公开(公告)号：US6410486B2

公开(公告)日：2002-06-25

申请号：US86752401

申请日：2001-05-31

Applicant: BASF AG

Inventor： WETTERICH FRANK ,  EICKEN KARL ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  ROSE INGO

IPC: A01N37/34 ,  C07C255/31 ,  C07C255/58 ,  C07C255/00

CPC classification number: C07C255/58 ,  A01N37/34 ,  C07C255/31 ,  C07C2601/02 ,  C07C2601/08

Abstract: The present invention relates to novel cycloalkylalkane-carboxamides of the formula Iwhere the substituents have the following meanings:A is C3-C6-cycloalkyl;R1 is C1-C6-alkyl or C2-C6-alkenyl;R2, R3 and R4 are hydrogen or, independently of this meaning, have one of the meanings of the radical R1;n is 0 or 1;Y is cyano or halogen;w is phenyl, naphthyl or heteroaryl.

Abstract translation: 本发明涉及式I的新的环烷基烷烃 - 甲酰胺，其中取代基具有以下含义：A为C 3 -C 6 - 环烷基; R 1为C 1 -C 6 - 烷基或C 2 -C 6 - 烯基; R 2，R 3和R 4为氢或 独立于该含义，具有基团R 1的含义之一; n为0或1; Y为氰基或卤素; w为苯基，萘基或杂芳基。

公开(公告)号：JP2002047262A

公开(公告)日：2002-02-12

申请号：JP2001207021

申请日：2001-07-06

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: C07C251/80 ,  A01N33/26 ,  A01N37/50 ,  C07C249/16 ,  C07C251/86

Abstract: PROBLEM TO BE SOLVED: To provide a compound that has increased controlling effect against harmful fungi. SOLUTION: The objective salicylic acid derivative is represented by formula I [wherein X is a halogen, NO2, cyano, an alkyl or an alkoxy; (m) is 0, 1, 2 or 3 where in the case m >=2, X may differ from each other; A is OH, an alkoxy, NH2, NHCH3 or N(CH3)2, R1 is phenyl, naphthyl, cycloalkyl, one to three N-atoms and/or one O or S atom or one or two O and/or S atoms- including 5-membered or 5-membered ring heteroaryl or 5-membered or 6-membered heterocyclyl where the ring structure may be unsubstituted or substituted; and R2 is H, cyano, an alkyl, an alkenyl, an alkynyl, a haloalkyl, an alkoxy or an alkylthio]. This invention further provides a method of producing the derivative, a composition including the derivative and the use of the composition for controlling harmful fungi.

公开(公告)号：JP2003206252A

公开(公告)日：2003-07-22

申请号：JP2002313232

申请日：2002-10-28

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  CARTER PAUL ,  CURTZE JUERGEN

IPC: A01N31/14 ,  A01N31/16 ,  A01N33/10 ,  A01N37/38 ,  A01N37/40 ,  C07B61/00 ,  C07C39/42 ,  C07C41/26 ,  C07C43/23 ,  C07C69/017 ,  C07C69/14 ,  C07C323/19 ,  C07C323/25

Abstract: PROBLEM TO BE SOLVED: To provide a benzhydryl derivative that exhibits high effect in the control of deleterious fungi. SOLUTION: The benzhydryl derivative is represented by formula I (wherein X is O or S; R 1 , R 3 are each a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkenyl, an alkynyl, an alkoxy, an alkenyloxy, an alkynyloxy, an alkyklcarbonyloxy, formyloxy or alkylthio or the like; R 2 is a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkoxy, a haloalkyl, or a haloalkoxy wherein in the case that n=2, R 2 may differ from each other; R 4 is an alkyl, an alkenyl or an alkynyl; R 5 and R 6 are each hydroxyl, an alkyl, an alkenyl, a haloalkyl, a haloalkenyl, an alkoxy or an alkenyloxy; m is 0, 1 or 2). COPYRIGHT: (C)2003,JPO

公开(公告)号：JP2003201289A

公开(公告)日：2003-07-18

申请号：JP2002272397

申请日：2002-09-19

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED

IPC: A01N43/16 ,  C07C45/46 ,  C07C45/54 ,  C07C49/84 ,  C07D311/86

Abstract: PROBLEM TO BE SOLVED: To provide a compound effective for controlling hazardous phytopathogenic fungi, to provide a method for producing the compound, to provide a composition containing the compound, and to provide a method for using the composition. SOLUTION: This compound comprises a xanthone derivative expressed by general formula (I) (n is 0, 1 or 2; R 1 is an alkyl or the like; R 2 and R 3 are each an alkoxy or the like, or together form an oxyalkyleneoxy which may be substituted; R 4 is a halogen or the like; R 5 is equal to the R 4 , provided that R 5 s may be different from each other when n is 2; and X and Y are each O or S). The method for producing the compound and the composition containing the compound are provided in the specification, respectively. The composition is used for controlling the hazardous phytopathogenic fungi. COPYRIGHT: (C)2003,JPO

