AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME
    1.
    发明申请
    AZOLYLMETHYLOXIRANES, USE THEREOF FOR CONTROLLING PLANT PATHOGENIC FUNGI, AND AGENTS CONTAINING THE SAME 审中-公开
    Azolylmethyloxiranes,及其用于防治病原真菌植物及代理人含

    公开(公告)号:WO2008012234A2

    公开(公告)日:2008-01-31

    申请号:PCT/EP2007057353

    申请日:2007-07-17

    CPC classification number: C07D405/14 A01N43/653 C07D409/14

    Abstract: The invention relates to azolylmethyloxiranes of general formula (I), wherein A or B is benzodioxolyl which is optionally substituted by between one and five of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio, and the respective other substituent A or B is phenyl or 5-membered or 6-membered heteroaryl, said substituents being optionally substituted by between one and three of the following substituents, halogen, CN, NO 2 , amino, C 1 -C 4 alkyl, C 1 -C 4 alkoxy, C 1 -C 4 halogenalkyl, C 1 -C 4 halogenalkoxy, C 1 -C 4 alkylamino, C 1 -C 4 dialkylamino, thio or C 1 -C 4 alkylthio. The invention also relates to the plant-tolerant acid addition salts or metal salts of said compounds, to the use of the compounds of formula (I) for controlling plant-pathogenic fungi, and to agents containing the same.

    Abstract translation: 本发明涉及通式(I),其中A或B是苯并二的azolylmethyloxirane其任选地被一个取代以下substi- tuenten卤素,CN,NO 2 ,氨基,C <五 SUB> 1 -C 4 烷基,C 1 -C 4 烷氧基,C 1 -C 4 - 卤代烷基,C 1 -C 4卤代烷,C 1 -C 4 烷基氨基, ç 1 -C 4 二烷基氨基,硫代,或C 1 -C 4 是烷硫基,被取代的,和 各其他取代基A或B为苯基或5元或6元杂芳基,所述取代基任选地被1-3个下列取代基取代:卤素,CN,NO 2 ,氨基,C < SUB> 1 -C 4 烷基,C 1 -C 4 烷氧基,C 1 -C 4 卤代烷基,C 1 -C 4 - 卤代烷氧基,C 1 -C 4 - 烷基氨基,C 1 -C 4 二烷基氨基,巯基或C 1 -C 4 - 烷硫基,被取代的,和它们的植物耐受的酸加成盐或金属盐,使用式(I)的用于控制植物病原真菌包含它们的化合物和试剂。

    USE OF 5-ALKYL-6-PHENYLALKYL-7-AMINO-AZOLOPYRIMIDINES, NOVEL AZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF, AND AGENTS CONTAINING THE SAME
    2.
    发明申请
    USE OF 5-ALKYL-6-PHENYLALKYL-7-AMINO-AZOLOPYRIMIDINES, NOVEL AZOLOPYRIMIDINES, METHODS FOR THE PRODUCTION THEREOF, AND AGENTS CONTAINING THE SAME 审中-公开
    使用5-烷基-6-苯基 - 7-氨基AZOLOPYRIMIDINEN,NEW azolopyrimidines,METHOD用于生产和AGENTS CONTAINING THE SAME

    公开(公告)号:WO2006114405A2

    公开(公告)日:2006-11-02

    申请号:PCT/EP2006061786

    申请日:2006-04-24

    CPC classification number: A01N43/90 C07D487/04

    Abstract: The invention relates to the use of 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines of formula I for controlling phytopathogenic fungi. The variables in formula I have the following designations: Y represents alkylene, alkenylene or alkinylene, optionally substituted by alkyl groups; R 1 represents halogen, cyano, nitro, hydroxy, mercapto, alkyl, halogenalkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxy, halogenalkoxy, alkenyloxy, alkinyloxy, alkylthio, NR A R B , alkylcarbonyl, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; R A , R B represent hydrogen, alkyl and alkylcarbonyl; n represents 0, 1, 2, 3 or 4; R 2 represents alkyl, alkenyl, cycloalkyl, alkoxyalkyl and alkylthioalkyl; R 3 represents hydrogen, halogen, cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, or alkyl-S(O) m- ; m represents 0, 1 or 2; A represents N and C-R a ; and R a represents hydrogen and alkyl. The carbon atoms in Y, R 1 , R 2 , R 3 and Ra can be substituted according to the description. The invention also relates to novel 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines, to methods for producing said compounds, and to agents containing the same.

