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公开(公告)号:CR9624A
公开(公告)日:2008-02-21
申请号:CR9624
申请日:2007-12-20
Applicant: BASF AG
Inventor: SCHMIDT THOMAS , PUHL MICHAEL , DICKHAUT JOACHIM , BASTIAANS HENRICUS MARIA MARTINUS , RACK MICHAEL , CULBERTSON DEBORAH , ANSPAUGH DOUGLAS , BRAUN FRANZ JOSEF , BUCCI TONI , COTTER HENRY , KUHN DAVID , OLOUMI-SADEGHI HASSAN
IPC: A01N43/56 , C07D401/04
Abstract: Compuestos de N-tio-antranilamida de la formula (I) en donde A es un grupo seleccionado de A1 y A2 en donde las variables y los indices son como se definen por la descripcion, procesos para preparar los compuestos I, composiciones pesticidas que comprenden los compuestos I, uso de los compuestos 1para el control de insectos, acaros o nematodos, y metodos para tratar, controlar, prevenir o proteger a los animales contra una infestacion o infeccion de parasitos con el uso de compuestos de la formula I.
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公开(公告)号:AT363829T
公开(公告)日:2007-06-15
申请号:AT02782789
申请日:2002-09-09
Applicant: BASF AG
Inventor: WOOD WILLIAM , KUHN DAVID , HU YULIN , TECLE BERHANE
IPC: A01N43/90 , A01N43/42 , A61K31/437 , A61P33/00 , C07D471/02 , C07D491/02 , C07D513/04
Abstract: Di- and trifluorosubstituted alkene compounds of formula I wherein X is hydrogen or fluorine; Y is oxygen, NR 1 or S(O) m ; R 1 is hydrogen or C 1 -C 6 -alkyl; m is 0, 1, or 2; A,B,D and E are selected from the following: a) A is N and B, D and E are CR 2 ; or b) B is N and A, D and E are CR 2 ; or c) D is N and A, B, and E are CR 2 ; or d) A and D are N and B and E are CR 2 ; or e) B and E are N and A and D are CR 2 ; R 2 is H, halogen, NH 2 , NO 2 , CN, alkyl, haloalkyl, alkenyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, aminosulfonyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl,alkylaminoalkyl, dialkylaminoalkyl, hydroxycarbonyl, or alkoxycarbonyl; or phenyl which may be substituted with halogen, CN, NO 2 , alkyl, haloalkyl, alkoxy, or haloalkoxy; or a 5- to 6-membered heteroaromatic ring system containing 1 to 3 heteroatoms selected from oxygen, sulfur and nitrogen, which may be substituted with halogen, CN, NO 2 , alkyl, haloalkyl, alkoxy, or haloalkoxy; n is 1, 2, 3 or 4, and the agriculturally and/or physiologically tolerable salts thereof, methods for the preparation of compounds I, and compositions and methods for the control of nematodes and arachnids, and for treating, controlling, preventing and protecting warm-blooded animals, fish and humans against infestation and infection by helminths, arachnids and arthropod endo- and ectoparasites.
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公开(公告)号:HU0402238A2
公开(公告)日:2005-02-28
申请号:HU0402238
申请日:2002-09-25
Applicant: BASF AG
Inventor: FURCH JOSEPH A , KUHN DAVID , SZUCS STEPHEN S , GU KUN-JIAN , VON DEYN WOLFGANG
IPC: A01N25/02 , A01N25/08 , A01N43/56 , A01N47/36 , C07D231/12 , C07D231/14 , C07D231/16 , C07D231/18 , C07D231/20 , C07D231/28 , C07D231/38 , C07D231/40 , C07D401/04
Abstract: Compounds of formula (I), wherein the variables and the index have the following meanings: R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or optionally substituted phenyl; R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR R , N=CHOR , or N=CHNR ; R , R H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl, diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R alkyl, haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy; M N or CR ; R H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestation and infection by arachnids and arthropod endo-and ectoparasites.
