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公开(公告)号:DE59208733D1
公开(公告)日:1997-08-28
申请号:DE59208733
申请日:1992-01-24
Applicant: BASF AG
Inventor: GRAMMENOS WASSILIOS DR , HARREUS ALBRECHT DR , SAUTER HUBERT DR , HELLENDAHL BEATE DR , DOETZER REINHARD DR , AMMERMANN EBERHARD DR , LORENZ GISELA DR
IPC: A01N37/50 , A01N43/54 , A01N43/58 , A01N43/76 , A01N43/836 , C07C69/65 , C07C69/653 , C07C69/734 , C07C69/738 , C07C251/48 , C07C251/50 , C07C251/52 , C07C251/54 , C07C251/56 , C07C251/58 , C07C251/60 , C07C251/86 , C07C255/15 , C07C255/57 , C07C255/58 , C07C255/62 , C07D213/77 , C07D239/42 , C07D241/20 , C07D263/32 , C07D333/28
Abstract: Iminoalkyl-phenylacrylic acid derivs. (I) ar new: R = H or 1-6C alkyl; R = H; 1-4C alkyl opt. substd. by halo; or opt. substd. aryl; Z ,Z = H; halo; CN; NO2;etc.;Y = O; NH; or NR ; and R = H; 1-4C alkoxycarbonyl-1-4C alkyl; or opt. substd. alkyl, cycloalkyl, etc.; or Y+R form a ring which is opt. substd. when Y = NH or NR ; R = 1-6C alkyl; X = CH-1-4C alkoxy or CH-1-4C alkylthio (also 1-4C alkylidene and 1-4C alkoxyimino in the description).
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公开(公告)号:DE19604732A1
公开(公告)日:1997-08-14
申请号:DE19604732
申请日:1996-02-09
Applicant: BASF AG
Inventor: GROTE THOMAS DR , SAUTER HUBERT DR , KIRSTGEN REINHARD DR , BAYER HERBERT DR , MUELLER RUTH DR , MUELLER BERND DR , OBERDORF KLAUS DR , GRAMMENOS WASSILIOS DR , GOETZ NORBERT DR , RACK MICHAEL DR , HARREUS ALBRECHT DR , ROEHL FRANZ DR , AMMERMANN EBERHARD DR , HARRIES VOLKER DR , LORENZ GISELA DR , STRATHMANN SIEGFRIED DR
IPC: C07C251/60 , A01N37/34 , A01N37/50 , A01N43/00 , C07C69/757 , C07C255/62 , C07C255/64 , C07C323/24
Abstract: 2-Iminooxyphenylacetic acid derivatives of formula (I) and their salts are new. R = C(CO2Me)=NOMe, C(CONHMe)=NOMe, C(CONH2)=NOMe, C(CO2Me)=COMe or C(CO2Me)=CHMe; R2 = CN, NO2, halo, 1-4C alkyl, 1-4C haloalkyl or 1-4C alkoxy; m = 0-2; R3 = H, CN, OH, halo, 1-6C alkyl (optionally substituted by halo or 1-6C alkoxy) 1-6C alkoxy, 1-6C haloalkoxy, 1-6C alkylthio, cyclopropyl, 2-6C alkenyl, or aryloxy-1-6C alkyl, benzyl or benzyloxy (all optionally ring-substituted by 1-3 CN, NO2, halo, 1-6C alkyl, 1-6C alkoxy, 1-6C haloalkyl or 1-6C haloalkoxy) or C(Me)=N-Y-Ra; Ra = 1-6C alkyl; Y = O, NH or NRa; R4 = H, CN, -Qp-C(R5)=N-Y'-R6 or -Q-O-N=CR7R8; or alkyl, alkenyl, alkynyl, cycloalkyl, heterocyclyl, aryl, heteroaryl, alkoxy, alkenyloxy, alkynyloxy, cycloalkoxy, heterocyclyloxy, aryloxy, heteroaryloxy, arylthio or heteroarylthio (all optionally substituted); or CR3R4 = 4-8 membered ring containing C atoms an optionally 1 or 2 of O, S, NH and/or N(1-4C alkyl) (optionally substituted on C by halo, 1-6C alkyl or 1-4C alkoxyimino), provided R3 and R4 are not both bonded to C via hetero atoms; Q = bond, CH2, CH(Me), CH(Et) or 1,1-cyclopropyl; p = 0 or 1; Y' = O, NH or N(1-4C alkyl); R5 = as for R3 or optionally substituted cycloalkoxy, heterocyclyloxy, aryloxy, heteroaryloxy, arylthio or heteroarylthio; R6 = optionally substituted 1-10C alkyl, 3-6C cycloalkyl, 2-10C alkenyl, 2-10C alkynyl, 1-10C alkylcarbonyl, 2-10C alkenylcarbonyl, 2-10C alkynylcarbonyl, 1-10C alkylsulphonyl, aryl, heteroaryl, arylcarbonyl, heteroarylcarbonyl, arylsulphonyl or heteroarylsulphonyl; R7, R8 = Me, Et, Ar or CH2Ar; Ar = phenyl (optionally mono-, di- or trisubstituted by CN, NO2, halo, 1-6C alkyl, 1-6C alkoxy, 1-6C haloalkyl or 1-6C haloalkoxy.
