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公开(公告)号:NO20004351D0
公开(公告)日:2000-09-01
申请号:NO20004351
申请日:2000-09-01
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: C07D251/22 , A61K31/192 , A61K31/216 , A61K31/505 , A61K31/506 , A61K31/519 , A61K31/53 , A61P9/04 , A61P9/06 , A61P9/10 , A61P9/12 , A61P11/06 , A61P13/08 , A61P13/12 , A61P35/00 , A61P43/00 , C07C59/66 , C07C59/68 , C07C69/734 , C07D213/63 , C07D239/34 , C07D239/52 , C07D239/60 , C07D405/12 , C07D491/048
Abstract: The invention relates to carboxylic acid derivatives of formula (I), wherein R -R , Q, W, X, Y and Z have the meanings given in the description. The novel compounds are suitable for combating diseases.
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公开(公告)号:NO20004351A
公开(公告)日:2000-09-01
申请号:NO20004351
申请日:2000-09-01
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: C07D251/22 , A61K31/192 , A61K31/216 , A61K31/505 , A61K31/506 , A61K31/519 , A61K31/53 , A61P9/04 , A61P9/06 , A61P9/10 , A61P9/12 , A61P11/06 , A61P13/08 , A61P13/12 , A61P35/00 , A61P43/00 , C07C59/66 , C07C59/68 , C07C69/734 , C07D213/63 , C07D239/34 , C07D239/52 , C07D239/60 , C07D405/12 , C07D491/048
CPC classification number: C07D239/52 , C07C59/68 , C07C69/734 , C07D239/34
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公开(公告)号:NO20002154A
公开(公告)日:2000-05-12
申请号:NO20002154
申请日:2000-04-27
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , HILLEN HEINZ , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILLIANE
IPC: C07D249/12 , A61K31/41 , A61K31/415 , A61K31/4164 , A61K31/42 , A61K31/421 , A61K31/422 , A61K31/4245 , A61K31/425 , A61K31/426 , A61K31/427 , A61K31/428 , A61K31/433 , A61P9/04 , A61P9/08 , A61P9/10 , A61P9/12 , A61P11/06 , A61P13/08 , A61P13/12 , A61P35/00 , A61P43/00 , C07D231/20 , C07D233/70 , C07D261/12 , C07D263/38 , C07D271/06 , C07D271/10 , C07D273/01 , C07D275/02 , C07D275/03 , C07D277/20 , C07D277/32 , C07D277/34 , C07D277/60 , C07D277/68 , C07D285/00 , C07D285/08 , C07D285/12 , C07D291/04 , C07D413/12 , C07D417/12 , C07D
CPC classification number: C07D275/03 , C07D261/12 , C07D263/38 , C07D277/34 , C07D277/60 , C07D277/68
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公开(公告)号:NO20002124L
公开(公告)日:2000-04-26
申请号:NO20002124
申请日:2000-04-26
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: A61K31/505 , A61K31/506 , A61K31/517 , A61K31/519 , A61K31/5377 , A61P9/02 , A61P9/10 , A61P9/12 , A61P13/08 , A61P13/12 , A61P35/00 , A61P43/00 , C07D239/34 , C07D239/36 , C07D239/52 , C07D239/60 , C07D239/70 , C07D401/12 , C07D403/12 , C07D491/048 , C07D
Abstract: The invention relates to carboxylic acid derivatives of formula (I), wherein the substituents have the meaning as commented in the description. It also relates to the production and use of same as endothelin receptor antagonists.
