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公开(公告)号:HK1146664A1
公开(公告)日:2011-06-30
申请号:HK10111467
申请日:2010-12-09
Applicant: ARRAY BIOPHARMA INC
Inventor: MARK MUNSON , DAVID A MARESKA A , YOUNGBOO KIM , ROBERT GRONEBERG , JAMES RIZZI , MARTHA RODRIGUEZ , GANGHYEOK KIM , GUY VIGERS , CHANG RAO , DEVAN BALACHARI , DARREN HARVEY
IPC: C07D20060101 , A61K20060101 , A61K31/4745 , A61K31/503 , A61K31/675 , A61P20060101 , C07D231/56 , C07D261/20 , C07D401/14 , C07D403/04 , C07D403/12 , C07D405/12 , C07D413/12 , C07D471/02 , C07D471/04 , C07D487/02 , C07D491/02 , C07D498/02
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公开(公告)号:HK1084673A1
公开(公告)日:2006-08-04
申请号:HK06107025
申请日:2006-06-21
Applicant: ARRAY BIOPHARMA INC
Inventor: MARK MUNSON , MARESKA DAVID A , YOUNGBOO KIM , ROBERT GRONEBERG , JAMES RIZZI , MARTHA RODRIGUEZ , GANGHYEOK KIM , GUY VIGERS , CHANG RAO , DEVAN BALACHARI , DARREN HARVEY
IPC: C07D20090101 , A61K20060101 , A61K31/4745 , A61K31/503 , A61K31/675 , A61P20090101 , C07D231/56 , C07D261/20 , C07D401/14 , C07D403/04 , C07D403/12 , C07D405/12 , C07D413/12 , C07D471/02 , C07D471/04 , C07D487/02 , C07D491/02 , C07D498/02
Abstract: Compounds having the Formula: wherein Y, A, W, B, U, V, X and Ar 1 have the meanings given in the specification, which compounds are useful in therapy as p38-inhibitors.
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公开(公告)号:BRPI0407993B8
公开(公告)日:2021-05-25
申请号:BRPI0407993
申请日:2004-02-25
Applicant: ARRAY BIOPHARMA INC
Inventor: CHANG RAO , DARREN HARVEY , DAVID A MARESKA , DEVAN BALACHARI , GANGHYEOK KIM , GUY VIGERS , JAMES RIZZI , MARK MUNSON , MARTHA RODRIGUEZ , ROBERT D GRONENBERG , YOUNGBOO KIM
IPC: C07D401/14 , A61K20060101 , A61K31/4745 , A61K31/503 , A61K31/675 , A61P29/00 , C07D20060101 , C07D231/56 , C07D261/20 , C07D403/04 , C07D403/12 , C07D405/12 , C07D413/12 , C07D471/02 , C07D471/04 , C07D487/02 , C07D491/02 , C07D498/02
Abstract: "inibidores de p38 e métodos para uso dos mesmos". a presente invenção refere-se a inibidores de p38 e métodos para produção desses inibidores. a invenção também provê composições farmacêuticas compreendendo os inibidores da invenção e métodos de utilização dos inibidores e composições farmacêuticas no tratamento e prevenção de vários distúrbios mediados por p38.
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公开(公告)号:ZA200806507B
公开(公告)日:2009-10-28
申请号:ZA200806507
申请日:2008-07-25
Applicant: ARRAY BIOPHARMA INC
Inventor: ROBERT GRONEBERG , BURGESS LAURENCE E , DARREN HARVEY , ELLEN LAIRD , MARK MUNSON , JAMES RIZZI , MARTHA RODRIGUEZ , TODD EARY CHARLES , DANIEL WATSON
IPC: A61K20100101 , A61P20100101 , C07D20100101
Abstract: The compound of Formula (I) and pharmaceutically acceptable salts and prodrugs thereof are useful in the treatment and prevention of various disorders mediated by kinases.
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公开(公告)号:BRPI0419305B8
公开(公告)日:2021-05-25
申请号:BRPI0419305
申请日:2004-02-25
Applicant: ARRAY BIOPHARMA INC
Inventor: CHANG RAO , DARREN HARVEY , DAVID A MARESKA , DEVAN BALACHARI , GANGHYEOK KIM , GUY P A VIGERS , JAMES RIZZI , MARK MUNSON , MARTHA RODRIGUEZ , ROBERT D GRONEBERG , YOUNGBOO KIM
IPC: C07D401/14 , A61K20060101 , A61K31/4745 , A61K31/503 , A61K31/675 , C07D20060101 , C07D231/56 , C07D261/20 , C07D403/04 , C07D403/12 , C07D405/12 , C07D413/12 , C07D471/02 , C07D471/04 , C07D487/02 , C07D491/02 , C07D498/02
Abstract: compostos inibidores de p38,composições farmacêuticas compreendendo o mesmos e usos dos referidos compostos na preparação de medicamentos. a presente invenção refere-se a compostos que apresentam a fórmula: em que y, a, w, b, u, v, x, e ar1 são definidos de acordo com o relatório descritivo. os referidos compostos são úteis em terapias como inibidores de p38.
