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1.
公开(公告)号:WO2014045263A3
公开(公告)日:2014-05-15
申请号:PCT/IB2013058808
申请日:2013-09-24
Applicant: REDDYS LAB LTD DR
Inventor: IQBAL JAVED , DAHANUKAR VILAS HARESHWAR , ORUGANTI SRINIVAS , KANDAGATLA BHASKAR , KUNHIMON SYAM KUMAR UNNIARAN , SAGYAM RAJESHWAR REDDY , IRENI BABU , KONDEPUDI VEERA VENKATA SATYANARAYANA MURTHY , MUTTAVARAPU MURALI MOHAN , BUCCHIKONDA RAVINDER , GANGIREDDY RAJENDAR REDDY
IPC: C07D209/52 , C07C205/28 , C07C217/14 , C07D317/16 , C07D317/28
CPC classification number: C07D209/52 , C07B2200/07 , C07C35/06 , C07C43/315 , C07C215/20 , C07C217/44 , C07C223/02 , C07C255/46 , C07C271/16 , C07C271/18 , C07C309/66 , C07C2601/08 , C07D317/18 , C07D317/28 , C07F7/1856 , C07K5/0202 , C07K5/1024
Abstract: Provided are novel processes for preparation of (1S, 3aR, 6aS)-octahydrocyclopenta[c]pyrrole-1-carboxylic acid and its derivatives; land their use in preparation of Telaprevir.
Abstract translation: 提供(1S,3aR,6aS) - 八氢环戊二烯并[c]吡咯-1-羧酸及其衍生物的制备方法; 将其用于制备特拉匹韦尔。
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公开(公告)号:WO2013190509A2
公开(公告)日:2013-12-27
申请号:PCT/IB2013055096
申请日:2013-06-21
Applicant: REDDYS LAB LTD DR
Inventor: NARIYAM SEKHAR MUNASWAMY , BHALERAO DINESH SHIVAJI , DAHANUKAR VILAS HARESHWAR , ORUGANTI SRINIVAS , RAPOLU RAJESH KUMAR , KANDAGATLA BHASKAR , IQBAL JAVED , KHOBARE SANDIP RAMDAS , KALLAM SRINIVASA REDDY , BANDA MALAVIKA , GARARE VIKAS SADASHIV , EDA VISHNUVARDHANA VEMA REDDY
CPC classification number: A61K38/06 , A61K38/55 , C07K5/0808
Abstract: The present application relates to processes for preparing intermediates of Boceprevir and their use in preparation of Boceprevir or its pharmaceutically acceptable salts thereof.
Abstract translation: 本申请涉及制备波普瑞韦中间体的方法及其在制备波普瑞韦或其药学上可接受的盐中的用途。
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公开(公告)号:WO2012146980A3
公开(公告)日:2012-12-27
申请号:PCT/IB2012000922
申请日:2012-04-27
Applicant: REDDYS LAB LTD DR , KATKAM SRINIVAS , SAGYAM RAJESWAR REDDY , MORTHALA RAGHAVENDAR RAO , IRENI BABU , VINIGARI KRISHNA , RAMDOSS SURESH KUMAR , RANGINENI SRINIVASULU , TUMMALA ARJUNKUMAR , IQBAL JAVED , ORUGANTI SRINIVAS , KANDAGATLA BHASKAR
Inventor: KATKAM SRINIVAS , SAGYAM RAJESWAR REDDY , MORTHALA RAGHAVENDAR RAO , IRENI BABU , VINIGARI KRISHNA , RAMDOSS SURESH KUMAR , RANGINENI SRINIVASULU , TUMMALA ARJUNKUMAR , IQBAL JAVED , ORUGANTI SRINIVAS , KANDAGATLA BHASKAR
IPC: C07C211/00 , C07D333/20
CPC classification number: C07C205/45 , C07C201/10 , C07C201/12 , C07C213/00 , C07C213/02 , C07C213/10 , C07C215/28 , C07C205/04
Abstract: The present application provide processes for the preparation of fingolimod and its pharmaceutically acceptable salts, process for the purification of fingolimod hydrochloride and process for the preparation of amorphous fingolimod hydrochloride.
Abstract translation: 本申请提供了芬戈莫德及其药学上可接受的盐的制备方法,盐酸芬戈莫德的纯化方法和用于制备无定形芬戈莫德盐酸盐的方法。
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公开(公告)号:EP2702034A4
公开(公告)日:2015-03-25
申请号:EP12777520
申请日:2012-04-27
Applicant: REDDYS LAB LTD DR
Inventor: KATKAM SRINIVAS , SAGYAM RAJESWAR REDDY , MORTHALA RAGHAVENDAR RAO , IRENI BABU , VINIGARI KRISHNA , RAMDOSS SURESH KUMAR , RANGINENI SRINIVASULU , TUMMALA ARJUNKUMAR , IQBAL JAVED , ORUGANTI SRINIVAS , KANDAGATLA BHASKAR
IPC: C07C211/00 , C07C201/10 , C07C201/12 , C07C213/02 , C07D333/20
CPC classification number: C07C205/45 , C07C201/10 , C07C201/12 , C07C213/00 , C07C213/02 , C07C213/10 , C07C215/28 , C07C205/04
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5.
公开(公告)号:CA2918451A1
公开(公告)日:2015-01-22
申请号:CA2918451
申请日:2014-07-15
Applicant: REDDYS LAB LTD DR
Inventor: IQBAL JAVED , DAHANUKAR VILAS HARESHWAR , ORUGANTI SRINIVAS , KANDAGATLA BHASKAR
IPC: A61K31/551 , C07D243/08
Abstract: A novel processes for the preparation of suvorexant (formula I), its related compounds and its intermediates that are simple, economical and commercially viable. (I)
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