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公开(公告)号:NO822313L
公开(公告)日:1983-01-03
申请号:NO822313
申请日:1982-07-01
Applicant: CIBA GEIGY AG
Inventor: MEYER ALFRED , NYFELER ROBERT , STURM ELMAR , MUELLER URS
IPC: A01N43/50 , A01N43/653 , C07D303/22 , C07D303/34 , C07D521/00 , C07D , A01N
Abstract: Novel 2-hydroxy-3-azolylpropane derivatives of the general formula I wherein R1 is an azolyl group, R2 is C1-C4alkyl or an aryl group which is unsubstituted or substituted by halogen, cyano, C1-C3alkyl, C1-C3alkoxy, nitro, thiocyano, C1-C3alkylthio and/or C1-C3haloalkyl, R3 and R4, each independently of the other, are hydrogen or C1-C4alkyl, R5 is an unsubstituted or mono- or polysubstituted radical selected from C1-C8alkyl, C3-C8cycloalkyl, C3-C6alkenyl, C3-C6alkynyl and aralkyl, said substituents being selected from the group consisting of halogen, cyano, C1-C3alkyl, C1-C5alkoxy, C1-C5haloalkoxy, C1-C3alkylthio, C1-C3haloalkyl, C1-C3haloalkylthio, nitro and/or thiocyano; and X is oxygen or sulfur, and the acid addition salts, quaternary azolium salts and metal complexes thereof, are useful in controlling phytopathogenic microorganisms and/or of regulating plant growth.
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公开(公告)号:AU5030879A
公开(公告)日:1980-03-06
申请号:AU5030879
申请日:1979-08-27
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , SCHEMPP HEINRICH , MARTIN HENRY
IPC: A01N25/32 , C07C67/00 , C07C313/00 , C07C317/28 , C07C317/44 , C07C317/48 , C07C323/12 , C07C325/00 , C07C327/58 , C07C327/60 , C07D307/40 , C07D307/56 , C07D307/68 , C07D333/38 , C07C147/06 , A01N5/00 , A01N9/12 , A01N9/14 , C07C147/14 , C07C149/415
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公开(公告)号:CA994782A
公开(公告)日:1976-08-10
申请号:CA133492
申请日:1972-01-31
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , CELLARIUS HANS-JOERG , VON BREDOW BRIGITTA , VOGEL CHRISTIAN
IPC: A01N47/16 , A01P13/00 , C07D221/04
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公开(公告)号:AU607993B2
公开(公告)日:1991-03-21
申请号:AU1550488
申请日:1988-05-02
Applicant: CIBA GEIGY AG
Inventor: NYFELER ROBERT , ZONDLER HELMUT , STURM ELMAR
IPC: C07D249/08 , A01N31/04 , A01N31/14 , A01N43/64 , A01N43/653 , B01J27/10 , B01J31/10 , B01J31/22 , C07B61/00 , C07C20060101 , C07C33/20 , C07C41/00 , C07C41/03 , C07C43/13 , C07C43/178 , C07C43/23 , C07C43/295 , C07C43/315 , C07C67/00 , C07C201/00 , C07C201/12 , C07C205/34 , C07C253/00 , C07C253/30 , C07C255/54 , C07D253/00 , C07D521/00
Abstract: Essentially, a process is described for the preparation of the 1-triazolylethyl ether derivatives, defined in claim 1, of the general formula I (I) which consists in (a) reacting an oxirane of the formula II (II) at temperatures of -20 DEG to +100 DEG C., in the presence of an acid catalyst or an acid condensation agent, with an alcohol of the formula III R3-OH (III) to give a glycol monoether of the formula IV (IV) and (b) subsequently reacting the glycol monoether of the formula IV or one of its esters, in the presence of an acid-binding agent or condensation agent, at temperatures of 0 DEG to 150 DEG C., with a triazole of the formula V (V) the substituents R1, R2 ; amd R3 in the formula II to IV being as defined under formula I and M in formula V being hydrogen or a metal atom. The novel compounds within the scope of formula I and their use are also described.
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公开(公告)号:AU603417B2
公开(公告)日:1990-11-15
申请号:AU1075288
申请日:1988-01-22
Applicant: CIBA GEIGY AG
Inventor: MEYER ALFRED , STURM ELMAR
IPC: A01N43/50 , A01N43/653 , A01P3/00 , C07C39/00 , C07C45/63 , C07C45/71 , C07D233/60 , C07D233/64 , C07D249/08 , C07D303/08 , C07D303/22 , C07D303/34 , C07D521/00 , A61K31/335
Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.
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公开(公告)号:PH24423A
公开(公告)日:1990-06-25
申请号:PH33405
申请日:1986-02-11
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , GALLAY JEAN JAQUES , KRISTINSSON HAUKUR , PISSIOTAS GEORG
IPC: C07D263/58 , A61K31/496 , A61K31/515 , A61P33/10 , C07D233/70 , C07D235/26 , C07D239/62 , C07D239/66 , C07D249/08 , C07D249/12 , C07D263/34 , C07D271/06 , C07D271/10 , C07D271/113 , C07D277/24 , C07D277/34 , C07D277/58 , C07D277/68 , C07D285/08 , C07D285/12 , C07D285/13 , C07D403/12 , C07D413/12 , C07D417/12
Abstract: The invention relates to novel 5-(azolyloxyphenylcarbamoyl)barbituric acid derivatives of the general formula I (I) wherein X is oxygen or sulfur; R1 is C1-C6alkyl, C1-C6alkoxy, C3-C6cycloalkyl or allyl; R2 is C1-C6alkyl or allyl; R3 is an unsubstituted or substituted five-membered azole ring which is bound through carbon and is selected from the group consisting of benzimadazole, benzoxazole, benzothiazole, imidazole, oxazole, thiazole, oxadiazole, thiadiazole and triazole; and R4 and R5 are each independently of the other hydrogen, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; and to the tautomers and salts thereof, as anthelmintic compounds. Together with suitable carriers and further assistants, these compounds may be used in particular for controlling helminths which are parasites of animals.
