公开(公告)号：ES2081314T3

公开(公告)日：1996-03-01

申请号：ES90107120

申请日：1990-04-12

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： UNEME HIDEKI ,  MINAMIDA ISAO ,  OKAUCHI TETSUO

IPC: C07D277/20 ,  A01N43/40 ,  A01N43/78 ,  C07D213/36 ,  C07D213/61 ,  C07D213/64 ,  C07D213/643 ,  C07D213/74 ,  C07D277/32 ,  C07D521/00 ,  C07D213/70 ,  C07D213/38

Abstract: Diaminoethylene derivatives of the formula: wherein R is a heterocyclic group which may be substituted, R , R and R are a hydrogen atom or a hydrocarbon group which may be substituted or R and R are combined to form a cyclic amino group together with the adjacent nitrogen atom; R is hydrogen atom or a hydrocarbon group or heterocyclic group which may be substituted; X is an electron attractive group; Y is a hydroxyl or substituted hydroxyl group, amino or substituted amino group or mercapto or substituted mercapto group; n is 0 or 1; or their salts, which are useful as insecticides.

公开(公告)号：DE69024397D1

公开(公告)日：1996-02-08

申请号：DE69024397

申请日：1990-04-12

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： UNEME HIDEKI ,  MINAMIDA ISAO ,  OKAUCHI TETSUO

IPC: C07D277/20 ,  A01N43/40 ,  A01N43/78 ,  C07D213/36 ,  C07D213/61 ,  C07D213/64 ,  C07D213/643 ,  C07D213/74 ,  C07D277/32 ,  C07D521/00 ,  C07D213/70 ,  C07D213/38

Abstract: Diaminoethylene derivatives of the formula: wherein R is a heterocyclic group which may be substituted, R , R and R are a hydrogen atom or a hydrocarbon group which may be substituted or R and R are combined to form a cyclic amino group together with the adjacent nitrogen atom; R is hydrogen atom or a hydrocarbon group or heterocyclic group which may be substituted; X is an electron attractive group; Y is a hydroxyl or substituted hydroxyl group, amino or substituted amino group or mercapto or substituted mercapto group; n is 0 or 1; or their salts, which are useful as insecticides.

公开(公告)号：ES2061569T3

公开(公告)日：1994-12-16

申请号：ES88112210

申请日：1988-07-28

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： MINAMIDA ISAO ,  IWANAGA KOICHI ,  OKAUCHI TETSUO

IPC: C07D213/61 ,  A01N33/18 ,  A01N35/08 ,  A01N43/40 ,  A01N43/42 ,  A01N43/60 ,  A01N43/78 ,  A01N47/24 ,  A01N55/00 ,  C07C211/22 ,  C07C211/29 ,  C07C229/34 ,  C07C243/10 ,  C07C311/50 ,  C07D20060101 ,  C07D213/24 ,  C07D213/38 ,  C07D213/40 ,  C07D213/42 ,  C07D213/64 ,  C07D213/70 ,  C07D213/74 ,  C07D213/77 ,  C07D215/12 ,  C07D215/38 ,  C07D239/26 ,  C07D241/12 ,  C07D277/20 ,  C07D277/22 ,  C07D277/28 ,  C07D277/32 ,  C07D277/38 ,  C07D277/42 ,  C07D295/13 ,  C07D295/30 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14 ,  C07D403/12 ,  C07D403/14 ,  C07D413/12 ,  C07D413/14 ,  C07D417/12 ,  C07D417/14 ,  C07F7/08 ,  C07D213/36 ,  C07D213/71

Abstract: α-Unsaturated amines of the formula:wherein X¹ and X² are such that one is an electron-attracting group with the other being a hydrogen atom or an electron-attracting group; R¹ is a group attached through a nitrogen atom; R² is a hydrogen atom or a group attached through a carbon, nitrogen or oxygen atom; n is an integer equal to 0, 1 or 2; A is a heterocyclic group or a cyclic hydrocarbon group, and salts thereof and their agrochemical use as insecticidal and/or miticidal agents are described.

