公开(公告)号：JP2002047262A

公开(公告)日：2002-02-12

申请号：JP2001207021

申请日：2001-07-06

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: C07C251/80 ,  A01N33/26 ,  A01N37/50 ,  C07C249/16 ,  C07C251/86

Abstract: PROBLEM TO BE SOLVED: To provide a compound that has increased controlling effect against harmful fungi. SOLUTION: The objective salicylic acid derivative is represented by formula I [wherein X is a halogen, NO2, cyano, an alkyl or an alkoxy; (m) is 0, 1, 2 or 3 where in the case m >=2, X may differ from each other; A is OH, an alkoxy, NH2, NHCH3 or N(CH3)2, R1 is phenyl, naphthyl, cycloalkyl, one to three N-atoms and/or one O or S atom or one or two O and/or S atoms- including 5-membered or 5-membered ring heteroaryl or 5-membered or 6-membered heterocyclyl where the ring structure may be unsubstituted or substituted; and R2 is H, cyano, an alkyl, an alkenyl, an alkynyl, a haloalkyl, an alkoxy or an alkylthio]. This invention further provides a method of producing the derivative, a composition including the derivative and the use of the composition for controlling harmful fungi.

公开(公告)号：JP2003201289A

公开(公告)日：2003-07-18

申请号：JP2002272397

申请日：2002-09-19

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED

IPC: A01N43/16 ,  C07C45/46 ,  C07C45/54 ,  C07C49/84 ,  C07D311/86

Abstract: PROBLEM TO BE SOLVED: To provide a compound effective for controlling hazardous phytopathogenic fungi, to provide a method for producing the compound, to provide a composition containing the compound, and to provide a method for using the composition. SOLUTION: This compound comprises a xanthone derivative expressed by general formula (I) (n is 0, 1 or 2; R 1 is an alkyl or the like; R 2 and R 3 are each an alkoxy or the like, or together form an oxyalkyleneoxy which may be substituted; R 4 is a halogen or the like; R 5 is equal to the R 4 , provided that R 5 s may be different from each other when n is 2; and X and Y are each O or S). The method for producing the compound and the composition containing the compound are provided in the specification, respectively. The composition is used for controlling the hazardous phytopathogenic fungi. COPYRIGHT: (C)2003,JPO

公开(公告)号：JP2002030058A

公开(公告)日：2002-01-29

申请号：JP2001182539

申请日：2001-06-15

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N37/28 ,  A01N37/34 ,  A01N37/40 ,  A01N37/46 ,  A01N47/20 ,  A01N47/30 ,  C07B61/00 ,  C07C249/16 ,  C07C251/86 ,  C07C253/30 ,  C07C255/59 ,  C07C255/64 ,  C07C255/66 ,  C07C269/04 ,  C07C271/28 ,  C07C273/18 ,  C07C275/42

Abstract: PROBLEM TO BE SOLVED: To provide a compound improved in controlling actions on noxious fungi. SOLUTION: This salicylohydrazide derivative is represented by the formula I (wherein, X is a halogen, NO2, cyano, a 1-4C alkyl or a 1-4C alkoxy; (m) is 0, 1, 2 or 3; R1 is NO2, NH2 or NH-CO-A; A is hydrogen, 1-4C alkyl, a 1-4C alkoxy, NH2, NHCH3 or N(CH3)2; R2 is hydrogen, cyano, a 1-6C alkyl, a 2-6C alkeiyl, a 2-6C alkynyl, a 1-6C haloalkyl, a 1-6C alkoxy or a 1-6C alkylthio; and R3 is phenyl, naphthyl, a 3-10C cycloalkyl, a 5- or a 6-membered ring heteroaryl or a 5- or a 6-membered ring heterocyclyl). The method for producing the salicylohydrazide derivative is provided and an intermediate for producing the derivative is obtained. The composition for controlling the noxious fungi comprises the derivative.

