公开(公告)号：WO0129033A3

公开(公告)日：2001-12-06

申请号：PCT/EP0010417

申请日：2000-10-23

Applicant: BASF CORP ,  BASF AG ,  IDEMITSU KOSAN CO

Inventor： SZUCS STEPHEN S

IPC: A01N43/56 ,  C07D409/06 ,  C07D405/06

CPC classification number: C07D409/06 ,  A01N43/56

Abstract: The present invention provides a compound of formula (I). Compounds of formula (I) are useful as herbicidal agents, particularly as agents for the control of undesirable plant species in the presence of a cereal crop.

Abstract translation: 本发明提供式（I）化合物。 式（I）化合物可用作除草剂，特别是作为在谷物作物存在下控制不期望的植物物种的试剂。

公开(公告)号：HU0402238A2

公开(公告)日：2005-02-28

申请号：HU0402238

申请日：2002-09-25

Applicant: BASF AG

Inventor： FURCH JOSEPH A ,  KUHN DAVID ,  SZUCS STEPHEN S ,  GU KUN-JIAN ,  VON DEYN WOLFGANG

IPC: A01N25/02 ,  A01N25/08 ,  A01N43/56 ,  A01N47/36 ,  C07D231/12 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18 ,  C07D231/20 ,  C07D231/28 ,  C07D231/38 ,  C07D231/40 ,  C07D401/04

Abstract: Compounds of formula (I), wherein the variables and the index have the following meanings: R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or optionally substituted phenyl; R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR R , N=CHOR , or N=CHNR ; R , R H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl, diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R alkyl, haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy; M N or CR ; R H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestation and infection by arachnids and arthropod endo-and ectoparasites.

公开(公告)号：EA007969B1

公开(公告)日：2007-02-27

申请号：EA200400413

申请日：2002-09-25

Applicant: BASF AG

Inventor： FURCH JOSEPH A ,  KUHN DAVID ,  SZUCS STEPHEN S ,  GU KUN-JIAN ,  VON DEYN WOLFGANG

IPC: C07D231/12 ,  A01N25/02 ,  A01N25/08 ,  A01N43/56 ,  A01N47/36 ,  A61K31/415 ,  A61K31/4155 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18 ,  C07D231/20 ,  C07D231/22 ,  C07D231/28 ,  C07D231/38 ,  C07D231/40 ,  C07D401/04

Abstract: Соединенияформулы Iвкоторойпеременныепараметрыи индексыимеютследующиезначения: R- водород, галоген, C-Салкил, C-Сгалоалкил, C-Салкенил, C-Сгалоалкенил; R- галоген; А - водород, циано, нитро, галоген, родано, C-Салкокси, C-Сгалоалкокси, C-Салкилтио, C-Сгалоалкилтио, аминотиокарбонил, гидроксикарбонил, С-Салкоксикарбонил, аминокарбонил; В - водород, гидрокси, амино, циано, нитро, галоген, C-С-алкил, незамещенныйилизамещенный 1-3 группами, выбраннымиизгалогенаи циано; C-Салкокси, незамещенныйилизамещенный 1-3 группами, выбраннымиизгалогена, циано, С-Салкенилаи C-Салкоксикарбонил-С-Салкенила; C-Салкенил, незамещенныйилизамещенный 1-3 группами, выбраннымиизгалогенаи циано; C-Салкенилокси, C-Салкилтио, C-Сгалоалкилтио, C-Салкокситиокарбонилтио, C-Салкоксикарбонил-C-Салкокси, C-Салкоксикарбонил-С-Салкилтио, C-Салкилсульфинил, C-Салкилсульфонил, аминотиокарбонил, NRR, N=CHORили N=CHNR; R,R- каждыйнезависимо, представляетсобойводород, C-Салкил, C-Салкоксикарбонил-C-Салкил, [(C-Салкоксикарбонил)(С-Салкенил)]C-Салкил, C-Салкоксикарбонил-С-Салкенил, C-Салкилкарбонил, С-Сциклоалкилкарбонил, C-Салкиламинокарбонил, ди(C-Салкил)аминокарбонил, C-Салкоксикарбонил, C-Салкоксиаминосульфонилилиди(C-С-алкокси)аминосульфонил; R- C-Салкил; Q - галоген; X - водород; Y - водород, галоген, C-С-галоалкил, C-С-алкоксиили C-С-галоалкокси; Z –водород; М - N или CR; R- галоген; n - 1, 2; приусловии, чтокогда Rозначаетводород, n неявляетсянулем, способыполучениясоединенийформулы I, композиции, содержащиеих, иихиспользованиедляборьбыс паукообразнымии членистоногиминасекомымии длязащитырастенийотэтихнасекомых, атакжеихиспользованиедлялечения, борьбы, профилактикии защитытеплокровныхживотныхи человекаотзараженияи инфицирования

公开(公告)号：BR0212385A

公开(公告)日：2004-08-17

申请号：BR0212385

申请日：2002-09-25

Applicant: BASF AG

Inventor： FURCH JOSEPH A ,  KUHN DAVID ,  SZUCS STEPHEN S ,  GU KUN-JIAN ,  DEYN WOLFGANG VON

IPC: A01N25/02 ,  A01N25/08 ,  A01N43/56 ,  A01N47/36 ,  C07D231/12 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18 ,  C07D231/20 ,  C07D231/28 ,  C07D231/38 ,  C07D231/40 ,  C07D401/04 ,  C07D231/22 ,  A61K31/415 ,  A61K31/4155

Abstract: Compounds of formula (I), wherein the variables and the index have the following meanings: R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or optionally substituted phenyl; R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR R , N=CHOR , or N=CHNR ; R , R H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl, diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R alkyl, haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy; M N or CR ; R H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestation and infection by arachnids and arthropod endo-and ectoparasites.

