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公开(公告)号:PL1682138T6
公开(公告)日:2013-03-29
申请号:PL04811727
申请日:2004-11-18
Applicant: ARRAY BIOPHARMA INC
Inventor: MARLOW ALLISON L , WALLACE ELI , SEO JEONGBEOB , LYSSIKATOS JOSEPH P , YANG HONG WOON , BLAKE JIM
IPC: C07D213/80 , A01N33/02 , A01N43/42 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/90 , A61K20060101 , A61K31/40 , A61K31/415 , A61K31/416 , A61K31/4353 , A61K31/44 , A61K31/4439 , A61K31/4745 , A61K31/495 , A61K31/50 , A61K31/501 , A61K31/502 , A61K31/5025 , A61K31/517 , A61K31/519 , A61K31/53 , A61K31/655 , A61P35/00 , C07D20060101 , C07D209/44 , C07D209/46 , C07D213/82 , C07D215/48 , C07D221/04 , C07D231/56 , C07D237/24 , C07D237/26 , C07D237/28 , C07D237/32 , C07D239/74 , C07D401/04 , C07D401/06 , C07D403/02 , C07D413/02 , C07D413/04 , C07D413/14 , C07D417/02 , C07D417/04 , C07D471/02 , C07D471/04 , C07D487/02 , C07D491/02 , C07D498/02
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公开(公告)号:RS52243B
公开(公告)日:2012-10-31
申请号:RSP20120090
申请日:2006-05-17
Applicant: ASTRAZENECA AB , ARRAY BIOPHARMA INC
Inventor: PITTAM JOHN DAVID , LYSSIKATOS JOSEPH P , MARLOW ALLISON L , WALLACE ELI , SEO JEONGBEOB , YANG HONG WOON , BLAKE JIM , STOREY RICHARD ANTHONY , BOOTH REBECCA JANE , LEONARD JOHN , FIELDING MARK RICHARD
IPC: C07D237/24 , A61K31/501 , A61P35/00 , C07D213/80 , C07D213/82 , C07D213/85
Abstract: This invention relates to a series of novel heterocyclic compounds that are useful in the treatment of hyperproliferative diseases, such as cancer and inflammation, in mammals. This invention also relates to a method of using such compounds in the treatment of hyperproliferative diseases in mammals, especially humans, and to pharmaceutical compositions containing such compounds.
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公开(公告)号:ZA200710318B
公开(公告)日:2012-09-26
申请号:ZA200710318
申请日:2007-04-28
Applicant: ARRAY BIOPHARMA INC , ASTRAZENECA AB
Inventor: MARLOW ALLISON L , WALLACE ELI , SEO JEONGBEIB , LYSSIKATOS JOSEPH P , YANG HONG , BLAKE JIM , STOREY RICHARD ANTHONY , BOOTH REBECCA JANE , PITTAM JOHN DAVID , LEONARD JOHN , FIELDING MARK RICHARD
IPC: C07D20060101 , A61K20060101
Abstract: This invention relates to a series of novel heterocyclic compounds that are useful in the treatment of hyperproliferative diseases, such as cancer and inflammation, in mammals. This invention also relates to a method of using such compounds in the treatment of hyperproliferative diseases in mammals, especially humans, and to pharmaceutical compositions containing such compounds.
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公开(公告)号:PL1922307T3
公开(公告)日:2012-07-31
申请号:PL06836069
申请日:2006-05-17
Applicant: ARRAY BIOPHARMA INC , ASTRAZENECA AB
Inventor: MARLOW ALLISON L , WALLACE ELI , SEO JEONGBEOB , LYSSIKATOS JOSEPH P , YANG HONG WOON , BLAKE JIM , STOREY RICHARD ANTHONY , BOOTH REBECCA JANE , PITTAM JOHN DAVID , LEONARD JOHN , FIELDING MARK RICHARD
IPC: C07D237/24 , A61K31/501 , A61P35/00 , C07D213/80 , C07D213/82 , C07D213/85
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公开(公告)号:UA98926C2
公开(公告)日:2012-07-10
申请号:UAA200705497
申请日:2005-10-18
Applicant: ARRAY BIOPHARMA INC
Inventor: HANS JEREMY , WALLACE ELI M , ZHAO QIAN , LYSSIKATOS JOSEPH P , AICHER TOM , LAIRD ELLEN , ROBINSON JOHN , ALLEN SHELLEY
IPC: A61K38/04 , A61K31/4245 , A61K31/433 , A61K31/4439 , A61K31/496 , A61K31/675 , C07D413/04 , C07D417/04
Abstract: Этоизобретениекасаетсяингибиторовмитотическихкинезинов, вчастности KSP, испособовполученияэтихингибиторов. Изобретениетакжеобеспечиваетфармацевтическиекомпозиции, которыесодержатингибиторысогласноизобретению, ииспользованиеэтихингибиторови фармацевтическихкомпозицийв лечениии предупрежденииразличныхнарушений.
