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公开(公告)号:NO20063132A
公开(公告)日:2006-09-11
申请号:NO20063132
申请日:2006-07-05
Applicant: VERTEX PHARMA
Inventor: MAKINGS LEWIS R , GROOTENHUIS PETER D J , BLANCO MIGUEL GARCIA-GUZMAN , LONDO PHILIP MARTIN
IPC: C07D471/04 , A61K31/4745 , C07D471/02
CPC classification number: C07D471/04
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公开(公告)号:CA2548009A1
公开(公告)日:2005-06-23
申请号:CA2548009
申请日:2004-12-07
Applicant: VERTEX PHARMA
Inventor: MAKINGS LEWIS R , LONDO PHILIP MARTIN , GROOTENHUIS PETER D J , GARCIA-GUZMAN BLANCO MIGUEL
IPC: C07D471/04 , A61K31/4745 , A61P25/00 , C07D471/02
Abstract: A compound of formula (I) wherein: Ring A is aryl or heteroaryl; one of V, W , Y or Z is nitrogen and the other of V, W, Y and Z are -C(R5)-; modulate muscarinic receptors and are useful for treating muscarinic receptor mediate d diseases.
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公开(公告)号:AU2004297241A1
公开(公告)日:2005-06-23
申请号:AU2004297241
申请日:2004-12-07
Applicant: VERTEX PHARMA
Inventor: MAKINGS LEWIS R , GROOTENHUIS PETER D J , LONDO PHILIP MARTIN , BLANCO MIGUEL GARCIA-GUZMAN
IPC: C07D471/04 , A61K31/4745 , C07D471/02
Abstract: The modulator compounds described herein modulate muscarinic receptors and are useful for treating muscarinic receptor mediated diseases.
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公开(公告)号:NO20063132L
公开(公告)日:2006-09-11
申请号:NO20063132
申请日:2006-07-05
Applicant: VERTEX PHARMA
Inventor: MAKINGS LEWIS R , GROOTENHUIS PETER D J , BLANCO MIGUEL GARCIA-GUZMAN , LONDO PHILIP MARTIN
IPC: C07D471/04 , A61K31/4745 , C07D471/02
Abstract: The modulator compounds described herein modulate muscarinic receptors and are useful for treating muscarinic receptor mediated diseases.
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公开(公告)号:MXPA06006532A
公开(公告)日:2006-08-23
申请号:MXPA06006532
申请日:2004-12-07
Applicant: VERTEX PHARMA
Inventor: LONDO PHILIP MARTIN
IPC: A61P25/00 , C07D471/02 , C07D471/04 , A61K31/4745
Abstract: Un compuesto de la Formula (I) en donde: el anillo A es arilo o heteroarilo, uno de V, W, Y o Z es nitrogeno y el otro de V, W, Y y Z son -C(R5)-; modulan los receptores muscarinicos y son utiles para tratar enfermedades mediadas por el receptor muscarinico.
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