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    SUBSTITUTED 5-HETARYLPYRIMIDINES
    2.
    发明申请
    SUBSTITUTED 5-HETARYLPYRIMIDINES 审中-公开
    取代的5 HETARYLPYRIMIDINE

    公开(公告)号：WO2007113322A2

    公开(公告)日：2007-10-11

    申请号：PCT/EP2007053332

    申请日：2007-04-04

    Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MUELLER BERND ,  ULMSCHNEIDER SARAH

    Inventor： RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MUELLER BERND ,  ULMSCHNEIDER SARAH

    CPC classification number: C07D401/04 ,  A01N43/54

    Abstract: The invention relates to 5-hetaryl-4-pyrimidines of formula (I) and to their salts and plant protection agents which contain at least one compound of said type as an active component, wherein W represents oxygen, sulphur, a group S=O or S(=O) 2 ; R 1 represents optionally substituted C 1 -C 8 -alkyl, C 3 -C 8 -cycloalkyl, C 5 -C 10 -bicycloalkyl, C 2 -C 8 -alkenyl, C 4 -C 10 -alkadienyl, C 3 -C 6 -cycloalkenyl, C 2 -C 8 -alkynyl, phenyl, naphthyl, or a C-bound five- or six-membered saturated, partially unsaturated or aromatic heterocycle containing one, two, three or four heteroatoms from the groups O, N or S as ring members; R 2 represents halogen, cyano, hydroxy, mercapto, N 3 , C 1 -C 6 -alkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkynyl, C 1 C 6 -halogenalkyl, C 1 C 6 -alkoxy, C 3 -C 8 -alkenyloxy, C 3 -C 8 -alkynyloxy, C 1 C 6 -halogenalkoxy, C 1 -C 6 -alkylthio, C 3 -C 8 -alkenylthio, C 3 -C 8 -alkynylthio, C 1 -C 6 -halogenalkylthio, or a radical of formulae C(=Z)OR 21 , C(=Z)NR 22 R 23 , C(=Z)NR 24 -NR 22 R 23 , C(=Z)R 25 , CR 26 R 27 -OR 28 , CR 26 R 27 -NR 22 R 23 , ON(=CR 29 R 30 ), O-C(=Z)R 25 , NR 22 R 23a , NR 31 (C(=Z)R 25 ), NR 31 (C(=Z)OR 21 ), NR 31 (C(=Z)-NR 22 R 23 ), NR 32a (N=CR 29 R 30 ), NR 32 NR 22 R 23 , NR 32 OR 21 , or C(=N-Z'-R 25 )SR 21 ; or a cyclic radical; R3 represents hydrogen, OH, halogen, cyano, NR 37 R 38 , C 1 -C--alkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylsulfinyl, C 1 -C--alkylsulfonyl, C 2 -C 8 -alkenyl or C 2 -C 8 -alkinyl, whereby the seven latter radicals can be partially or totally halogenated and/or optionally can support one, two or three substitutes, selected among nitro, cyano, OH, C 1 -C 2 -alkoxy, C 1 -C 4 -alkoxycarbonyl, amino, C 1 -C 4 -alkylamino and Di-C 1 -C 4 -alkylamino, Het represents a substituted C- or N-bound, 5-or 6-membered aromatic heterocycle which comprises 1, 2, 3 or 4 heteroatoms as ring members selected among nitrogen, oxygen and sulphur. The invention also relates to the use of 5-hetaryl-4-pyrimidines of formula (I) and there salts for combating plant pathogenic fungi.

