公开(公告)号：DE59302595D1

公开(公告)日：1996-06-20

申请号：DE59302595

申请日：1993-10-14

Applicant: BAYER AG

Inventor： WAGNER KLAUS DR ,  ERDELEN CHRISTOPH DR ,  HARTWIG JUERGEN DR ,  LEICHT WOLFGANG DR ,  STENDEL WILHELM DR

IPC: A01N43/08 ,  A01N43/10 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01N43/824 ,  A01N43/836 ,  A01N47/44 ,  A01N51/00 ,  C07D213/24 ,  C07D213/26 ,  C07D213/30 ,  C07D213/61 ,  C07D277/20 ,  C07D277/32 ,  C07D401/06 ,  C07D403/06 ,  C07D405/06 ,  C07D409/06 ,  C07D413/06 ,  C07D417/06

Abstract: The present invention relates to the novel substituted aza(cyclo)alkanes of the general formula (I) in which R represents a five- or six-membered heterocyclic group which contains 1, 2, 3 or 4 nitrogen atoms and/or one or two oxygen or sulphur atoms as hetero atom ring members, the number of hetero atoms being 1, 2, 3 or 4, and which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, alkoxy, haloalkoxy, alkenyloxy, haloalkenyloxy, alkynyloxy, alkylthio, haloalkylthio, alkenylthio, haloalkenylthio, alkynylthio, alkylsulphinyl, haloalkylsulphinyl, alkylsulphonyl, haloalkylsulphonyl, amino, alkylamino, dialkylamino, aryl, arylthio, arylamino, aralkyl, formylamino, alkylcarbonylamino, formyl, carbamoyl, alkylcarbonyl and/or alkoxycarbonyl, R represents hydroxyalkyl, polyhydroxyalkyl, alkoxyalkyl or polyalkoxyalkyl, R represents hydrogen, alkyl, hydroxyalkyl, dihydroxyalkyl, alkoxyalkyl or dialkoxyalkyl, R and R together represent hydroxyalkanediyl, dihydroxyalkanediyl, alkoxyalkanediyl, dialkoxyalkanediyl, oxoalkanediyl or dioxoalkanediyl, R represents hydrogen, alkyl (which is optionally substituted by halogen, cyano, alkoxy, alkylthio, dialkylamino, trialkylsilyl, alkoxycarbonyl, carboxyl, carbamoyl, alkylaminocarbonyl, dialkylaminocarbonyl or by the radical R , R having the abovementioned meaning) or represents alkenyl (which is optionally substituted by halogen), alkynyl, benzyl (which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy or alkoxycarbonyl), formyl, alkylcarbonyl (which is optionally substituted by halogen, cyano, phenyl, phenoxy or alkoxy), cycloalkylcarbonyl (which is optionally substituted by halogen and/or alkyl), alkenylcarbonyl (which is optionally substituted by halogen), phenylcarbonyl or naphthylcarbonyl (which are optionally substituted by halogen, alkyl, haloalkyl, cyano, nitro, alkoxy and/or alkoxycarbonyl), alkoxycarbonyl, benzyloxycarbonyl, phenoxycarbonyl, alkylthiocarbonyl, benzylthiocarbonyl, phenylthiocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, phenylaminocarbonyl (which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio or alkoxycarbonyl), benzoylaminocarbonyl (which is optionally substituted by halogen, alkyl or haloalkyl), phenylsulphonylaminocarbonyl (which is optionally substituted by halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or alkoxycarbonyl), alkylthio (which is optionally substituted by halogen), phenylthio (which is optionally substituted by halogen, nitro or alkyl), alkylsulphinyl, alkylsulphonyl (which is optionally substituted by halogen), phenylsulphinyl (which is optionally substituted by halogen, nitro or alkyl), phenylsulphonyl or naphthylsulphonyl (which are optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy and/or alkoxycarbonyl), dialkyl(thio)phosphoryl, alkylalkoxy(thio)phosphoryl or dialkoxy(thio)phosphoryl, Y represents nitrogen or a CH group and Z represents cyano or nitro, to processes for their preparation and to their use as pesticides.

公开(公告)号：DE4012338A1

公开(公告)日：1991-10-24

申请号：DE4012338

申请日：1990-04-18

Applicant: BAYER AG

Inventor： WEISSMUELLER JOACHIM DR ,  ERDELEN CHRISTOPH DR ,  WACHENDORFF-NEUMANN ULRIKE DR ,  STENDEL WILHELM DR ,  LEICHT WOLFGANG DR

IPC: A01N43/58 ,  C07D311/14 ,  C07D311/58 ,  C07D405/12

Abstract: There are provided novel substituted pyridazinones of the general formula (I) in which R is alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, (di)alkylaminoalkyl, alkenyl, haloalkenyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl or aralkyl, R is halogen or alkyl, R and R independently of one another in each case represent hydrogen or alkyl, R and R are hydrogen, carboxyl, in each case optionally substituted straight-chain or branched alkyl, alkenyl, alkoxycarbonyl, aryl, aralkyl, or together with the carbon atom to which they are bonded an optionally substituted saturated or unsaturated carbocycle, R , R , R , R and R independently of one another in each case represent hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio or haloalkylthio and X is oxygen or sulphur. The novel compounds of the formula (I) have a highly pronounced activity against pests, in particular a good insecticidal, acaricidal and ovicidal activity.

