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公开(公告)号:WO0132655A2
公开(公告)日:2001-05-10
申请号:PCT/US0030551
申请日:2000-11-06
Applicant: ABBOTT LAB
Inventor: ELMORE STEVEN W , COOPER CURT S , SCHULTZ COLLEEN C , HUTCHINSON DOUGLAS K , DONNER PAMELA L , GREEN BRIAN E , ANDERSON DAVID D , XIE QINGHUA , DINGES JURGEN , LYNCH LINDA M
IPC: A61K31/4375 , A61K31/4436 , A61K31/444 , A61K31/4725 , A61K31/496 , A61K31/542 , A61P31/04 , A61P43/00 , C07B61/00 , C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04 , C07D519/00 , C07D409/00
CPC classification number: C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04
Abstract: Compounds having formula (I), or pharmaceutically acceptable salts or prodrugs thereof, wherein A is nitrogen or (II), wherein W is selected from the group consisting of (1) hydrogen and (2) optionally substituted alkyl; A is selected from the group consisting of (1) -S-, (2) -O-, and (3) -N(R )-, wherein R is hydrogen or C1-C6 alkyl; and R and R together are a carbocyclic or a heterocyclic ring, are useful as antibacterial agents.
Abstract translation: 具有式(I)化合物或其药学上可接受的盐或前药,其中A 1是氮或(II),其中W选自(1)氢和(2)任选取代的烷基; A 2选自(1)-S-,(2)-O-和(3)-N(R 7) - ,其中R 7是氢或C 1 -C 6 烷基; R 5和R 6一起是碳环或杂环,可用作抗菌剂。
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公开(公告)号:BR0010728A
公开(公告)日:2004-02-17
申请号:BR0010728
申请日:2000-11-06
Applicant: ABBOTT LAB
Inventor: ELMORE STEVEN W , COOPER CURT S , SCHULTZ COLLEEN C , HUTCHINSON DOUGLAS K , DONNER PAMELA L , GREEN BRIAN E , ANDERSON DAVID D , XIE QUINGHUA , DINGES JURGEN , LYNCH LINDA M
IPC: A61K31/4375 , A61K31/4436 , A61K31/444 , A61K31/4725 , A61K31/496 , A61K31/542 , A61P31/04 , A61P43/00 , C07B61/00 , C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04 , C07D519/00 , C07D409/00
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公开(公告)号:NO20022156A
公开(公告)日:2002-07-04
申请号:NO20022156
申请日:2002-05-06
Applicant: ABBOTT LAB
Inventor: ELMORE STEVEN W , COOPER CURT S , SCHULTZ COLLEEN C , HUTCHINSON DOUGLAS K , DONNER PAMELA L , GREEN BRIAN E , ANDERSON DAVID D , XIE QINGHUA , DINGES JURGEN , LYNCH LINDA M
IPC: A61K31/4375 , A61K31/4436 , A61K31/444 , A61K31/4725 , A61K31/496 , A61K31/542 , A61P31/04 , A61P43/00 , C07B61/00 , C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04 , C07D519/00 , A61K31/4709
CPC classification number: C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04
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公开(公告)号:CZ20021531A3
公开(公告)日:2002-09-11
申请号:CZ20021531
申请日:2000-11-06
Applicant: ABBOTT LAB
Inventor: GREEN BRIAN E , ANDERSON DAVID D , XIE QINGHUA , DINGES JURGEN , LYNCH LINDA M , ELMORE STEVEN W , COOPER CURT S , SCHULTZ COLLEEN C , HUTCHINSON DOUGLAS K , DONNER PAMELA L
IPC: A61K31/4375 , A61K31/4436 , A61K31/444 , A61K31/4725 , A61K31/496 , A61K31/542 , A61P31/04 , A61P43/00 , C07B61/00 , C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04 , C07D519/00 , C07D409/10 , A61K31/381 , A61K31/47 , C07D405/10 , C07D417/10 , C07D495/10
