公开(公告)号：JP2002047262A

公开(公告)日：2002-02-12

申请号：JP2001207021

申请日：2001-07-06

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: C07C251/80 ,  A01N33/26 ,  A01N37/50 ,  C07C249/16 ,  C07C251/86

Abstract: PROBLEM TO BE SOLVED: To provide a compound that has increased controlling effect against harmful fungi. SOLUTION: The objective salicylic acid derivative is represented by formula I [wherein X is a halogen, NO2, cyano, an alkyl or an alkoxy; (m) is 0, 1, 2 or 3 where in the case m >=2, X may differ from each other; A is OH, an alkoxy, NH2, NHCH3 or N(CH3)2, R1 is phenyl, naphthyl, cycloalkyl, one to three N-atoms and/or one O or S atom or one or two O and/or S atoms- including 5-membered or 5-membered ring heteroaryl or 5-membered or 6-membered heterocyclyl where the ring structure may be unsubstituted or substituted; and R2 is H, cyano, an alkyl, an alkenyl, an alkynyl, a haloalkyl, an alkoxy or an alkylthio]. This invention further provides a method of producing the derivative, a composition including the derivative and the use of the composition for controlling harmful fungi.

公开(公告)号：JP2003206252A

公开(公告)日：2003-07-22

申请号：JP2002313232

申请日：2002-10-28

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  CARTER PAUL ,  CURTZE JUERGEN

IPC: A01N31/14 ,  A01N31/16 ,  A01N33/10 ,  A01N37/38 ,  A01N37/40 ,  C07B61/00 ,  C07C39/42 ,  C07C41/26 ,  C07C43/23 ,  C07C69/017 ,  C07C69/14 ,  C07C323/19 ,  C07C323/25

Abstract: PROBLEM TO BE SOLVED: To provide a benzhydryl derivative that exhibits high effect in the control of deleterious fungi. SOLUTION: The benzhydryl derivative is represented by formula I (wherein X is O or S; R 1 , R 3 are each a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkenyl, an alkynyl, an alkoxy, an alkenyloxy, an alkynyloxy, an alkyklcarbonyloxy, formyloxy or alkylthio or the like; R 2 is a halogen, cyano, nitro, hydroxyl, mercapto, an amino, an alkyl, an alkoxy, a haloalkyl, or a haloalkoxy wherein in the case that n=2, R 2 may differ from each other; R 4 is an alkyl, an alkenyl or an alkynyl; R 5 and R 6 are each hydroxyl, an alkyl, an alkenyl, a haloalkyl, a haloalkenyl, an alkoxy or an alkenyloxy; m is 0, 1 or 2). COPYRIGHT: (C)2003,JPO

公开(公告)号：JPH11335361A

公开(公告)日：1999-12-07

申请号：JP2568099

申请日：1999-02-03

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  SAUTER HUBERT ,  BAYER HERBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GOETZ ROLAND ,  MUELLER BERND ,  PTOCK ARNE ,  ROEHL FRANZ ,  HARRIES VOLKER ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED

IPC: A01N43/653 ,  A01N43/76 ,  C07C271/10 ,  C07D249/12 ,  C07D263/44 ,  C07D403/12 ,  C07D413/12

Abstract: PROBLEM TO BE SOLVED: To obtain the subject new compound useful for controlling harmful animals and harmful fungi. SOLUTION: This compound is shown by formula I Y is a halogen, a 1-4C alkyl or the like; (n) is 0-2; E is a group of formula II (V is O or the like); T is O or oxymethylene; Z is a group X [X is a (substituted) heterocyclyl, a (substituted) aryl or the like], N=CWR [W is a (substituted) 1-6C alkyl or the like; R is H, cyano or the like] or the like} such as N-methyl-5-[2-(o-tolyloxymethylene)phenyl]-1,3- oxazolidine-2,4-dione.The compound of formula I, for example, in the case in which it is a compound of formula III, is obtained by a process for acylating an alkyl α- hydroxy-α-phenylacetate with phosgene or the like to give a compound of formula IV and further reacting the compound with a primary amine of the formula H2 N-R αto cause a ring formation and in the case of not advancing the ring formation by the strength of the amine, by a process for hydrolyzing an ester amide of formula V, then treating the resultant substance with an acid and reacting the treated substance with a compound of the formula Z-OH.