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公开(公告)号:SI1922307T1
公开(公告)日:2012-04-30
申请号:SI200631291
申请日:2006-05-17
Applicant: ARRAY BIOPHARMA INC , ASTRAZENECA AB
Inventor: MARLOW ALLISON L , WALLACE ELI , SEO JEONGBEOB , LYSSIKATOS JOSEPH P , YANG HONG WOON , BLAKE JIM , STOREY RICHARD ANTHONY , BOOTH REBECCA JANE , PITTAM JOHN DAVID , LEONARD JOHN , FIELDING MARK RICHARD
IPC: C07D237/00 , A61K31/00 , A61P35/00 , C07D213/00
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公开(公告)号:DK1922307T3
公开(公告)日:2012-04-02
申请号:DK06836069
申请日:2006-05-17
Applicant: ARRAY BIOPHARMA INC , ASTRAZENECA AB
Inventor: MARLOW ALLISON L , WALLACE ELI , SEO JEONGBEOB , LYSSIKATOS JOSEPH P , YANG HONG WOON , BLAKE JIM , STOREY RICHARD ANTHONY , BOOTH REBECCA JANE , PITTAM JOHN DAVID , LEONARD JOHN , FIELDING MARK RICHARD
IPC: C07D237/24 , A61K31/501 , A61P35/00 , C07D213/80 , C07D213/82 , C07D213/85
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公开(公告)号:HK1153139A1
公开(公告)日:2012-03-23
申请号:HK11107302
申请日:2011-07-13
Applicant: ARRAY BIOPHARMA INC
Inventor: WALLACE ELI M , LYSSIKATOS JOSEPH P , HURLEY BRIAN T , MARLOW ALLISON L
IPC: A61K20060101 , C07D235/08 , A61K31/4184 , A61K31/422 , A61K31/4245 , A61K31/427 , A61K31/4439 , A61K31/454 , A61K31/496 , A61K31/5377 , A61K31/541 , A61P20060101 , A61P1/00 , A61P1/18 , A61P3/10 , A61P9/08 , A61P9/10 , A61P13/08 , A61P13/12 , A61P17/00 , A61P17/04 , A61P17/06 , A61P19/02 , A61P27/02 , A61P29/00 , A61P35/00 , A61P43/00 , C07D20060101 , C07D235/04 , C07D235/06 , C07D401/06 , C07D401/12 , C07D401/14 , C07D403/04 , C07D403/06 , C07D403/12 , C07D405/06 , C07D413/04 , C07D413/06 , C07D417/06 , C07D417/12
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公开(公告)号:AU2010284240A1
公开(公告)日:2012-03-08
申请号:AU2010284240
申请日:2010-08-18
Applicant: ARRAY BIOPHARMA INC , VENTIRX PHARMACEUTICALS INC
Inventor: HOWBERT JAMES JEFFRY , DIETSCH GREGORY , HERSHBERG ROBERT , BURGESS LAURENCE E , LYSSIKATOS JOSEPH P , NEWHOUSE BRAD , YANG HONG WOON
IPC: C07D401/14 , A61K31/4025 , A61K31/454 , A61K31/55 , A61P31/00 , A61P35/00 , C07D223/14 , C07D403/10
Abstract: Provided are compositions and methods useful for modulation of signaling through the Toll-like receptors TLR7 and/or TLR8. The compositions and methods have use in treating or preventing disease, including cancer, autoimmune disease, infectious disease, inflammatory disorder, graft rejection, and graft-verses-host disease.
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公开(公告)号:PL1689387T3
公开(公告)日:2012-02-29
申请号:PL04811726
申请日:2004-11-18
Applicant: ARRAY BIOPHARMA INC
Inventor: WALLACE ELI , YANG HONG WOON , LYSSIKATOS JOSEPH P
IPC: C07D213/80 , A01N33/02 , A01N43/42 , A01N43/54 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/90 , A61K20060101 , A61K31/40 , A61K31/415 , A61K31/416 , A61K31/4353 , A61K31/44 , A61K31/4439 , A61K31/4745 , A61K31/495 , A61K31/50 , A61K31/501 , A61K31/502 , A61K31/5025 , A61K31/517 , A61K31/519 , A61K31/53 , A61K31/655 , A61P35/00 , C07D20060101 , C07D209/44 , C07D209/46 , C07D213/82 , C07D215/48 , C07D221/04 , C07D231/56 , C07D237/24 , C07D237/26 , C07D237/28 , C07D237/32 , C07D239/74 , C07D401/04 , C07D401/06 , C07D403/02 , C07D413/02 , C07D413/04 , C07D413/14 , C07D417/02 , C07D417/04 , C07D471/02 , C07D471/04 , C07D487/02 , C07D491/02 , C07D498/02
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