公开(公告)号：ES2058057T3

公开(公告)日：1994-11-01

申请号：ES86116752

申请日：1986-12-02

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： MINAMIDA ISAO ,  HASHIMOTO NAOTO

IPC: A61K31/365 ,  A61K31/40 ,  A61K31/44 ,  A61K31/445 ,  A61K31/495 ,  A61K31/535 ,  A61K31/54 ,  A61P31/00 ,  C07D311/00 ,  C07D313/00 ,  C07D493/08 ,  C07H15/00

公开(公告)号：CA1307269C

公开(公告)日：1992-09-08

申请号：CA524507

申请日：1986-12-04

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： MINAMIDA ISAO ,  HASHIMOTO NAOTO

IPC: A61K31/365 ,  A61K31/40 ,  A61K31/44 ,  A61K31/445 ,  A61K31/495 ,  A61K31/535 ,  A61K31/54 ,  A61P31/00 ,  C07D311/00 ,  C07D313/00 ,  C07D493/08 ,  C07H15/00 ,  A61K31/395

Abstract: The present invention provides lankacidin derivative of the formula ¢1! ¢1! In the formula, one of R1 and R2 is H and the other is -C(=X)R5 ¢where X is O or S and R5 are an organic residue! or R1 and R2 together form ¢where R6 is acyl, sulfonyl or alkoxycarbonyl and R7 is alkyl!; R3 and R4 are OH, halogen, azido or an organic residue. The lankacidin derivative ¢1! shows excellent antimicrobial activities and thus can be used for prophylaxis and treatment of infectious disease in animals.

公开(公告)号：DK161081C

公开(公告)日：1991-11-11

申请号：DK621189

申请日：1989-12-08

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： NUMATA MITSUO ,  MINAMIDA ISAO ,  TSUSHIMA SUSUMU

IPC: A61K20060101 ,  A61K31/545 ,  A61K31/546 ,  A61P31/04 ,  C07D20060101 ,  C07D257/04 ,  C07D277/38 ,  C07D277/40 ,  C07D277/46 ,  C07D499/00 ,  C07D501/00 ,  C07D501/20 ,  C07D501/22 ,  C07D501/24 ,  C07D501/28 ,  C07D501/34 ,  C07D501/36 ,  C07D501/38 ,  C07D501/46 ,  C07D501/56 ,  C07D501/60

Abstract: Disclosed are 2-(syn)-hydroxyimino-acetamide derivatives of the formula: wherein Y is hydrogen, hydroxyl, an acyloxy, carbamoyloxy, a quaternary ammonium or a nitrogen-containing heterocyclic ring-substituted thio group; or pharmaceutically acceptable salts or esters thereof are useful as antibacterial agents. Also disclosed are processes for producing them.

公开(公告)号：BR9001734A

公开(公告)日：1991-06-04

申请号：BR9001734

申请日：1990-04-11

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： UNEME HIDEKI ,  MINAMIDA ISAO ,  OKAUCHI TETSUO

IPC: C07D277/20 ,  A01N43/40 ,  A01N43/78 ,  C07D213/36 ,  C07D213/61 ,  C07D213/64 ,  C07D213/643 ,  C07D213/74 ,  C07D277/32 ,  C07D521/00 ,  C07D401/00 ,  C07D405/00 ,  C07D407/00 ,  C07D409/00 ,  A01N43/00

Abstract: Diaminoethylene derivatives of the formula: wherein R is a heterocyclic group which may be substituted, R , R and R are a hydrogen atom or a hydrocarbon group which may be substituted or R and R are combined to form a cyclic amino group together with the adjacent nitrogen atom; R is hydrogen atom or a hydrocarbon group or heterocyclic group which may be substituted; X is an electron attractive group; Y is a hydroxyl or substituted hydroxyl group, amino or substituted amino group or mercapto or substituted mercapto group; n is 0 or 1; or their salts, which are useful as insecticides.