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公开(公告)号:GR3021583T3
公开(公告)日:1997-02-28
申请号:GR960402957
申请日:1996-11-07
Applicant: BASF AG
Inventor: OBERDORF KLAUS DR , SAUTER HUBERT DR , GRAMMENOS WASSILIOS DR , KIRSTGEN REINHARD DR , HARRIES VOLKER DR , LORENZ GISELA DR , AMMERMANN EBERHARD DR , GOLD RANDALL EVAN DR , SIEGEL WOLFGANG DR , HARREUS ALBRECHT DR
IPC: A01N37/18 , A01N37/34 , A01N37/36 , A01N37/38 , A01N37/50 , C07C251/40 , C07C251/48 , C07C251/50 , C07C251/52 , C07C251/54 , C07C251/58 , C07C251/60 , C07C255/32 , C07C255/62 , C07D213/63 , C07D333/32 , C07D521/00
Abstract: Substituted oxime ethers of the general formula I in which R denotes alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxyalkyl, cycloalkyl, cycloalkylalkyl, cyanoalkyl, alkoxycarbonylalkyl, arylalkyl, heteroarylalkyl, arylalkenyl or aryloxyalkyl, the aromatic or heteroaromatic ring optionally being substituted, R and R denote hydrogen, alkyl, haloalkyl, alkoxy, haloalkoxy, halogen, cyano or nitro, R denotes hydrogen, alkyl, cycloalkyl, haloalkyl or aryl, the aromatic ring optionally being substituted and R and R are identical or different and denote hydrogen or alkyl, and X denotes CH or N, and fungicides and pesticides containing these compounds.
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公开(公告)号:ES2094842T3
公开(公告)日:1997-02-01
申请号:ES92107059
申请日:1992-04-24
Applicant: BASF AG
Inventor: GRAMMENOS WASSILIOS DR , KIRSTGEN REINHARD DR , OBERDORF KLAUS DR , SAUTER HUBERT DR , ROEHL FRANZ DR , OTTER RAINER DR
IPC: A01N35/10 , A01N43/54 , A01N43/56 , A01N43/78 , C07C59/64 , C07C69/145 , C07C69/618 , C07C69/65 , C07C69/73 , C07C69/732 , C07C69/734 , C07C69/738 , C07C69/76 , C07C69/767 , C07C69/92 , C07C69/94 , C07C251/48 , C07C251/52 , C07C251/54 , C07C323/62 , C07D207/337 , C07D209/18 , C07D209/30 , C07D213/64 , C07D231/12 , C07D231/18 , C07D235/26 , C07D235/28 , C07D239/26 , C07D239/34 , C07D239/38 , C07D239/46 , C07D239/52 , C07D239/56 , C07D239/60 , C07D239/88 , C07D239/90 , C07D261/08 , C07D261/10 , C07D261/12 , C07D261/20 , C07D263/16 , C07D263/38 , C07D263/40 , C07D263/46 , C07D263/56 , C07D263/58 , C07D271/10 , C07D271/113 , C07D275/02 , C07D277/20 , C07D277/30 , C07D277/32 , C07D277/34 , C07D277/36 , C07D277/64 , C07D277/74 , C07D285/08 , C07D285/12 , C07D285/125 , C07D307/54 , C07D317/30 , C07D333/24 , C07F9/40
