公开(公告)号：US6087542B1

公开(公告)日：2000-07-11

申请号：US14271597

申请日：1997-03-06

Applicant: BASF AG

Inventor： EICKEN KARL ,  GEBBARDT JOACHIM ,  RANG HARALD ,  RACK MICHAEL ,  SCHAEFER PETER

IPC: B01J31/24 ,  C07B37/04 ,  C07B61/00 ,  C07C201/12 ,  C07C205/06 ,  C07C205/11 ,  C07C205/12 ,  C07C205/35 ,  C07C253/30 ,  C07C205/00 ,  C07C43/00

CPC classification number: C07B37/04 ,  C07C201/12 ,  C07C253/30 ,  C07C205/11

公开(公告)号：JP2003206252A

公开(公告)日：2003-07-22

申请号：JP2002313232

申请日：2002-10-28

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  CARTER PAUL ,  CURTZE JUERGEN

IPC: A01N31/14 ,  A01N31/16 ,  A01N33/10 ,  A01N37/38 ,  A01N37/40 ,  C07B61/00 ,  C07C39/42 ,  C07C41/26 ,  C07C43/23 ,  C07C69/017 ,  C07C69/14 ,  C07C323/19 ,  C07C323/25

Abstract: PROBLEM TO BE SOLVED: To provide a benzhydryl derivative that exhibits high effect in the control of deleterious fungi. SOLUTION: The benzhydryl derivative is represented by formula I (wherein X is O or S; R 1 , R 3 are each a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkenyl, an alkynyl, an alkoxy, an alkenyloxy, an alkynyloxy, an alkyklcarbonyloxy, formyloxy or alkylthio or the like; R 2 is a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkoxy, a haloalkyl, or a haloalkoxy wherein in the case that n=2, R 2 may differ from each other; R 4 is an alkyl, an alkenyl or an alkynyl; R 5 and R 6 are each hydroxyl, an alkyl, an alkenyl, a haloalkyl, a haloalkenyl, an alkoxy or an alkenyloxy; m is 0, 1 or 2). COPYRIGHT: (C)2003,JPO

公开(公告)号：JP2003201289A

公开(公告)日：2003-07-18

申请号：JP2002272397

申请日：2002-09-19

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED

IPC: A01N43/16 ,  C07C45/46 ,  C07C45/54 ,  C07C49/84 ,  C07D311/86

Abstract: PROBLEM TO BE SOLVED: To provide a compound effective for controlling hazardous phytopathogenic fungi, to provide a method for producing the compound, to provide a composition containing the compound, and to provide a method for using the composition. SOLUTION: This compound comprises a xanthone derivative expressed by general formula (I) (n is 0, 1 or 2; R 1 is an alkyl or the like; R 2 and R 3 are each an alkoxy or the like, or together form an oxyalkyleneoxy which may be substituted; R 4 is a halogen or the like; R 5 is equal to the R 4 , provided that R 5 s may be different from each other when n is 2; and X and Y are each O or S). The method for producing the compound and the composition containing the compound are provided in the specification, respectively. The composition is used for controlling the hazardous phytopathogenic fungi. COPYRIGHT: (C)2003,JPO

公开(公告)号：JP2002030058A

公开(公告)日：2002-01-29

申请号：JP2001182539

申请日：2001-06-15

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N37/28 ,  A01N37/34 ,  A01N37/40 ,  A01N37/46 ,  A01N47/20 ,  A01N47/30 ,  C07B61/00 ,  C07C249/16 ,  C07C251/86 ,  C07C253/30 ,  C07C255/59 ,  C07C255/64 ,  C07C255/66 ,  C07C269/04 ,  C07C271/28 ,  C07C273/18 ,  C07C275/42

Abstract: PROBLEM TO BE SOLVED: To provide a compound improved in controlling actions on noxious fungi. SOLUTION: This salicylohydrazide derivative is represented by the formula I (wherein, X is a halogen, NO2, cyano, a 1-4C alkyl or a 1-4C alkoxy; (m) is 0, 1, 2 or 3; R1 is NO2, NH2 or NH-CO-A; A is hydrogen, 1-4C alkyl, a 1-4C alkoxy, NH2, NHCH3 or N(CH3)2; R2 is hydrogen, cyano, a 1-6C alkyl, a 2-6C alkeiyl, a 2-6C alkynyl, a 1-6C haloalkyl, a 1-6C alkoxy or a 1-6C alkylthio; and R3 is phenyl, naphthyl, a 3-10C cycloalkyl, a 5- or a 6-membered ring heteroaryl or a 5- or a 6-membered ring heterocyclyl). The method for producing the salicylohydrazide derivative is provided and an intermediate for producing the derivative is obtained. The composition for controlling the noxious fungi comprises the derivative.

