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公开(公告)号:PL367615A1
公开(公告)日:2005-03-07
申请号:PL36761502
申请日:2002-07-08
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , SAUTER HUBERT , MULLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAFER PETER , SCHIEWECK FRANK , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC: A01N25/04 , A01N43/90 , C07D487/04
Abstract: 6-(2,6-Difluoro-phenyl)-triazolopyrimidines of formula (I), in which R and R independently denote hydrogen or Alkyl, Alkyl, Alkenyl, Alkynyl, or alkadienyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulphur or oxygen atom. Or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulphur or xygen atom where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered hetericyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulphur or oxygen atom, which may be substituted; X is halogen, cyano, alkoxy, haloalkoxy or alkenyloxy; Processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.
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公开(公告)号:PT1353554E
公开(公告)日:2004-11-30
申请号:PT02710012
申请日:2002-01-17
Applicant: BASF AG
Inventor: LORENZ GISELA , STRATHMANN SIEGFRIED , LEYENDECKER JOACHIM , SCHERER MARIA , AMMERMANN EBERHARD , SCHELBERGER KLAUS , HADEN EGON , MULLER BERND , ROSE INGO , STIERL REINHARD
IPC: A01N35/04 , A01N43/653 , A01N47/24
Abstract: Fungicidal mixtures comprising a) a benzophenone of the formula I, b) a carbamate of the formula II, and c) an azole derivative of the formula III in a synergistically effective amount, and a method for controlling harmful fungi using mixtures of the compounds I, II and III are described. The active compounds of the formulae I, II and III are defined in the description.
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公开(公告)号:AT279110T
公开(公告)日:2004-10-15
申请号:AT01919332
申请日:2001-02-23
Applicant: BASF AG
Inventor: RHEINHEIMER JOACHIM , EICKEN KARL , ROSE INGO , GROTE THOMAS , AMMERMANN EBERHARD , SPEAKMAN JOHN-BRYAN , STRATHMANN SIEGFRIED , LORENZ GISELA
Abstract: Agrochemical compositions having fungicidal action and comprising as active compounds compounds of the formula IwhereR1 is hydrogen, C1-C6-alkyl, C1-C6-alkylcarbonyl, formyl or C1-C6-haloalkylcarbonyl;R2 is halogen, C1-C6-alkylthio, C1-C6-alkoxy, C3-C6-cycloalkyl-C1-C6-alkoxy, C1-C6-alkoxy-C1-C6-alkyl, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, C1-C6-alkylsulfinyl, halo-C1-C6-alkylsulfonyl, cyano or a radical NR13R14;R3-R12 are hydrogen, halogen, C1-C8-cycloalkyl, C1-C6-alkyl, halo-C1-C6-alkyl, C1-C6-alkoxy, halo-C1-C6-alkoxy, C1-C6-alkylsulfonyl, halo-C1-C6-alkylsulfonyl, formyl, C1-C6-alkylcarbonyl, cyano, C1-C6-alkylthio or phenyl, which may be unsubstituted or substituted by halogen, C1-C6-alkyl or halo-C1-C6-alkyl,R13 is hydrogen, C1-C6-alkyl,R14 is C1-C6-alkyl, C1-C8-cycloalkyl or, together with R13 and the nitrogen atom to which they are attached, a saturated or unsaturated heterocyclic five- or six-membered ring which contains one or two heteroatoms selected from the group consisting of nitrogen and oxygen,and their agriculturally useful salts are described.