Abstract: alpha -Phenylacrylic acid derivatives I in which n = 0 to 4; y = 0 or 1; R = H; alkyl; alkenyl; alkynyl; optionally substituted cycloalkyl; vinyl or ethynyl if W represents a direct bond; R = CN; alkenyl; alkynyl; optionally substituted cycloalkyl; optionally substituted alkyl; R = H; NO2; CN; halogen; alkyl; alkoxy; haloalkyl; haloalkoxy; alkylthio; or, in the event that n represents 2, 3 or 4, two adjacent substituents R together are optionally substituted 1,3-butadiene-1,4-diyl; R = H; CHO; optionally substituted alkyl; optionally substituted alkenyl; optionally substituted alkynyl; an optionally substituted saturated or unsaturated cyclic radical; (phenyl)3P-; (phenyl)2PO-; (alkoxy)2PO-; an optionally substituted (hetero)aromatic system; W = a direct bond; oxygen; sulphur; optionally substituted nitrogen; A = -O-; -C(=O)-; -O-C(=O)-; -C(=O)-O-; -S-; -S(=O)-; -O-S(=0)--S(=O)-O-; -S(=O)2-; -O-S(=O)2-; -S(=O)2-O-; -NR -; -O-NR -; -NR -C(=O)-; -C(=O)-NR -; -NR -C(=O)-NR -; -NR -S(=O)-; -S(=O)-NR -; -NR -S-(=O)-NR -; -NR -S(=O)2-; -S(=O)2-NR -; -NR -S(=O)2-NR -; -N=N-; -NR -NR -; -NR -NR -C(=O)-; -C(=O)-NR -NR -; -NR -NR -S(=O)-; -S(=O)-NR -NR -; -NR -NR -S(=O)2-; -S(=O)2-NR -NR -; -O-(alkylene)-O-; -C-(=O)-(alkylene)-O-; -O-C(=O)-(alkylene)-O-; -C(=O)-O-(alkylene)-O-; -S-(alkylene)-O-; -S(=0)2-(alkylene)-O-; -O-S-(=O)2-(alkylene)-O-; -S(=O)2-O-(alkylene)-O-; -NR -(alkylene)-O-; -O-NR -(alkylene)-O-; -NR -C(=O)-(alkylene)-O-; -C(=O)-NR -(alkylene)-O-; -NR -C(=O)-NR -(alkylene)-O-; -N=N-(alkylene)-O-; -NR -NR -(alkylene)-O-; -NR -NR -C(=O)-(alkylene)-O-; -C(=O)-NR -NR -(alkylene)-O-; optionally substituted alkylene, alkenylene or alkynylene, it being possible for these carbon chains to be interrupted by one of the following groups or to be bonded to R or to the phenyl ring by one of the following groups: O, S, NR , CO, CO-O, O-CO, SO, SO2, SO2-O, O-SO2, NR -CO, CO-NR , NR -CO-NR , N=N, NR -NR , NR -NR -CO, CO-NR -NR ; R , R = H, alkyl or alkoxy, their preparation, fungicides and pesticides containing them, and their use.
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公开(公告)号:GR3021280T3
公开(公告)日:1997-01-31
申请号:GR960402642
申请日:1996-10-09
Applicant: BASF AG
Inventor: WINGERT HORST DR , WOLF BERND DR , BENOIT REMY DR , SAUTER HUBERT DR , HEPP MICHAEL DR , GRAMMENOS WASSILIOS DR , KUEKENHOEHNER THOMAS DR
IPC: C07C69/736 , C07C20060101 , C07C51/09 , C07C51/367 , C07C59/68 , C07C65/21 , C07C65/24 , C07C67/22 , C07C69/738 , C07C69/76 , C07C235/34 , C07C235/78 , C07C249/08 , C07C251/48 , C07C253/14 , C07C255/17 , C07C255/40 , C07C317/24
Abstract: Prepn. of 2-phenoxymethyl benzoic acid derivs. of formula (I) comprises (a) converting a phenol of formula (II) to the phenolate in the presence of a basic diluent; (b) mixing the mixt. with a lactone of formula (III); (c) distilling off the diluent; (d) reacting the mixt. at 50-250 degrees C in the melt; and (e) dissolving the liq. melt with water and acidifying. X, Y = halogen, 1-4C alkyl, 1-4C alkoxy or CF3; m = 0-4; n = 0-3.
