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公开(公告)号:DE69824332T2
公开(公告)日:2005-06-16
申请号:DE69824332
申请日:1998-03-26
Applicant: SERVIER LAB
Inventor: PEGLION JEAN-LOUIS , GOUMENT BERTRAND , MILLAN MARK , GOBERT ALAIN , AUDINOT VALERIE
IPC: A61K31/443 , A61K31/4433 , A61K31/445 , A61P3/00 , A61P9/00 , A61P25/04 , A61P25/18 , A61P25/30 , C07D405/04 , C07D409/04 , C07D411/04 , C07D471/04 , A61K31/40
Abstract: N-Aryl piperidine derivatives of formula (I), their racemic mixtures, optical isomers and acid addition salts are new. m = 1-5; n = 1 or 2; R = H, 1-5C alkyl or aryl(1-5C) alkyl; E = H or Me; Ar = bicyclic heteroaryl (optionally substituted by halo); and A = adamantyl or bicyclic aryl or tricyclic heteroaryl (both optionally substituted).
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公开(公告)号:MA27070A1
公开(公告)日:2004-12-20
申请号:MA27596
申请日:2004-03-26
Applicant: SERVIER LAB
Inventor: POISSONNIER-DURIEUX SOPHIE , WALLEZ VALERIE , GASNEREAU ANNE , YOUS SAID , LESIEUR DANIEL , DELAGRANGE PHILIPPE , RENARD PIERRE , BENNEJEAN CAROLINE , BOUTIN JEAN ALBERT , AUDINOT VALERIE
IPC: C07D217/14 , A61K31/472 , A61P1/00 , A61P3/02 , A61P3/04 , A61P3/10 , A61P9/00 , A61P15/00 , A61P25/00 , A61P25/02 , A61P25/06 , A61P25/08 , A61P25/16 , A61P25/20 , A61P25/22 , A61P25/24 , A61P25/28 , A61P35/00 , A61P37/02 , A61P43/00 , C07D217/16 , C07D217/24
Abstract: Nouveaux dérivés d'isoquinoleine, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent
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公开(公告)号:DE69630854T2
公开(公告)日:2004-08-26
申请号:DE69630854
申请日:1996-10-10
Applicant: SERVIER LAB
Inventor: PEGLION JEAN-LOUIS , GOUMENT BERTRAND , HARMANGE JEAN-CHRISTOPHE , VIAN JOEL , DESSINGES AIMEE , MILLAN MARK , AUDINOT VALERIE
IPC: A61K31/35 , A61K31/352 , A61K31/38 , A61K31/381 , A61K31/40 , A61P25/00 , A61P25/18 , A61P25/24 , A61P25/26 , A61P25/28 , A61P25/30 , C07C225/20 , C07D311/78 , C07D311/92 , C07D311/94 , C07D333/74 , C07D405/12
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公开(公告)号:ES2213171T3
公开(公告)日:2004-08-16
申请号:ES96402044
申请日:1996-09-26
Applicant: SERVIER LAB
Inventor: PEGLION JEAN-LOUIS , VIAN JOEL , DESSINGES AIMEE , MILLAN MARK , AUDINOT VALERIE
IPC: C07D307/77 , A61K31/34 , A61K31/343 , A61K31/40 , A61P25/00 , A61P25/18 , A61P25/24 , A61P25/26 , A61P25/28 , C07D307/92 , C07D405/12
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公开(公告)号:AT268767T
公开(公告)日:2004-06-15
申请号:AT98400711
申请日:1998-03-26
Applicant: SERVIER LAB
Inventor: PEGLION JEAN-LOUIS , GOUMENT BERTRAND , MILLAN MARK , GOBERT ALAIN , AUDINOT VALERIE
IPC: A61K31/443 , A61K31/4433 , A61K31/445 , A61P3/00 , A61P9/00 , A61P25/04 , A61P25/18 , A61P25/30 , C07D405/04 , C07D409/04 , C07D411/04 , C07D471/04 , A61K31/40 , C07D221/00
Abstract: N-Aryl piperidine derivatives of formula (I), their racemic mixtures, optical isomers and acid addition salts are new. m = 1-5; n = 1 or 2; R = H, 1-5C alkyl or aryl(1-5C) alkyl; E = H or Me; Ar = bicyclic heteroaryl (optionally substituted by halo); and A = adamantyl or bicyclic aryl or tricyclic heteroaryl (both optionally substituted).
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公开(公告)号:PL187005B1
公开(公告)日:2004-04-30
申请号:PL32032597
申请日:1997-06-03
Applicant: SERVIER LAB
Inventor: PEGLION JEAN-LOUIS , MILLAN MARK , BROCCO MAURICETTE , AUDINOT VALERIE
IPC: A61K31/445 , A61K31/495 , A61P25/18 , A61P25/20 , A61P43/00 , C07D413/12 , C07D413/14 , A61K31/42
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公开(公告)号:DK0765877T3
公开(公告)日:2004-04-19
申请号:DK96402044
申请日:1996-09-26
Applicant: SERVIER LAB
Inventor: DESSINGES AIMEE , AUDINOT VALERIE , PEGLION JEAN-LOUIS , VIAN JOEL , MILLAN MARK
IPC: C07D307/77 , A61K31/34 , A61K31/343 , A61K31/40 , A61P25/00 , A61P25/18 , A61P25/24 , A61P25/26 , A61P25/28 , C07D307/92 , C07D405/12
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公开(公告)号:DK0768307T3
公开(公告)日:2004-04-05
申请号:DK96402148
申请日:1996-10-10
Applicant: SERVIER LAB
Inventor: PEGLION JEAN-LOUIS , GOUMENT BERTRAND , HARMANGE JEAN-CHRISTOPHE , VIAN JOEL , DESSINGES AIMEE , MILLAN MARK , AUDINOT VALERIE
IPC: A61K31/35 , A61K31/352 , A61K31/38 , A61K31/381 , A61K31/40 , A61P25/00 , A61P25/18 , A61P25/24 , A61P25/26 , A61P25/28 , A61P25/30 , C07C225/20 , C07D311/78 , C07D311/92 , C07D311/94 , C07D333/74 , C07D405/12
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公开(公告)号:PT768307E
公开(公告)日:2004-03-31
申请号:PT96402148
申请日:1996-10-10
Applicant: SERVIER LAB
Inventor: PEGLION JEAN-LOUIS , AUDINOT VALERIE , GOUMENT BERTRAND , HARMANGE JEAN-CHRISTOPHE , VIAN JOEL , DESSINGES AIMEE , MILLAN MARK
IPC: A61K31/35 , A61K31/352 , A61K31/38 , A61K31/381 , A61K31/40 , A61P25/00 , A61P25/18 , A61P25/24 , A61P25/26 , A61P25/28 , A61P25/30 , C07C225/20 , C07D311/78 , C07D311/92 , C07D311/94 , C07D333/74 , C07D405/12
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公开(公告)号:AT256675T
公开(公告)日:2004-01-15
申请号:AT96402044
申请日:1996-09-26
Applicant: SERVIER LAB
Inventor: PEGLION JEAN-LOUIS , VIAN JOEL , DESSINGES AIMEE , MILLAN MARK , AUDINOT VALERIE
IPC: C07D307/77 , A61K31/34 , A61K31/343 , A61K31/40 , A61P25/00 , A61P25/18 , A61P25/24 , A61P25/26 , A61P25/28 , C07D307/92 , C07D405/12
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