    Abstract translation: 本发明涉及式（I）的包含至少一种这样的化合物作为有效成分的5-杂芳基-4-嘧啶和它们的盐和杀虫剂。 其中W = O或S（= O） 2 表示氧，硫，基团S; [R 1 表示任选subsitituiert.esç 1 -C 8 烷基，C 3 -C 8 环烷基，C 5 -C 10 双环，C 2 -C 8 - 烯基，C 4 -C 10 链二烯基，C 3 -C 6 环烯基，C 2 -C 8 是炔基，苯基，萘基或C-连接的五元或六元饱和，部分不饱和或芳族的含有一个，两个，三个或四个杂原子的从杂环 包含基团的O，N或S作为环成员; [R 2 表示卤素，氰基，羟基，巯基，N 3 ，C 1 -C 6 烷基， ç 2 -C 8 烯基，C 2 -C 8 - 炔基，C 1 < / SUB> C 6 卤代烷基，C 1 C 6 烷氧基，C 3 -C 8 烯，C 3 -C 8 炔氧基，C 1 C 6 卤代烷氧基 ，C 1 -C 6 烷硫基，C 3 -C 8 烯，C 3 -C 8 炔硫基，C 1 -C 6 卤代烷硫基，或一个基团，式C（= Z） OR 21 ，C（= Z）NR 22 - [R 23 ，C（= Z）NR 24 -NR 22 - [R 23 ，C（= Z）R 25 ，CR 26 - [R 27 -OR 28 ，CR 26 - [R 27 -NR 22 - [R 23 ， ON（= CR 29 - [R 30 ），OC（= Z）R 25 ，NR 22 - [R 图23A ，NR 31 （C（= Z）R 25 ），NR 31 （C（= Z）OR < SUP> 21 ）NR 31 （ C（= Z）-NR 22 - [R 23 ），NR 32A （N = CR 29 - [R 30 ），NR 32 NR 22 - [R 23 ，NR 32 OR 21 ，或C（= N-Z'-R 25 ）SR 21 ; 或环状基团; R 3是氢，OH，卤素，氰基，NR 37 - [R 38 ，C 1 -C - 烷基，C 1 -C 8 烷氧基，C 1 -C 8 烷硫基，C 1 -C 8 烷基亚磺酰基，C 1 -C - 烷基磺酰基，C 2 -C 8 链烯基或C 2 -C 8 炔基，其中所述7最后提到的基团可以部分或完全卤化和/或选自硝基一个，两个或三个取代基，氰基，OH，C 1 -C 2 烷氧基，C 1 -C 4 烷氧基羰基，氨基，C 1 -C 4 烷基氨基和二C 1 -C 4可携带>烷基氨基，

    AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME
    4.
    发明申请
    AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME 审中-公开
    Azolylmethyloxiranes，及其用于防治病原真菌植物及代理人含

    公开(公告)号：WO2008012234A2

    公开(公告)日：2008-01-31

    申请号：PCT/EP2007057353

    申请日：2007-07-17

    Applicant: BASF AG ,  DIETZ JOCHEN ,  GROTE THOMAS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH ,  GLAETTLI ALICE

    Inventor： DIETZ JOCHEN ,  GROTE THOMAS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH ,  GLAETTLI ALICE

    IPC: C07D405/14 ,  A01N43/707 ,  C07D409/14

    CPC classification number: C07D405/14 ,  A01N43/653 ,  C07D409/14

    Abstract: The invention relates to azolylmethyloxiranes of general formula (I), wherein A or B is benzodioxolyl which is optionally substituted by between one and five of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, said substituents being optionally substituted by between one and three of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio. The invention also relates to the plant-tolerant acid addition salts or metal salts of said compounds, to the use of the compounds of formula (I) for controlling plant-pathogenic fungi, and to agents containing the same.

    Abstract translation: 本发明涉及通式（I），其中A或B是苯并二的azolylmethyloxirane其任选地被一个取代以下substi- tuenten卤素，CN，NO 2 ，氨基，C <五 SUB> 1 -C 4 烷基，C 1 -C 4 烷氧基，C 1 -C 4 - 卤代烷基，C 1 -C 4卤代烷，C 1 -C 4 烷基氨基， ç 1 -C 4 二烷基氨基，硫代，或C 1 -C 4 是烷硫基，被取代的，和 各其他取代基A或B为苯基或5元或6元杂芳基，所述取代基任选地被1-3个下列取代基取代：卤素，CN，NO 2 ，氨基，C < SUB> 1 -C 4 烷基，C 1 -C 4 烷氧基，C 1 -C 4 卤代烷基，C 1 -C 4 - 卤代烷氧基，C 1 -C 4 - 烷基氨基，C 1 -C 4 二烷基氨基，巯基或C 1 -C 4 - 烷硫基，被取代的，和它们的植物耐受的酸加成盐或金属盐，使用式（I）的用于控制植物病原真菌包含它们的化合物和试剂。