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公开(公告)号:DE59206443D1
公开(公告)日:1996-07-11
申请号:DE59206443
申请日:1992-01-24
Applicant: BASF AG
Inventor: GRAMMENOS WASSILIOS DR , HARREUS ALBRECHT DR , SAUTER HUBERT DR , HELLENDAHL BEATE DR , DOETZER REINHARD DR , AMMERMANN EBERHARD DR , LORENZ GISELA DR
IPC: A01N37/50 , A01N43/54 , A01N43/58 , A01N43/76 , A01N43/836 , C07C69/65 , C07C69/653 , C07C69/734 , C07C69/738 , C07C251/48 , C07C251/50 , C07C251/52 , C07C251/54 , C07C251/56 , C07C251/58 , C07C251/60 , C07C251/86 , C07C255/15 , C07C255/57 , C07C255/58 , C07C255/62 , C07D213/77 , C07D239/42 , C07D241/20 , C07D263/32 , C07D333/28
Abstract: Iminoalkyl-phenylacrylic acid derivs. (I) ar new: R = H or 1-6C alkyl; R = H; 1-4C alkyl opt. substd. by halo; or opt. substd. aryl; Z ,Z = H; halo; CN; NO2;etc.;Y = O; NH; or NR ; and R = H; 1-4C alkoxycarbonyl-1-4C alkyl; or opt. substd. alkyl, cycloalkyl, etc.; or Y+R form a ring which is opt. substd. when Y = NH or NR ; R = 1-6C alkyl; X = CH-1-4C alkoxy or CH-1-4C alkylthio (also 1-4C alkylidene and 1-4C alkoxyimino in the description).
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公开(公告)号:GR3017716T3
公开(公告)日:1996-01-31
申请号:GR950402825
申请日:1995-10-11
Applicant: BASF AG
Inventor: SAUTER HUBERT DR , BAYER HERBERT DR , OBERDORF KLAUS DR , WINGERT HORST DR , VON DEYN WOLFGANG DR , GRAMMENOS WASSILIOS DR , KOENIG HARTMANN DR , RANG HARALD DR , ROEHL FRANZ DR , LORENZ GISELA DR , AMMERMANN EBERHARD DR
IPC: A01N37/36 , A01N37/38 , A01N37/44 , A01N37/48 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/56 , A01N43/74 , A01N43/78 , A01N43/80 , A01N43/82 , C07C69/618 , A61K31/21 , A61K31/40 , A61K31/505 , C07C67/343 , C07C69/65 , C07C69/734 , C07C69/736 , C07C69/738 , C07C69/75 , C07C69/76 , C07C69/84 , C07C69/86 , C07C69/92 , C07C69/94 , C07C205/34 , C07C205/38 , C07C205/56 , C07C229/40 , C07C229/44 , C07C233/11 , C07C235/32 , C07C235/34 , C07C251/38 , C07C251/48 , C07C251/52 , C07C251/60 , C07C251/66 , C07C255/57 , C07C255/64 , C07C275/64 , C07C309/66 , C07C309/73 , C07C311/09 , C07C311/21 , C07C311/29 , C07C313/04 , C07C313/06 , C07C317/44 , C07C317/46 , C07C323/56 , C07C323/62 , C07C327/22 , C07C327/48 , C07D207/32 , C07D207/335 , C07D207/337 , C07D213/53 , C07D213/64 , C07D213/643 , C07D213/66 , C07D213/68 , C07D213/70 , C07D215/22 , C07D215/227 , C07D215/233 , C07D215/36 , C07D231/12 , C07D233/84 , C07D235/28 , C07D239/52 , C07D249/12 , C07D257/04 , C07D261/08 , C07D263/32 , C07D263/34 , C07D263/58 , C07D271/06 , C07D271/10 , C07D271/113 , C07D277/28 , C07D277/30 , C07D277/36 , C07D277/68 , C07D277/74 , C07D285/12 , C07D285/125 , C07D307/46 , C07D307/52 , C07D307/54 , C07D309/06 , C07D333/24 , C07D409/04 , C07D413/04 , C07D513/04 , C07D521/00 , C07F7/08
