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公开(公告)号：AU2004272507B2
公开(公告)日：2011-05-12
申请号：AU2004272507
申请日：2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor： DHARANIPRAGADA RAMALINGA M , BARRAGUE MATTHIEU , DU YAN , MUSICK KWON YON , PARKAR ASHFAQ AHMED , EDWARDS MICHAEL LOUIS , JURCAK JOHN GERARD , GILLESPY TIMOTHY ALAN , WEINTRAUB PHILIP MARVIN
IPC: C07D495/04 , C07D519/00
Abstract: Thienopyrazoles of formula I, their preparation, pharmaceutical compositions comprising these compounds, and their pharmaceutical uses in the treatment of disease states capable of being modulated by the inhibition of the protein kinases, in particular interleukin-2 inducible tyrosine kinase (ITK).
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公开(公告)号：PL1682553T3
公开(公告)日：2010-10-29
申请号：PL04779049
申请日：2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor： JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
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公开(公告)号：CA2465247C
公开(公告)日：2010-05-18
申请号：CA2465247
申请日：2002-10-24
Applicant: AVENTIS PHARMA INC
Inventor： EDWARDS MICHAEL LOUIS , COX PAUL JOSEPH , AMENDOLA SHELLEY , DEPRETS STEPHANIE DANIELE , GILLESPY TIMOTHY ALAN , EDLIN CHRISTOPHER DAVID , MORLEY ANDREW DAVID , GARDNER CHARLES J , PEDGRIFT BRIAN , BOUCHARD HERVE , BABIN DIDIER , GAUZY LAURENCE , LE BRUN ALAIN , MAJID TAHIR NEDEEM , READER JOHN C , PAYNE LLOYD J , KHAN NAWAZ M , CHERRY MICHAEL
IPC: C07D403/04 , A61K31/4184 , A61K31/4188 , A61K31/42 , A61K31/437 , A61K31/4439 , A61K31/454 , A61K31/496 , A61K31/4985 , A61K31/5377 , A61P1/04 , A61P3/04 , A61P3/10 , A61P7/00 , A61P9/00 , A61P9/04 , A61P9/10 , A61P11/00 , A61P11/02 , A61P11/06 , A61P17/00 , A61P17/06 , A61P19/00 , A61P19/02 , A61P19/10 , A61P21/00 , A61P25/00 , A61P25/16 , A61P25/18 , A61P25/24 , A61P25/28 , A61P27/02 , A61P29/00 , A61P31/04 , A61P31/12 , A61P33/00 , A61P35/00 , A61P37/02 , A61P37/06 , A61P37/08 , A61P39/02 , A61P43/00 , C07D401/14 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/04 , C07D413/14 , C07D471/04 , C07D487/04 , C07D491/04 , C07D491/056 , C07D521/00
Abstract: The invention is directed to physiologically active compounds of the general formula (Ix) and compositions containing such compounds, and their prodrugs, and pharmaceutically acceptable salts and solvates of such compounds and their prodrugs, as well as to novel compounds within the scope of formula (Ix), and to processes for their preparation. Such compounds and compositions have valuable pharmaceutical properties, in particular the ability to inhibit kinases.
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公开(公告)号：AU2002334217B2
公开(公告)日：2008-07-03
申请号：AU2002334217
申请日：2002-10-24
Applicant: AVENTIS PHARMA INC
Inventor： MORLEY ANDREW DAVID , BABIN DIDIER , READER JOHN C , AMENDOLA SHELLEY , CHERRY MICHAEL , GARDNER CHARLES J , MAJID TAHIR NEDEEM , COX PAUL JOSEPH , GILLESPY TIMOTHY ALAN , KHAN NAWAZ M , BRUN ALAIN LE , DEPRETS STEPHANIE DANIELE , PEDGRIFT BRIAN , EDWARDS MICHAEL LOUIS , PAYNE LLOYD J , GAUZY LAURENCE , EDLIN CHRISTOPHER DAVID , BOUCHARD HERVE
IPC: A61K31/4184 , A61K31/4188 , A61K31/42 , A61K31/437 , A61K31/4439 , A61K31/454 , A61K31/496 , A61K31/4985 , A61K31/5377 , A61P1/04 , A61P3/04 , A61P3/10 , A61P7/00 , A61P9/00 , A61P9/04 , A61P9/10 , A61P11/00 , A61P11/02 , A61P11/06 , A61P17/00 , A61P17/06 , A61P19/00 , A61P19/02 , A61P19/10 , A61P21/00 , A61P25/00 , A61P25/16 , A61P25/18 , A61P25/24 , A61P25/28 , A61P27/02 , A61P29/00 , A61P31/04 , A61P31/12 , A61P33/00 , A61P35/00 , A61P37/02 , A61P37/06 , A61P37/08 , A61P39/02 , A61P43/00 , C07D401/14 , C07D403/04 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/04 , C07D413/14 , C07D471/04 , C07D487/04 , C07D491/04 , C07D491/056 , C07D521/00
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公开(公告)号：RS20060162A
公开(公告)日：2008-06-05
申请号：YUP20060162
申请日：2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor： JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , DU YAN , DHARANIPRAGADA RAMALINGA , PARKAR ASHFAQ AHMED , WEINTRAUB PHILIP MARVIN
IPC: C07D495/04 , C07D519/00
Abstract: Tienopirazoli, njihova priprema, farmaceutski preparati koji sadrže ova jedinjenja, i njihova farmaceutsko upotreba u lečenju bolesnih stanja koja se mogu menjati inhibicijom protein kinaze, naročito tirozin kinaze koja se može indukovati interleukinom-2.