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公开(公告)号:BG106679A
公开(公告)日:2003-01-31
申请号:BG10667902
申请日:2002-05-09
Applicant: ABBOTT LAB
Inventor: ELMORE STEVEN W , COOPER CURT S , SCHULTZ COLLEEN C , HUTCHINSON DOUGLAS K , DONNER PAMELA L , GREEN BRIAN E , ANDERSON DAVID D , XIE QINGHUA , DINGES JURGEN , LYNCH LINDA M
IPC: A61K31/4375 , A61K31/4436 , A61K31/444 , A61K31/4725 , A61K31/496 , A61K31/542 , A61P31/04 , A61P43/00 , C07B61/00 , C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04 , C07D519/00 , A61K31/4709 , C07D417/04
Abstract: Compounds having the formula are pharmaceutically acceptable salts or prodrugs thereof, are useful as antibacterial agents. 21 claims
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公开(公告)号:AU1468901A
公开(公告)日:2001-05-14
申请号:AU1468901
申请日:2000-11-06
Applicant: ABBOTT LAB
Inventor: ELMORE STEVEN W , COOPER CURT S , SCHULTZ COLLEEN C , HUTCHINSON DOUGLAS K , DONNER PAMELA L , GREEN BRIAN E , ANDERSON DAVID D , XIE QINGHUA , DINGES JURGEN , LYNCH LINDA M
IPC: A61K31/4375 , A61K31/4436 , A61K31/444 , A61K31/4725 , A61K31/496 , A61K31/542 , A61P31/04 , A61P43/00 , C07B61/00 , C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04 , C07D519/00 , C07D409/00
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公开(公告)号:ZA200202187B
公开(公告)日:2004-11-17
申请号:ZA200202187
申请日:2002-03-18
Applicant: ABBOTT LAB
Inventor: ELMORE STEVEN W , SCHULTZ COLLEEN C , DONNER PAMELA L , ANDERSON DAVID D , DINGES JURGEN , COOPER CURT S , HUTCHINSON DOUGLAS K , GREEN BRIAN E , XIE QINGHUA , LYNCH LINDA M
IPC: A61K20060101 , A61P20060101 , C07D20060101 , C07D , A61K , A61P
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公开(公告)号:NO20022156L
公开(公告)日:2002-07-04
申请号:NO20022156
申请日:2002-05-06
Applicant: ABBOTT LAB
Inventor: ELMORE STEVEN W , COOPER CURT S , SCHULTZ COLLEEN C , HUTCHINSON DOUGLAS K , DONNER PAMELA L , GREEN BRIAN E , ANDERSON DAVID D , XIE QINGHUA , DINGES JURGEN , LYNCH LINDA M
IPC: A61K31/4375 , A61K31/4436 , A61K31/444 , A61K31/4725 , A61K31/496 , A61K31/542 , A61P31/04 , A61P43/00 , C07B61/00 , C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04 , C07D519/00 , A61K31/4709
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公开(公告)号:NO20022156D0
公开(公告)日:2002-05-06
申请号:NO20022156
申请日:2002-05-06
Applicant: ABBOTT LAB
Inventor: ELMORE STEVEN W , COOPER CURT S , SCHULTZ COLLEEN C , HUTCHINSON DOUGLAS K , DONNER PAMELA L , GREEN BRIAN E , ANDERSON DAVID D , XIE QINGHUA , DINGES JURGEN , LYNCH LINDA M
IPC: A61K31/4375 , A61K31/4436 , A61K31/444 , A61K31/4725 , A61K31/496 , A61K31/542 , A61P31/04 , A61P43/00 , C07B61/00 , C07D405/04 , C07D409/04 , C07D409/14 , C07D413/14 , C07D417/14 , C07D471/04 , C07D495/04 , C07D513/04 , C07D519/00 , C07D
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