Abstract: Derivatives of beta -substituted cinnamic acid of the general formula 1 in which R denotes optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and in which R can also denote chlorine or bromine, -X- represents the groups -O-, -S-, m denotes 0 or 1, -Y represents the groups -OR , -O-N=CR R , -NR R , -N(OR )R or -Sr , where the abovementioned substituents R to R denote optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and for the radicals R , R and R to R can also denote hydrogen, Z denotes halogen, nitro, cyano, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aralkyl, optionally substituted aryloxyalkyl, optionally substituted arylthioalkyl, optionally substituted heteroarylalkyl, optionally substituted heteroaryloxyalkyl, optionally substituted heteroarylthioalkyl, optionally substituted alkenyl, optionally substituted aralkenyl, optionally substituted aryloxyalkenyl, optionally substituted arylthioalkenyl, optionally substituted heteroarylalkenyl, optionally substituted heteroaryloxyalkenyl, optionally substituted heteroarylthioalkenyl, optionally substituted alkynyl, optionally substituted arylalkynyl, optionally substituted heteroarylalkynyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted arylazo, optionally substituted acylamino, -OR , -SR ,-SOR , -SO2R , -COOR , -CONR R , -COR , -CR =NR , -N=CR R , -CR =N-OR , -CR R -O-N=CR R , -CH2-OCOR or -NR R , where the groups R to R , and R and R denote hydrogen, optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted cycloalkyl, optionally substituted cycloalkylalkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted aralkyl, optionally substituted heteroarylalkyl, optionally substituted aryloxyalkyl, optionally substituted arylthioalkyl, optionally substituted heteroaryloxyalkyl or optionally substituted heteroarylthioalkyl and R denotes hydrogen or C1-C4-alkyl and in which U, V, W denote hydrogen or have one of the meanings mentioned for Z or in which two of the groups Z, U, V or W in adjacent positions of the phenyl ring optionally together form an optionally substituted five- or six-membered, aromatic or aliphatic ring fused to the phenyl ring, which can optionally contain one to three heteroatoms (N, S, O).
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公开(公告)号:ES2078602T3
公开(公告)日:1995-12-16
申请号:ES92112086
申请日:1992-07-15
Applicant: BASF AG
Inventor: SAUTER HUBERT DR , BAYER HERBERT DR , OBERDORF KLAUS DR , WINGERT HORST DR , VON DEYN WOLFGANG DR , GRAMMENOS WASSILIOS DR , KOENIG HARTMANN DR , RANG HARALD DR , ROEHL FRANZ DR , LORENZ GISELA DR , AMMERMANN EBERHARD DR
IPC: A01N37/36 , A01N37/38 , A01N37/44 , A01N37/48 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/56 , A01N43/74 , A01N43/78 , A01N43/80 , A01N43/82 , C07C69/618 , A61K31/21 , A61K31/40 , A61K31/505 , C07C67/343 , C07C69/65 , C07C69/734 , C07C69/736 , C07C69/738 , C07C69/75 , C07C69/76 , C07C69/84 , C07C69/86 , C07C69/92 , C07C69/94 , C07C205/34 , C07C205/38 , C07C205/56 , C07C229/40 , C07C229/44 , C07C233/11 , C07C235/32 , C07C235/34 , C07C251/38 , C07C251/48 , C07C251/52 , C07C251/60 , C07C251/66 , C07C255/57 , C07C255/64 , C07C275/64 , C07C309/66 , C07C309/73 , C07C311/09 , C07C311/21 , C07C311/29 , C07C313/04 , C07C313/06 , C07C317/44 , C07C317/46 , C07C323/56 , C07C323/62 , C07C327/22 , C07C327/48 , C07D207/32 , C07D207/335 , C07D207/337 , C07D213/53 , C07D213/64 , C07D213/643 , C07D213/66 , C07D213/68 , C07D213/70 , C07D215/22 , C07D215/227 , C07D215/233 , C07D215/36 , C07D231/12 , C07D233/84 , C07D235/28 , C07D239/52 , C07D249/12 , C07D257/04 , C07D261/08 , C07D263/32 , C07D263/34 , C07D263/58 , C07D271/06 , C07D271/10 , C07D271/113 , C07D277/28 , C07D277/30 , C07D277/36 , C07D277/68 , C07D277/74 , C07D285/12 , C07D285/125 , C07D307/46 , C07D307/52 , C07D307/54 , C07D309/06 , C07D333/24 , C07D409/04 , C07D413/04 , C07D513/04 , C07D521/00 , C07F7/08
Abstract: Derivatives of beta -substituted cinnamic acid of the general formula 1 in which R denotes optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and in which R can also denote chlorine or bromine, -X- represents the groups -O-, -S-, m denotes 0 or 1, -Y represents the groups -OR , -O-N=CR R , -NR R , -N(OR )R or -Sr , where the abovementioned substituents R to R denote optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and for the radicals R , R and R to R can also denote hydrogen, Z denotes halogen, nitro, cyano, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aralkyl, optionally substituted aryloxyalkyl, optionally substituted arylthioalkyl, optionally substituted heteroarylalkyl, optionally substituted heteroaryloxyalkyl, optionally substituted heteroarylthioalkyl, optionally substituted alkenyl, optionally substituted aralkenyl, optionally substituted aryloxyalkenyl, optionally substituted arylthioalkenyl, optionally substituted heteroarylalkenyl, optionally substituted heteroaryloxyalkenyl, optionally substituted heteroarylthioalkenyl, optionally substituted alkynyl, optionally substituted arylalkynyl, optionally substituted heteroarylalkynyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted arylazo, optionally substituted acylamino, -OR , -SR ,-SOR , -SO2R , -COOR , -CONR R , -COR , -CR =NR , -N=CR R , -CR =N-OR , -CR R -O-N=CR R , -CH2-OCOR or -NR R , where the groups R to R , and R and R denote hydrogen, optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted cycloalkyl, optionally substituted cycloalkylalkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted aralkyl, optionally substituted heteroarylalkyl, optionally substituted aryloxyalkyl, optionally substituted arylthioalkyl, optionally substituted heteroaryloxyalkyl or optionally substituted heteroarylthioalkyl and R denotes hydrogen or C1-C4-alkyl and in which U, V, W denote hydrogen or have one of the meanings mentioned for Z or in which two of the groups Z, U, V or W in adjacent positions of the phenyl ring optionally together form an optionally substituted five- or six-membered, aromatic or aliphatic ring fused to the phenyl ring, which can optionally contain one to three heteroatoms (N, S, O).