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公开(公告)号:ZA200402932B
公开(公告)日:2005-04-19
申请号:ZA200402932
申请日:2004-04-19
Applicant: BASF AG
Inventor: FURCH JOSEPH A , GU KUN-JIAN , KUHN DAVID , SZUCS STEPHEN S , DEYN WOLFGANG VON
IPC: A01N25/02 , A01N25/08 , A01N43/56 , A01N47/36 , C07D231/12 , C07D231/14 , C07D231/16 , C07D231/18 , C07D231/20 , C07D231/28 , C07D231/38 , C07D231/40 , C07D401/04 , C07D , A61K
Abstract: Compounds of formula (I), wherein the variables and the index have the following meanings: R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or optionally substituted phenyl; R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR R , N=CHOR , or N=CHNR ; R , R H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl, diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R alkyl, haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy; M N or CR ; R H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestation and infection by arachnids and arthropod endo-and ectoparasites.
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公开(公告)号:CA2460906A1
公开(公告)日:2003-04-10
申请号:CA2460906
申请日:2002-09-25
Applicant: BASF AG
Inventor: VON DEYN WOLFGANG , FURCH JOSEPH A , GU KUN-JIAN , KUHN DAVID , SZUCS STEPHEN S
IPC: A01N25/02 , A01N25/08 , A01N43/56 , A01N47/36 , C07D231/12 , C07D231/14 , C07D231/16 , C07D231/18 , C07D231/20 , C07D231/28 , C07D231/38 , C07D231/40 , C07D401/04 , C07D231/22 , A61K31/415 , A61K31/4155
Abstract: Compounds of formula (I), wherein the variables and the index have the following meanings: R1 H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or optionally substituted phenyl; R2 H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR3R4, N=CHOR5, or N=CHNR5; R3, R4 H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl , diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R5 alkyl, haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy;M N or CR6; R6 H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R1 is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestatio n and infection by arachnids and arthropod endo-and ectoparasites.
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公开(公告)号:EA007969B1
公开(公告)日:2007-02-27
申请号:EA200400413
申请日:2002-09-25
Applicant: BASF AG
Inventor: FURCH JOSEPH A , KUHN DAVID , SZUCS STEPHEN S , GU KUN-JIAN , VON DEYN WOLFGANG
IPC: C07D231/12 , A01N25/02 , A01N25/08 , A01N43/56 , A01N47/36 , A61K31/415 , A61K31/4155 , C07D231/14 , C07D231/16 , C07D231/18 , C07D231/20 , C07D231/22 , C07D231/28 , C07D231/38 , C07D231/40 , C07D401/04
Abstract: Соединенияформулы Iвкоторойпеременныепараметрыи индексыимеютследующиезначения: R- водород, галоген, C-Салкил, C-Сгалоалкил, C-Салкенил, C-Сгалоалкенил; R- галоген; А - водород, циано, нитро, галоген, родано, C-Салкокси, C-Сгалоалкокси, C-Салкилтио, C-Сгалоалкилтио, аминотиокарбонил, гидроксикарбонил, С-Салкоксикарбонил, аминокарбонил; В - водород, гидрокси, амино, циано, нитро, галоген, C-С-алкил, незамещенныйилизамещенный 1-3 группами, выбраннымиизгалогенаи циано; C-Салкокси, незамещенныйилизамещенный 1-3 группами, выбраннымиизгалогена, циано, С-Салкенилаи C-Салкоксикарбонил-С-Салкенила; C-Салкенил, незамещенныйилизамещенный 1-3 группами, выбраннымиизгалогенаи циано; C-Салкенилокси, C-Салкилтио, C-Сгалоалкилтио, C-Салкокситиокарбонилтио, C-Салкоксикарбонил-C-Салкокси, C-Салкоксикарбонил-С-Салкилтио, C-Салкилсульфинил, C-Салкилсульфонил, аминотиокарбонил, NRR, N=CHORили N=CHNR; R,R- каждыйнезависимо, представляетсобойводород, C-Салкил, C-Салкоксикарбонил-C-Салкил, [(C-Салкоксикарбонил)(С-Салкенил)]C-Салкил, C-Салкоксикарбонил-С-Салкенил, C-Салкилкарбонил, С-Сциклоалкилкарбонил, C-Салкиламинокарбонил, ди(C-Салкил)аминокарбонил, C-Салкоксикарбонил, C-Салкоксиаминосульфонилилиди(C-С-алкокси)аминосульфонил; R- C-Салкил; Q - галоген; X - водород; Y - водород, галоген, C-С-галоалкил, C-С-алкоксиили C-С-галоалкокси; Z –водород; М - N или CR; R- галоген; n - 1, 2; приусловии, чтокогда Rозначаетводород, n неявляетсянулем, способыполучениясоединенийформулы I, композиции, содержащиеих, иихиспользованиедляборьбыс паукообразнымии членистоногиминасекомымии длязащитырастенийотэтихнасекомых, атакжеихиспользованиедлялечения, борьбы, профилактикии защитытеплокровныхживотныхи человекаотзараженияи инфицирования