公开(公告)号：JP2003201289A

公开(公告)日：2003-07-18

申请号：JP2002272397

申请日：2002-09-19

Applicant: BASF AG

Inventor： ROSE INGO ,  BLASCO JORDI TORMO I ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  GROTE THOMAS ,  GYPSER ANDREAS ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED

IPC: A01N43/16 ,  C07C45/46 ,  C07C45/54 ,  C07C49/84 ,  C07D311/86

Abstract: PROBLEM TO BE SOLVED: To provide a compound effective for controlling hazardous phytopathogenic fungi, to provide a method for producing the compound, to provide a composition containing the compound, and to provide a method for using the composition. SOLUTION: This compound comprises a xanthone derivative expressed by general formula (I) (n is 0, 1 or 2; R 1 is an alkyl or the like; R 2 and R 3 are each an alkoxy or the like, or together form an oxyalkyleneoxy which may be substituted; R 4 is a halogen or the like; R 5 is equal to the R 4 , provided that R 5 s may be different from each other when n is 2; and X and Y are each O or S). The method for producing the compound and the composition containing the compound are provided in the specification, respectively. The composition is used for controlling the hazardous phytopathogenic fungi. COPYRIGHT: (C)2003,JPO

公开(公告)号：JP2002030058A

公开(公告)日：2002-01-29

申请号：JP2001182539

申请日：2001-06-15

Applicant: BASF AG

Inventor： GYPSER ANDREAS ,  GROTE THOMAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  MUELLER BERND ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N37/28 ,  A01N37/34 ,  A01N37/40 ,  A01N37/46 ,  A01N47/20 ,  A01N47/30 ,  C07B61/00 ,  C07C249/16 ,  C07C251/86 ,  C07C253/30 ,  C07C255/59 ,  C07C255/64 ,  C07C255/66 ,  C07C269/04 ,  C07C271/28 ,  C07C273/18 ,  C07C275/42

Abstract: PROBLEM TO BE SOLVED: To provide a compound improved in controlling actions on noxious fungi. SOLUTION: This salicylohydrazide derivative is represented by the formula I (wherein, X is a halogen, NO2, cyano, a 1-4C alkyl or a 1-4C alkoxy; (m) is 0, 1, 2 or 3; R1 is NO2, NH2 or NH-CO-A; A is hydrogen, 1-4C alkyl, a 1-4C alkoxy, NH2, NHCH3 or N(CH3)2; R2 is hydrogen, cyano, a 1-6C alkyl, a 2-6C alkeiyl, a 2-6C alkynyl, a 1-6C haloalkyl, a 1-6C alkoxy or a 1-6C alkylthio; and R3 is phenyl, naphthyl, a 3-10C cycloalkyl, a 5- or a 6-membered ring heteroaryl or a 5- or a 6-membered ring heterocyclyl). The method for producing the salicylohydrazide derivative is provided and an intermediate for producing the derivative is obtained. The composition for controlling the noxious fungi comprises the derivative.

公开(公告)号：JP2001226339A

公开(公告)日：2001-08-21

申请号：JP2001008676

申请日：2001-01-17

Applicant: BASF AG

Inventor： GRAMMENOS WASSILOS DR ,  SAUTER HUBERT DR ,  GYPSER ANDREAS ,  GEWEHR MARKUS DR ,  TORMO I BLASCO JORDI ,  PTOCK ARNE DR ,  MUELLER BERND DR ,  CULLMANN OLIVER DR ,  GROTE THOMAS DR ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED DR ,  LORENZ GISELA

IPC: A01N37/50 ,  B27K3/38 ,  B27K3/40 ,  C07C249/08 ,  C07C251/48

Abstract: PROBLEM TO BE SOLVED: To obtain a compound having enhanced activity as a crop-protecting agent. SOLUTION: This iminoxy-substituted benzyl phenyl ether is expressed by formula I [wherein Y expresses H or the like; Q expresses C(= NOCH3)-CONHCH3 or the like; X expresses a 1-4C alkyl; m expresses 1 or 2; R1 expresses an alkyl; R2 expresses H or the like; R3 expresses an alkyl or the like and R4 expresses an alkyl, an alkenyl, an alkynyl or the like].