公开(公告)号：WO0238565A3

公开(公告)日：2003-10-09

申请号：PCT/EP0112977

申请日：2001-11-09

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07B53/00 ,  C07C209/62 ,  C07C211/03 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: The invention relates to 7-(R) aminotriazolopyrimidines of formula (I), in which the substituents and index have the following definitions: R represents hydrogen or methyl; R represents methyl; R represents C2-C10 alkyl, C1-C4 alkoxymethyl, or C3-C10 cycloalkyl; R represents halogen, C1-C4 alkyl, C1-C4 haloalkyl or C1-C4 alkoxy; n represents a number between 1 and 5; Y represents halogen, cyano, C1-C4 alkyl or C1-C4 alkoxy; whereby * is a chirality centre with an R-configuration. The invention also relates to a method for producing said compounds, to agents containing the compounds and to the use thereof for combating harmful fungi.

Abstract translation: 7-（R）式（I）的-aminotriazolopyrimidine其中取代基和指数具有以下含义：R t <1>是氢或甲基; [R <2>是甲基; [R <3> C2-C10烷基，C1-C4烷氧基，C3-C10环烷基; [R <4>为卤素，C1-C4烷基，C1-C4卤代烷基或C1-C4烷氧基; n是从1到5的数; Y是卤素，氰基，C1-C4烷基或C1-C4烷氧基; 其中*是R构型的手性中心。 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO2005087770A3

公开(公告)日：2005-12-08

申请号：PCT/EP2005002424

申请日：2005-03-08

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD ,  HUENGER UDO

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  NIEDENBRUECK MATTHIAS ,  SCHERER MARIA ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD ,  HUENGER UDO

IPC: C07D487/04

CPC classification number: C07D487/04

Abstract: The invention relates to 5,6-dialkyl-7-amino-triazolopyrimidines of formula (I), in which the substituents are defined as follows: R represents alkyl, alkoxyalkyl, alkenyl or alkynyl; R represents alkyl, alkoxyalkyl, alkenyl or alkynyl, R and/or R being substituted according to the description. The invention also relates to a method for producing said compounds, to agents containing the latter and to their use for controlling plant-pathogenic fungi.

Abstract translation: 5,6-二烷基 - 7-氨基三唑并嘧啶，其中取代基具有式（I）的以下含义：R t <1>是烷基，烷氧基烷基，烯基或炔基; [R <2>是烷基，烷氧基烷基，烯基或炔基; 其中R <1>和/或R <2>取代根据描述; 一种用于制备这些化合物，含有它们和它们在防治植物病原性有害真菌的用途的组合物的过程。

公开(公告)号：WO2004041824A2

公开(公告)日：2004-05-21

申请号：PCT/EP0312276

申请日：2003-11-04

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07C69/65 ,  C07C69/76 ,  C07D487/04

CPC classification number: C07C69/65 ,  A01N43/90 ,  C07D487/04

Abstract: Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula (I) in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R and R radicals may be substituted as defined in the description, R denote hydrogen, or a group mentioned for R ; or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L , L independently denote hydrogen, halogen, or alkyl; L is hydrogen, halogen, haloalkyl, or NH2, NHR , or N(Rb)2, wherein Rb is as defined in the description,wherein at least one from L , L , and L is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 取代的式（I）的6-（2-卤代苯基） - 三唑并嘧啶，其中R1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元饱和，不饱和或 芳族杂环，其含有1-4个氮原子或一至三个氮原子和一个硫或氧原子，其中R 1和R 2基团可以如说明书中所定义地被取代，R 2表示氢，或 R 1中提到的基团; 或R 1和R 2连同相邻的氮原子表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环，该环可以被取代 如说明书中所定义的; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或N（R b）2，其中R b如说明书中所定义，其中至少一个L 1，L 2， 而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基，它们的制备方法，含有它们的组合物和它们用于防治植物病原性真菌的用途。