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公开(公告)号:IS2959B
公开(公告)日:2017-02-15
申请号:IS8810
申请日:2009-03-16
Applicant: ARRAY BIOPHARMA INC
Inventor: MARK MUNSON , DAVID A MARESKA , YOUNGBOO KIM , ROBERT GRONEBERG , JAMES RIZZI , MARTHA RODRIGUEZ , GANGHYEOK KIM , GUY VIGERS , CHANG RAO , DEVAN BALACHARI , DARREN HARVEY
IPC: C07D401/14 , A61K20060101 , A61K31/4745 , A61K31/503 , A61K31/675 , C07D20060101 , C07D231/56 , C07D261/20 , C07D403/04 , C07D403/12 , C07D405/12 , C07D413/12 , C07D471/02 , C07D471/04 , C07D487/02 , C07D491/02 , C07D498/02
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公开(公告)号:MY151835A
公开(公告)日:2014-07-14
申请号:MYPI20082836
申请日:2007-01-26
Applicant: ARRAY BIOPHARMA INC
Inventor: ROBERT GRONEBERG , BURGESS LAURENCE E , DARREN HARVEY , ELLEN LAIRD , MARK MUNSON , JAMES RIZZI , MARTHA RODRIGUEZ , TODD EARY CHARLES , DANIEL WATSON
IPC: A61P29/00
Abstract: THE COMPOUND OF FORMULA I AND PHARMACEUTICALLY ACCEPTABLE SALTS AND PRODRUGS THEREOF ARE USEFUL IN THE TREATMENT AND PREVENTION OF VARIOUS DISORDERS MEDIATED BY KINASES.
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公开(公告)号:BRPI0707401B8
公开(公告)日:2022-12-20
申请号:BRPI0707401
申请日:2007-01-26
Applicant: ARRAY BIOPHARMA INC
Inventor: ROBERT D GRONEBERG , LAURENCE E BURGESS , DARREN HARVEY , ELLEN LAIRD , MARK MUNSON , JAMES RIZZI , MARTHA RODRIGUEZ , CHARLES TODD EARY , DANIEL J WATSON
IPC: C07D231/40 , A61K31/416 , A61P29/00 , C07D231/56
Abstract: INIBIDORES DE CINASE E MÉTODOS DE USO DOS MESMOS. Composto de Fórmula I e sais farmaceuticamente aceitáveis e pró-fármacos dos mesmos são úteis no tratamento e prevenção de vários distúrbios mediados por cinases.
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公开(公告)号:AU2007210073B2
公开(公告)日:2011-10-06
申请号:AU2007210073
申请日:2007-01-26
Applicant: ARRAY BIOPHARMA INC
Inventor: MARTHA RODRIGUEZ , BURGESS LAURENCE E , MARK MUNSON , ELLEN LAIRD , ROBERT GRONEBERG , TODD EARY CHARLES , JAMES RIZZI , DANIEL WATSON , DARREN HARVEY
IPC: C07D231/40 , A61K31/416 , A61P29/00 , C07D231/56
Abstract: The compound of Formula (I) and pharmaceutically acceptable salts and prodrugs thereof are useful in the treatment and prevention of various disorders mediated by kinases.
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公开(公告)号:BRPI0707401B1
公开(公告)日:2020-09-15
申请号:BRPI0707401
申请日:2007-01-26
Applicant: ARRAY BIOPHARMA INC
Inventor: CHARLES TODD EARY , DANIEL J WATSON , DARREN HARVEY , ELLEN LAIRD , JAMES RIZZI , LAURENCE E BURGESS , MARK MUNSON , MARTHA RODRIGUEZ , ROBERT D GRONEBERG
IPC: C07D231/56 , A61K31/416 , A61P29/00 , C07D231/40
Abstract: inibidores de cinase e métodos de uso dos mesmos. composto de fórmula i e sais farmaceuticamente aceitáveis e pró-fármacos dos mesmos são úteis no tratamento e prevenção de vários distúrbios mediados por cinases.
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