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公开(公告)号:BR0212385A
公开(公告)日:2004-08-17
申请号:BR0212385
申请日:2002-09-25
Applicant: BASF AG
Inventor: FURCH JOSEPH A , KUHN DAVID , SZUCS STEPHEN S , GU KUN-JIAN , DEYN WOLFGANG VON
IPC: A01N25/02 , A01N25/08 , A01N43/56 , A01N47/36 , C07D231/12 , C07D231/14 , C07D231/16 , C07D231/18 , C07D231/20 , C07D231/28 , C07D231/38 , C07D231/40 , C07D401/04 , C07D231/22 , A61K31/415 , A61K31/4155
Abstract: Compounds of formula (I), wherein the variables and the index have the following meanings: R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl, alkylthio, alkoxyalkyl, alkylthioalkyl, or optionally substituted phenyl; R H, halogen, alkyl, haloalkyl, alkenyl, haloalkenyl or optionally substituted phenyl; A H, OH, CN, NO2, halogen, SCN, alkoxy, haloalkoxy, alkenyloxy, alkylthio, haloalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, hydroxycarbonyl, alkoxycarbonyl, or aminocarbonyl; B H, OH, NH2, CN, NO2, halogen, optionally substituted alkyl, optionally substituted alkoxy, optionally substituted alkenyl, alkenyloxy, alkylthio, haloalkylthio, alkoxythiocarbonylthio, alkoxycarbonylalkoxy, alkoxycarbonylalkylthio, alkylsulfinyl, alkylsulfonyl, aminothiocarbonyl, NR R , N=CHOR , or N=CHNR ; R , R H, alkyl, alkoxycarbonylalkyl, [(alkoxycarbonyl)(alkenyl)]alkyl, alkoxycarbonylalkenyl, alkylcarbonyl, cycloalkylcarbonyl, alkylaminocarbonyl, diaminocarbonyl, alkoxycarbonyl, alkoxyaminosulfonyl, or di(alkoxy)aminosulfonyl; R alkyl, haloalkyl, or phenylalkyl; Q H, NO2, halogen, haloalkyl, alkylamino, dialkylamino, alkoxy, haloalkoxy, or alkenyloxy; X H, halogen, haloalkyl, alkoxy or haloalkoxy; Y H, halogen, haloalkyl, alkoxy or haloalkoxy; Z H, halogen, haloalkyl, alkoxy or haloalkoxy; M N or CR ; R H, NO2, halogen or haloalkyl; n 0, 1, 2, 3, or 4, with the proviso that, when R is hydrogen, n is not zero, processes for the preparation of compounds of formula (I), compositions containing them and their use for the control of insect and acarid pests and for the protection of plants from those pests as well as their use for treating, controlling, preventing and protecting warm-blooded animals and humans against infestation and infection by arachnids and arthropod endo-and ectoparasites.
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8.
公开(公告)号:CR7259A
公开(公告)日:2004-05-28
申请号:CR7259
申请日:2004-02-24
Applicant: BASF AG
Inventor: KUHN DAVID , HU YULIN , TECLE BERHANE , WOOD WILLIAM WAKEFIELD
IPC: A01N43/42 , A01N43/90 , A61K31/437 , A61P33/00 , C07D471/02 , C07D491/02 , C07D513/04
Abstract: Un objetivo de la presente invencion proveer compuestos que tienen una actividad mejorada para el control de nematodos y acaridos, insectos nocivos y parasitos, para la proteccion del crecimiento y del dano causado por nematodos y ataque de acaridos e infestacion en cultivos cosechados. Proveer un metodo para tratar, controlar, prevenir y proteger animales de sangre caliente, peces y humanos contra la infestacion e infeccion por helmitos, acaridos y artropodos endo y ectoparasitos. Estos objetivos son logrados por los compuestos alqueno di- y tri-fluorosubstituido de formula I. Ademas, hemos encontrado procesos para preparar los compuestos de formula I.
