中科微点-全球专利检索

  1. Login
  2. Sign Up

Search Results

196 records (took 0.023 seconds)

    New pyrazine compounds useful in the fungicidal agent, for combating plant pathogenic fungus in protecting materials, plants, ground or seeds and to treat cancer
    83.
    发明专利
    New pyrazine compounds useful in the fungicidal agent, for combating plant pathogenic fungus in protecting materials, plants, ground or seeds and to treat cancer 未知

    公开(公告)号：DE102008000872A1

    公开(公告)日：2008-11-13

    申请号：DE102008000872

    申请日：2008-03-28

    Applicant: BASF SE

    Inventor： DIETZ JOCHEN ,  VRETTOU MARIANNA ,  MUELLER BERND ,  RENNER JENS ,  ULMSCHNEIDER SARAH ,  LOHMANN JAN KLAAS

    IPC: C07D237/06 ,  A01N43/58 ,  A61K31/50

    Abstract: Pyrazine compounds (I) and their salts are new. Pyrazine compounds of formula (I) and their salts are new. R1>, R4>halo (preferred), CN, 1-8C alkoxy or phenyl-1-4C alkyl; R2>1-12C alkyl, 1-10C haloalkyl, 2-10C alkenyl, 2-10C haloalkenyl, 2-10C alkynyl, 2-10C haloalkynyl, 3-6C cycloalkyl, 3-8C cycloalkenyl, 3-12C cycloalkenyl, 3-6C halocycloalkyl, 3-12C halocycloalkenyl, aryl (preferred) or aromatic heterocycle (containing 1-4 R1a group and other than carbon atoms, up to 4 N or 0-2 N, S or O as a ring atoms, where the aromatic groups are 5-10 membered ring system); R1a : CN, nitro, OH, carboxyl, 1-6C alkyl, 2-6C alkynyl, 3-6C cycloalkyl, 3-8C cycloalkenyl, 1-6C alkoxy, 2-6C alkenyloxy, 3-6C alkynyloxy, 3-6C cycloalkoxy, 3-6C cycloalkenyloxy, C(O)R1n, C(O)OR1n, C(S)OR1n, C(O)SR1n, C(S)SR, OC(O)OR1n, 1-6C alkylthio, amino, 1-6C alkylamino, di-1-6C alkylamino, 1-6C alkylene, oxy-1-4C alkylene, oxy-1-3C alkylenoxy, where the divalent groups are bonded to the same atom or at the adjacent atoms, phenyl, naphthyl, 5-10 membered saturated, partially unsaturated or aromatic heterocycle (containing other than the carbon atoms, an up to 4 N or up to 3 N, S or O as a ring atom); R1n : 1-8C alkyl, 3-8C alkenyl, 3-8C alkynyl, 3-6C cycloalkyl or 3-6C cycloalkenyl, where the aliphatic, alicyclic or aromatic groups in R1a and R1n are halogenated partially or completely and carries 1-3 groups of R1b; R1b : halo, CN, nitro, OH, mercapto, amino, carboxyl, alkyl, haloalkyl, alkenyl, alkoxy, haloalkoxy, alkenyloxy, alkynyloxy, alkylthio, alkylamino, dialkylamino, formyl, alkylcarbonyl, alkylsulfonyl, alkylsulfoxyl, alkoxycarbonyl, alkylcarbonyloxy, alkoxycarbonyloxy, aminocarbonyl, aminothiocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkylaminothiocarbonyl, dialkylaminothiocarbonyl, where the alkyl group contains 1-6 carbon atom and the alkenyl- or alkynyl group contains 2-8 carbon atoms, cycloalkyl, cycloalkoxy, heterocyclyl, heterocyclyloxy, where the cyclic system contains 3-10 ring member, aryl, aryloxy, arylthio, aryl-1-6C alkoxy, aryl-1-6C alkyl, hetaryl, hetaryloxy, hetarylthio, where the aryl residue is preferably 6-10 ring members containing 5-6 membered hetaryl residues, where the cyclic systems are partially or completely halogenated and/or substituted by alkyl- or haloalkyl group; R3>aryl (preferred) or heteroaryl, containing other than carbon atom, up to 4 N or 0-2 N, S or as a ring atom, where the group is 5-10 membered ring system, containing a group L1> in ortho position to the bonding to the pyridazine-basic unit and at least a further group Lm; L1>halo, 1-4C alkyl, 1-4C haloalkyl; L : halo, OH, OCN, CN, nitro, 1-8C alkyl, 1-8C haloalkyl, 2-10C alkenyl, 2-10C haloalkenyl, 2-10C alkynyl, 3-6C cycloalkyl, 3-6C halocycloalkyl, 3-6C cycloalkenyl, 1-8C alkoxy, 1-8C haloalkoxy, 2-10C alkenyloxy, 2-10C alkynyloxy, 3-6C cycloalkyloxy, 3-6C cycloalkenyloxy, amino, 1-4C alkylamino, di-(1-4C)-alkylamino, C(O)-R1z, C(S)-R1z, S(O)n-R1z, 1-8C alkoxyimino- (1-8C)-alkyl, 2-10C alkenyloxyimino-(1-8C)-alkyl, 2-10C alkynyloxyimino-(1-8C)-alkyl, 2-10C alkynylcarbonyl, 3-6C cycloalkylcarbonyl, or 5-10 membered saturated, partially unsaturated or aromatic heterocyclic containing 1-4 heteroatoms of O, N or S; R1z : H, 1-4C alkyl, 1-2C haloalkyl, 1-4C alkoxy, 2-4C alkenyloxy, 2-4C alkynyloxy, where the group R1z is substituted with 1-3 R1b group; n : 0-2; and m : 1-4. Independent claims are included for: (1) the preparation of (I); (2) 1,2-dihydro-pyridazine-3,6-dione compound of formula (II); a fungicidal agent containing a solid or liquid carrier and (I); and (3) a seed containing (I) in a quantity of 1-1000 g/100 kg. [Image] [Image] ACTIVITY : Fungicide; Cytostatic. MECHANISM OF ACTION : None given.

