Microbiocidal N-phenyl-N-[4-(4-pyridyl-2-pyrimidin-2-YL]-amine derivatives

    公开(公告)号:AU2002236101B2

    公开(公告)日:2006-09-14

    申请号:AU2002236101

    申请日:2001-12-20

    Abstract: The invention relates to novel N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives of the general formula (I) wherein the sum of (m+p) together is 0, 1, 2 or 3; n and q are independently of each other 0 or 1, and the sum of (m+p+q) together is 1, 2, 3 or 4; R 1 is hydrogen, halogen, alkoxy, haloalkyl, haloalkoxy or alkyl; R 2 is hydrogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl or C 1 -C 6 -alkoxy; R 2A is hydrogen, C 1 -C 6 -alkyl, C 3 -C 4 -alkenyl or C 3 -C 4 -alkynyl; each of R 3 , R 4 , R 5 and R 6 is, independently of the others, hydrogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, hydroxy-C 1 -C 6 -alkyl or C 1 -C 6 -alkoxy-C 1 -C 6 -alkyl, or the ring members CR 3 R 4 or CR 5 R 6 or CR 2 R 2A are independently of each other a carbonyl group (C-O) or a group C-S; X is C-O, C-S, S-O or O-S-O; Y is O, S, C-O, CH 2 , -N(R 8 )-, -O-N(R 8 )-, -N(R 8 )-O- or NH-; R 7 is hydrogen, C 1 -C 4 -alkyl, C 3 -C 4 -alkenyl, C 3 -C 4 -alkynyl, -CH 2 OR 8 , CH 2 SR 8 , -C(O)R 8 , -C(O)OR 8 , SO2R 8 , SOR 8 or SR 8 ; and R 8 is C 1 -C 8 -alkyl, C 1 -C 8 -alkoxyalkyl, C 1 -C 8 haloalkyl or phenylC 1 -C 2 -alkyl wherein the phenyl may be substituted by up to three groups selected from halo or C 1 -C 4 -alkyl; or a salt thereof. The invention also relates to the preparation of the compounds and to agrochemical compositions comprising at least one of those compounds as active ingredient as well as the preparation of the said compositions and to the use of the compounds or of the compositions in controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.

    50.
    发明专利
    未知

    公开(公告)号:DE60105646T2

    公开(公告)日:2005-11-17

    申请号:DE60105646

    申请日:2001-12-20

    Abstract: The invention relates to novel N-phenyl-4-(4-pyridyl)-2-pyrimidineamine derivatives of the general formula (I) wherein the sum of (m+p) together is 0, 1, 2 or 3; n and q are independently of each other 0 or 1, and the sum of (m+p+q) together is 1, 2, 3 or 4; R 1 is hydrogen, halogen, alkoxy, haloalkyl, haloalkoxy or alkyl; R 2 is hydrogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl or C 1 -C 6 -alkoxy; R 2A is hydrogen, C 1 -C 6 -alkyl, C 3 -C 4 -alkenyl or C 3 -C 4 -alkynyl; each of R 3 , R 4 , R 5 and R 6 is, independently of the others, hydrogen, C 1 -C 6 -alkyl, C 1 -C 6 -haloalkyl, hydroxy-C 1 -C 6 -alkyl or C 1 -C 6 -alkoxy-C 1 -C 6 -alkyl, or the ring members CR 3 R 4 or CR 5 R 6 or CR 2 R 2A are independently of each other a carbonyl group (C-O) or a group C-S; X is C-O, C-S, S-O or O-S-O; Y is O, S, C-O, CH 2 , -N(R 8 )-, -O-N(R 8 )-, -N(R 8 )-O- or NH-; R 7 is hydrogen, C 1 -C 4 -alkyl, C 3 -C 4 -alkenyl, C 3 -C 4 -alkynyl, -CH 2 OR 8 , CH 2 SR 8 , -C(O)R 8 , -C(O)OR 8 , SO2R 8 , SOR 8 or SR 8 ; and R 8 is C 1 -C 8 -alkyl, C 1 -C 8 -alkoxyalkyl, C 1 -C 8 haloalkyl or phenylC 1 -C 2 -alkyl wherein the phenyl may be substituted by up to three groups selected from halo or C 1 -C 4 -alkyl; or a salt thereof. The invention also relates to the preparation of the compounds and to agrochemical compositions comprising at least one of those compounds as active ingredient as well as the preparation of the said compositions and to the use of the compounds or of the compositions in controlling or preventing the infestation of plants by phytopathogenic microorganisms, especially fungi.

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