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1.MODULATION OF ENDOGENOUS AMPK LEVELS FOR THE TREATMENT OF OBESITY 审中-公开
Title translation: 内源性AMPK水平的调节用于治疗肥胖公开(公告)号:WO2009019600A3
公开(公告)日:2009-12-30
申请号:PCT/IB2008002140
申请日:2008-08-08
Applicant: REDDYS LAB LTD DR , MISRA PARIMAL , CHAKRABARTI RANJAN , MADHURAREKHA CHINNABOINA , HASHAM SUMERA NIKHAT , POTLURI VIJAY KUMAR , SASMAL PRADIP KUMAR , DAS SAIBAL KUMAR , IQBAL JAVED
Inventor: MISRA PARIMAL , CHAKRABARTI RANJAN , MADHURAREKHA CHINNABOINA , HASHAM SUMERA NIKHAT , POTLURI VIJAY KUMAR , SASMAL PRADIP KUMAR , DAS SAIBAL KUMAR , IQBAL JAVED
IPC: G01N33/00
CPC classification number: C12Q1/485 , G01N2800/044
Abstract: A method for identifying an AMPK activator is provided. The method includes providing a sample of cells that include AMPK and perilipin, providing a sample of an AMPK activator-candidate, contacting the cell sample and the activator-candidate, and measuring a quantitative indicator of the AMPK activation within the cell sample after the contacting step.
Abstract translation: 提供了一种用于鉴定AMPK激活剂的方法。 该方法包括提供包含AMPK和肾上腺素的细胞样品,提供AMPK激活剂候选物的样品,接触细胞样品和活化剂候选物,并测量接触后细胞样品中AMPK活化的定量指标 步。
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公开(公告)号:WO2007005785B1
公开(公告)日:2007-03-22
申请号:PCT/US2006025898
申请日:2006-06-30
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR , POTLURI VIJAY KUMAR , DAS SAIBAL KUMAR , SASMAL PRADIP KUMAR , IQBAL JAVED , MISRA PARIMAL , CHAKRABARTI RANJAN , TALWAR RASHMI
Inventor: POTLURI VIJAY KUMAR , DAS SAIBAL KUMAR , SASMAL PRADIP KUMAR , IQBAL JAVED , MISRA PARIMAL , CHAKRABARTI RANJAN , TALWAR RASHMI
IPC: C07D277/14 , A61K31/426 , A61K31/5377 , C07D265/32
CPC classification number: C07D277/42
Abstract: The present application provides novel thiazole derivatives that are useful as activators of Adenosine 5'-Monophosphate-Activated Protein Kinase and pharmaceutical compositions containing such compounds.
Abstract translation: 本申请提供了可用作腺苷5'-单磷酸激活蛋白激酶的激活剂的新型噻唑衍生物和含有这些化合物的药物组合物。
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公开(公告)号:EP1907369A4
公开(公告)日:2009-07-22
申请号:EP06774435
申请日:2006-06-30
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR
Inventor: POTLURI VIJAY KUMAR , DAS SAIBAL KUMAR , SASMAL PRADIP KUMAR , IQBAL JAVED , MISRA PARIMAL , CHAKRABARTI RANJAN , TALWAR RASHMI
IPC: C07D277/14 , A61K31/426 , A61K31/5377 , C07D265/32
CPC classification number: C07D277/42
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公开(公告)号:BRPI0613555A2
公开(公告)日:2011-01-18
申请号:BRPI0613555
申请日:2006-06-30
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR
Inventor: POTLURI VIJAY KUMAR , DAS SAIBAL KUMAR , SASMAL PRADIP KUMAR , IQBAL JAVED , MISRA PARIMAL , CHAKRABARTI RANJAN , TALWAR RASHMI
IPC: C07D277/14 , A61K31/426 , A61K31/5377 , C07D265/32
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公开(公告)号:NO20080629A
公开(公告)日:2008-02-19
申请号:NO20080629
申请日:2008-02-04
Applicant: REDDYS LAB LTD DR
Inventor: POTLURI VIJAY KUMAR , DAS SAIBAL KUMAR , SASMAL PRADIP KUMAR , IQBAL JAVED , MISRA PARIMAL , CHAKRABARTI RANJAN , TALWAR RASHMI
IPC: C07D277/14
CPC classification number: C07D277/42
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公开(公告)号:NO20080629L
公开(公告)日:2008-02-19
申请号:NO20080629
申请日:2008-02-04
Applicant: REDDYS LAB LTD DR
Inventor: POTLURI VIJAY KUMAR , DAS SAIBAL KUMAR , SASMAL PRADIP KUMAR , IQBAL JAVED , MISRA PARIMAL , CHAKRABARTI RANJAN , TALWAR RASHMI
IPC: C07D277/14
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公开(公告)号:CA2614098A1
公开(公告)日:2007-01-11
申请号:CA2614098
申请日:2006-06-30
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR
Inventor: DAS SAIBAL KUMAR , TALWAR RASHMI , POTLURI VIJAY KUMAR , IQBAL JAVED , CHAKRABARTI RANJAN , SASMAL PRADIP KUMAR , MISRA PARIMAL
IPC: C07D277/14 , A61K31/426 , A61K31/5377 , C07D265/32
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