公开(公告)号：JP2003206252A

公开(公告)日：2003-07-22

申请号：JP2002313232

申请日：2002-10-28

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  CARTER PAUL ,  CURTZE JUERGEN

IPC: A01N31/14 ,  A01N31/16 ,  A01N33/10 ,  A01N37/38 ,  A01N37/40 ,  C07B61/00 ,  C07C39/42 ,  C07C41/26 ,  C07C43/23 ,  C07C69/017 ,  C07C69/14 ,  C07C323/19 ,  C07C323/25

Abstract: PROBLEM TO BE SOLVED: To provide a benzhydryl derivative that exhibits high effect in the control of deleterious fungi. SOLUTION: The benzhydryl derivative is represented by formula I (wherein X is O or S; R 1 , R 3 are each a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkenyl, an alkynyl, an alkoxy, an alkenyloxy, an alkynyloxy, an alkyklcarbonyloxy, formyloxy or alkylthio or the like; R 2 is a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkoxy, a haloalkyl, or a haloalkoxy wherein in the case that n=2, R 2 may differ from each other; R 4 is an alkyl, an alkenyl or an alkynyl; R 5 and R 6 are each hydroxyl, an alkyl, an alkenyl, a haloalkyl, a haloalkenyl, an alkoxy or an alkenyloxy; m is 0, 1 or 2). COPYRIGHT: (C)2003,JPO

公开(公告)号：JPH11335361A

公开(公告)日：1999-12-07

申请号：JP2568099

申请日：1999-02-03

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  SAUTER HUBERT ,  BAYER HERBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GOETZ ROLAND ,  MUELLER BERND ,  PTOCK ARNE ,  ROEHL FRANZ ,  HARRIES VOLKER ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

IPC: A01N43/653 ,  A01N43/76 ,  C07C271/10 ,  C07D249/12 ,  C07D263/44 ,  C07D403/12 ,  C07D413/12

Abstract: PROBLEM TO BE SOLVED: To obtain the subject new compound useful for controlling harmful animals and harmful fungi. SOLUTION: This compound is shown by formula I Y is a halogen, a 1-4C alkyl or the like; (n) is 0-2; E is a group of formula II (V is O or the like); T is O or oxymethylene; Z is a group X [X is a (substituted) heterocyclyl, a (substituted) aryl or the like], N=CWR [W is a (substituted) 1-6C alkyl or the like; R is H, cyano or the like] or the like} such as N-methyl-5-[2-(o-tolyloxymethylene)phenyl]-1,3- oxazolidine-2,4-dione.The compound of formula I, for example, in the case in which it is a compound of formula III, is obtained by a process for acylating an alkyl α- hydroxy-α-phenylacetate with phosgene or the like to give a compound of formula IV and further reacting the compound with a primary amine of the formula H2 N-R αto cause a ring formation and in the case of not advancing the ring formation by the strength of the amine, by a process for hydrolyzing an ester amide of formula V, then treating the resultant substance with an acid and reacting the treated substance with a compound of the formula Z-OH.

公开(公告)号：WO2007113322A2

公开(公告)日：2007-10-11

申请号：PCT/EP2007053332

申请日：2007-04-04

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MUELLER BERND ,  ULMSCHNEIDER SARAH

Inventor： RHEINHEIMER JOACHIM ,  GROTE THOMAS ,  MUELLER BERND ,  ULMSCHNEIDER SARAH

CPC classification number: C07D401/04 ,  A01N43/54

Abstract: The invention relates to 5-hetaryl-4-pyrimidines of formula (I) and to their salts and plant protection agents which contain at least one compound of said type as an active component, wherein W represents oxygen, sulphur, a group S=O or S(=O) 2 ; R 1 represents optionally substituted C 1 -C 8 -alkyl, C 3 -C 8 -cycloalkyl, C 5 -C 10 -bicycloalkyl, C 2 -C 8 -alkenyl, C 4 -C 10 -alkadienyl, C 3 -C 6 -cycloalkenyl, C 2 -C 8 -alkynyl, phenyl, naphthyl, or a C-bound five- or six-membered saturated, partially unsaturated or aromatic heterocycle containing one, two, three or four heteroatoms from the groups O, N or S as ring members; R 2 represents halogen, cyano, hydroxy, mercapto, N 3 , C 1 -C 6 -alkyl, C 2 -C 8 -alkenyl, C 2 -C 8 -alkynyl, C 1 C 6 -halogenalkyl, C 1 C 6 -alkoxy, C 3 -C 8 -alkenyloxy, C 3 -C 8 -alkynyloxy, C 1 C 6 -halogenalkoxy, C 1 -C 6 -alkylthio, C 3 -C 8 -alkenylthio, C 3 -C 8 -alkynylthio, C 1 -C 6 -halogenalkylthio, or a radical of formulae C(=Z)OR 21 , C(=Z)NR 22 R 23 , C(=Z)NR 24 -NR 22 R 23 , C(=Z)R 25 , CR 26 R 27 -OR 28 , CR 26 R 27 -NR 22 R 23 , ON(=CR 29 R 30 ), O-C(=Z)R 25 , NR 22 R 23a , NR 31 (C(=Z)R 25 ), NR 31 (C(=Z)OR 21 ), NR 31 (C(=Z)-NR 22 R 23 ), NR 32a (N=CR 29 R 30 ), NR 32 NR 22 R 23 , NR 32 OR 21 , or C(=N-Z'-R 25 )SR 21 ; or a cyclic radical; R3 represents hydrogen, OH, halogen, cyano, NR 37 R 38 , C 1 -C--alkyl, C 1 -C 8 -alkoxy, C 1 -C 8 -alkylthio, C 1 -C 8 -alkylsulfinyl, C 1 -C--alkylsulfonyl, C 2 -C 8 -alkenyl or C 2 -C 8 -alkinyl, whereby the seven latter radicals can be partially or totally halogenated and/or optionally can support one, two or three substitutes, selected among nitro, cyano, OH, C 1 -C 2 -alkoxy, C 1 -C 4 -alkoxycarbonyl, amino, C 1 -C 4 -alkylamino and Di-C 1 -C 4 -alkylamino, Het represents a substituted C- or N-bound, 5-or 6-membered aromatic heterocycle which comprises 1, 2, 3 or 4 heteroatoms as ring members selected among nitrogen, oxygen and sulphur. The invention also relates to the use of 5-hetaryl-4-pyrimidines of formula (I) and there salts for combating plant pathogenic fungi.

Abstract translation: 本发明涉及式（I）的包含至少一种这样的化合物作为有效成分的5-杂芳基-4-嘧啶和它们的盐和杀虫剂。 其中W = O或S（= O） _{2 表示氧，硫，基团S; [R ^{1 表示任选subsitituiert.esç 1 -C 8 烷基，C 3 -C 8 环烷基，C 5 -C 10 双环，C 2 -C 8 - 烯基，C 4 -C 10 链二烯基，C 3 -C 6 环烯基，C 2 -C 8 是炔基，苯基，萘基或C-连接的五元或六元饱和，部分不饱和或芳族的含有一个，两个，三个或四个杂原子的从杂环 包含基团的O，N或S作为环成员; [R 2 表示卤素，氰基，羟基，巯基，N 3 ，C 1 -C 6 烷基， ç 2 -C 8 烯基，C 2 -C 8 - 炔基，C 1 < / SUB> C 6 卤代烷基，C 1 C 6 烷氧基，C 3 -C 8 烯，C 3 -C 8 炔氧基，C 1 C 6 卤代烷氧基 ，C 1 -C 6 烷硫基，C 3 -C 8 烯，C 3 -C 8 炔硫基，C 1 -C 6 卤代烷硫基，或一个基团，式C（= Z） OR 21 ，C（= Z）NR 22 - [R 23 ，C（= Z）NR 24 -NR 22 - [R 23 ，C（= Z）R 25 ，CR 26 - [R 27 -OR 28 ，CR 26 - [R 27 -NR 22 - [R 23 ， ON（= CR 29 - [R 30 ），OC（= Z）R 25 ，NR 22 - [R 图23A ，NR 31 （C（= Z）R 25 ），NR 31 （C（= Z）OR < SUP> 21 ）NR 31 （ C（= Z）-NR 22 - [R 23 ），NR 32A （N = CR 29 - [R 30 ），NR 32 NR 22 - [R 23 ，NR 32 OR 21 ，或C（= N-Z'-R 25 ）SR 21 ; 或环状基团; R 3是氢，OH，卤素，氰基，NR 37 - [R 38 ，C 1 -C - 烷基，C 1 -C 8 烷氧基，C 1 -C 8 烷硫基，C 1 -C 8 烷基亚磺酰基，C 1 -C - 烷基磺酰基，C 2 -C 8 链烯基或C 2 -C 8 炔基，其中所述7最后提到的基团可以部分或完全卤化和/或选自硝基一个，两个或三个取代基，氰基，OH，C 1 -C 2 烷氧基，C 1 -C 4 烷氧基羰基，氨基，C 1 -C 4 烷基氨基和二C 1 -C 4可携带>烷基氨基，}}

