公开(公告)号：SI1414302T1

公开(公告)日：2007-08-31

申请号：SI200230527

申请日：2002-07-16

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD ,  KRUMMEL GUNTER

IPC: A01N43/90 ,  A01N43/00 ,  C07D487/00 ,  C07D487/04

公开(公告)号：DE50209786D1

公开(公告)日：2007-05-03

申请号：DE50209786

申请日：2002-07-16

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD ,  KRUMMEL GUENTER

IPC: A01N43/90 ,  C07D487/04

Abstract: The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R 1 , R 2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R 1 and R 2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R 3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R 3 and R 2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by R a . The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.

公开(公告)号：AT357142T

公开(公告)日：2007-04-15

申请号：AT02790165

申请日：2002-07-16

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD ,  KRUMMEL GUENTER

IPC: A01N43/90 ,  C07D487/04

Abstract: The invention relates to 7-amino triazolopyrimidines of formula (I), in which the substituents have the following meanings: R 1 , R 2 represent hydrogen, alkyl, alkenyl, alkynyl, cycloalkyl, phenyl, naphthyl; or 5-membered or 6-membered heterocyclyl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; or 5-membered or 6-membered heteroaryl containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or R 1 and R 2 can, together with the nitrogen atom, which binds them, form a 5-membered or 6-membered ring containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom; R 3 represents alkyl, alkenyl, alkynyl, cycloalkyl, phenylalkyl and alkyl halide; whereby R 3 and R 2 can be unsubstituted or partially or completely substituted according to the description; X represents halogen, cyano, alkoxy, alkyl halide, phenyl or phenyl that is substituted by R a . The invention also relates to methods and intermediate products for producing said compounds, to agents containing the same, and to their use.

公开(公告)号：AT353901T

公开(公告)日：2007-03-15

申请号：AT02758297

申请日：2002-07-03

Applicant: BASF AG

Inventor： MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  TORMO I BLASCO JORDI ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

Abstract: 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines (I) are new. 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines of formula (I) are new. [Image] n : 0-5; R : halo, CN, OH or OCN, or alkyl, alkenyl, alkynyl, T', haloalkenyl, OT, alkenyloxy, alkynyloxy, OT', cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, CONH 2, mono- or dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); T : 1-6C alkyl; T' : 1-6C haloalkyl; Het : 5-10 membered, saturated, partially unsaturated or aromatic heterocycle containing 1-4 of O, N and/or S heteroatoms; R 11-10C alkyl, alkenyl, alkynyl, 3-12C cycloalkyl, 3-10C cycloalkenyl, phenyl, naphthyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); R ahalo, CN, NO 2, OH, T, T', COT, cycloalkyl, OT, OT', COOT, NHT, NT 2, 2-6C alkenyl, 2-6C alkenyloxy, 3-6C alkynyloxy, alkoximino, alkenyloximino, alkynyloximino, aralkoximino, alkynyl, alkynyloxycarbonyl, phenyl, naphthyl or Het (where all aliphatic, alicyclic or aromatic groups are optionally partially or completely halogenated and optionally substituted by 1-3 R aand/or 1-3 R c); R bhalo, CN, NO 2, OH, SH, NH 2, COOH, CONH 2, CSNH 2, T, T', 2-8C alkenyl, 2-8C alkenyloxy, 2-8C alkynyloxy, OT, OT', ST, NHT, NT 2, CHO, COT, SO 2T, SOT, COOT, OCOT, CONHT, CONT 2, CSNHT or CSNT 2; R ccycloalkyl, -O-cycloalkyl, heterocyclyl, -O-heterocyclyl, aryl, -O-aryl, -S-aryl, -O-T-aryl, -T-aryl, heteroaryl, -O-heteroaryl or -S-heteroaryl (where cycloalkyl or heterocyclyl rings are 3-10 membered, aryl rings are preferably 6-10 membered and heteroaryl rings are preferably 5-6 membered; and all rings are optionally partially or completely halogenated and optionally substituted by alkyl or haloalkyl); and R 21-4C alkyl, 2-4C alkynyl or 2-4C alkynyl (all optionally substituted by halo, CN, NO 2, OMe, OEt or 1-4C alkoxycarbonyl; Unless specified otherwise alkyl moieties have 1-8C, alkenyl or alkynyl moieties 2-10C and cycloalkyl or cycloalkenyl moieties 3-6C. Independent claims are also included for: (1) preparation of (I); and (2) dicarbonyl compound intermediates of formula (III), provided that n is not 0 and R 1and R 2are not both Me. [Image] ACTIVITY : Fungicide. 7-Cyclohexyl-5-methyl-6-(2-chloro-6-fluorophenyl)-1,2,4-triazolo[1,5-a]pyrimidine (Ia) at a concentration of 63 ppm gave at least 90 % protection of tomato plants against Alternaria solani. MECHANISM OF ACTION : None given.

公开(公告)号：AU2002302359B2

公开(公告)日：2006-12-21

申请号：AU2002302359

申请日：2002-01-17

Applicant: BASF AG

Inventor： ROSE INGO ,  STIERL REINHARD ,  LORENZ GISELA ,  SCHERER MARIA ,  AMMERMANN EBERHARD ,  HADEN EGON ,  EICKEN KARL ,  SCHELBERGER KLAUS ,  STRATHMANN SIEGFRIED

IPC: A01N35/04 ,  A01N25/02 ,  A01N25/08 ,  A01N37/52 ,  A01N43/08 ,  A01N43/10 ,  A01N43/36 ,  A01N43/50 ,  A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/78

Abstract: Fungicidal mixtures, comprising a) benzophenones of the formula I in which R is chlorine, methyl, methoxy, acetoxy, pivaloyloxy or hydroxyl; R is chlorine or methyl; R is hydrogen, halogen or methyl; and R is C1-C6-alkyl or benzyl, where the phenyl moiety of the benzyl radical may carry a halogen or methyl substituent, and b) oxime ether derivatives of the formula II where the substituents X to X and Y to Y are as defined in the description; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II and compositions comprising them are described.