公开(公告)号：ES2087926T3

公开(公告)日：1996-08-01

申请号：ES91105395

申请日：1991-04-05

Applicant: BAYER AG

Inventor： WEISSMULLER JOACHIM DR ,  ERDELEN CHRISTOPH DR ,  WACHENDORFF-NEUMANN ULRIKE DR ,  STENDEL WILHELM DR ,  LEICHT WOLFGANG DR

IPC: A01N43/58 ,  C07D311/14 ,  C07D311/58 ,  C07D405/12

Abstract: There are provided novel substituted pyridazinones of the general formula (I) in which R is alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, (di)alkylaminoalkyl, alkenyl, haloalkenyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl or aralkyl, R is halogen or alkyl, R and R independently of one another in each case represent hydrogen or alkyl, R and R are hydrogen, carboxyl, in each case optionally substituted straight-chain or branched alkyl, alkenyl, alkoxycarbonyl, aryl, aralkyl, or together with the carbon atom to which they are bonded an optionally substituted saturated or unsaturated carbocycle, R , R , R , R and R independently of one another in each case represent hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio or haloalkylthio and X is oxygen or sulphur. The novel compounds of the formula (I) have a highly pronounced activity against pests, in particular a good insecticidal, acaricidal and ovicidal activity.

公开(公告)号：DE59107939D1

公开(公告)日：1996-07-25

申请号：DE59107939

申请日：1991-04-05

Applicant: BAYER AG

Inventor： WEISSMUELLER JOACHIM DR ,  ERDELEN CHRISTOPH DR ,  WACHENDORFF-NEUMANN ULRIKE DR ,  STENDEL WILHELM DR ,  LEICHT WOLFGANG DR

IPC: A01N43/58 ,  C07D311/14 ,  C07D311/58 ,  C07D405/12

Abstract: There are provided novel substituted pyridazinones of the general formula (I) in which R is alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, (di)alkylaminoalkyl, alkenyl, haloalkenyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl or aralkyl, R is halogen or alkyl, R and R independently of one another in each case represent hydrogen or alkyl, R and R are hydrogen, carboxyl, in each case optionally substituted straight-chain or branched alkyl, alkenyl, alkoxycarbonyl, aryl, aralkyl, or together with the carbon atom to which they are bonded an optionally substituted saturated or unsaturated carbocycle, R , R , R , R and R independently of one another in each case represent hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio or haloalkylthio and X is oxygen or sulphur. The novel compounds of the formula (I) have a highly pronounced activity against pests, in particular a good insecticidal, acaricidal and ovicidal activity.

公开(公告)号：GR3020295T3

公开(公告)日：1996-09-30

申请号：GR960401575

申请日：1996-06-20

Applicant: BAYER AG

Inventor： WEISSMUELLER JOACHIM DR ,  ERDELEN CHRISTOPH DR ,  WACHENDORFF-NEUMANN ULRIKE DR ,  STENDEL WILHELM DR ,  LEICHT WOLFGANG DR

IPC: A01N43/58 ,  C07D311/14 ,  C07D311/58 ,  C07D405/12

Abstract: There are provided novel substituted pyridazinones of the general formula (I) in which R is alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, (di)alkylaminoalkyl, alkenyl, haloalkenyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl or aralkyl, R is halogen or alkyl, R and R independently of one another in each case represent hydrogen or alkyl, R and R are hydrogen, carboxyl, in each case optionally substituted straight-chain or branched alkyl, alkenyl, alkoxycarbonyl, aryl, aralkyl, or together with the carbon atom to which they are bonded an optionally substituted saturated or unsaturated carbocycle, R , R , R , R and R independently of one another in each case represent hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio or haloalkylthio and X is oxygen or sulphur. The novel compounds of the formula (I) have a highly pronounced activity against pests, in particular a good insecticidal, acaricidal and ovicidal activity.

公开(公告)号：ES2086849T3

公开(公告)日：1996-07-01

申请号：ES93116618

申请日：1993-10-14

Applicant: BAYER AG

Inventor： WAGNER KLAUS DR ,  ERDELEN CHRISTOPH DR ,  HARTWIG JURGEN DR ,  LEICHT WOLFGANG DR ,  STENDEL WILHELM DR

IPC: A01N43/08 ,  A01N43/10 ,  A01N43/36 ,  A01N43/40 ,  A01N43/50 ,  A01N43/54 ,  A01N43/58 ,  A01N43/60 ,  A01N43/647 ,  A01N43/653 ,  A01N43/76 ,  A01N43/78 ,  A01N43/80 ,  A01N43/824 ,  A01N43/836 ,  A01N47/44 ,  A01N51/00 ,  C07D213/24 ,  C07D213/26 ,  C07D213/30 ,  C07D213/61 ,  C07D277/20 ,  C07D277/32 ,  C07D401/06 ,  C07D403/06 ,  C07D405/06 ,  C07D409/06 ,  C07D413/06 ,  C07D417/06