公开(公告)号：WO9502590A3

公开(公告)日：1995-06-01

申请号：PCT/EP9402264

申请日：1994-07-11

Applicant: BASF AG ,  SCHAEFER PETER ,  HAMPRECHT GERHARD ,  HEISTRACHER ELISABETH ,  KOENING HARTMANN ,  KLINTZ RALF ,  MUENSTER PETER ,  RANG HARALD ,  WESTPHALEN KARL OTTO ,  GERBER MATTHIAS ,  WALTER HELMUT

Inventor： SCHAEFER PETER ,  HAMPRECHT GERHARD ,  HEISTRACHER ELISABETH ,  KOENING HARTMANN ,  KLINTZ RALF ,  MUENSTER PETER ,  RANG HARALD ,  WESTPHALEN KARL-OTTO ,  GERBER MATTHIAS ,  WALTER HELMUT

IPC: A01N43/40 ,  A01N43/42 ,  A01N43/60 ,  A01N43/647 ,  A01N43/76 ,  A01N43/78 ,  A01N43/84 ,  A01N47/22 ,  C07D213/30 ,  C07D213/61 ,  C07D213/65 ,  C07D213/70 ,  C07D213/89 ,  C07D265/36 ,  C07D401/04 ,  C07D405/04 ,  C07D405/14 ,  C07D409/04 ,  C07D409/12 ,  C07D413/04 ,  C07D417/04

CPC classification number: C07D213/30 ,  C07D213/61 ,  C07D265/36 ,  C07D409/12

Abstract: A substituted 2-phenylpyridine of formula (I), where Ar is a radical (A) or (B) and where the ring R is a fused heterocyclic ring which, together with the phenyl ring, forms one of the following bicyclic rings (a) to (l) and the N-oxides of (I) and the agriculturally utilizable salts of (I) if these exist. Use: herbicides, desiccation/defoliation of plants.

公开(公告)号：WO9502580A3

公开(公告)日：1995-03-16

申请号：PCT/EP9402263

申请日：1994-07-11

Applicant: BASF AG ,  SCHAEFER PETER ,  HAMPRECHT GERHARD ,  HEISTRACHER ELISABETH ,  KOENIG HARTMANN ,  KLINTZ RALF ,  MUENSTER PETER ,  RANG HARALD ,  WESTPHALEN KARL OTTO ,  GERBER MATTHIAS ,  WALTER HELMUT

Inventor： SCHAEFER PETER ,  HAMPRECHT GERHARD ,  HEISTRACHER ELISABETH ,  KOENIG HARTMANN ,  KLINTZ RALF ,  MUENSTER PETER ,  RANG HARALD ,  WESTPHALEN KARL-OTTO ,  GERBER MATTHIAS ,  WALTER HELMUT

IPC: A01N43/40 ,  A01N43/42 ,  A01N43/60 ,  A01N43/647 ,  A01N43/76 ,  A01N43/78 ,  A01N43/84 ,  A01N47/22 ,  C07D213/30 ,  C07D213/61 ,  C07D213/65 ,  C07D213/70 ,  C07D213/89 ,  C07D265/36 ,  C07D401/04 ,  C07D405/04 ,  C07D405/14 ,  C07D409/04 ,  C07D409/12 ,  C07D413/04 ,  C07D417/04 ,  C07D213/68