公开(公告)号：JP2002030058A

公开(公告)日：2002-01-29

申请号：JP2001182539

申请日：2001-06-15

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N37/28 ,  A01N37/34 ,  A01N37/40 ,  A01N37/46 ,  A01N47/20 ,  A01N47/30 ,  C07B61/00 ,  C07C249/16 ,  C07C251/86 ,  C07C253/30 ,  C07C255/59 ,  C07C255/64 ,  C07C255/66 ,  C07C269/04 ,  C07C271/28 ,  C07C273/18 ,  C07C275/42

Abstract: PROBLEM TO BE SOLVED: To provide a compound improved in controlling actions on noxious fungi. SOLUTION: This salicylohydrazide derivative is represented by the formula I (wherein, X is a halogen, NO2, cyano, a 1-4C alkyl or a 1-4C alkoxy; (m) is 0, 1, 2 or 3; R1 is NO2, NH2 or NH-CO-A; A is hydrogen, 1-4C alkyl, a 1-4C alkoxy, NH2, NHCH3 or N(CH3)2; R2 is hydrogen, cyano, a 1-6C alkyl, a 2-6C alkeiyl, a 2-6C alkynyl, a 1-6C haloalkyl, a 1-6C alkoxy or a 1-6C alkylthio; and R3 is phenyl, naphthyl, a 3-10C cycloalkyl, a 5- or a 6-membered ring heteroaryl or a 5- or a 6-membered ring heterocyclyl). The method for producing the salicylohydrazide derivative is provided and an intermediate for producing the derivative is obtained. The composition for controlling the noxious fungi comprises the derivative.

公开(公告)号：WO03004465A2

公开(公告)日：2003-01-16

申请号：PCT/EP0207340

申请日：2002-07-03

Applicant: BASF AG ,  MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

Inventor： MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04 ,  C07D ,  A01N ,  C07C

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: Triazolopyrimidines of formula (I), wherein the index and substituents have the following meaning: n = 0 or a whole number of 1 - 5; R = halogen, cyano, hydroxy, cyanate, alkyl, alkenyl, alkinyl, halogenalkyl, halogenalkenyl, alkoxy, alkenyloxy, alkinyloxy, halogenalkoxy, cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkinyloxycarbonyl, aminocarbonyl, alkylaminocarbonyl, dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkinyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkinylcarbonyl, cycloalkylcarbonyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S; R = alkyl, alkenyl, alkinyl, cycloalkyl, cycloalkenyl, phenyl, naphthyl or a five to ten membered saturated, partially unsaturated or aromatic heterocycle, containing one to four heteroatoms from the group O, N or S, R and/or R being able to be substituted according to the description; R = alkyl, alkenyl or alkinyl which can be substituted by halogen, cyano, nitro, alkoxy or alkoxycarbonyl. The invention also relates to a method for the production of said compounds, agents containing same, and the use thereof in controlling noxious fungi.

Abstract translation: 式（I），其中所述索引和所述取代基具有以下含义的三唑并嘧啶：n是0或1〜5的整数; R是卤素，氰基，羟基，氰酸酯，烷基，烯基，炔基，卤代烷基，卤代烯基，烷氧基，链烯氧基，炔氧基，卤代烷氧基，环烷基，环烯基，环烷氧基，烷氧基羰基，烯氧基羰基，炔氧基羰基，氨基羰基，烷基氨基羰基，二烷基氨基羰，alkoximinoalkyl，Alkenyloximinocarbonyl，Alkinyloximinoalkyl 羰基，烯基，炔基羰基，环烷基羰基，或5至10元的饱和，其包含选自一至四个杂原子的部分不饱和或芳族杂环O，N或S; [R <1>是烷基，烯基，炔基，环烷基，环烯基，苯基，萘基，或5至10元饱和，部分不饱和或芳族，其包含从O型一至四个杂原子的杂环，N或S，其中R和/ 或者R 1可以如上所述被取代; [R <2>是烷基，烯基或炔基，可被卤素，氰基，硝基，烷氧基或烷氧羰基取代; 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO0162087A3

公开(公告)日：2002-02-14

申请号：PCT/EP0102059

申请日：2001-02-23

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  EICKEN KARL ,  ROSE INGO ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

