New acylated 5-amino-isothiazole derivatives

    公开(公告)号:DE19736545A1

    公开(公告)日:1999-02-25

    申请号:DE19736545

    申请日:1997-08-22

    Applicant: BAYER AG

    Abstract: Acylated 5-aminoisothiazole derivatives (I) are new. Acylated 5-aminoisothiazole derivatives of formula (I) are new. R1 = alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, alkoxy, alkylthio, alkylamino, dialkylamino or optionally substituted cycloalkyl; R2 = H, halo, CN, NO2, thiocyanato, alkoxycarbonyl, alkenyloxycarbonyl, alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, alkylsulfonyl, haloalkylsulfonyl, thiocarbamoyl, alkoxy, formyl, alkylcarbonyl or CR7=NOR8; R7, R8 = H, alkyl, haloalkyl, alkenyl, optionally substituted cycloalkyl or cycloalkylalkyl or optionally substituted aryl or arylalkyl; R3 = alkyl, haloalkyl, alkoxyalkyl, alkylthioalkyl, alkenyl, alkynyl, alkylcarbonyloxyalkyl, alkoxycarbonyloxyalkyl, optionally substituted aryl, aralkyl or arylalkoxyalkyl, optionally substituted cycloalkyl, cycloalkylalkyl, cycloalkoxyalkyl or cycloalkylthioalkyl or N=CR5R6; R5, R6 = H, alkyl, haloalkyl, alkenyl, optionally substituted cycloalkyl or cycloalkylalkyl or optionally substituted aryl or arylalkyl; or R5+R6 = an optionally substituted carbocyclic ring; R4 = optionally substituted aryl, cycloalkyl, cycloalkenyl or heterocyclyl; A, Z = O or S; Y = optionally substituted alkylene, alkenylene or alkyleneoxy. Independent claims are included for the following: (a) the preparation of (I); and (b) intermediates of formula (IV) and (VIA). R21 = R, CO-R71 or CR71=NOR7; R = alkylthio, haloalkylthio, alkylsulfinyl, haloalkylsulfinyl, akylsulfonyl or haloalkylsulfonyl; R71 = H or alkyl; R8 = H, 1-4C alkyl, 1-4C haloalkyl, 2-4C alkenyl, 3-6C cycloalkyl or 3-6C cycloalkyl-(1-4C alkyl) (both optionally substituted by 1-3 from 1-4C alkyl or halo groups) or phenyl or phenyl-(1-4C alkyl) (both optionally ring-substituted by 1-3 from halo, NO2, CN, 1-4C alkyl, 1- or 2C haloalkyl, 1-4C alkoxy, 1-4C alkylthio, 1- or 2C haloalkoxy or 1- or 2C haloalkylthio groups) or (1-4C alkoxy)carbonyl or (1-4C alkyl)carbonyloxy.

    9.
    发明专利
    未知

    公开(公告)号:DE19545638A1

    公开(公告)日:1997-06-12

    申请号:DE19545638

    申请日:1995-12-07

    Applicant: BAYER AG

    Abstract: The invention relates to the use of partially known 1,2,3-thiadiazole carboxylic acid (thio)esters of formula (I), in which R is hydrogen, optionally substituted alkyl or optionally substituted aryl; R is optionally substituted alkyl, optionally substituted cycloalkyl, optionally substituted cycloalkenyl or optionally substituted aryl; and Q is oxygen or sulphur, and the use of acid addition salts and metal salt complexes of said esters to protect plants well from attack by undesirable micro-organisms and to control animal pests. Particular 1,2,3-thiadiazole carboxylic acid (thio)esters of formula (I) are novel.

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