    2-(PIRIDIN-2-IL)-PIRIMIDINAS COMO FUNGICIDAS.
    84.
    发明专利
    2-(PIRIDIN-2-IL)-PIRIMIDINAS COMO FUNGICIDAS. 未知

    公开(公告)号：MX2008012513A

    公开(公告)日：2008-10-10

    申请号：MX2008012513

    申请日：2007-04-11

    Applicant: BASF SE

    Inventor： MUELLER BERND ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  DIETZ JOCHEN ,  LOHMANN JAN KLAAS ,  RENNER JENS ,  ULMSCHNEIDER SARAH

    IPC: C07D401/04 ,  A01N43/54 ,  A01N43/90 ,  C07D401/14 ,  C07D405/14 ,  C07D409/14 ,  C07D491/048 ,  C07D491/052 ,  C07D491/056

    Abstract: La presente invención se refiere a 2-(piridin-2-il)-pirimidinas y su uso para el combate de hongos dañinos, así como a agentes fitoprotectores, que contienen estos compuestos como componente eficaz. (ver fórmula I) en donde: Q es un carbociclo condensado, saturado, de 5, 6 6 7 miembros o un heterociclo de 5, 6 ó 7 miembros que presenta, además de los miembros del anillo de carbono, uno o dos heteroátomos seleccionados entre oxígeno y azufre como miembros del anillo, en donde el carbociclo y el heterociclo no están sustituidos o presentan 1, 2, 3 ó 4 grupos alquilo C1-C4 como sustituyentes; es hidrógeno, OH, alquilo C1-C4, alcoxi C1-C4, halogenalquilo C1-C4, halogenalcoxi C1-C4 o halógeno; R2 es hidrógeno, NO2, halógeno, alquilo C1-C6, cicloalquilo C3-C6, alcoxi C1-C6, halogenalquilo Ci-C6 O halogenalcoxi C1-C6 R3 es hidrógeno, halógeno, alquilo Ci-C4, alcoxi C1- C4, halogenalquilo C1-C4 o halogenalcoxi C1-C4 es fenilo, heteroarilo de 5 miembros que presenta 1, 2, 3 ó 4 átomos de nitrógeno o 1 heteroátomo seleccionado entre oxígeno y azufre y eventualmente 1, 2 ó 3 átomos de nitrógeno como átomos del anillo, o hetarilo de 6 miembros, que presenta 1, 2, 3 ó 4 átomos de nitrógeno como miembros del anillo, en donde el fenilo, el hetarilo de 5 y 6 miembros pueden presentar 1, 2, 3 ó 4 sustituyentes Ra.