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公开(公告)号:ZA989312B
公开(公告)日:2000-04-13
申请号:ZA989312
申请日:1998-10-13
Applicant: BASF AG
Inventor: PUHL MICHAEL , ZECHEL JOHANN-CHRISTIAN , DITRICH KLAUS , HILLEN HEINZ , KOHL TANJA , ERHARDT MELANIE , HERGENROEDER STEFAN , MARKERT CLAUS OTTO
IPC: C07D333/40 , A61K31/198 , A61K31/27 , A61K31/381 , A61K31/4704 , A61K31/498 , A61P1/04 , A61P1/18 , A61P7/02 , A61P9/04 , A61P9/10 , A61P9/12 , A61P13/08 , A61P13/12 , A61P25/06 , A61P35/00 , C07C271/12 , C07C271/20 , C07C323/56 , C07D215/48 , C07D241/44 , C07D333/38 , C07D , A61K , C07C
Abstract: Pharmaceutically active compounds are prepared as described and used to produce pharmaceutical preparations for treating diseases.
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公开(公告)号:NO20001846A
公开(公告)日:2000-04-10
申请号:NO20001846
申请日:2000-04-10
Applicant: BASF AG
Inventor: PUHL MICHAEL , ZECHEL JOHANN-CHRISTIAN , DITRICH KLAUS , HILLEN HEINZ , KOHL TANJA , ERHARDT MELANIE , HERGENROEDER STEFAN , MARKERT CLAUS OTTO
IPC: C07D333/40 , A61K31/198 , A61K31/27 , A61K31/381 , A61K31/4704 , A61K31/498 , A61P1/04 , A61P1/18 , A61P7/02 , A61P9/04 , A61P9/10 , A61P9/12 , A61P13/08 , A61P13/12 , A61P25/06 , A61P35/00 , C07C271/12 , C07C271/20 , C07C323/56 , C07D215/48 , C07D241/44 , C07D333/38 , C07D333/16 , A61K31/38 , A61K31/47 , A61K31/495 , C07C271/22 , C07D215/14 , C07D241/42
CPC classification number: C07C271/20 , C07C323/56 , C07C2603/18 , C07D241/44 , C07D333/38
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公开(公告)号:NO20001077L
公开(公告)日:2000-03-02
申请号:NO20001077
申请日:2000-03-02
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: A61K31/421 , A61K31/426 , A61K31/428 , A61K31/496 , A61K31/505 , A61P9/10 , A61P9/12 , A61P43/00 , C07D239/34 , C07D239/52 , C07D263/38 , C07D277/20 , C07D277/34 , C07D277/68 , C07D409/12 , C07D239/04
Abstract: The invention relates to carboxylic acid derivatives of formula (I) wherein the radicals are defined in the description, and to the use of these derivatives as ETA/ETB endothelin-receptor antagonists.
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公开(公告)号:CZ61999A3
公开(公告)日:2000-02-16
申请号:CZ61999
申请日:1997-09-02
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , KLING ANDREAS , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: A61K31/505 , A61P9/12 , C07D237/22 , C07D239/34 , C07D239/60 , C07D239/70 , C07D491/04
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公开(公告)号:PL331998A1
公开(公告)日:1999-08-16
申请号:PL33199897
申请日:1997-09-02
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , KLING ANDREAS , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: A61K31/505 , A61K31/506 , A61K31/519 , A61P9/04 , A61P9/08 , A61P9/12 , A61P43/00 , C07C59/66 , C07C69/734 , C07D239/34 , C07D239/52 , C07D239/60 , C07D239/70 , C07D491/04 , C07D491/048
Abstract: The invention relates to carboxylic acid derivatives of the formula Iwhere the radicals have the meanings stated in the description, and to their use as drugs.
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50.
公开(公告)号:ZA9711305B
公开(公告)日:1999-06-17
申请号:ZA9711305
申请日:1997-12-17
Applicant: BASF AG
Inventor: AMBERG WILHELM , JANSEN ROLF , KLING ANDREAS , KLINGE DAGMAR , RIECHERS HARTMUT , HERGENROEDER STEFAN , RASCHACK MANFRED , UNGER LILIANE
IPC: C07D237/14 , C07D237/16 , C07D241/18 , C07D253/07 , C07D253/075 , C07D253/10 , C07D491/04 , C07D , A61K
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