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公开(公告)号:DE60201089D1
公开(公告)日:2004-09-30
申请号:DE60201089
申请日:2002-04-06
Applicant: BASF AG
Inventor: TORMO I BLASCO JORDI , SAUTER HUBERT , MUELLER BERND , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAEFER PETER , SCHIEWECK FRANK , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC: A01N25/02 , A01N25/08 , A01N43/90 , C07D487/04
Abstract: 6-(2-Chloro-6-fluoro-phenyl)-triazolopyrimidines of formula (I), in which R 1 and R 2 independently denote hydrogen or alkyl, alkenyl, alkynyl, alkadienyl, or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R 1 and R 2 radicals may be unsubstituted or partially or fully halogenated or may be substituted as defined in the description. R 1 and R 2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; X is cyano, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi
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公开(公告)号:HU0400210A2
公开(公告)日:2004-08-30
申请号:HU0400210
申请日:2002-03-13
Applicant: BASF AG
Inventor: AMMERMANN EBERHARD , GEWEHR MARKUS , GROTE THOMAS , GYPSER ANDREAS , LORENZ GISELA , MUELLER BERND , RHEINHEIMER JOACHIM , ROSE INGO , SAUTER HUBERT , SCHIEWECK FRANK , SCHAEFER PETER , STIERL REINHARD , STRATHMANN SIEGFRIED , TORMO I BLASCO JORDI
IPC: A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/647 , A01N43/653 , A01N43/713 , A01N43/90 , C07D239/42 , C07D401/14 , C07D403/04 , C07D471/04 , C07D473/06 , C07D487/04 , C07D521/00
Abstract: 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.
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公开(公告)号:BR0211180A
公开(公告)日:2004-08-10
申请号:BR0211180
申请日:2002-07-08
Applicant: BASF AG
Inventor: BLASCO JORDI TORMO I , SAUTER HUBERT , LLER BERND M , GEWEHR MARKUS , GRAMMENOS WASSILIOS , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHOFER PETER , SCHIEWECK FRANK , RACK MICHAEL , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC: A01N43/90 , C07D487/04
Abstract: Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.
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公开(公告)号:BR0210858A
公开(公告)日:2004-06-29
申请号:BR0210858
申请日:2002-07-03
Applicant: BASF AG
Inventor: MUELLER BERND , SAUTER HUBERT , GEWEHR MARKUS , GRAMMENOS WASSILIOS , BLASCO JORDI TORMO I , GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHOFER PETER , SCHIEWECK FRANK , RACK MICHAEL , LORENZ GISELA , STRATHMANN SIEGFRIED , AMMERMANN EBERHARD , STIERL REINHARD
IPC: A01N43/90 , C07D487/04 , A01N43/653
Abstract: 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines (I) are new. 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines of formula (I) are new. [Image] n : 0-5; R : halo, CN, OH or OCN, or alkyl, alkenyl, alkynyl, T', haloalkenyl, OT, alkenyloxy, alkynyloxy, OT', cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, CONH 2, mono- or dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); T : 1-6C alkyl; T' : 1-6C haloalkyl; Het : 5-10 membered, saturated, partially unsaturated or aromatic heterocycle containing 1-4 of O, N and/or S heteroatoms; R 11-10C alkyl, alkenyl, alkynyl, 3-12C cycloalkyl, 3-10C cycloalkenyl, phenyl, naphthyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); R ahalo, CN, NO 2, OH, T, T', COT, cycloalkyl, OT, OT', COOT, NHT, NT 2, 2-6C alkenyl, 2-6C alkenyloxy, 3-6C alkynyloxy, alkoximino, alkenyloximino, alkynyloximino, aralkoximino, alkynyl, alkynyloxycarbonyl, phenyl, naphthyl or Het (where all aliphatic, alicyclic or aromatic groups are optionally partially or completely halogenated and optionally substituted by 1-3 R aand/or 1-3 R c); R bhalo, CN, NO 2, OH, SH, NH 2, COOH, CONH 2, CSNH 2, T, T', 2-8C alkenyl, 2-8C alkenyloxy, 2-8C alkynyloxy, OT, OT', ST, NHT, NT 2, CHO, COT, SO 2T, SOT, COOT, OCOT, CONHT, CONT 2, CSNHT or CSNT 2; R ccycloalkyl, -O-cycloalkyl, heterocyclyl, -O-heterocyclyl, aryl, -O-aryl, -S-aryl, -O-T-aryl, -T-aryl, heteroaryl, -O-heteroaryl or -S-heteroaryl (where cycloalkyl or heterocyclyl rings are 3-10 membered, aryl rings are preferably 6-10 membered and heteroaryl rings are preferably 5-6 membered; and all rings are optionally partially or completely halogenated and optionally substituted by alkyl or haloalkyl); and R 21-4C alkyl, 2-4C alkynyl or 2-4C alkynyl (all optionally substituted by halo, CN, NO 2, OMe, OEt or 1-4C alkoxycarbonyl; Unless specified otherwise alkyl moieties have 1-8C, alkenyl or alkynyl moieties 2-10C and cycloalkyl or cycloalkenyl moieties 3-6C. Independent claims are also included for: (1) preparation of (I); and (2) dicarbonyl compound intermediates of formula (III), provided that n is not 0 and R 1and R 2are not both Me. [Image] ACTIVITY : Fungicide. 7-Cyclohexyl-5-methyl-6-(2-chloro-6-fluorophenyl)-1,2,4-triazolo[1,5-a]pyrimidine (Ia) at a concentration of 63 ppm gave at least 90 % protection of tomato plants against Alternaria solani. MECHANISM OF ACTION : None given.
