 10-membered heterocyclyl, optionally substituted. Full definitions are given in the Definitions Field (Full Definitions). Independent claims are also included for: (1) compounds (I) in which Y and Z are not both optionally substituted phenyl, excluding 7-chloro-5-cycloheptyl-6-(2,4,6-trifluorophenyl)-imidazo[1,2-a]pyrimidine, 3-(4-(7-chloro-5-cycloheptyl-imidazo[1,2-a]pyrimidin-6-yl)-3,5-difluorophenoxy)-N,N-dimethyl-1-propanamine and N-(3-(4-(7-chloro-5-cyclohexyl-imidazo[1,2-a]pyrimidin-6-yl)-3,5-difluorophenoxy)propyl)-N,N-dimethylamine; (2) two processes for preparing (I); (3) imidazopyrimidine derivatives of formula (VI) and their hydrolysis products. X" : H or 1-7C alkyl; R : 1-4C alkyl. [Image] [Image] ACTIVITY : Plant antifungal. No biological data given. MECHANISM OF ACTION : None given.

    New amino-pyridinoazine derivatives, useful as fungicides for protection of plants and materials, also new intermediates in their synthesis

    公开(公告)号:DE102005051514A1

    公开(公告)日:2007-05-03

    申请号:DE102005051514

    申请日:2005-10-26

    Applicant: BASF AG

    Abstract: Amino-substituted pyridinoazines (I) are new. Amino-substituted pyridinoazines of formula (I) are new. R1>1-14C alkyl, 1-12C alkoxy(1-12C)alkyl, 1-6C alkoxy(2-12C)-alkenyl or -alkynyl, 5-8C cycloalkyl, phenyl, phenyl(1-4C)alkyl, 2-12C alkenyl or alkynyl, where the carbon chain may be substituted by 1-3, same or different, Ra> and/or Rb>; Ra>halo, cyano, nitro, hydroxy, 1-6C alkylthio, 3-12C alkenyloxy or alkynyloxy, NR11>R12>, or phenyl or 3-6C cycloalkyl optionally substituted by 1-4, same or different, Rb>, and carbon chains in Ra> may themselves be halogenated; Rb>halo, cyano, hydroxy, mercapto, 1-6C (halo)alkyl, 3-8C cycloalkyl, 2-10C alkenyl or alkynyl, 1-6C alkoxy or alkylthio, 1-6C alkoxy(1-6C)alkyl or NR11>R12>; R11> and R12>hydrogen or 1-6C alkyl; R2>1-12C alkyl, or 2-12C alkenyl or alkynyl, optionally substituted by 1-3 Rc>; Rc>cyano, nitro, hydroxy, NR11>R12> or 3-6C cycloalkyl (optionally substituted by 1-4 of, same or different, 1-4C alkyl, halo, cyano, nitro, hydroxy, 1-6C alkoxy or alkylthio, 3-6C alkenyloxy or alkynyloxy, or NR11>R12>; W1 and X1, W1 and Y1, W1 and Z1, X1 and Y1, X1 and Z1, or Y1 and Z1 each : N and the others CR3>, or W1, Z1 and one of X1 and Y1 = N and the other CR3>; each R3>hydrogen, halo, or 1-4C alkyl or alkoxy . Independent claims are included for the following: (1) several methods for preparing (I); (2) intermediates of formulae (V), (VI), (VII) and (IX); and (3) seeds treated with (I) at 1-1000 g per 100 kg. in (VI) and (VII) X on the pyrido ring : halo; R22>hydrogen or 1-11C alkyl; R : 1-4C alkyl . [Image] [Image] ACTIVITY : Plant Antifungal. No details of tests for antifungal activity are given. MECHANISM OF ACTION : None given.

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