公开(公告)号：AU7790100A

公开(公告)日：2001-04-30

申请号：AU7790100

申请日：2000-10-23

Applicant: BASF AG ,  BASF CORP ,  IDEMITSU KOSAN CO

Inventor： SZUCS STEPHEN S

IPC: A01N43/56 ,  C07D409/06 ,  C07D409/00

Abstract: The present invention provides a compound of formula I:wherein X is O or S(O)n; n is zero, 1 or 2; and Y is CR7R8, CHOR9, C(OR9)2, C=NOR10 or C=NNR20R21.Compounds of formula I are useful as herbicidal agents, particularly as agents for the control of undesirable plant species in the presence of a cereal crop.

公开(公告)号：UA79758C2

公开(公告)日：2007-07-25

申请号：UA20040403076

申请日：2002-09-25

Applicant: BASF AG

Inventor： FURCH JOSEPH A ,  KUHN DAVID ,  SZUCS STEPHEN S ,  GU KUN-JIAN ,  VON DEYN WOLFGANG

IPC: A01N25/02 ,  A01N25/08 ,  A01N43/56 ,  A01N47/36 ,  C07D231/12 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18 ,  C07D231/20 ,  C07D231/28 ,  C07D231/38 ,  C07D231/40 ,  C07D401/04

Abstract: Compounds of formula (1), wherein the variables and the index have the following meanings: R1 H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or opieonally substituted phenyl; R2 H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR3R4, N=CHOR5, or N=CHNR5; R3, R4 H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl, diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R5 alkyl,haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy; M N or CR6; R6 H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R1 is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestation and infection by arachnids and arthropod endo- and ectoparasites. (I)

公开(公告)号：PL370353A1

公开(公告)日：2005-05-16

申请号：PL37035302

申请日：2002-09-25

Applicant: BASF AG

Inventor： FURCH JOSEPH A ,  KUHN DAVID ,  SZUCS STEPHEN S ,  GU KUN-JIAN ,  VON DEYN WOLFGANG

IPC: A01N25/02 ,  A01N25/08 ,  A01N43/56 ,  A01N47/36 ,  C07D231/12 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18 ,  C07D231/20 ,  C07D231/28 ,  C07D231/38 ,  C07D231/40 ,  C07D401/04 ,  A61K31/415

Abstract: Compounds of formula (I), wherein the variables and the index have the following meanings: R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or optionally substituted phenyl; R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR R , N=CHOR , or N=CHNR ; R , R H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl, diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R alkyl, haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy; M N or CR ; R H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestation and infection by arachnids and arthropod endo-and ectoparasites.

公开(公告)号：CA2416039A1

公开(公告)日：2002-01-24

申请号：CA2416039

申请日：2001-07-13

Applicant: BASF AG

Inventor： SINGH BIJAY K ,  PEDERSEN MARIANNE K ,  TECLE BERHANE ,  KAMESWARAN VENKATARAMAN ,  BIRK IWONA T ,  ORTH ANN B ,  SZUCS STEPHEN S

IPC: A01N43/56 ,  C07D231/20 ,  C07D231/32 ,  C07D401/12 ,  C07D409/12 ,  G01N33/50 ,  C12Q1/37

Abstract: This invention relates to a method for identifying compounds that specifical ly inhibit a metabolic target site or pathway in plants. Enzymes which are specifically affected by the method of the invention include plant pyramidin e biosynthetic pathway enzymes, and particularly the enzymes involved in the conversion of orotate to uridine-5'-monophosphate (UMP). Further, the invention relates to a method for control of undesirable monocotyledonous an d dicotyledenous plant species.

公开(公告)号：ZA200402932B

公开(公告)日：2005-04-19

申请号：ZA200402932

申请日：2004-04-19

Applicant: BASF AG

Inventor： FURCH JOSEPH A ,  GU KUN-JIAN ,  KUHN DAVID ,  SZUCS STEPHEN S ,  DEYN WOLFGANG VON

IPC: A01N25/02 ,  A01N25/08 ,  A01N43/56 ,  A01N47/36 ,  C07D231/12 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18 ,  C07D231/20 ,  C07D231/28 ,  C07D231/38 ,  C07D231/40 ,  C07D401/04 ,  C07D ,  A61K

Abstract: Compounds of formula (I), wherein the variables and the index have the following meanings: R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or optionally substituted phenyl; R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR R , N=CHOR , or N=CHNR ; R , R H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl, diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R alkyl, haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy; M N or CR ; R H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestation and infection by arachnids and arthropod endo-and ectoparasites.

公开(公告)号：CA2460906A1

公开(公告)日：2003-04-10

申请号：CA2460906

申请日：2002-09-25

Applicant: BASF AG

Inventor： VON DEYN WOLFGANG ,  FURCH JOSEPH A ,  GU KUN-JIAN ,  KUHN DAVID ,  SZUCS STEPHEN S

IPC: A01N25/02 ,  A01N25/08 ,  A01N43/56 ,  A01N47/36 ,  C07D231/12 ,  C07D231/14 ,  C07D231/16 ,  C07D231/18 ,  C07D231/20 ,  C07D231/28 ,  C07D231/38 ,  C07D231/40 ,  C07D401/04 ,  C07D231/22 ,  A61K31/415 ,  A61K31/4155

Abstract: Compounds of formula (I), wherein the variables and the index have the following meanings: R1 H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or optionally substituted phenyl; R2 H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR3R4, N=CHOR5, or N=CHNR5; R3, R4 H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl , diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R5 alkyl, haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy;M N or CR6; R6 H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R1 is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestatio n and infection by arachnids and arthropod endo-and ectoparasites.