    Abstract translation: 式的5-烷基-6-苯基-7-氨基azolopyrimidinen的使用I:其中各变量具有以下含义:Y是任选被烷基取代的亚烷基,亚烯基或亚炔基; [R 1 为卤素,氰基,硝基,羟基,巯基,烷基,卤代烷基,链烯基,环烷基,环烯基,烷氧基,卤代烷氧基,烯氧基,炔氧基,烷硫基,NR - [R < SUP>乙,烷基羰基,苯基,萘基或五 - 或六元饱和环,其包含选自一至四个杂原子的部分不饱和或罗马杂环O,N或S; [R ,R 是氢,烷基和烷基羰基; n是零,1,2,3或4; [R 2 烷基,烯基,环烷基,烷氧基烷基和烷硫基烷基; [R 3 为氢,卤素,氰基,NR - [R ,羟基,巯基,烷基,卤代烷基,环烷基,烷氧基,烷硫基,环烷氧基, 环烷硫基,羧基,甲酰基,烷基羰基,烷氧基羰基,烯氧基羰基,炔氧基羰基,苯基,苯氧基,苯硫基,苄氧基,苄硫基,烷基-S(O)米 - ; m是0,1或2; A N和C-R ; [R 氢和烷基; 其中Y中的碳原子,R 1 ,R 2 ,R 3 和R a可以按照该描述被取代; 防治植物病原性有害真菌; 新5-烷基-6-苯基-7- aminoazolopyrimidines,处理用于制备这些化合物和含有它们的组合物。

    2-SUBSTITUTED 7-AMINO-AZOLOPYRIMIDINE, A METHOD FOR THE PRODUCTION AND USE THEREOF FOR CONTROLLING PATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUND
    6.
    发明申请
    2-SUBSTITUTED 7-AMINO-AZOLOPYRIMIDINE, A METHOD FOR THE PRODUCTION AND USE THEREOF FOR CONTROLLING PATHOGENIC FUNGI AND AGENTS CONTAINING SAID COMPOUND 审中-公开
    2-取代的7- aminoazolopyrimidines,METHOD用于生产和它们用于防治有害真菌和代理含

    公开(公告)号:WO2006092428A2

    公开(公告)日:2006-09-08

    申请号:PCT/EP2006060399

    申请日:2006-03-02

    CPC classification number: C07D487/04

    Abstract: The invention relates to 2-substituted 7-amino-azolopyrimidine of formula (I), wherein substituents have the following meanings: R 1 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, Cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or akoxyalkinyl; R 2 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, wherein a carbon chain in R 1 and/or R 2 are substitutable according to a description; R 3 is halogen, Cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phe- nylthio, benzyloxy, benzylthio, alkyl-S(O) m- ; A N and CR x ; R x is hydrogen or one of above groups for R 3 . A method and intermediate products for producing said compounds, agents containing said compounds and the use thereof for combating plant-pathogen fungi are also disclosed.

    Abstract translation: 2-取代的式(I)其中取代基具有以下含义的7-氨基azolopyrimidines:R t 1 为氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基, benzyloxyalkyl,烷氧基烯基或alkoxyalkynyl; [R 2 为氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基和烷硫基烷基,其中在R中的碳链 1 和/或R 2 可以根据描述被取代; [R 3 为卤素,氰基,NR - [R ,羟基,巯基,烷基,卤代烷基,环烷基,烷氧基,烷硫基,环烷氧基,环烷硫基, 羧基,甲酰基,烷基羰基,烷氧基羰基,烯氧基羰基,炔氧基羰基,苯基,苯氧基,苯丙氨酸nylthio,苄氧基,苄硫基,烷基-S(O)米 - ; A N和CR X ; ,R 3 X 是氢或其中R 称作; 的方法和中间体制备这些化合物,含有它们和它们在防治植物病原性有害真菌的组合物。

    8.
    发明专利
    未知

    公开(公告)号:BRPI0712704A2

    公开(公告)日:2012-07-03

    申请号:BRPI0712704

    申请日:2007-06-15

    Applicant: BASF AG

    Abstract: The present invention relates to azolylmethyloxiranes of the general formula I in which A is phenyl which is substituted by two F, B is unsubstituted pyridyl, thienyl, thiazolyl, oxazolyl or furyl or is phenyl which is optionally substituted by one to three of the following substituents: halogen, NO2, amino, C1-C4-alkyl, C1-C4alkoxy, C1-C4-haloalkyl, C1-C4-haloalkoxy, C1-C4-alkylamino, thio or C1-C4-alkylthio, with the proviso that B is not o-methylphenyl if A is 2,4-difluorophenyl, and to the plant-compatible acid addition salts or metal salts thereof, to the use of the compounds of the formula I for controlling phytopathogenic fungi and to compositions comprising these compounds.

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