Abstract: The present invention relates to the novel substituted aza(cyclo)alkanes of the general formula (I) in which R represents a five- or six-membered heterocyclic group which contains 1, 2, 3 or 4 nitrogen atoms and/or one or two oxygen or sulphur atoms as hetero atom ring members, the number of hetero atoms being 1, 2, 3 or 4, and which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, alkoxy, haloalkoxy, alkenyloxy, haloalkenyloxy, alkynyloxy, alkylthio, haloalkylthio, alkenylthio, haloalkenylthio, alkynylthio, alkylsulphinyl, haloalkylsulphinyl, alkylsulphonyl, haloalkylsulphonyl, amino, alkylamino, dialkylamino, aryl, arylthio, arylamino, aralkyl, formylamino, alkylcarbonylamino, formyl, carbamoyl, alkylcarbonyl and/or alkoxycarbonyl, R represents hydroxyalkyl, polyhydroxyalkyl, alkoxyalkyl or polyalkoxyalkyl, R represents hydrogen, alkyl, hydroxyalkyl, dihydroxyalkyl, alkoxyalkyl or dialkoxyalkyl, R and R together represent hydroxyalkanediyl, dihydroxyalkanediyl, alkoxyalkanediyl, dialkoxyalkanediyl, oxoalkanediyl or dioxoalkanediyl, R represents hydrogen, alkyl (which is optionally substituted by halogen, cyano, alkoxy, alkylthio, dialkylamino, trialkylsilyl, alkoxycarbonyl, carboxyl, carbamoyl, alkylaminocarbonyl, dialkylaminocarbonyl or by the radical R , R having the abovementioned meaning) or represents alkenyl (which is optionally substituted by halogen), alkynyl, benzyl (which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy or alkoxycarbonyl), formyl, alkylcarbonyl (which is optionally substituted by halogen, cyano, phenyl, phenoxy or alkoxy), cycloalkylcarbonyl (which is optionally substituted by halogen and/or alkyl), alkenylcarbonyl (which is optionally substituted by halogen), phenylcarbonyl or naphthylcarbonyl (which are optionally substituted by halogen, alkyl, haloalkyl, cyano, nitro, alkoxy and/or alkoxycarbonyl), alkoxycarbonyl, benzyloxycarbonyl, phenoxycarbonyl, alkylthiocarbonyl, benzylthiocarbonyl, phenylthiocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, phenylaminocarbonyl (which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio or alkoxycarbonyl), benzoylaminocarbonyl (which is optionally substituted by halogen, alkyl or haloalkyl), phenylsulphonylaminocarbonyl (which is optionally substituted by halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or alkoxycarbonyl), alkylthio (which is optionally substituted by halogen), phenylthio (which is optionally substituted by halogen, nitro or alkyl), alkylsulphinyl, alkylsulphonyl (which is optionally substituted by halogen), phenylsulphinyl (which is optionally substituted by halogen, nitro or alkyl), phenylsulphonyl or naphthylsulphonyl (which are optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy and/or alkoxycarbonyl), dialkyl(thio)phosphoryl, alkylalkoxy(thio)phosphoryl or dialkoxy(thio)phosphoryl, Y represents nitrogen or a CH group and Z represents cyano or nitro, to processes for their preparation and to their use as pesticides.

公开(公告)号：BR9101524A

公开(公告)日：1991-12-10

申请号：BR9101524

申请日：1991-04-16

Applicant: BAYER AG

Inventor： WEISSMUELLER JOACHIM DR ,  ERDELEN CHRISTOPH DR ,  WACHENDORFF-NEUMANN ULRIKE DR ,  STENDEL WILHELM DR ,  LEICHT WOLFGANG DR

IPC: A01N43/58 ,  C07D311/14 ,  C07D311/58 ,  C07D405/12 ,  C07D237/14 ,  C07D237/18 ,  C07D237/12 ,  C07D405/14

Abstract: There are provided novel substituted pyridazinones of the general formula (I) in which R is alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, (di)alkylaminoalkyl, alkenyl, haloalkenyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl or aralkyl, R is halogen or alkyl, R and R independently of one another in each case represent hydrogen or alkyl, R and R are hydrogen, carboxyl, in each case optionally substituted straight-chain or branched alkyl, alkenyl, alkoxycarbonyl, aryl, aralkyl, or together with the carbon atom to which they are bonded an optionally substituted saturated or unsaturated carbocycle, R , R , R , R and R independently of one another in each case represent hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio or haloalkylthio and X is oxygen or sulphur. The novel compounds of the formula (I) have a highly pronounced activity against pests, in particular a good insecticidal, acaricidal and ovicidal activity.