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Patent Agency Ranking
公开(公告)号：CA2538032A1
公开(公告)日：2005-03-24
申请号：CA2538032
申请日：2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor： BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , JURCAK JOHN GERARD , DHARANIPRAGADA RAMALINGA M , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , DU YAN , WEINTRAUB PHILIP MARVIN , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
Abstract: Thienopyrazoles, their preparation, pharmaceutical compositions comprising these compounds, and their pharmaceutical uses in the treatment of disease states capable of being modulated by the inhibition of the protein kinases, in particular interleukin-2 inducible tyrosine kinase (ITK).
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公开(公告)号：AU2004272507A1
公开(公告)日：2005-03-24
申请号：AU2004272507
申请日：2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor： DHARANIPRAGADA RAMALINGA M , BARRAGUE MATTHIEU , DU YAN , MUSICK KWON YON , PARKAR ASHFAQ AHMED , EDWARDS MICHAEL LOUIS , JURCAK JOHN GERARD , GILLESPY TIMOTHY ALAN , WEINTRAUB PHILIP MARVIN
IPC: C07D495/04 , C07D519/00
Abstract: Thienopyrazoles of formula I, their preparation, pharmaceutical compositions comprising these compounds, and their pharmaceutical uses in the treatment of disease states capable of being modulated by the inhibition of the protein kinases, in particular interleukin-2 inducible tyrosine kinase (ITK).
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公开(公告)号：PA8557101A1
公开(公告)日：2003-12-10
申请号：PA8557101
申请日：2002-10-25
Applicant: AVENTIS PHARMA INC
Inventor： COX PAUL JOSEPH , DEPRETS STEPHANIE DANIELE , GARDNER CHARLES J , GILLESPY TIMOTHY ALAN , BOUCHARD HERVE , EDWARDS MICHAEL LOUIS , AMENDOLA SHELLEY , EDLIN CHRISTOPHER DAVID , MORLEY ANDREW DAVID , PEDGRIFT BRIAN , BABIN DIDIER , GAUZY LAURENCE , LE BRUN ALAIN , MAJID TAHIR , READER JOHN C , PAYNE LLOYD J , KHAN NAWAZ M , CHERRY MICHAEL
IPC: A61K31/4184 , A61P35/00 , C07D401/14 , C07D403/04 , C07D403/14 , C07D405/14 , C07D409/14 , C07D413/04 , C07D413/14 , C07D471/04 , C07D487/04 , C07D491/04 , C07D521/00
Abstract: LA INVENCION SE REFIERE A COMPUESTOS FISIOLOGICAMENTE ACTIVOS LA FORMULA GENERAL (lX) Y COMPOSICIONES QUE CONTIENEN DICHOS COMPUESTOS, Y SUS PROFARMACOS Y LAS SALES Y LOS SOLVATOS ACEPTABLES PARA USO FARMACEUTICO DE DICHOS COMPUESTOS Y SUS PROFARMACOS, COMO TAMBIEN A NUEVOS COMPUESTOS DENTRO DEL ALCANCE DE LA FORMULA (lX), Y A PROCESOS PARA SU PREPARACION. DICHOS COMPUESTOS Y COMPOSICIONES TIENEN VALIOSAS PROPIEDADES FARMACEUTICAS, EN PARTICULAR LA CAPACIDAD DE INHIBIR LAS QUINASAS.
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公开(公告)号：PT1682553E
公开(公告)日：2010-07-29
申请号：PT04779049
申请日：2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor： JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
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公开(公告)号：DE602004027288D1
公开(公告)日：2010-07-01
申请号：DE602004027288
申请日：2004-07-23
Applicant: AVENTIS PHARMA INC
Inventor： JURCAK JOHN GERARD , BARRAGUE MATTHIEU , GILLESPY TIMOTHY ALAN , EDWARDS MICHAEL LOUIS , MUSICK KWON YON , WEINTRAUB PHILIP MARVIN , DU YAN , DHARANIPRAGADA RAMALINGA M , PARKAR ASHFAQ AHMED
IPC: C07D495/04 , C07D519/00
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