公开(公告)号：WO2004041824A2

公开(公告)日：2004-05-21

申请号：PCT/EP0312276

申请日：2003-11-04

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  BLETTNER CARSTEN ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  SCHWOEGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  SCHOEFL ULRICH ,  STIERL REINHARD

IPC: A01N43/90 ,  C07C69/65 ,  C07C69/76 ,  C07D487/04

CPC classification number: C07C69/65 ,  A01N43/90 ,  C07D487/04

Abstract: Substituted 6-(2-halogenphenyl)-triazolopyrimidines of formula (I) in which R1 denote alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or a 5- or 6-membered saturated, unsaturated, or aromatic heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, wherein R and R radicals may be substituted as defined in the description, R denote hydrogen, or a group mentioned for R ; or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocycle, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which ring may be substituted as defined in the description; Hal is halogen; L , L independently denote hydrogen, halogen, or alkyl; L is hydrogen, halogen, haloalkyl, or NH2, NHR , or N(Rb)2, wherein Rb is as defined in the description,wherein at least one from L , L , and L is not hydrogen; X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

Abstract translation: 取代的式（I）的6-（2-卤代苯基） - 三唑并嘧啶，其中R1表示烷基，烯基，炔基，链二烯基，卤代烷基，卤代烯基，环烷基，苯基，萘基或5-或6-元饱和，不饱和或 芳族杂环，其含有1-4个氮原子或一至三个氮原子和一个硫或氧原子，其中R 1和R 2基团可以如说明书中所定义地被取代，R 2表示氢，或 R 1中提到的基团; 或R 1和R 2连同相邻的氮原子表示含有1-4个氮原子或1-3个氮原子和一个硫或氧原子的5-或6-元杂环，该环可以被取代 如说明书中所定义的; 卤素是卤素; L 1，L 3独立地表示氢，卤素或烷基; L 2是氢，卤素，卤代烷基或NH 2，NHR b或N（R b）2，其中R b如说明书中所定义，其中至少一个L 1，L 2， 而L 3不是氢; X是卤素，氰基，烷基，烷氧基，卤代烷氧基或烯氧基，它们的制备方法，含有它们的组合物和它们用于防治植物病原性真菌的用途。

公开(公告)号：WO9959982A3

公开(公告)日：2000-03-16

申请号：PCT/EP9903003

申请日：1999-05-04

Applicant: BASF AG ,  BAYER HERBERT ,  GOETZ ROLAND ,  KEIL MICHAEL ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  HARRIES VOLKER

Inventor： BAYER HERBERT ,  GOETZ ROLAND ,  KEIL MICHAEL ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GYPSER ANDREAS ,  MUELLER BERND ,  PTOCK ARNE ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  HARRIES VOLKER

IPC: C07C251/38 ,  A01N37/40 ,  C07C49/303 ,  C07C251/42 ,  C07C251/50 ,  C07C251/52 ,  C07C251/60 ,  A01N37/50 ,  C07C49/35

CPC classification number: C07C251/60 ,  C07C2601/14

Abstract: The invention relates to bisoximether derivatives of formula (I) in which the variables have the following meanings: R represents halogen, C1-C4 alkyl, C1-C4 alkyl halide, C1-C4 alkoxy or C1-C4 alkoxy halide; n is 1 to 5, whereby the radicals R can be different if n is not equal to 1; R represents C1-C4 alkyl, C3-C6 alkenyl or C3-C6 alkynyl, whereby these groups can be partially or completely halogenated; Q represents C(=CHOCH3)-COOCH3, C(=CHCH3)-COOCH3, C(=NOCH3)-COOCH3 or C(=NOCH3)-CONHCH3. The invention also relates to the salts of the bisoximether derivatives, to methods and intermediate products for the production of these compounds and to their use for combating animal pests and fungicidal pests.

Abstract translation: 式（I），其中各变量具有以下含义的双肟醚衍生物，R <1>为卤素，C1-C4烷基，C1-C4卤代烷基，C1-C4烷氧基或C1-C4卤代烷氧基; n为1至5，其中基团可以是与R <1>不同的，当n不为1; [R <2> C1-C4烷基，C3-C6链烯基或C3-C6炔基，其中这些基团可以部分或完全被卤代; Q为C（= CHOCH 3）-COOCH 3，C（= CHCH 3）-COOCH 3，C（= NOCH 3）-COOCH 3或C（= NOCH 3）-CONHCH 3; 和它们的盐，方法和中间体制备这些化合物和它们用于控制动物害虫和有害真菌中的用途。

