-
公开(公告)号:GR880300092T1
公开(公告)日:1988-10-21
申请号:GR880300092
申请日:1988-10-21
Applicant: BASF AG
IPC: A61K31/05 , A61K31/047 , A61K31/085 , A61K31/135 , A61K31/16 , A61K31/19 , A61K31/195 , A61K31/215 , A61K31/22 , A61K31/357 , A61K31/36 , A61P17/00 , A61P29/00 , A61P35/00 , C07C27/00 , C07C39/23 , C07C39/42 , C07C41/00 , C07C43/168 , C07C43/20 , C07C43/215 , C07C51/00 , C07C59/125 , C07C59/68 , C07C59/72 , C07C62/38 , C07C67/00 , C07C69/07 , C07C69/157 , C07C69/24 , C07C69/712 , C07C69/78 , C07C213/00 , C07C217/18 , C07D317/50 , C07D325/00
-
公开(公告)号:HU220875B1
公开(公告)日:2002-06-29
申请号:HU9603067
申请日:1995-04-26
Applicant: BASF AG
Inventor: DR AMBERG WILHELM , DR BERNARD HARALD , DR BUSCHMANN ERNST , DR DE POTZOLLI BERND , DR HAUPT ANDREAS , DR JANITSCHKE LOTHAR , DR JANSSEN BERND , DR KARL ULRICH , DR KLING ANDREAS , DR MUELLER STEFAN , DR RITTER KURT , DR THYES MARCO , DR ZIERKE THOMAS
Abstract: PCT No. PCT/EP95/01577 Sec. 371 Date Nov. 4, 1996 Sec. 102(e) Date Nov. 4, 1996 PCT Filed Apr. 26, 1995 PCT Pub. No. WO95/30691 PCT Pub. Date Nov. 16, 1995The compound Me2Val-Val-MeVal-Pro-Pro-NHBzlxHCl is described. It is prepared from Z-Val-Val-MeVal-Pro-OR1 where Z and R1 have the meanings stated in the description. The compound shows antineoplastic activity.
-
公开(公告)号:HU220862B1
公开(公告)日:2002-06-29
申请号:HU9603068
申请日:1995-04-26
Applicant: BASF AG
Inventor: DR AMBERG WILHELM , DR BERNARD HARALD , DR BUSCHMANN ERNST , DR DE POTZOLLI BERND , DR HAUPT ANDREAS , DR JANITSCHKE LOTHAR , DR JANSSEN BERND , DR KARL ULRICH , DR KLING ANDREAS , DR MUELLER STEFAN , DR RITTER KURT , DR THYES MARCO , DR ZIERKE THOMAS
Abstract: Compounds of the formulawhere R1, R2, R3 and R4 have the meaning stated in the description, and a process for preparing them are described. The compounds are suitable as starting material for synthesizing substances which are active against tumors.
-
-