CPC classification number: C07D213/30 ,  C07D213/61 ,  C07D265/36 ,  C07D409/12

Abstract: Substituted 2-phenylpyridines have formula (I) wherein R1, R3 = H, halogen, alkyl, haloalkyl, alkoxyalkyl, alkoxy, alkoxyalkoxy, OH, haloalkoxy, alkylcarbonyloxy, haloalkylcarbonyloxy, SH, alkylthio, alkylsulfinyl, alkylsulfonyl, haloalkylthio, haloalkylsulfinyl, haloalkylsulfonyl, CHO, CN, CO¿2?H, alkoxycarbonyl, alkoxyalkoxycarbonyl, haloalkoxycarbonyl, alkylcarbonyl, haloalkylcarbonyl, alkoxyalkylcarbonyl, CONH2, alkylaminocarbonyl, dialkylaminocarbonyl, pyrrolidinylcarbonyl, piperidylcarbonyl, morpholinylcarbonyl, NO2, NH2, alkylamino, dialkylamino, pyrrolidinyl, piperidinyl, morpholinyl, alkylcarbonylamino, haloalkylcarbonylamino, alkylsulfonylamino; R?2¿ = halogen, CN, NO¿2?, alkyl, haloalkyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio; or R?1 + R2 or R2 + R3¿ = trimethylene or tetramethylene chain; R4 = halogen, alkyl, haloalkyl, alkoxyalkyl, alkoxy, alkoxyalkoxy, OH, haloalkoxy, alkylcarbonyloxy, haloalkylcarbonyloxy, SH, alkylthio, alkylsulfinyl, alkylsulfonyl, haloalkylthio, haloalkylsulfinyl, haloalkylsulfonyl, CHO, CN, CO¿2?H, alkoxycarbonyl, alkoxyalkoxycarbonyl, haloalkoxycarbonyl, alkylcarbonyl, haloalkylcarbonyl, alkoxyalkylcarbonyl, NO2, NH2, alkylamino, dialkylamino, pyrrolidinyl, piperidinyl, morpholinyl, alkylcarbonylamino, haloalkylcarbonylamino, alkylsulfonylamino; R?5¿ = hydrogen or halogen; R6 = halogen, CN, NO¿2?, OH, CF3, C1-C6-alkyl, C1-C4-alkoxy; R?7¿ = various radicals; and the N-oxides of (I) and the agriculturally utilizable salts of (I) where these exist, excepting those compounds (I) where R2 is C1-C4-alkoxy and R1 and/or R3 is carboxyl or the salt, ester or amide thereof. Use: herbicides; desiccation/defoliation of plants.

公开(公告)号：WO2005113555A8

公开(公告)日：2006-12-14

申请号：PCT/EP2005005270

申请日：2005-05-13

Applicant: BASF AG ,  BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

Inventor： BLETTNER CARSTEN ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHWOEGLER ANJA ,  WAGNER OLIVER ,  SPEAKMAN JOHN-BRYAN ,  JABS THORSTEN ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  SCHERER MARIA ,  STIERL REINHARD

IPC: C07D487/04 ,  A01N43/90

CPC classification number: A01N43/90 ,  C07D487/04

Abstract: The invention relates to novel triazolopyrimidine compounds of general formula (I), to their use for controlling pathogenic fungi and to agricultural pesticides containing compounds of this type as active constituents. In formula (I), X, Y, L, m, Ar and A are defined as follows: X represents halogen, cyano, C 1 -C 4 alkyl, C 1 -C 4 haloalkyl, C 1 -C 4 alkoxy or C 1 -C 4 haloalkoxy; Y represents halogen, C 1 -C 4 alkyl or C 1 -C 4 haloalkyl; L represents independently of one another halogen, C 1 -C 6 alkyl, C 2 -C 6 alkenyl, C 1 -C 6 haloalkyl, C 1 -C 6 alkoxy, C 1 -C 6 haloalkoxy, nitro, amino, NHR, NR 2 , cyano, S(=O) n A 1 or C(=O)A 2 ; m represents 0, 1, 2, 3 or 4; A stands for a chemical bond or a CR 4 R 5 group; Ar represents phenyl or a 5- or 6-membered heteroaromatic group comprising 1, 2 or 3 heteroatoms selected from O, S and N as ring members, whereby the phenyl and the heteroaromatic group can comprise a fused benzole ring and can have 1, 2, 3, 4 or 5 R a substituents. R 1 to R 3 are defined as cited in claim 1.

Abstract translation: 本发明涉及如下通式的新型三唑并嘧啶化合物I和它们在防治有害真菌中的用途，以及植物保护剂，这样的化合物作为活性成分enthalten.In式I，X，Y，L，M，Ar和A具有下列含义：X 卤素，氰基，C _{1 -C 4 烷基，C 1 -C 4 卤代烷基，C < SUB> 1 -C 4 - 烷氧基或C 1 -C 4 卤代烷氧基; Y是卤素，C 1 -C 4 烷基或C 1 -C 4 卤代烷基; 独立地为卤素，C 1 -C 6 烷基，C 2 -C 6 烯基，C 1 -C ç 6 卤代烷基，C 1 -C 6 烷氧基，C 1 -C 6 < / SUB>卤代烷氧基，硝基，氨基，NHR，NR 2 ，氰基，S（= O）名词 A“或C（= O）A ^{2 ; m是0，1，2，3或4; A是一个化学键或基团CR 4 - [R 5 是; Ar是苯基或5-或6-元杂芳基具有1个，选自O，S和N的杂原子作为环成员，其中苯基和杂芳基可以具有一个稠合的苯环和1，2，3 2或3 ，4或5个取代基R 一可以包括;. R“至R 3 具有权利要求1中给出的含义。}}