    5.
    发明专利
    未知

    公开(公告)号：BRPI0712704A2

    公开(公告)日：2012-07-03

    申请号：BRPI0712704

    申请日：2007-06-15

    Applicant: BASF AG

    Inventor： DIETZ JOCHEN ,  GROTE THOMAS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH ,  GLOTTLI ALICE

    IPC: C07D405/06 ,  A01N43/653 ,  A01N43/74 ,  A01P3/00 ,  C07D405/14 ,  C07D409/14 ,  C07D413/14 ,  C07D417/14

    Abstract: The present invention relates to azolylmethyloxiranes of the general formula I in which A is phenyl which is substituted by two F, B is unsubstituted pyridyl, thienyl, thiazolyl, oxazolyl or furyl or is phenyl which is optionally substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, thio or C1-C4-alkylthio, with the proviso that B is not o-methylphenyl if A is 2,4-difluorophenyl, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

    New 2-substituted pyrimidine derivatives, useful for controlling phytopathogenic fungi and for controlling animal pests in agriculture
    10.
    发明专利
    New 2-substituted pyrimidine derivatives, useful for controlling phytopathogenic fungi and for controlling animal pests in agriculture 未知

    公开(公告)号：DE102005046592A1

    公开(公告)日：2007-03-29

    申请号：DE102005046592

    申请日：2005-09-28

    Applicant: BASF AG

    Inventor： RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MUELLER BERND ,  LOHMANN JAN KLAAS ,  GRAMMENOS WASSILIOS ,  HUENGER UDO ,  SCHIEWECK FRANK ,  ULMSCHNEIDER SARAH ,  DIETZ JOCHEN ,  RENNER JENS ,  SPEAKMAN JOHN-BRYAN ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  STIERL REINHARD