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157.
公开(公告)号:HU196978B
公开(公告)日:1989-02-28
申请号:HU433483
申请日:1983-12-13
Applicant: CIBA GEIGY AG
Inventor: STURM ELMAR , MEYER ALFRED
IPC: A01N43/50 , A01N43/653 , A01P3/00 , C07C39/00 , C07C45/63 , C07C45/71 , C07D233/60 , C07D233/64 , C07D249/08 , C07D303/08 , C07D303/22 , C07D303/34 , C07D521/00 , A01N43/20
Abstract: 1-Azolyl-2-aryl-3-fluoro-alkan-2- ols of the general formula I in which Az is 1H-1,2,4-triazole, 4H-1,2,4-triazole or 1H-imidazole; Ar is an unsubstituted or substituted aromatic radical from the series comprising phenyl, biphenyl, phenoxyphenyl and naphthyl; R1 is hydrogen, C1-C4-alkyl, C3-C5-alkenyl or benzyl; R2 is hydrogen, fluorine or C1-C6-alkyl and R3 is hydrogen, fluorine, C1-C6-alkyl, C1-C6-haloalkyl, C1-C6-alkoxy, C1-C6-alkylthio, phenyl, phenoxy, phenylthio or C3-C7-cycloalkyl, and each aromatic substituent or aromatic moiety of a substituent is unsubstituted or mono- or poly-substituted by halogen, C1-C4-alkyl, C1-C4-alkoxy, C1-C4-haloalkyl, nitro and/or cyano; including the acid addition salts, quaternary azolium salts and metal complexes, are useful for controlling phytopathogenic microorganisms.
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公开(公告)号:AU570653B2
公开(公告)日:1988-03-24
申请号:AU2158183
申请日:1983-11-22
Applicant: CIBA GEIGY AG
Inventor: KUNZ WALTER , STURM ELMAR
IPC: A01N43/50 , A01N43/653 , A61K31/4164 , A61K31/4196 , A61P31/10 , C07C45/61 , C07C45/68 , C07C45/71 , C07D233/60 , C07D249/08 , C07D303/22 , C07D303/32 , C07D405/06 , C07D407/04 , C07D407/06 , C07D521/00 , A01N43/64
Abstract: Novel 1-carbonyl-1-phenoxyphenyl-2-azolylethanol derivatives of the general formula I wherein R1 and R2 are each independently hydrogen, halogen C1-C4 alkyl or CF3, and Rn denotes one to three alkyl, alkoxy, haloalkoxy, haloalkyl, halogen and/or cyano groups, R4 is hydrogen, C1-C10 alkyl, C3-C6 cycloalkyl or unsubstituted or substituted phenyl, X is -CH= or -N=, R5 is hydrogen, C1-C12 alkyl, C2-C4 alkenyl, C2-C4 alkynyl, or unsubstituted or substituted benzyl; and A is the radical wherein R6 and R7 are each independently C1-C12 alkyl, unsubstituted or substituted phenyl, or both together form a C2-C4 alkylene bridge which is unsubstituted or substituted by one or more identical or different members selected from the group consisting of C1-C4 alkyl, C2-C4 alkenyloxymethyl or C1-C3 alkoxymethyl; and to the acid addition salts, quaternary azolium salts and metal complexes thereof, are useful for controlling phytopathogenic microorganisms and/or regulating plant growth.
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公开(公告)号:PH21667A
公开(公告)日:1988-01-13
申请号:PH32973
申请日:1985-10-25
Applicant: CIBA GEIGY AG
Inventor: NYFELER ROBERT , ZONDLER HELMUT , STURM ELMAR
IPC: A01N31/04 , A01N31/14 , C07D249/08 , A01N43/64 , A01N43/653 , B01J27/10 , B01J31/10 , B01J31/22 , C07B61/00 , C07C20060101 , C07C33/20 , C07C41/00 , C07C41/03 , C07C43/13 , C07C43/178 , C07C43/23 , C07C43/295 , C07C43/315 , C07C67/00 , C07C201/00 , C07C201/12 , C07C205/34 , C07C253/00 , C07C253/30 , C07C255/54 , C07D253/00 , C07D521/00
Abstract: Essentially, a process is described for the preparation of the 1-triazolylethyl ether derivatives, defined in claim 1, of the general formula I (I) which consists in (a) reacting an oxirane of the formula II (II) at temperatures of -20 DEG to +100 DEG C., in the presence of an acid catalyst or an acid condensation agent, with an alcohol of the formula III R3-OH (III) to give a glycol monoether of the formula IV (IV) and (b) subsequently reacting the glycol monoether of the formula IV or one of its esters, in the presence of an acid-binding agent or condensation agent, at temperatures of 0 DEG to 150 DEG C., with a triazole of the formula V (V) the substituents R1, R2 ; amd R3 in the formula II to IV being as defined under formula I and M in formula V being hydrogen or a metal atom. The novel compounds within the scope of formula I and their use are also described.
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公开(公告)号:MX154686A
公开(公告)日:1987-11-25
申请号:MX636382
申请日:1982-04-14
Applicant: CIBA GEIGY AG
Inventor: FANKHAUSER ERNST , STURM ELMAR
IPC: A01N41/10 , C07C147/06
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