    SUBSTITUTED 5-HETARYL-4-AMINOPYRIMIDINES
    86.
    发明专利
    SUBSTITUTED 5-HETARYL-4-AMINOPYRIMIDINES 未知

    公开(公告)号：CA2645779A1

    公开(公告)日：2007-10-04

    申请号：CA2645779

    申请日：2007-03-26

    Applicant: BASF SE

    Inventor： MUELLER BERND ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  STIERL REINHARD ,  RENNER JENS ,  ULMSCHNEIDER SARAH ,  GRAMMENOS WASSILIOS

    IPC: A01N43/54 ,  A01N43/56 ,  A01N43/653 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01P3/00 ,  A01P5/00 ,  A01P7/00 ,  A61K31/506 ,  C07D401/04 ,  C07D403/04 ,  C07D405/04 ,  C07D409/04 ,  C07D413/04 ,  C07D417/04

    Abstract: The present invention relates to the use of 5-hetaryl-4-aminopyrimidines of the formula I and their salts for controlling plant-damaging fungi. The invention also relates to novel 5-hetaryl-4-aminopyrimidines and to crop protection compositions comprising at least one such compound as active component. Het is an optionally substituted 5- or 6-membered aromatic heterocycle which has 1, 2, 3 or 4 heteroatoms selected from the group consisting of nitrogen, oxygen and sulfur as ring members, where the 5- or 6-membered heteroaromatic radical may have 1, 2, 3 or 4 identical or different substituents L, R1, R2 are inter alia hydrogen, C1-C8-alkyl, C3-C8-cycloalkyl, C5-C10-bicycloalkyl, C2-C8-alkenyl, C4-C10-alkadienyl, C3-C6-cycloalkenyl, C2-C8-alkynyl, phenyl, naphthyl or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle which has one, two, three or four heteroatoms from the group consisting of O, N or S as ring members; or together form a ring; R3 is inter alia hydrogen, OH, halogen, cyano, NR31R32, C1-C8-alkyl, C1-C8-alkoxy, C1-C8-alkylthio, C1-C8-alkylsulfinyl, C1-C8-alkylsulfonyl, C2-C8-alkenyl or C2-C8-alkynyl, and R4 is halogen, cyano, hydroxyl, mercapto, N3, C1-C6-alkyl, C2-C8-alkenyl, C2-C8-alkynyl, C1-C6-haloalkyl, C1-C6-alkoxy, C3-C8-alkenyloxy, C3-C8-alkynyloxy, C1-C6-haloalkoxy, C1-C6-alkylthio, C3-C8-alkenylthio, C3-C8-alkinylthio, C1-C6-haloalkylthio, or is a radical of the formula C(═Z)OR41, C(═Z)NR42R43, C(═Z)NR44—NR42R43, C(═Z)R45, CR46R47—OR48, CR46R47—NR42R43, ON(═CR49R50), O—C(═Z)R45, NR42R43a, NR51(C(═Z)R45), NR51(C(═Z)OR41), NR51(C(═Z)—NR42R43), NR52a(N═CR49R50), NR52NR42R43, NR52OR41 or C(═N—X—R45)SR41.

Patent Agency Ranking