Abstract:
The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R and/or R being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.
Abstract:
The invention relates to the use of 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines of formula I for controlling phytopathogenic fungi. The variables in formula I have the following designations: Y represents alkylene, alkenylene or alkinylene, optionally substituted by alkyl groups; R 1 represents halogen, cyano, nitro, hydroxy, mercapto, alkyl, halogenalkyl, alkenyl, cycloalkyl, cycloalkenyl, alkoxy, halogenalkoxy, alkenyloxy, alkinyloxy, alkylthio, NR A R B , alkylcarbonyl, phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group O, N or S; R A , R B represent hydrogen, alkyl and alkylcarbonyl; n represents 0, 1, 2, 3 or 4; R 2 represents alkyl, alkenyl, cycloalkyl, alkoxyalkyl and alkylthioalkyl; R 3 represents hydrogen, halogen, cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phenylthio, benzyloxy, benzylthio, or alkyl-S(O) m- ; m represents 0, 1 or 2; A represents N and C-R a ; and R a represents hydrogen and alkyl. The carbon atoms in Y, R 1 , R 2 , R 3 and Ra can be substituted according to the description. The invention also relates to novel 5-alkyl-6-phenylalkyl-7-amino-azolopyrimidines, to methods for producing said compounds, and to agents containing the same.
Abstract:
The invention relates to 2-substituted 7-amino-azolopyrimidine of formula (I), wherein substituents have the following meanings: R 1 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, Cycloalkyl, alkoxy, alkoxyalkyl, benzyloxyalkyl, alkoxyalkenyl or akoxyalkinyl; R 2 is hydrogen, halogen, cyano, alkyl, halogenalkyl, alkenyl, alkynyl, cycloalkyl, alkoxy, alkoxyalkyl and alkylthioalkyl, wherein a carbon chain in R 1 and/or R 2 are substitutable according to a description; R 3 is halogen, Cyano, NR A R B , hydroxy, mercapto, alkyl, halogenalkyl, cycloalkyl, alkoxy, alkylthio, cycloalkoxy, cycloalkylthio, carboxyl, formyl, alkylcarbonyl, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, phenyl, phenoxy, phe- nylthio, benzyloxy, benzylthio, alkyl-S(O) m- ; A N and CR x ; R x is hydrogen or one of above groups for R 3 . A method and intermediate products for producing said compounds, agents containing said compounds and the use thereof for combating plant-pathogen fungi are also disclosed.
Abstract translation:2-取代的式(I)其中取代基具有以下含义的7-氨基azolopyrimidines:R t 1 SUP>为氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基, benzyloxyalkyl,烷氧基烯基或alkoxyalkynyl; [R 2 SUP>为氢,卤素,氰基,烷基,卤代烷基,烯基,炔基,环烷基,烷氧基,烷氧基烷基和烷硫基烷基,其中在R中的碳链 1 SUP>和/或R 2 SUP>可以根据描述被取代; [R 3 SUP>为卤素,氰基,NR 一 SUP> - [R 乙 SUP>,羟基,巯基,烷基,卤代烷基,环烷基,烷氧基,烷硫基,环烷氧基,环烷硫基, 羧基,甲酰基,烷基羰基,烷氧基羰基,烯氧基羰基,炔氧基羰基,苯基,苯氧基,苯丙氨酸nylthio,苄氧基,苄硫基,烷基-S(O)米 - SUB>; A N和CR X SUP>; ,R 3 SUP>基 X SUP>是氢或其中R 称作; 的方法和中间体制备这些化合物,含有它们和它们在防治植物病原性有害真菌的组合物。
Abstract:
The invention relates to 6-(2,6-dichlorophenyl)-triazolopyrimidines of formula (I) wherein the substituents have the following designations: R and R represent hydrogen, alkyl, halogenalkyl, cycloalkyl, halogencycloalkyl, alkenyl, halogenalkenyl, cycloalkenyl, halogencycloalkenyl, alkinyl, halogenalkinyl or phenyl, naphthyl, or a five-membered or six-membered saturated, partially unsaturated or aromatic heterocycle containing between one and four heteroatoms from the group containing O, N or S; R and R can also form, together with the nitrogen atom to which they are bound, a five-membered or six-membered heterocycle or heteroaryl which is bound by N and contains between one and three other heteroatoms from the group containing O, N and S as a cyclic member and is substituted according to the description; and X represents alkyl, cyano, alkoxy, halogenalkoxy, alkenyloxy or halogenalkenyloxy, but does not represent C1-C4 alkyl when R and R together represent piperidin-1-yl or 4-methylpiperidin-1-yl. The invention also relates to a method for producing said compounds, agents containing the same, and the use thereof for controlling plant pathogenic fungi.
