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公开(公告)号:ZA971184B
公开(公告)日:1997-08-27
申请号:ZA971184
申请日:1997-02-12
Applicant: ABBOTT LAB
Inventor: TASKER ANDREW S , VONGELDERN THOMAS W , JAE HWAN-SOO , SORENSEN BRYAN K , WINN MARTIN , BOYD STEVEN A , HENRY KENNETH J
IPC: A61K31/395 , A61K31/40 , A61K31/4025 , A61K31/675 , A61P1/00 , A61P7/00 , A61P9/00 , A61P11/00 , A61P13/12 , A61P25/04 , A61P35/00 , A61P43/00 , C07D20060101 , C07D207/16 , C07D401/04 , C07D403/04 , C07D405/04 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14 , C07D419/14 , C07D453/02 , C07F9/572 , C07D , A61K , C07F
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公开(公告)号:DK0776324T3
公开(公告)日:2002-10-07
申请号:DK95928323
申请日:1995-08-04
Applicant: ABBOTT LAB
Inventor: WINN MARTIN , BOYD STEVEN A , HUTCHINS CHARLES W , JAE HWAN-SOO , TASKER ANDREW S , VONGELDERN THOMAS W , KESTER JEFFREY A , SORENSEN BRYAN K
IPC: A61K31/40 , A61K31/402 , A61K31/4025 , A61K31/403 , A61K31/41 , A61K31/415 , A61K31/422 , A61K31/435 , A61K31/44 , A61K31/4439 , A61K31/445 , A61K31/454 , A61K31/47 , A61K31/505 , A61K31/506 , A61K31/535 , A61K31/5377 , A61P9/00 , A61P9/04 , A61P9/08 , A61P9/10 , A61P9/12 , A61P29/00 , A61P35/00 , A61P43/00 , C07D20060101 , C07D207/14 , C07D207/16 , C07D401/04 , C07D403/04 , C07D405/04 , C07D405/10 , C07D405/14 , C07D413/04 , C07D419/04 , C07D471/04 , C07F9/572 , C07F9/59
Abstract: Processes for preparing endothelin antagonists of formula (I) and pharmaceutically acceptable salts thereof and processes for preparing intermediates thereof.
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公开(公告)号:ZA9805209B
公开(公告)日:1999-01-06
申请号:ZA9805209
申请日:1998-06-15
Applicant: ABBOTT LAB
Inventor: TASKER ANDREW S , WINN MARTIN , BOYD STEVEN A , JAE HWAN-SOO , VONGELDERN THOMAS W , SORENSEN BRYAN K , HENRY KENNETH J
IPC: C07D207/16 , C07D405/04 , C07D , A61K , C07F
CPC classification number: C07D405/04 , C07D207/16
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公开(公告)号:CA2195677C
公开(公告)日:2005-11-08
申请号:CA2195677
申请日:1995-08-04
Applicant: ABBOTT LAB
Inventor: WINN MARTIN , BOYD STEVEN A , HUTCHINS CHARLES W , JAE HWAN-SOO , TASKER ANDREW S , VONGELDERN THOMAS W , KESTER JEFFREY A , SORENSEN BRYAN K
IPC: A61K31/40 , A61K31/402 , A61K31/4025 , A61K31/403 , A61K31/41 , A61K31/415 , A61K31/422 , A61K31/435 , A61K31/44 , A61K31/4439 , A61K31/445 , A61K31/454 , A61K31/47 , A61K31/505 , A61K31/506 , A61K31/535 , A61K31/5377 , A61P9/00 , A61P9/04 , A61P9/08 , A61P9/10 , A61P9/12 , A61P29/00 , A61P35/00 , A61P43/00 , C07D20060101 , C07D207/14 , C07D207/16 , C07D401/04 , C07D403/04 , C07D405/04 , C07D405/10 , C07D405/14 , C07D413/04 , C07D419/04 , C07D471/04 , C07F9/572 , C07F9/59
Abstract: A compound of formula (I) or a pharmaceutically acceptable salt thereof is disclosed, as well as processes for and intermediates in the preparation thereof, and a method of antagonizing endothelin.