公开(公告)号：WO0238565A3

公开(公告)日：2003-10-09

申请号：PCT/EP0112977

申请日：2001-11-09

Applicant: BASF AG ,  TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

Inventor： TORMO I BLASCO JORDI ,  DITRICH KLAUS ,  SAUTER HUBERT ,  CULLMANN OLIVER ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MUELLER BERND ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07B53/00 ,  C07C209/62 ,  C07C211/03 ,  C07D487/04

CPC classification number: C07D487/04 ,  A01N43/90

Abstract: The invention relates to 7-(R) aminotriazolopyrimidines of formula (I), in which the substituents and index have the following definitions: R represents hydrogen or methyl; R represents methyl; R represents C2-C10 alkyl, C1-C4 alkoxymethyl, or C3-C10 cycloalkyl; R represents halogen, C1-C4 alkyl, C1-C4 haloalkyl or C1-C4 alkoxy; n represents a number between 1 and 5; Y represents halogen, cyano, C1-C4 alkyl or C1-C4 alkoxy; whereby * is a chirality centre with an R-configuration. The invention also relates to a method for producing said compounds, to agents containing the compounds and to the use thereof for combating harmful fungi.

Abstract translation: 7-（R）式（I）的-aminotriazolopyrimidine其中取代基和指数具有以下含义：R t <1>是氢或甲基; [R <2>是甲基; [R <3> C2-C10烷基，C1-C4烷氧基，C3-C10环烷基; [R <4>为卤素，C1-C4烷基，C1-C4卤代烷基或C1-C4烷氧基; n是从1到5的数; Y是卤素，氰基，C1-C4烷基或C1-C4烷氧基; 其中*是R构型的手性中心。 一种用于制备这些化合物，含有它们以及它们在防治有害真菌中的用途的组合物的过程。

公开(公告)号：WO9940082A3

公开(公告)日：1999-10-21

申请号：PCT/EP9900470

申请日：1999-01-26

Applicant: BASF AG ,  PTOCK ARNE ,  SAUTER HUBERT ,  KIRSTGEN REINHARD ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  BAYER HERBERT ,  GEWEHR MARKUS ,  CULLMANN OLIVER ,  MUELLER BERND ,  GOETZ ROLAND ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  HARRIES VOLKER ,  STRATHMANN SIEGFRIED

Inventor： PTOCK ARNE ,  SAUTER HUBERT ,  KIRSTGEN REINHARD ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  BAYER HERBERT ,  GEWEHR MARKUS ,  CULLMANN OLIVER ,  MUELLER BERND ,  GOETZ ROLAND ,  ROEHL FRANZ ,  AMMERMANN EBERHARD ,  LORENZ GISELA ,  HARRIES VOLKER ,  STRATHMANN SIEGFRIED

IPC: A01N43/56 ,  C07D401/12 ,  C07D401/14 ,  A01N43/48

CPC classification number: C07D401/12 ,  A01N43/56

Abstract: The present invention relates to compounds of the general formula (I) and to the salts thereof, wherein the substituents and the n index have the following values: Q represents -C(=CHCH3)-COOCH3, -C(=CHOCH3)-COOCH3, -C(=NOCH3)-COOCH3 or -C(=NOCH3)-CONH(CH3); R represents hydrogen, halogen, C1-C4 alkyl, C1-C2 halogenalkyl, C1-C4 alkoxy or C1-C2 halogenalkoxy; R represents halogen, C1-C4 alkyl, C1-C2 halogenalkyl or C1-C4 alkoxy; n is 0, 1 or 2, wherein the R substituents can be different when n = 2; and R represents phenyl, pyridyle or pyrimidyle. This invention also relates to agents containing these compounds as well as to the use of said compounds (I) and agents against noxious fungi and animal parasites.

Abstract translation: 通式（I）和它们的盐，其中取代基和指数n具有以下含义的化合物：Q是-C（= CHCH 3）-COOCH 3，-C（= CHOCH 3）-COOCH 3，C（= NOCH 3） - COOCH 3或-C（= NOCH 3）-CONH（CH 3）; R 1是氢，卤素，C 1 -C 4烷基，C 1 -C 2卤代烷基，C 1 -C 4烷氧基或C 1 -C 2卤代烷氧基; R 2是卤素，C 1 -C 4烷基，C 1 -C 2卤代烷基，C 1 -C 4烷氧基; n是0,1或2，其中当n = 2时取代基R 2可以不同; R 3苯基，吡啶基或嘧啶基，含有它们的试剂以及化合物（I）和防治有害真菌和动物害虫的试剂的用途。