    IPC: C07D413/04 ,  A01N43/54 ,  A01N43/72 ,  A01N43/80 ,  C07D239/42 ,  C07D413/14

    Abstract: 2-Substituted pyrimidine derivatives (I) are new. 2-Substituted pyrimidine derivatives of formula (I) and their salts are new. R 1>, R 11>1-8C (halo)alkyl, 2-8C (halo)alkenyl, 2-8C (halo)alkynyl, 3-6C (halo)cycloalkyl or 4-6C (halo)cycloalkenyl, or R 1>+R 11>forms a 5- to 7-membered ring optionally containing another heteroatom (O, N or S); R 1>and R 11>are optionally substituted with 1-4 of R 2>and two substituents on adjacent ring atoms can form 1-6C alkylene, 2-4C oxyalkylene or 1-3C alkylenedioxy; R 2>halo, CN, 1-6C (halo)alkyl, 3-6C (halo)cycloalkyl, 4-6C cycloalkenyl, OH, 1-6C (halo)alkoxy, 2-8C alkenyloxy, 2-8C alkynyloxy, 3-6C cycloalkoxy, 4-6C cycloalkenyloxy, 1-6C alkylthio, =CH 2, =C(1-4C alkyl) 2, COA, COOA, CONAA', C(A')(NOA), NAA', NA'COA, NA"CONAA', SO mA, SO mOA, SO mNAA', Si(1-6C alkyl) 3, or phenyl optionally substituted with 1-3 of halo, 1-6C (halo)alkyl, 2-6C alkenyl, 2-6C alkynyl, 3-6C cycloalkyl, 1-6C alkoxy, CN, NO 2, COA, COOA, CONAA', C(A')(NOA), NAA'; m : 0-2; A, A', A" : H, 1-6C alkyl, 2-6C alkenyl, 2-6C alkynyl, 3-6C cycloalkyl, 3-8C cycloalkenyl or phenyl, all optionally halogenated and/or substituted with NO 2, OCN, CN, 1-4C alkoxy, or A+A' forms a 5- or 6-membered ring with 1-4 heteroatoms (O, N, S); R 3>halo, CN, N 3, 1-4C (halo)alkyl, 2-4C (halo)alkenyl, 2-4C (halo)alkynyl, 3-6C (halo)cycloalkyl, 1-4C alkoxy, 3-4C alkenyloxy, 3-4C alkynyloxy, 1-6C alkylthio, di(1-6C alkyl)amino or 1-6C alkylamino, all optionally substituted with 1-4 of halo, CN,, NO 2, 1-2C alkoxy and 1-4C alkoxycarbonyl; R 4>5- or 6-membered heterocyclyl with 1-4 heteroatoms (O, N, S), optionally halogenated and/or substituted with 1-4 of Ru; or CN, CZORa, CZNRzRb, CZNRaNRzRb, CZRa, CRaRbORz, CRaRbNRzRc, ON=CRaRb, OCZRa, NRaRb', NRaCZRb, NRaCZORb, NRaCZNRzRb, NRaN=CRcRb, NRaNRzRb or NRzORa; Ru : halo, CN, 1-8C (halo)alkyl, 2-8C (halo)alkenyl, 2-8C (halo)alkynyl, 1-6C (halo)alkoxy, 3-6C (halo)cycloalkyl, 2-8C alkenyloxy, 2-8C alkynyloxy, 4-6C cycloalkenyl, 3-6C cycloalkoxy, 4-6C cycloalkenyloxy, COA, COOA, CONAA', C(A')(NOA), NAA', NA'COA, NA"CONAA', SO mA, SO mOA, SO mNAA'; Z : O, S, NRd, NORd or NNRzRc; Rb' : 1-6C alkyl, 2-6C alkynyl, 2-6C alkynyl, 3-6C cycloalkyl or 4-6C cycloalkenyl; Ra, Rb, Rc, Rd : H or Rb'; Rz : Ra, CORd or COORd; B : 5- or 6-membered heteroaryl with 1-4 heteroatoms (O, N, S), or phenyl; L : halo, CN, OCN, 1-8C (halo)alkyl, 2-8C (halo)alkenyl, 2-8C (halo)alkynyl, 1-6C (halo)alkoxy, 3-6C (halo)cycloalkyl, 2-8C alkenyloxy, 2-8C alkynyloxy, 4-6C cycloalkenyl, 3-6C cycloalkoxy, 4-6C cycloalkenyloxy, COA, COOA, CONAA', C(A')(NOA), NAA', NA'COA, NA"CONAA', SO mA, SO mOA, SO mNAA', optionally substituted with 1-4 of RL; RL : halo, CN, 1-6C alkoxy, 3-6C cycloalkyl, 2-8C alkenyloxy, 2-8C alkynyloxy, 4-6C cycloalkenyl, 3-6C cycloalkoxy, 4-6C cycloalkenyloxy, COA, COOA, CONAA', C(A')(NOA), NAA', NA'COA, NA"CONAA', SO mA, SO mOA, SO mNAA'; and n : 1-5. Ra, Rb, Rc, Rd, Rb', Rz Are optionally halogenated and/or substituted with 1-4 of halo, CN, 1-8C alkyl, 2-10C alkenyl, 2-10C alkynyl, 1-6C alkoxy, 2-10C alkenyloxy, 2-10C alkynyloxy, 3-6C cycloalkyl, 3-6C cycloalkenyl, 3-6C cycloalkoxy, 3-6C cycloalkenyloxy; and two of Ra, Rb, Rc, Rz can form a 5- or 6-membered ring with 1-4 heteroatoms (O, N, S). Independent claims are also included for: (1) combination of at least one compound (I) and at least one other fungicide, insecticide and/or herbicide; (2) controlling phytopathogenic fungi by treating the fungi and/or materials, plants, soil or seeds to be protected from fungal attack with at least one compound (I); (3) controlling animal pests in agriculture by treating the pests and/or materials, plants, soil or seeds to be protected from them with at least one compound (I); (4) seeds comprising a compound (I) in an amount of 1-1000 g/100 kg. [Image] ACTIVITY : Plant antifungal. In a protective test against Alternaria solanion tomato plants, plants treated with 2-(1,2,4-triazol-1-yl)-4-chloro-5-(2-chloro-4-fluorophenyl)-6-(N-methoxy-N-methylamino)-pyrimidine (250 ppm) showed no more than 20% attack after 5 days, compared with 90% for control plants. MECHANISM OF ACTION : None given.

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