SUBSTITUTED AZA (CYCLO) ALKANES
    2.
    发明专利

    公开(公告)号:IL107380A

    公开(公告)日:1997-09-30

    申请号:IL10738093

    申请日:1993-10-25

    Applicant: BAYER AG

    Abstract: The present invention relates to the novel substituted aza(cyclo)alkanes of the general formula (I) in which R represents a five- or six-membered heterocyclic group which contains 1, 2, 3 or 4 nitrogen atoms and/or one or two oxygen or sulphur atoms as hetero atom ring members, the number of hetero atoms being 1, 2, 3 or 4, and which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, alkoxy, haloalkoxy, alkenyloxy, haloalkenyloxy, alkynyloxy, alkylthio, haloalkylthio, alkenylthio, haloalkenylthio, alkynylthio, alkylsulphinyl, haloalkylsulphinyl, alkylsulphonyl, haloalkylsulphonyl, amino, alkylamino, dialkylamino, aryl, arylthio, arylamino, aralkyl, formylamino, alkylcarbonylamino, formyl, carbamoyl, alkylcarbonyl and/or alkoxycarbonyl, R represents hydroxyalkyl, polyhydroxyalkyl, alkoxyalkyl or polyalkoxyalkyl, R represents hydrogen, alkyl, hydroxyalkyl, dihydroxyalkyl, alkoxyalkyl or dialkoxyalkyl, R and R together represent hydroxyalkanediyl, dihydroxyalkanediyl, alkoxyalkanediyl, dialkoxyalkanediyl, oxoalkanediyl or dioxoalkanediyl, R represents hydrogen, alkyl (which is optionally substituted by halogen, cyano, alkoxy, alkylthio, dialkylamino, trialkylsilyl, alkoxycarbonyl, carboxyl, carbamoyl, alkylaminocarbonyl, dialkylaminocarbonyl or by the radical R , R having the abovementioned meaning) or represents alkenyl (which is optionally substituted by halogen), alkynyl, benzyl (which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy or alkoxycarbonyl), formyl, alkylcarbonyl (which is optionally substituted by halogen, cyano, phenyl, phenoxy or alkoxy), cycloalkylcarbonyl (which is optionally substituted by halogen and/or alkyl), alkenylcarbonyl (which is optionally substituted by halogen), phenylcarbonyl or naphthylcarbonyl (which are optionally substituted by halogen, alkyl, haloalkyl, cyano, nitro, alkoxy and/or alkoxycarbonyl), alkoxycarbonyl, benzyloxycarbonyl, phenoxycarbonyl, alkylthiocarbonyl, benzylthiocarbonyl, phenylthiocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, phenylaminocarbonyl (which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio or alkoxycarbonyl), benzoylaminocarbonyl (which is optionally substituted by halogen, alkyl or haloalkyl), phenylsulphonylaminocarbonyl (which is optionally substituted by halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or alkoxycarbonyl), alkylthio (which is optionally substituted by halogen), phenylthio (which is optionally substituted by halogen, nitro or alkyl), alkylsulphinyl, alkylsulphonyl (which is optionally substituted by halogen), phenylsulphinyl (which is optionally substituted by halogen, nitro or alkyl), phenylsulphonyl or naphthylsulphonyl (which are optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy and/or alkoxycarbonyl), dialkyl(thio)phosphoryl, alkylalkoxy(thio)phosphoryl or dialkoxy(thio)phosphoryl, Y represents nitrogen or a CH group and Z represents cyano or nitro, to processes for their preparation and to their use as pesticides.

    Substituted pyridazinones, process for their preparation and their use as parasiticide

    公开(公告)号:GR3020295T3

    公开(公告)日:1996-09-30

    申请号:GR960401575

    申请日:1996-06-20

    Applicant: BAYER AG

    Abstract: There are provided novel substituted pyridazinones of the general formula (I) in which R is alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, (di)alkylaminoalkyl, alkenyl, haloalkenyl, in each case optionally substituted cycloalkyl, cycloalkylalkyl, aryl or aralkyl, R is halogen or alkyl, R and R independently of one another in each case represent hydrogen or alkyl, R and R are hydrogen, carboxyl, in each case optionally substituted straight-chain or branched alkyl, alkenyl, alkoxycarbonyl, aryl, aralkyl, or together with the carbon atom to which they are bonded an optionally substituted saturated or unsaturated carbocycle, R , R , R , R and R independently of one another in each case represent hydrogen, halogen, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio or haloalkylthio and X is oxygen or sulphur. The novel compounds of the formula (I) have a highly pronounced activity against pests, in particular a good insecticidal, acaricidal and ovicidal activity.