Abstract:
The invention relates to fungicidal mixtures containing in the form of active components 1) 5-methyl-7-amino-triazolopyrimidine of formula (I), wherein R is alkyl, halogenalkyl, alkenyl or cyclopentyl, R is hydrogen or alkyl, R and R together with the nitrogen atom to which they are bound may form a piperidinyl cycle substitutable by a methyl group, L is fluorine or chlorine, L , L are independently from each other hydrogen, fluorine or chlorine and 2) at least one type of active substance selected from groups A) azoles, B) strobilurins, C) acyl alanines, D) amine derivatives, E) anilinopyrimidines; F) dicarboximides; G) cinnamic acid amides and analogues thereof, H) antibiotics, K) dithiocarbamates, L) heterocyclic compounds, M) sulphur and copper fungicides, N) nitrophenyl derivatives, O) phenylpyrroles, P) sulfenic acid derivatives, Q) other fungicides and R) growth retardants according to the descriptions, wherein said mixtures contain the compounds in a synergically efficient amount. Novel triazolopyrimidines, methods for controlling pathogenic fungi using the mixtures of the compound (I) with active substances of the groups A) and R), the use the compounds (I) with the active substances of the groups A) and R) for producing said mixtures and agents containing said mixtures are also disclosed.
Abstract:
Fungicidal mixtures, comprising as active components 1) the strobilurin derivative of the formula I, and 2) at least one active compound II selected from the group of the carbamates in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with active compounds II, the use of the compound I with active compounds II for preparing such mixtures and compositions comprising these mixtures.
Abstract:
Fungicidal mixtures, comprising as active components 1) the strobilurin derivative of the formula I, and 2) at least one active compound II selected from the group of the guanidines, antibiotics, nitrophenyl derivatives, sulfur-containing heterocyclyl compounds, organometallic compounds, organophosphorus compounds, organochlorine compounds, inorganic active compounds, cyflufenamid, cymoxanil, dimethirimol, ethirimol, furalaxyl, metrafenone and spiroxamine, in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compound I with active compounds II, the use of the compound I with active compounds II for preparing such mixtures and compositions comprising these mixtures.
Abstract:
Substituted triazolopyrimidines of the formula I in which the substituents are as defined below: R 1 is alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, halocycloalkenyl, alkynyl, haloalkynyl or phenyl, naphthyl, or a five- or six-membered saturated, partially unsaturated or aromatic heterocycle comprising one to four heteroatoms from the group consisting of O, N and S, R 2 is hydrogen or a group R 1 , R 1 and R 2 together with the nitrogen atom, to which they are attached, may also form a five- or six-membered heterocyclyl or heteroaryl which is attached via N and which may comprise one to three further heteroatoms from the groups consisting of O, N and S as ring member and/or may be substituted according to the description; L is fluorine, chlorine or methyl; X is cyano, C 1 -C 4 -alkyl, C 1 -C 4 -alkoxy or C 1 -C 2 -haloalkoxy, where X is not methyl if R 1 and R 2 together are n-pentylene or 3-methyl-n-pentylene and L is fluorine, or R 1 and R 2 together are 3-methyl-n-pentylene and L is chlorine; processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi.