公开(公告)号：RU2151142C1

公开(公告)日：2000-06-20

申请号：RU97102108

申请日：1995-06-21

Applicant: BASF AG

Inventor： BERND MJULLER ,  KHARTMANN KENIG ,  REJNKHARD KIRSTGEN ,  KLAUS OBERDORF ,  FRANTS REL ,  NORBERT GETTS ,  KHUBERT ZAUTER ,  GIZELA LORENTS ,  EHBERKHARD AMMERMANN

IPC: C07D231/06 ,  A01N20060101 ,  A01N43/40 ,  A01N43/56 ,  A01N47/22 ,  A01N47/24 ,  A01N47/30 ,  A01P3/00 ,  C07C239/10 ,  C07C271/28 ,  C07C271/58 ,  C07D20060101 ,  C07D231/08 ,  C07D231/20 ,  C07D231/22 ,  C07D231/30 ,  C07D401/04 ,  C07D403/04

Abstract: agriculture. SUBSTANCE: described are new compounds, namely 2- [(dihydro)pyrazolyl-3'-oxymethylene] anilides of formula I wherein -- denotes single or double bond, and indexes and substituents are defined as follows: n is 0,1 or 2; m is 0,1 or 2, R2 substituents are different if m is more than 1; X is straight bond, 0 or NRa; Ra are hydrogen; R1 is C1-C4 alkyl, halogen or in case wherein n is 2, is hydrocarbon bridge additionally bonded with two adjacent ring atoms, said bridge containing 3 or 4 carbon atoms; R2 in nitro, halogen, C1-C4 alkyl, C1-C4 halogenalkyl or C1-C4 alkoxycarbonyl; R3 is optionally substituted alkyl, optionally substituted saturated ring or optionally substituted single or binuclear aromatic radical which, in addition to carbon atoms contains one to four nitrogen atoms as ring members; R4 is hydrogen or optionally substituted alkyl; R5 is alkyl, or in case X is NRa is additionally hydrogen. Compounds of formula I are useful for controlling pests and harmful fungi. Also described are method of preparation thereof and, intermediate compounds, agent for controlling agricultural pests and harmful fungi, and control method. EFFECT: increased efficiency of the title compounds and agents for controlling agricultural pests and harmful fungi. 12 cl, 6 tbl

公开(公告)号：RU2166500C2

公开(公告)日：2001-05-10

申请号：RU97110060

申请日：1995-11-07

Applicant: BASF AG

Inventor： REJNKHARD KIRSTGEN ,  KLAUS OBERDORF ,  FRANTS SHJUTTS ,  KHANS TEOBAL D ,  FOL KER KHARRIES

IPC: C07D239/54 ,  A01N43/54 ,  A01P7/02 ,  C07D239/52 ,  C07D239/56

Abstract: organic chemistry, insecticides. SUBSTANCE: invention relates to novel derivatives of 2-[(2-alkoxy-6-trifluoromethyl- pyrimidine-4-yl)-oxymethylene]-phenylacetic acid of the general formula (I) where R is -C1-C6-alkyl; R1 is halogen atom; n = 0-1; V is O or NH; U is CH or N. Claimed compounds show fungicide, insecticide and acaricide activity and can be used for protection of plants, protection from storehouse pests and for protection of foodstuffs stores and in the field of hygiene and veterinary also. Invention relates to also method of synthesis of compounds of the general formula (I) using compounds of the general formula (II) as intermediate compounds. Method of synthesis involves interaction of compound of the formula (II) where R has the above indicated value with compound of the formula (III) where X means nucleophilic group to be removed. Invention relates to also agent containing liquid filling agent and compound of the formula (I) of acaricide class used for control of pests, harmful fungi and insects with exception in the latter case of compounds of the general formula (I) when U is CH and V is NH. EFFECT: new compounds indicated above, improved method of synthesis, valuable properties. 9 cl, 15 tbl, 5 ex