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公开(公告)号:BR0209835A
公开(公告)日:2004-06-15
申请号:BR0209835
申请日:2002-05-17
Applicant: BASF AG
Inventor: RHEINHEIMER JOACHIM , GYPSER ANDREAS , ROSE INGO , GROTE THOMAS , SCHOFER PETER , SCHIEWECK FRANK , AMMERMANN EBERHARD , SPEAKMAN JOHN-BRYAN , STRATHMANN SIEGFRIED , LORENZ GISELA
IPC: A01N43/86 , A01N43/90 , C07D265/24 , C07D498/04 , C07D513/04
Abstract: Oxazin(ethi)one compounds of the formula I: in which the variables Z, R 1 , R 2 , R 3 and n are as defined in claim 1 and A is a 5- or 6-membered carbocycle or a 5- or 6-membered heterocycle having 1, 2 or 3 heteroatoms selected from the group consisting of N, O and S, each of which cycles is attached via two carbon atoms to the oxazin(ethi)one ring, and the agriculturally useful salts of the oxazin(ethi)one compounds I are described. Moreover, the invention describes the use of compounds I and their salts for controlling phytopathogenic fungi, compositions which comprise the compounds I and/or their salts in a fungicidally effective amount and a method for controlling phytopathogenic fungi which comprises treating the fungi or the materials, plants, seeds or the soil threatened by fungal attack with a fungicidally effective amount of at least one compound of the formula I as claimed in claim 1 and/or a salt of I.
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公开(公告)号:BR0207975A
公开(公告)日:2004-06-15
申请号:BR0207975
申请日:2002-03-13
Applicant: BASF AG
Inventor: GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHOFER PETER , SCHIEWECK FRANK , SAUTER HUBERT , GEWEHR MARKUS , MUELLER BERND , BLASCO JORDI TORMO I , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC: A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/647 , A01N43/653 , A01N43/713 , A01N43/90 , C07D239/42 , C07D401/14 , C07D403/04 , C07D471/04 , C07D473/06 , C07D487/04 , C07D521/00 , C07D473/00
Abstract: 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.
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公开(公告)号:SK11422003A3
公开(公告)日:2004-04-06
申请号:SK11422003
申请日:2002-03-13
Applicant: BASF AG
Inventor: GROTE THOMAS , GYPSER ANDREAS , RHEINHEIMER JOACHIM , ROSE INGO , SCHAFER PETER , SCHIEWECK FRANK , SAUTER HUBERT , GEWEHR MARKUS , MULLER BERND , TORMO I BLASCO JORDI , AMMERMANN EBERHARD , STRATHMANN SIEGFRIED , LORENZ GISELA , STIERL REINHARD
IPC: A01N43/54 , A01N43/56 , A01N43/58 , A01N43/60 , A01N43/64 , A01N43/647 , A01N43/653 , A01N43/713 , A01N43/90 , C07D239/42 , C07D401/14 , C07D403/04 , C07D471/04 , C07D473/06 , C07D487/04 , C07D521/00 , C07D473/00
Abstract: 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.
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