公开(公告)号：WO2005018328A8

公开(公告)日：2006-03-09

申请号：PCT/EP2004007397

申请日：2004-07-07

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： TORMO I BLASCO JORDI ,  GROTE THOMAS ,  SCHERER MARIA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  A01N43

CPC classification number: A01N43/90 ,  A01N2300/00

Abstract: Disclosed are fungicidal mixtures containing 1) a triazolopyrimidine derivative of formula (I) and 2) epoxiconazole of formula (II) as active components at a synergistically effective quantity, a method for controlling harmful fungi of the class

Abstract translation: 一种杀真菌混合物，其包含作为活性组分1）式（I）的三唑并嘧啶衍生物，以及2）在协同有效量的式（II）的氟环唑，对于从类<我的防治有害真菌的方法

公开(公告)号：WO2005087770A3

公开(公告)日：2005-12-08

申请号：PCT/EP2005002424

申请日：2005-03-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD ,  HUENGER UDO

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD ,  HUENGER UDO

IPC: C07D487/04

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R and/or R being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

Abstract translation: 5,6-二烷基 - 7-氨基三唑并嘧啶，其中取代基具有式（I）的以下含义：R t <1>是烷基，烷氧基烷基，烯基或炔基; [R <2>是烷基，烷氧基烷基，烯基或炔基; 其中R <1>和/或R <2>取代根据描述; 一种用于制备这些化合物，含有它们和它们在防治植物病原性有害真菌的用途的组合物的过程。

公开(公告)号：WO2004045288A2

公开(公告)日：2004-06-03

申请号：PCT/EP0312769

申请日：2003-11-14

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

Inventor： TORMO I BLASCO JORDI ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH

IPC: A01N43/90 ,  A01N35/00

CPC classification number: A01N43/90 ,  A01N35/04 ,  A01N2300/00

Abstract: Disclosed are fungicidal mixtures for controlling rice pathogens, containing a synergistically effective amount of 1) a compound of formula (I), and 2) a compound of formula (II) as active components, methods for controlling destructive fungi by means of mixtures of compound I and compound II, the use of compounds I and II for producing such mixtures, and agents containing said mixtures.

Abstract translation: 一种用于在协同有效量控制水稻病原体，其包含作为活性组分：1）式（I的化合物），和2）式（II化合物）的杀真菌混合物，用于控制使用I的化合物的混合物与化合物有害真菌的方法 II，使用化合物I和II在制备该类混合物和包含这些混合物的组合物。

公开(公告)号：WO2004041824A2

公开(公告)日：2004-05-21

申请号：PCT/EP0312276

申请日：2003-11-04

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07C69/65 ,  C07C69/76 ,  C07D487/04

CPC classification number: C07C69/65 ,  A01N43/90 ,  C07D487/04

Abstract: Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula (I) in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R and R radicals may be substituted as defined in the description, R denote hydrogen, or a group mentioned for R ; or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L , L independently denote hydrogen, halogen, or alkyl; L is hydrogen, halogen, haloalkyl, or NH2, NHR , or N(Rb)2, wherein Rb is as defined in the description,wherein at least one from L , L , and L is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 取代的式（I）的6-（2-卤代苯基） - 三唑并嘧啶，其中R1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元饱和，不饱和或 芳族杂环，其含有1-4个氮原子或一至三个氮原子和一个硫或氧原子，其中R 1和R 2基团可以如说明书中所定义地被取代，R 2表示氢，或 R 1中提到的基团; 或R 1和R 2连同相邻的氮原子表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环，该环可以被取代 如说明书中所定义的; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或N（R b）2，其中R b如说明书中所定义，其中至少一个L 1，L 2， 而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基，它们的制备方法，含有它们的组合物和它们用于防治植物病原性真菌的用途。