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公开(公告)号:DE59203812D1
公开(公告)日:1995-11-02
申请号:DE59203812
申请日:1992-07-15
Applicant: BASF AG
Inventor: SAUTER HUBERT DR , BAYER HERBERT W- LUDWIGSHAFEN , OBERDORF KLAUS DR , WINGERT HORST DR , VON DEYN WOLFGANG DR , GRAMMENOS WASSILIOS DR , KOENIG HARTMANN DR , RANG HARALD DR , ROEHL FRANZ DR , LORENZ GISELA DR , AMMERMANN EBERHARD DR
IPC: A01N37/36 , A01N37/38 , A01N37/44 , A01N37/48 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/56 , A01N43/74 , A01N43/78 , A01N43/80 , A01N43/82 , C07C69/618 , A61K31/21 , A61K31/40 , A61K31/505 , C07C67/343 , C07C69/65 , C07C69/734 , C07C69/736 , C07C69/738 , C07C69/75 , C07C69/76 , C07C69/84 , C07C69/86 , C07C69/92 , C07C69/94 , C07C205/34 , C07C205/38 , C07C205/56 , C07C229/40 , C07C229/44 , C07C233/11 , C07C235/32 , C07C235/34 , C07C251/38 , C07C251/48 , C07C251/52 , C07C251/60 , C07C251/66 , C07C255/57 , C07C255/64 , C07C275/64 , C07C309/66 , C07C309/73 , C07C311/09 , C07C311/21 , C07C311/29 , C07C313/04 , C07C313/06 , C07C317/44 , C07C317/46 , C07C323/56 , C07C323/62 , C07C327/22 , C07C327/48 , C07D207/32 , C07D207/335 , C07D207/337 , C07D213/53 , C07D213/64 , C07D213/643 , C07D213/66 , C07D213/68 , C07D213/70 , C07D215/22 , C07D215/227 , C07D215/233 , C07D215/36 , C07D231/12 , C07D233/84 , C07D235/28 , C07D239/52 , C07D249/12 , C07D257/04 , C07D261/08 , C07D263/32 , C07D263/34 , C07D263/58 , C07D271/06 , C07D271/10 , C07D271/113 , C07D277/28 , C07D277/30 , C07D277/36 , C07D277/68 , C07D277/74 , C07D285/12 , C07D285/125 , C07D307/46 , C07D307/52 , C07D307/54 , C07D309/06 , C07D333/24 , C07D409/04 , C07D413/04 , C07D513/04 , C07D521/00 , C07F7/08
Abstract: Derivatives of beta -substituted cinnamic acid of the general formula 1 in which R denotes optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and in which R can also denote chlorine or bromine, -X- represents the groups -O-, -S-, m denotes 0 or 1, -Y represents the groups -OR , -O-N=CR R , -NR R , -N(OR )R or -Sr , where the abovementioned substituents R to R denote optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and for the radicals R , R and R to R can also denote hydrogen, Z denotes halogen, nitro, cyano, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aralkyl, optionally substituted aryloxyalkyl, optionally substituted arylthioalkyl, optionally substituted heteroarylalkyl, optionally substituted heteroaryloxyalkyl, optionally substituted heteroarylthioalkyl, optionally substituted alkenyl, optionally substituted aralkenyl, optionally substituted aryloxyalkenyl, optionally substituted arylthioalkenyl, optionally substituted heteroarylalkenyl, optionally substituted heteroaryloxyalkenyl, optionally substituted heteroarylthioalkenyl, optionally substituted alkynyl, optionally substituted arylalkynyl, optionally substituted heteroarylalkynyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted arylazo, optionally substituted acylamino, -OR , -SR ,-SOR , -SO2R , -COOR , -CONR R , -COR , -CR =NR , -N=CR R , -CR =N-OR , -CR R -O-N=CR R , -CH2-OCOR or -NR R , where the groups R to R , and R and R denote hydrogen, optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted cycloalkyl, optionally substituted cycloalkylalkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted aralkyl, optionally substituted heteroarylalkyl, optionally substituted aryloxyalkyl, optionally substituted arylthioalkyl, optionally substituted heteroaryloxyalkyl or optionally substituted heteroarylthioalkyl and R denotes hydrogen or C1-C4-alkyl and in which U, V, W denote hydrogen or have one of the meanings mentioned for Z or in which two of the groups Z, U, V or W in adjacent positions of the phenyl ring optionally together form an optionally substituted five- or six-membered, aromatic or aliphatic ring fused to the phenyl ring, which can optionally contain one to three heteroatoms (N, S, O).
