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公开(公告)号:PT1682553E
公开(公告)日:2010-07-29
申请号:PT04779049
申请日:2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
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公开(公告)号:DE602004027288D1
公开(公告)日:2010-07-01
申请号:DE602004027288
申请日:2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
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公开(公告)号:NZ545421A
公开(公告)日:2010-03-26
申请号:NZ54542104
申请日:2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , A61P11/06 , C07D519/00
Abstract: Disclosed is a compound of formula I wherein X is N, or C-R7; X1 is N, or C-R1 and wherein the rest of the substituents are disclosed within the specification. Also disclosed is the use of a compound of formula I in the manufacture of a medicament for treating a patient with a pathological condition related to overproduction of Th2 cytokine, such as asthma.
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公开(公告)号:ECSP066411A
公开(公告)日:2006-09-18
申请号:ECSP066411
申请日:2006-03-06
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
Abstract: Tienopirazoles, su preparación, composiciones farmacéuticas que comprenden estos compuestos, y sus usos farmacéuticos en el tratamiento de estados de enfermedad capaces de ser modulados por la inhibición de las proteína quinasas, en particular la tirosina quinasa inducible por interleuquina-2 (ITK).
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公开(公告)号:RS51846B
公开(公告)日:2012-02-29
申请号:RSP16206
申请日:2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DHARANIPRAGADA RAMALINGA M , DU YAN , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
Abstract: Thienopyrazoles of formula I, their preparation, pharmaceutical compositions comprising these compounds, and their pharmaceutical uses in the treatment of disease states capable of being modulated by the inhibition of the protein kinases, in particular interleukin-2 inducible tyrosine kinase (ITK).
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公开(公告)号:HRP20100398T1
公开(公告)日:2010-09-30
申请号:HRP20100398
申请日:2010-07-20
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
Abstract: Thienopyrazoles of formula I, their preparation, pharmaceutical compositions comprising these compounds, and their pharmaceutical uses in the treatment of disease states capable of being modulated by the inhibition of the protein kinases, in particular interleukin-2 inducible tyrosine kinase (ITK).
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公开(公告)号:SI1682553T1
公开(公告)日:2010-08-31
申请号:SI200431462
申请日:2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/00 , C07D495/04 , C07D519/00
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公开(公告)号:MEP20908A
公开(公告)日:2010-06-10
申请号:MEP20908
申请日:2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
Abstract: Thienopyrazoles of formula I, their preparation, pharmaceutical compositions comprising these compounds, and their pharmaceutical uses in the treatment of disease states capable of being modulated by the inhibition of the protein kinases, in particular interleukin-2 inducible tyrosine kinase (ITK).
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公开(公告)号:TNSN06058A1
公开(公告)日:2007-10-03
申请号:TNSN06058
申请日:2006-02-15
Applicant: AVENTIS PHARMA INC
Inventor: EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED , JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN
IPC: C07D495/04 , C07D519/00
Abstract: THIENOPYRAZOLES, THEIR PREPARATION, PHARMACEUTICAL COMPOSITIONS COMPRISING THESE COMPOUNDS, AND THEIR PHARMACEUTICAL USES IN THE TREATMENT OF DISEASE STATES CAPABLE OF BEING MODULATED BY THE INHIBITION OF THE PROTEIN KINASES, IN PARTICULAR INTERLEUKIN-2 INDUCIBLE TYROSINE KINASE (ITK).
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公开(公告)号:NO20061626A
公开(公告)日:2006-04-10
申请号:NO20061626
申请日:2006-04-10
Applicant: AVENTIS PHARMA INC
Inventor: JURCAK JOHN G , WEINTRAUB PHILIP MARVIN , EDWARDS MICHAEL LOUIS , DHARANIPRAGADA RAMALINGA M , BARRAGUE MATTHICU , GILLESPY TIMOTHY ALAN , MUSICK KWON YON , DU YAN , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
CPC classification number: C07D495/04
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