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公开(公告)号:WO0174787A3
公开(公告)日:2002-02-07
申请号:PCT/US0109112
申请日:2001-03-21
Applicant: ABBOTT LAB
Inventor: DICKMAN DANIEL A , CHEMBURKAR SANJAY , FORT JAMES J , HENRY RODGER F , LECHUGA-BALLESTEROS DAVID , NIU YUPING , PORTER WILLIAM
IPC: A61K31/513 , A61P31/18 , A61P43/00 , C07D239/10 , A61K31/505
CPC classification number: C07D239/10
Abstract: New crystalline forms of lopinavir are disclosed.
Abstract translation: 公开了新的结晶形式的洛匹那韦。
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公开(公告)号:HU0302675A2
公开(公告)日:2003-12-29
申请号:HU0302675
申请日:2001-03-21
Applicant: ABBOTT LAB
Inventor: CHEMBURKAR SANJAY , DICKMAN DANIEL A , FORT JAMES J , HENRY RODGER F , LECHUGA-BALLESTEROS DAVID , NIU YUPING , PORTER WILLIAM
IPC: A61K20060101 , A61K31/513 , A61P20060101 , A61P31/18 , A61P43/00 , C07D20060101 , C07D239/10
Abstract: New crystalline forms of lopinavir are disclosed.
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公开(公告)号:AU5092001A
公开(公告)日:2001-10-15
申请号:AU5092001
申请日:2001-03-21
Applicant: ABBOTT LAB
Inventor: DICKMAN DANIEL A , CHEMBURKAR SANJAY , FORT JAMES J , HENRY RODGER F , LECHUGA-BALLESTEROS DAVID , NIU YUPING , PORTER WILLIAM
IPC: A61K20060101 , A61K31/513 , A61P20060101 , A61P31/18 , A61P43/00 , C07D20060101 , C07D239/10 , C07D239/00
Abstract: New crystalline forms of lopinavir are disclosed.
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公开(公告)号:MY128296A
公开(公告)日:2007-01-31
申请号:MYPI20011034
申请日:2001-03-07
Applicant: ABBOTT LAB
Inventor: DICKMAN DANIEL A , CHEMBURKAR SANJAY , FORT JAMES J , HENRY RODGER F , LECHUGA-BALLESTEROS DAVID , NIU YUPING , PORTER WILLIAM
IPC: C07D239/36 , A61K20060101 , A61K31/513 , A61P20060101 , A61P31/18 , A61P43/00 , C07D20060101 , C07D239/10
Abstract: THERE IS DISCLOSED A NON-SOLVATED CRYSTALLINE FORM OF THE COMPOUND (2S,3S,5S)-2-(2,6 DIMETHYLPHENOXYACETYL)AMINO-3-HYDROXY-5-(2-(1-TETRAHYDRO PYRIMID-2-ONYL)-3-METHYLBUTANOYL)) AMINO-1,6-DIPHENYLHEXANE WITH A PEAK IN THE SOLID STATE INFRARED SPECTRUM AT A POSITION WITHIN THE RANGE 1680-1685 CM¯¹ AND A PEAK IN THE SOLID STATE INFRARED SPECTRUM AT A POSITION WITHIN THE RANGE 1625-1630 CM¯¹.(FIG 1)
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公开(公告)号:SA1573B1
公开(公告)日:2006-11-14
申请号:SA01220270
申请日:2001-08-07
Applicant: ABBOTT LAB
Inventor: DICKMAN DANIEL A , CHEMBURKAR SANJAY , FORT JAMES J , HENRY RODGER F , LECHUGA-BALLESTEROS DAVID , NIU YUPING , PORTER WILLIAM
IPC: A61K20060101 , A61K31/513 , A61P20060101 , A61P31/18 , A61P43/00 , C07D20060101 , C07D239/10
Abstract: الملخص: يصفالاختراعالراهنأشكالبلورية crystalline forms جديدةمنلوبينافير lopinavir.
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公开(公告)号:AU2006222711A1
公开(公告)日:2006-10-19
申请号:AU2006222711
申请日:2006-09-27
Applicant: ABBOTT LAB
Inventor: PORTER WILLIAM , FORT JAMES J , NIU YUPING , CHEMBURKAR SANJAY , HENRY RODGER F , LECHUGA-BALLESTEROS DAVID , DICKMAN DANIEL A
IPC: C07D239/10 , A61K20060101 , A61K31/513 , A61P20060101 , A61P31/18 , A61P43/00 , C07D20060101
Abstract: New crystalline forms of lopinavir are disclosed.
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公开(公告)号:BG107165A
公开(公告)日:2003-07-31
申请号:BG10716502
申请日:2002-10-03
Applicant: ABBOTT LAB
Inventor: DICKMAN DANIEL A , CHEMBURKAR SANJAY , FORT JAMES J , HENRY RODGER F , LECHUGA-BALLESTEROS DAVID , NIU YUPING , PORTER WILLIAM
IPC: A61K20060101 , A61K31/513 , A61P20060101 , A61P31/18 , A61P43/00 , C07D20060101 , C07D239/10
Abstract: The invention relates to new crystalline forms of lopinavir with peaks in the solid phase infrared spectrum in the interval 1652-1666 cm-1 and 1606-1615 cm-1, and to methods for their preparation. The crystalline forms are used for the purification or isolation of lopinavir or for the production of pharmaceutical preparations. 23 claims, 31 figures
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公开(公告)号:NO20024679L
公开(公告)日:2002-09-30
申请号:NO20024679
申请日:2002-09-30
Applicant: ABBOTT LAB
Inventor: DICKMAN DANIEL A , CHEMBURKAR SANJAY , FORT JAMES J , HENRY RODGER F , LECHUGA-BALLESTEROS DAVID , NIU YUPING , PORTER WILLIAM
IPC: A61K20060101 , A61K31/513 , A61P20060101 , A61P31/18 , A61P43/00 , C07D20060101 , C07D239/10
Abstract: New crystalline forms of lopinavir are disclosed.
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公开(公告)号:NO325005B1
公开(公告)日:2008-01-14
申请号:NO20024679
申请日:2002-09-30
Applicant: ABBOTT LAB
Inventor: CHEMBURKAR SANJAY , LECHUGA-BALLESTEROS DAVID , DICKMAN DANIEL A , FORT JAMES J , HENRY RODGER F , NIU YUPING , PORTER WILLIAM
IPC: C07D239/10 , A61K20060101 , A61K31/513 , A61P20060101 , A61P31/18 , A61P43/00 , C07D20060101
Abstract: New crystalline forms of lopinavir are disclosed.
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公开(公告)号:NO20024679D0
公开(公告)日:2002-09-30
申请号:NO20024679
申请日:2002-09-30
Applicant: ABBOTT LAB
Inventor: DICKMAN DANIEL A , CHEMBURKAR SANJAY , FORT JAMES J , HENRY RODGER F , LECHUGA-BALLESTEROS DAVID , NIU YUPING , PORTER WILLIAM
IPC: A61K20060101 , A61K31/513 , A61P20060101 , A61P31/18 , A61P43/00 , C07D20060101 , C07D239/10 , C07D
Abstract: New crystalline forms of lopinavir are disclosed.
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