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公开(公告)号:AT372674T
公开(公告)日:2007-09-15
申请号:AT04819647
申请日:2004-12-02
Applicant: BASF AG
Inventor: VON DEYN WOLFGANG , OLOUOMI-SADEGHI HASSAN , KUHN DAVID , ARMES NIGEL , COTTER HENRY , HICKS CAROL
IPC: A01N37/52
Abstract: Use of compounds of formula I wherein Q is X 1 is chlorine, bromine, or fluorine; R 1 , R 2 are each independently H, alkyl, alkenyl, alkynyl, or cycloalkyl, alkylamino, dialkylamino, alkylcarbonylamino, alkylsulfonyl, or alkylsulfinyl, wherein the carbon atoms in these groups may be substituted, or R 1 and R 2 may be taken together to form a ring represented by the structure p, m are 1, 2 or 3; X' is oxygen, sulfur, amino, alkylamino, phenylamino, or methylene; Z is alkyl or phenyl; R 3 is H, alkyl, alkenyl, alkynyl, cycloalkyl, wherein the carbon atoms in these groups may be substituted; R, R 4 are H or alkyl, alkoxycarbonyl, alkylaminocarbonyl, or dialkylaminocarbonyl, wherein the carbon atoms in the these groups may be substituted; A is C-R 5 or N; B is C-R 6 or N; W is C-R 7 or N; with the proviso that one of A, B and W is other than N; R 5 , R 6 , R 7 are H, halogen, nitro, cyano, amino, mercapto, hydroxy, alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkylamino, dialkylamino, alkylthio, alkylsulfonyl, or alkylsulfinyl, wherein the carbon atoms in these groups may be substituted, a 5 to 6-membered aromatic ringsystem which may contain 1 to 4 heteroatoms selected from oxygen, sulfur and nitrogen and which may be substituted; Y is hydrogen, halogen, cyano, nitro, amino, hydroxy, mercapto, alkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkylamino, dialkylamino, alkylthio, alkylsulfonyl, or alkylsulfinyl, wherein the carbon atoms in these groups may be substituted; n is 0, 1, or 2; for combating parasites in and on animals.
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公开(公告)号:ZA200402746B
公开(公告)日:2005-04-08
申请号:ZA200402746
申请日:2004-04-08
Applicant: BASF AG
Inventor: HU YULIN , KUHN DAVID , TECLE BERHANE , WAKEFIELD WOOD WILLIAM
IPC: A01N43/42 , A01N43/90 , A61K31/437 , A61P33/00 , C07D471/02 , C07D491/02 , C07D513/04 , A01N , C07D
Abstract: Di- and trifluorosubstituted alkene compounds of formula I wherein X is hydrogen or fluorine; Y is oxygen, NR 1 or S(O) m ; R 1 is hydrogen or C 1 -C 6 -alkyl; m is 0, 1, or 2; A,B,D and E are selected from the following: a) A is N and B, D and E are CR 2 ; or b) B is N and A, D and E are CR 2 ; or c) D is N and A, B, and E are CR 2 ; or d) A and D are N and B and E are CR 2 ; or e) B and E are N and A and D are CR 2 ; R 2 is H, halogen, NH 2 , NO 2 , CN, alkyl, haloalkyl, alkenyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, aminosulfonyl, alkoxyalkyl, alkylthioalkyl, alkylsulfinylalkyl, alkylsulfonylalkyl,alkylaminoalkyl, dialkylaminoalkyl, hydroxycarbonyl, or alkoxycarbonyl; or phenyl which may be substituted with halogen, CN, NO 2 , alkyl, haloalkyl, alkoxy, or haloalkoxy; or a 5- to 6-membered heteroaromatic ring system containing 1 to 3 heteroatoms selected from oxygen, sulfur and nitrogen, which may be substituted with halogen, CN, NO 2 , alkyl, haloalkyl, alkoxy, or haloalkoxy; n is 1, 2, 3 or 4, and the agriculturally and/or physiologically tolerable salts thereof, methods for the preparation of compounds I, and compositions and methods for the control of nematodes and arachnids, and for treating, controlling, preventing and protecting warm-blooded animals, fish and humans against infestation and infection by helminths, arachnids and arthropod endo- and ectoparasites.
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