Inventor： RHEINHEIMER JOACHIM ,  EICKEN KARL ,  ROSE INGO ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A01N37/32 ,  A01N37/36 ,  A01N37/38 ,  A01N41/02 ,  A01N41/10 ,  A01N43/36 ,  C07D207/50

CPC classification number: C07D207/50 ,  A01N37/32 ,  A01N37/36 ,  A01N37/38 ,  A01N41/02 ,  A01N41/10 ,  A01N43/36

Abstract: The invention relates to agrochemical compositions with a fungicidal action, containing compounds of formula (I) as their active agents. The radicals of said formula have the following meanings: R means hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-halogenalkylcarbonyl; R means halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halogen-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halogen-C1-C6-alkylsulfonyl, cyano or a radical NR R ; R -R mean hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halogen-C1-C6-alkyl, C1-C6-alkoxy, halogen-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halogen-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which can optionally be substituted by halogen atoms, C1-C6-alkyl or halogen-C1-C6-alkyl groups; R means hydrogen, C1-C6-alkyl; and R means C1-C6-alkyl, C1-C8-cycloalkyl or together with R and the nitrogen atom to which they are bonded, a saturated or unsaturated heterocyclic five or six-membered ring which has one or two heteroatoms selected from a group consisting of nitrogen atoms and oxygen atoms. The invention also relates to salts of said compositions which are suitable for agricultural use.

Abstract translation: 本发明的目的是具有包含（I），其中各基团具有以下含义的式作为活性成分的化合物的杀真菌作用的农药组合物，R <1>是氢，C1-C6烷基，C1-C6烷基羰基，甲酰基或C1-C6 卤代; [R <2>为卤素，C1-C6-烷硫基，C1-C6烷氧基，C3-C6环烷基-C1-C6-烷氧基，C1-C6烷氧基C1-C6烷基，卤代C1-C6烷氧基， C1-C6烷基磺酰基，C1-C6-烷基亚磺酰基，卤代C1-C6烷基磺酰基，氰基或基团NR <13> - [R <14>; [R <3> -R <12>为氢，卤素，C1-C8环烷基，C1-C6-烷基，卤代C1-C6烷基，C1-C6-烷氧基，卤代C1-C6烷氧基，C1-C6 烷基磺酰基，卤代C1-C6烷基磺酰基，甲酰基，C1-C6烷基羰基，氰基，C1-C6烷硫基或苯基，其是任选地被卤素原子，C1-C6烷基或烷基 - 卤素-C 1 -C 6 - 取代的 基团可被取代，R <13>为氢，C1-C6烷基，R <14> C1-C6-烷基，C1-C8环烷基，或一起为R <13>和的氮原子它们所连接形成其 意味着饱和或ungesätttigten杂环五元或含有从包含氮原子或氧原子，和它们的可农用可用的盐的组中选择的一个或两个杂原子的六元环。

公开(公告)号：WO0012465A3

公开(公告)日：2000-06-22

申请号：PCT/EP9906251

申请日：1999-08-26

Applicant: BASF AG ,  ROSE INGO ,  WETTERICH FRANK ,  EICKEN KARL ,  RHEINHEIMER JOACHIM ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  STRATHMANN SIEGFRIED

Inventor： ROSE INGO ,  WETTERICH FRANK ,  EICKEN KARL ,  RHEINHEIMER JOACHIM ,  LORENZ GISELA ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  STRATHMANN SIEGFRIED

IPC: C07C233/61 ,  A01N25/02 ,  A01N25/08 ,  A01N37/18 ,  A01N53/00 ,  A01N53/12 ,  C07C233/58 ,  C07C255/48 ,  C07C271/24

CPC classification number: A01N53/00 ,  C07C233/58 ,  C07C255/48 ,  C07C271/24 ,  C07C2601/02

Abstract: The invention relates to novel cycloalkylalkane carboxylic acid amides of the general formula (I), as well as salts thereof which are suitable for use in agriculture, in which the substituents have the following meanings: A is C3-C6 cycloalkyl which can carry one or more substituents; Alk is straight-chain or branched C1-C6-alkylene; R is C1-C6-alkyl or C2-C6-alkenyl, which can carry one or more substituents; R , R are hydrogen, C1-C6-alkyl or C2-C6-alkenyl, which rests can be partly or fully halogenated; and W is a fused bicyclic ring system with six ring atoms each. The invention also relates to fungicidal agents containing a compound of formula (I) as plant protectant.