    5.
    发明专利
    未知

    公开(公告)号:ES2086849T3

    公开(公告)日:1996-07-01

    申请号:ES93116618

    申请日:1993-10-14

    Applicant: BAYER AG

    Abstract: The present invention relates to the novel substituted aza(cyclo)alkanes of the general formula (I) in which R represents a five- or six-membered heterocyclic group which contains 1, 2, 3 or 4 nitrogen atoms and/or one or two oxygen or sulphur atoms as hetero atom ring members, the number of hetero atoms being 1, 2, 3 or 4, and which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkenyl, haloalkenyl, alkynyl, alkoxy, haloalkoxy, alkenyloxy, haloalkenyloxy, alkynyloxy, alkylthio, haloalkylthio, alkenylthio, haloalkenylthio, alkynylthio, alkylsulphinyl, haloalkylsulphinyl, alkylsulphonyl, haloalkylsulphonyl, amino, alkylamino, dialkylamino, aryl, arylthio, arylamino, aralkyl, formylamino, alkylcarbonylamino, formyl, carbamoyl, alkylcarbonyl and/or alkoxycarbonyl, R represents hydroxyalkyl, polyhydroxyalkyl, alkoxyalkyl or polyalkoxyalkyl, R represents hydrogen, alkyl, hydroxyalkyl, dihydroxyalkyl, alkoxyalkyl or dialkoxyalkyl, R and R together represent hydroxyalkanediyl, dihydroxyalkanediyl, alkoxyalkanediyl, dialkoxyalkanediyl, oxoalkanediyl or dioxoalkanediyl, R represents hydrogen, alkyl (which is optionally substituted by halogen, cyano, alkoxy, alkylthio, dialkylamino, trialkylsilyl, alkoxycarbonyl, carboxyl, carbamoyl, alkylaminocarbonyl, dialkylaminocarbonyl or by the radical R , R having the abovementioned meaning) or represents alkenyl (which is optionally substituted by halogen), alkynyl, benzyl (which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy or alkoxycarbonyl), formyl, alkylcarbonyl (which is optionally substituted by halogen, cyano, phenyl, phenoxy or alkoxy), cycloalkylcarbonyl (which is optionally substituted by halogen and/or alkyl), alkenylcarbonyl (which is optionally substituted by halogen), phenylcarbonyl or naphthylcarbonyl (which are optionally substituted by halogen, alkyl, haloalkyl, cyano, nitro, alkoxy and/or alkoxycarbonyl), alkoxycarbonyl, benzyloxycarbonyl, phenoxycarbonyl, alkylthiocarbonyl, benzylthiocarbonyl, phenylthiocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, phenylaminocarbonyl (which is optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio or alkoxycarbonyl), benzoylaminocarbonyl (which is optionally substituted by halogen, alkyl or haloalkyl), phenylsulphonylaminocarbonyl (which is optionally substituted by halogen, alkyl, haloalkyl, alkoxy, haloalkoxy or alkoxycarbonyl), alkylthio (which is optionally substituted by halogen), phenylthio (which is optionally substituted by halogen, nitro or alkyl), alkylsulphinyl, alkylsulphonyl (which is optionally substituted by halogen), phenylsulphinyl (which is optionally substituted by halogen, nitro or alkyl), phenylsulphonyl or naphthylsulphonyl (which are optionally substituted by halogen, cyano, nitro, alkyl, haloalkyl, alkoxy, haloalkoxy and/or alkoxycarbonyl), dialkyl(thio)phosphoryl, alkylalkoxy(thio)phosphoryl or dialkoxy(thio)phosphoryl, Y represents nitrogen or a CH group and Z represents cyano or nitro, to processes for their preparation and to their use as pesticides.

    7.
    发明专利
    未知

    公开(公告)号:DE59008063D1

    公开(公告)日:1995-02-02

    申请号:DE59008063

    申请日:1990-08-18

    Applicant: BAYER AG

    Abstract: There are described novel 3-aryl-pyrrolidine-2,4-dione derivatives of the formula (I) in which A-B represents -S-CH2-, -SO-CH2-, -SO2CH2-, -CH2-S-, -CH2SO-, -CH2SO2-, -S-, -SO- or -SO2-, X represents alkyl, halogen or alkoxy, Y represents hydrogen, alkyl, halogen, alkoxy or haloalkyl, Z represents alkyl, halogen or alkoxy, n represents a number from 0-3, R represents hydrogen or the groups -CO-R or -CO-O-R , where E represents a metal cation equivalent or an ammonium ion, R represents optionally halogen-substituted alkyl, alkenyl, alkoxyalkyl, alkylthioalkyl, polyalkoxyalkyl and optionally substituted cycloalkyl which can be interrupted by hetero atoms, or represents optionally substituted phenyl, optionally substituted phenylalkyl, substituted hetaryl, substituted phenoxyalkyl and substituted hetaryloxyalkyl, and R represents optionally halogen-substituted alkyl, cycloalkyl, alkenyl, alkoxyalkyl, polyalkoxyalkyl and optionally substituted phenyl, and several processes for their preparation. The novel compounds of the formula (I) can be used for controlling insects and arachnids and as weedkillers.

    10.
    发明专利
    未知

    公开(公告)号:AT111298T

    公开(公告)日:1994-09-15

    申请号:AT91112643

    申请日:1991-07-27

    Applicant: BAYER AG

    Abstract: The present invention relates to a method and agent for controlling fleas on and in the surroundings of domestic animals, which is characterised in that the domestic animals are treated with collars which contain active substances which inhibit the development of insects.

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