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公开(公告)号:AT128454T
公开(公告)日:1995-10-15
申请号:AT92112086
申请日:1992-07-15
Applicant: BASF AG
Inventor: SAUTER HUBERT DR , BAYER HERBERT DR , OBERDORF KLAUS DR , WINGERT HORST DR , VON DEYN WOLFGANG DR , GRAMMENOS WASSILIOS DR , KOENIG HARTMANN DR , RANG HARALD DR , ROEHL FRANZ DR , LORENZ GISELA DR , AMMERMANN EBERHARD DR
IPC: C07C69/618 , A01N37/36 , A01N37/38 , A01N37/44 , A01N37/48 , A01N43/08 , A01N43/10 , A01N43/36 , A01N43/56 , A01N43/74 , A01N43/78 , A01N43/80 , A01N43/82 , A61K31/21 , A61K31/40 , A61K31/505 , C07C67/343 , C07C69/65 , C07C69/734 , C07C69/736 , C07C69/738 , C07C69/75 , C07C69/76 , C07C69/84 , C07C69/86 , C07C69/92 , C07C69/94 , C07C205/34 , C07C205/38 , C07C205/56 , C07C229/40 , C07C229/44 , C07C233/11 , C07C235/32 , C07C235/34 , C07C251/38 , C07C251/48 , C07C251/52 , C07C251/60 , C07C251/66 , C07C255/57 , C07C255/64 , C07C275/64 , C07C309/66 , C07C309/73 , C07C311/09 , C07C311/21 , C07C311/29 , C07C313/04 , C07C313/06 , C07C317/44 , C07C317/46 , C07C323/56 , C07C323/62 , C07C327/22 , C07C327/48 , C07D207/32 , C07D207/335 , C07D207/337 , C07D213/53 , C07D213/64 , C07D213/643 , C07D213/66 , C07D213/68 , C07D213/70 , C07D215/22 , C07D215/227 , C07D215/233 , C07D215/36 , C07D231/12 , C07D233/84 , C07D235/28 , C07D239/52 , C07D249/12 , C07D257/04 , C07D261/08 , C07D263/32 , C07D263/34 , C07D263/58 , C07D271/06 , C07D271/10 , C07D271/113 , C07D277/28 , C07D277/30 , C07D277/36 , C07D277/68 , C07D277/74 , C07D285/12 , C07D285/125 , C07D307/46 , C07D307/52 , C07D307/54 , C07D309/06 , C07D333/24 , C07D409/04 , C07D413/04 , C07D513/04 , C07D521/00 , C07F7/08
Abstract: Derivatives of beta -substituted cinnamic acid of the general formula 1 in which R denotes optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and in which R can also denote chlorine or bromine, -X- represents the groups -O-, -S-, m denotes 0 or 1, -Y represents the groups -OR , -O-N=CR R , -NR R , -N(OR )R or -Sr , where the abovementioned substituents R to R denote optionally substituted alkyl, alkenyl, alkynyl, cycloalkyl or cycloalkenyl, and for the radicals R , R and R to R can also denote hydrogen, Z denotes halogen, nitro, cyano, optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted aralkyl, optionally substituted aryloxyalkyl, optionally substituted arylthioalkyl, optionally substituted heteroarylalkyl, optionally substituted heteroaryloxyalkyl, optionally substituted heteroarylthioalkyl, optionally substituted alkenyl, optionally substituted aralkenyl, optionally substituted aryloxyalkenyl, optionally substituted arylthioalkenyl, optionally substituted heteroarylalkenyl, optionally substituted heteroaryloxyalkenyl, optionally substituted heteroarylthioalkenyl, optionally substituted alkynyl, optionally substituted arylalkynyl, optionally substituted heteroarylalkynyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted arylazo, optionally substituted acylamino, -OR , -SR ,-SOR , -SO2R , -COOR , -CONR R , -COR , -CR =NR , -N=CR R , -CR =N-OR , -CR R -O-N=CR R , -CH2-OCOR or -NR R , where the groups R to R , and R and R denote hydrogen, optionally substituted alkyl, optionally substituted alkenyl, optionally substituted alkynyl, optionally substituted cycloalkyl, optionally substituted cycloalkylalkyl, optionally substituted aryl, optionally substituted heteroaryl, optionally substituted aralkyl, optionally substituted heteroarylalkyl, optionally substituted aryloxyalkyl, optionally substituted arylthioalkyl, optionally substituted heteroaryloxyalkyl or optionally substituted heteroarylthioalkyl and R denotes hydrogen or C1-C4-alkyl and in which U, V, W denote hydrogen or have one of the meanings mentioned for Z or in which two of the groups Z, U, V or W in adjacent positions of the phenyl ring optionally together form an optionally substituted five- or six-membered, aromatic or aliphatic ring fused to the phenyl ring, which can optionally contain one to three heteroatoms (N, S, O).
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