Abstract translation: 本发明涉及新的cycloalkylalkanecarboxamides通式（I），其中取代基具有以下含义：A，C 3 -C 6环烷基，其可带有一个或多个取代基; ALK的直链或支链C1-C6亚烷基; [R <1>，C1-C6烷基或C2-C6链烯基，其可以带有一个或nehrere取代基; [R <2>，R <3>为氢，C1-C6烷基或C2-C6链烯基，其中这些基团可以部分或完全被卤代; 具有六个环原子W，稠合的双环环系; 及其可农用可用的盐。 此外，本发明涉及包含式（I）的化合物用作植物保护剂的杀真菌组合物。

公开(公告)号：WO0238565A3

公开(公告)日：2003-10-09

申请号：PCT/EP0112977

申请日：2001-11-09

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07B53/00 ,  C07C209/62 ,  C07C211/03 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: The invention relates to 7-(R) aminotriazolopyrimidines of formula (I), in which the substituents and index have the following definitions: R represents hydrogen or methyl; R represents methyl; R represents C2-C10 alkyl, C1-C4 alkoxymethyl, or C3-C10 cycloalkyl; R represents halogen, C1-C4 alkyl, C1-C4 haloalkyl or C1-C4 alkoxy; n represents a number between 1 and 5; Y represents halogen, cyano, C1-C4 alkyl or C1-C4 alkoxy; whereby * is a chirality centre with an R-configuration. The invention also relates to a method for producing said compounds, to agents containing the compounds and to the use thereof for combating harmful fungi.

Abstract translation: 7-（R）式（I）的-aminotriazolopyrimidine其中取代基和指数具有以下含义：R t <1>是氢或甲基; [R <2>是甲基; [R <3> C2-C10烷基，C1-C4烷氧基，C3-C10环烷基; [R <4>为卤素，C1-C4烷基，C1-C4卤代烷基或C1-C4烷氧基; n是从1到5的数; Y是卤素，氰基，C1-C4烷基或C1-C4烷氧基; 其中*是R构型的手性中心。 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO0130154A3

公开(公告)日：2002-04-11

申请号：PCT/EP0010468

申请日：2000-10-24

Applicant: BASF AG ,  RHEINHEIMER JOACHIM ,  EICKEN KARL ,  ROSE INGO ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

Inventor： RHEINHEIMER JOACHIM ,  EICKEN KARL ,  ROSE INGO ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A01N43/56

CPC classification number: A01N43/56

Abstract: The invention relates to agrochemical compositions with a fungicidal action, containing compounds of formula (I) as their active agents, the radicals having the following meanings: R is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, C1-C4-alkoxy-C1-C6-alkyl, C1-C6-halogenalkyl, C3-C6-alkenyl, C3-C6-halogenalkenyl or phenyl-C1-C6-alkyl, wherein the phenyl group can be substituted by C1-C6-alkyl, halogen or C1-C6-halogenalkyl; R is hydrogen, C1-C6-alkyl, C1-C6-halogenalkyl, C1-C6-alkoxy, C1-C6-halogenalkoxy or halogen; R is phenyl that is optionally substituted by halogen, C1-C6-alkyl, C1-C6-halogenalkyl, C1-C6-alkoxy, C1-C6-halogenalkoxy, C1-C6-alkylthio, C1-C6-alkylsulfonyl, C1-C6-halogenalkylsulfonyl; and R is a heterocyclic radical with one or two nitrogen atoms - said heterocyclic radical can be substituted by halogen, C1-C6-alkyl or C1-C6-halogenalkyl. The invention also relates to methods for combating harmful fungi on plants using this fungicidal agent.

Abstract translation: 本发明涉及具有含有（I），其中各基团具有以下含义的式作为活性成分的化合物的杀真菌活性农业化学组合物，R <1>是氢，C1-C6烷基，C1-C6烷基羰基，C1-C4烷氧基 -C1-C6-烷基，C1-C6卤代烷基，C3-C6烯基，C3-C6卤代链烯基或苯基-C 1 -C 6 - 烷基，其中，由C1-C6烷基，卤素或C 1 -C 6卤代烷基的苯基 可以被取代; [R <2>是氢，C1-C6烷基，C1-C6卤代烷基，C1-C6-烷氧基，C1-C6卤代烷氧基或卤素; [R <3>是其任选地被卤素取代的，C1-C6-烷基，C1-C6卤代烷基，C1-C6-烷氧基，C1-C6卤代烷氧基，C1-C6-烷硫基，C1-C6-烷基磺酰基，C1苯基 C6卤代烷基磺酰基; [R <4>杂环基团具有一个或两个氮原子，其中杂环部分可以被卤素，C1-C6烷基或C1-C6卤代烷基。 此外，本发明提供用于在植物中防治有害真菌涉及使用这些杀真菌剂的方法。