公开(公告)号：DK159783B

公开(公告)日：1990-12-03

申请号：DK270377

申请日：1977-06-17

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： NUMATA MITSUO ,  MINAMIDA ISAO ,  TSUSHIMA SUSUMU

IPC: A61K20060101 ,  A61K31/545 ,  A61K31/546 ,  A61P31/04 ,  C07D20060101 ,  C07D257/04 ,  C07D277/38 ,  C07D277/40 ,  C07D277/46 ,  C07D499/00 ,  C07D501/00 ,  C07D501/20 ,  C07D501/22 ,  C07D501/24 ,  C07D501/28 ,  C07D501/34 ,  C07D501/36 ,  C07D501/38 ,  C07D501/46 ,  C07D501/56 ,  C07D501/60

Abstract: Disclosed are 2-(syn)-hydroxyimino-acetamide derivatives of the formula: wherein Y is hydrogen, hydroxyl, an acyloxy, carbamoyloxy, a quaternary ammonium or a nitrogen-containing heterocyclic ring-substituted thio group; or pharmaceutically acceptable salts or esters thereof are useful as antibacterial agents. Also disclosed are processes for producing them.

公开(公告)号：HUT52751A

公开(公告)日：1990-08-28

申请号：HU60990

申请日：1990-01-31

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： AOKI ISAO ,  TABUCHI TAKANORI ,  MINAMIDA ISAO

IPC: A01N33/18 ,  A01N35/08 ,  A01N37/52 ,  A01N43/40 ,  A01N43/42 ,  A01N43/60 ,  A01N43/78 ,  C07C201/06 ,  C07C201/14 ,  C07C205/08 ,  C07C205/09 ,  C07C209/08 ,  C07C211/27 ,  C07C211/29 ,  C07D213/38 ,  C07D213/61 ,  C07D213/64 ,  C07D213/70 ,  C07D213/74 ,  C07D215/08 ,  C07D215/12 ,  C07D239/26 ,  C07D277/20 ,  C07D277/28 ,  C07D277/32 ,  C07D277/42 ,  C07D277/22 ,  C07D241/12 ,  C07D213/36 ,  C07C211/24 ,  C07C209/06 ,  C07D401/12 ,  C07D403/12 ,  C07D413/12

Abstract: Methods for the production of 1,1,1,-trihalogeno-2-nitroethanes from 1,1-dihalogenoethylene by using nitric acid or its salt and hydrogen chloride or hydrogen bromide or its salt, and for the production of alpha-unsaturated amines from the 1,1,1-trihalogeno-2-nitroethanes which are useful as insecticides.

公开(公告)号：HU900722D0

公开(公告)日：1990-04-28

申请号：HU72288

申请日：1988-07-29

Applicant: TAKEDA CHEMICAL INDUSTRIES LTD

Inventor： MINAMIDA ISAO ,  IWANAGA KOICHI ,  OKAUCHI TETSUO

IPC: C07D213/61 ,  A01N33/18 ,  A01N35/08 ,  A01N43/40 ,  A01N43/42 ,  A01N43/60 ,  A01N43/78 ,  A01N47/24 ,  A01N55/00 ,  C07C211/22 ,  C07C211/29 ,  C07C229/34 ,  C07C243/10 ,  C07C311/50 ,  C07D20060101 ,  C07D213/24 ,  C07D213/38 ,  C07D213/40 ,  C07D213/42 ,  C07D213/64 ,  C07D213/70 ,  C07D213/74 ,  C07D213/77 ,  C07D215/12 ,  C07D215/38 ,  C07D239/26 ,  C07D241/12 ,  C07D277/20 ,  C07D277/22 ,  C07D277/28 ,  C07D277/32 ,  C07D277/38 ,  C07D277/42 ,  C07D295/13 ,  C07D295/30 ,  C07D401/06 ,  C07D401/12 ,  C07D401/14 ,  C07D403/12 ,  C07D403/14 ,  C07D413/12 ,  C07D413/14 ,  C07D417/12 ,  C07D417/14 ,  C07F7/08

Abstract: α-Unsaturated amines of the formula:wherein X¹ and X² are such that one is an electron-attracting group with the other being a hydrogen atom or an electron-attracting group; R¹ is a group attached through a nitrogen atom; R² is a hydrogen atom or a group attached through a carbon, nitrogen or oxygen atom; n is an integer equal to 0, 1 or 2; A is a heterocyclic group or a cyclic hydrocarbon group, and salts thereof and their agrochemical use as insecticidal and/or miticidal agents are described.