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公开(公告)号:AT219077T
公开(公告)日:2002-06-15
申请号:AT95928323
申请日:1995-08-04
Applicant: ABBOTT LAB
Inventor: WINN MARTIN , BOYD STEVEN A , HUTCHINS CHARLES W , JAE HWAN-SOO , TASKER ANDREW S , VONGELDERN THOMAS W , KESTER JEFFREY A , SORENSEN BRYAN K
IPC: A61K31/40 , A61K31/402 , A61K31/4025 , A61K31/403 , A61K31/41 , A61K31/415 , A61K31/422 , A61K31/435 , A61K31/44 , A61K31/4439 , A61K31/445 , A61K31/454 , A61K31/47 , A61K31/505 , A61K31/506 , A61K31/535 , A61K31/5377 , A61P9/00 , A61P9/04 , A61P9/08 , A61P9/10 , A61P9/12 , A61P29/00 , A61P35/00 , A61P43/00 , C07D20060101 , C07D207/14 , C07D207/16 , C07D401/04 , C07D403/04 , C07D405/04 , C07D405/10 , C07D405/14 , C07D413/04 , C07D419/04 , C07D471/04 , C07F9/572 , C07F9/59
Abstract: Processes for preparing endothelin antagonists of formula (I) and pharmaceutically acceptable salts thereof and processes for preparing intermediates thereof.
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公开(公告)号:ZA985209B
公开(公告)日:1999-01-06
申请号:ZA985209
申请日:1998-06-15
Applicant: ABBOTT LAB
Inventor: TASKER ANDREW S , WINN MARTIN , BOYD STEVEN A , JAE HWAN-SOO , VONGELDERN THOMAS W , SORENSEN BRYAN K , HENRY KENNETH J
IPC: C07D207/16 , C07D405/04 , C07D , A61K , C07F
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公开(公告)号:ZA9701184B
公开(公告)日:1997-08-27
申请号:ZA9701184
申请日:1997-02-12
Applicant: ABBOTT LAB
Inventor: TASKER ANDREW S , VONGELDERN THOMAS W , JAE HWAN-SOO , SORENSEN BRYAN K , WINN MARTIN , BOYD STEVEN A , HENRY KENNETH J
IPC: A61K31/395 , A61K31/40 , A61K31/4025 , A61K31/675 , A61P1/00 , A61P7/00 , A61P9/00 , A61P11/00 , A61P13/12 , A61P25/04 , A61P35/00 , A61P43/00 , C07D20060101 , C07D207/16 , C07D401/04 , C07D403/04 , C07D405/04 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14 , C07D419/14 , C07D453/02 , C07F9/572 , C07D , A61K , C07F
CPC classification number: C07D405/04 , A61K9/2059 , A61K9/4866
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公开(公告)号:ZA95892B
公开(公告)日:1996-01-24
申请号:ZA95892
申请日:1995-02-03
Applicant: ABBOTT LAB
Inventor: ROSENBERG SAUL H , SULLIVAN GERARD M , VONGELDERN THOMAS W , ZYDOWSKY THOMAS M , TASKER ANDREW S
IPC: A61K20060101 , C07C20060101 , C07D20060101 , A61K , C07C , C07D
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公开(公告)号:ZA9500892B
公开(公告)日:1996-01-24
申请号:ZA9500892
申请日:1995-02-03
Applicant: ABBOTT LAB
Inventor: ROSENBERG SAUL H , SULLIVAN GERARD M , VONGELDERN THOMAS W , ZYDOWSKY THOMAS M , TASKER ANDREW S
IPC: A61K20060101 , C07C20060101 , C07D20060101 , A61K , C07C , C07D
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公开(公告)号:PT888340E
公开(公告)日:2002-12-31
申请号:PT97905897
申请日:1997-02-10
Applicant: ABBOTT LAB
Inventor: SORENSEN BRYAN K , TASKER ANDREW S , WINN MARTIN , JAE HWAN-SOO , VONGELDERN THOMAS W , BOYD STEVEN A , HENRY KENNETH J
IPC: A61K31/395 , A61K31/40 , A61K31/4025 , A61K31/675 , A61P1/00 , A61P7/00 , A61P9/00 , A61P11/00 , A61P13/12 , A61P25/04 , A61P35/00 , A61P43/00 , C07D20060101 , C07D207/16 , C07D401/04 , C07D403/04 , C07D405/04 , C07D405/14 , C07D409/14 , C07D413/14 , C07D417/14 , C07D419/14 , C07D453/02 , C07F9/572
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