公开(公告)号：AU2002229712B2

公开(公告)日：2006-12-21

申请号：AU2002229712

申请日：2002-01-17

Applicant: BASF AG

Inventor： SCHERER MARIA ,  LORENZ GISELA ,  EICKEN KARL ,  HAMPEL MANFRED ,  SCHELBERGERD KLAUS ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  ROSE INGO ,  STIERL REINHARD ,  HADEN EGON

IPC: C07C49/84 ,  A01N35/04 ,  A01N37/06 ,  A01N43/40 ,  C07C69/157

Abstract: Fungicidal mixtures, comprising a) benzophenones of the formula I, in which R 1 is chlorine, methyl, methoxy, acetoxy, pivaloyloxy or hydroxyl; R 2 is chlorine or methyl; R 3 is hydrogen, halogen or methyl; and R 4 is C 1 -C 6 -alkyl or benzyl, where the phenyl moiety of the benzyl radical may carry a halogen or methyl substituent, and b) amide compounds of the formula II in which R 6 and R 7 are halogen nitro, cyano, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, haloalkynyl, alkoxy, haloalkoxy, alkylthio, haloalkylthio, alkylsulfinyl or alkylsulfonyl; x is 1, 2, 3 or 4; and y is 1, 2, 3, 4 or 5; in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II and compositions comprising them are described.

公开(公告)号：NZ533265A

公开(公告)日：2006-05-26

申请号：NZ53326502

申请日：2002-11-15

Applicant: BASF AG

Inventor： GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  MULLER BERND ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD ,  GYPSER ANDREAS ,  GROTE THOMAS ,  SCHWOGLER ANJA ,  RHEINHEIMER JOACHIM ,  SCHIEWECK FRANK ,  TORMO I BLASCO JORDI ,  ROSE INGO ,  SCHAFER PETER

IPC: A01N43/54 ,  C07D239/42 ,  C07D239/46 ,  C07D239/47 ,  C07D239/48 ,  C07D239/52 ,  C07D401/06 ,  C07D401/14 ,  C07D403/12

Abstract: Disclosed are 5-phenylpyrimidine compounds of formula (I), wherein: R1 and R2 are independently H, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, alkynyl or haloalkynyl, R1 and R2 together may form an optionally substituted five or six membered ring optionally interrupted by an ether, thio, sulfoxyl or sulfenyl group, R3 is H, halo, cyano, alkyl, haloalkyl, alkoxy, haloalkoxy or alkenyloxy, and the remaining substituents are defined herein. The compounds are used as in fungicidal compositions for controlling phytopathogenic fungi.

公开(公告)号：DE50203896D1

公开(公告)日：2005-09-15

申请号：DE50203896

申请日：2002-05-17

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  GYPSER ANDREAS ,  ROSE INGO ,  GROTE THOMAS ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A01N43/86 ,  A01N43/90 ,  C07D265/24 ,  C07D498/04 ,  C07D513/04

Abstract: Oxazin(ethi)one compounds of the formula I: in which the variables Z, R 1 , R 2 , R 3 and n are as defined in claim 1 and A is a 5- or 6-membered carbocycle or a 5- or 6-membered heterocycle having 1, 2 or 3 heteroatoms selected from the group consisting of N, O and S, each of which cycles is attached via two carbon atoms to the oxazin(ethi)one ring, and the agriculturally useful salts of the oxazin(ethi)one compounds I are described. Moreover, the invention describes the use of compounds I and their salts for controlling phytopathogenic fungi, compositions which comprise the compounds I and/or their salts in a fungicidally effective amount and a method for controlling phytopathogenic fungi which comprises treating the fungi or the materials, plants, seeds or the soil threatened by fungal attack with a fungicidally effective amount of at least one compound of the formula I as claimed in claim 1 and/or a salt of I.

公开(公告)号：NZ531065A

公开(公告)日：2005-04-29

申请号：NZ53106502

申请日：2002-07-08

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04 ,  C07D249/00 ,  C07D239/00

Abstract: Disclosed are 6-(2-tolyl)-triazolopyrimidines of formula I, wherein: R1 and R2 are independently H, alkyl, alkenyl, alkynyl, alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, heterocyclyl, or heteroaryl, and are optionally substituted, R1 and R2 may together form an optionally substituted heterocyclic ring, R3 is halogen, cyano, alkyl, alkoxy, haloalkyl or C(=O)A, n is from 1 to 4, and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkneyloxy. The compounds are used in a method for controlling phytopathogenic fungi, comprising treating the fungi, materials, plants, soil or seed with an effective amount of the compounds.

公开(公告)号：ZA200401256B

公开(公告)日：2005-03-10

申请号：ZA200401256

申请日：2004-02-17

Applicant: BASF AG

Inventor： AMMERMANN EBERHARD ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  LORENZ GISELA ,  MUELLER BERND ,  RACK MICHAEL ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SAUTER HUBERT ,  SCHIEWECK FRANK ,  SCHAEFER PETER ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  BLASCO JORDI TORMO I

IPC: A01N43/90 ,  C07D487/04 ,  C07D ,  A01N

Abstract: Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.