-
11.
公开(公告)号:WO2014045263A3
公开(公告)日:2014-05-15
申请号:PCT/IB2013058808
申请日:2013-09-24
Applicant: REDDYS LAB LTD DR
Inventor: IQBAL JAVED , DAHANUKAR VILAS HARESHWAR , ORUGANTI SRINIVAS , KANDAGATLA BHASKAR , KUNHIMON SYAM KUMAR UNNIARAN , SAGYAM RAJESHWAR REDDY , IRENI BABU , KONDEPUDI VEERA VENKATA SATYANARAYANA MURTHY , MUTTAVARAPU MURALI MOHAN , BUCCHIKONDA RAVINDER , GANGIREDDY RAJENDAR REDDY
IPC: C07D209/52 , C07C205/28 , C07C217/14 , C07D317/16 , C07D317/28
CPC classification number: C07D209/52 , C07B2200/07 , C07C35/06 , C07C43/315 , C07C215/20 , C07C217/44 , C07C223/02 , C07C255/46 , C07C271/16 , C07C271/18 , C07C309/66 , C07C2601/08 , C07D317/18 , C07D317/28 , C07F7/1856 , C07K5/0202 , C07K5/1024
Abstract: Provided are novel processes for preparation of (1S, 3aR, 6aS)-octahydrocyclopenta[c]pyrrole-1-carboxylic acid and its derivatives; land their use in preparation of Telaprevir.
Abstract translation: 提供(1S,3aR,6aS) - 八氢环戊二烯并[c]吡咯-1-羧酸及其衍生物的制备方法; 将其用于制备特拉匹韦尔。
-
12.IMPROVED PROCESS FOR PREPARATION OF SAXAGLIPTIN AND ITS SALTS 审中-公开
Title translation: 改进萨伐他汀及其盐的制备方法公开(公告)号:WO2013175395A3
公开(公告)日:2014-01-30
申请号:PCT/IB2013054167
申请日:2013-05-21
Applicant: REDDYS LAB LTD DR
Inventor: VARANASI GANESH , MACHARLA PRABHAKAR , VEMPATI CHANDRASEKHAR , BANDICHHOR RAKESHWAR , DAHANUKAR VILAS HARESHWAR , IQBAL JAVED , ORUGANTI SRINIVAS , RAPOLU RAJESH KUMAR , NARIYAM MUNASWAMY SEKHAR , NETI SRINIVASAN
IPC: C07D209/02 , A61K31/403 , C07C13/615 , C07D209/52
CPC classification number: C07D209/52
Abstract: Improved processes for preparing saxagliptin or its salt and intermediates thereof are provided.
Abstract translation: 提供了制备沙格列汀或其盐及其中间体的改进方法。
-
13.TRIAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM 审中-公开
Title translation: 三唑化合物作为抗菌剂和含有它们的药物组合物公开(公告)号:WO2005082892A3
公开(公告)日:2006-03-23
申请号:PCT/IB2005000343
申请日:2005-02-11
Applicant: REDDYS LAB LTD DR , DAS JAGATTARAN , TAKHI MOHAMED , NATESAN SELVAKUMAR , TREHAN SANJAY , IQBAL JAVED , MAGADI SITARAM KUMAR , KANDEPU SREENIVAS
Inventor: DAS JAGATTARAN , TAKHI MOHAMED , NATESAN SELVAKUMAR , TREHAN SANJAY , IQBAL JAVED , MAGADI SITARAM KUMAR , KANDEPU SREENIVAS
IPC: C07D249/06 , C07D401/10 , C07D401/14 , C07D403/00 , C07D403/06 , C07D403/12 , C07D405/12 , C07D405/14 , C07D413/12
CPC classification number: C07D403/06 , C07D249/06 , C07D401/10 , C07D401/14 , C07D403/12 , C07D405/12 , C07D405/14 , C07D413/12
Abstract: The present invention relates to novel triazole compounds of formula (I), where all symbols are as defined in the detailed description; their pharmaceutically acceptable salts their stereosiomers thereof, their prodrugs, their rotamers, their pharmaceutical compositions containing them. The present invention also relates to a process for the preparation of the above said novel compounds.
Abstract translation: 本发明涉及新的式(I)三唑化合物,其中所有符号如详细描述中所定义; 其药学上可接受的盐,它们的立体异构体,它们的前药,它们的旋转异构体,它们含有它们的药物组合物。 本发明还涉及制备上述新化合物的方法。
-
公开(公告)号:WO2013190509A2
公开(公告)日:2013-12-27
申请号:PCT/IB2013055096
申请日:2013-06-21
Applicant: REDDYS LAB LTD DR
Inventor: NARIYAM SEKHAR MUNASWAMY , BHALERAO DINESH SHIVAJI , DAHANUKAR VILAS HARESHWAR , ORUGANTI SRINIVAS , RAPOLU RAJESH KUMAR , KANDAGATLA BHASKAR , IQBAL JAVED , KHOBARE SANDIP RAMDAS , KALLAM SRINIVASA REDDY , BANDA MALAVIKA , GARARE VIKAS SADASHIV , EDA VISHNUVARDHANA VEMA REDDY
CPC classification number: A61K38/06 , A61K38/55 , C07K5/0808
Abstract: The present application relates to processes for preparing intermediates of Boceprevir and their use in preparation of Boceprevir or its pharmaceutically acceptable salts thereof.
Abstract translation: 本申请涉及制备波普瑞韦中间体的方法及其在制备波普瑞韦或其药学上可接受的盐中的用途。
-
公开(公告)号:WO2012146980A3
公开(公告)日:2012-12-27
申请号:PCT/IB2012000922
申请日:2012-04-27
Applicant: REDDYS LAB LTD DR , KATKAM SRINIVAS , SAGYAM RAJESWAR REDDY , MORTHALA RAGHAVENDAR RAO , IRENI BABU , VINIGARI KRISHNA , RAMDOSS SURESH KUMAR , RANGINENI SRINIVASULU , TUMMALA ARJUNKUMAR , IQBAL JAVED , ORUGANTI SRINIVAS , KANDAGATLA BHASKAR
Inventor: KATKAM SRINIVAS , SAGYAM RAJESWAR REDDY , MORTHALA RAGHAVENDAR RAO , IRENI BABU , VINIGARI KRISHNA , RAMDOSS SURESH KUMAR , RANGINENI SRINIVASULU , TUMMALA ARJUNKUMAR , IQBAL JAVED , ORUGANTI SRINIVAS , KANDAGATLA BHASKAR
IPC: C07C211/00 , C07D333/20
CPC classification number: C07C205/45 , C07C201/10 , C07C201/12 , C07C213/00 , C07C213/02 , C07C213/10 , C07C215/28 , C07C205/04
Abstract: The present application provide processes for the preparation of fingolimod and its pharmaceutically acceptable salts, process for the purification of fingolimod hydrochloride and process for the preparation of amorphous fingolimod hydrochloride.
Abstract translation: 本申请提供了芬戈莫德及其药学上可接受的盐的制备方法,盐酸芬戈莫德的纯化方法和用于制备无定形芬戈莫德盐酸盐的方法。
-
公开(公告)号:WO2005035528A3
公开(公告)日:2005-06-02
申请号:PCT/IB2004003360
申请日:2004-10-14
Applicant: REDDYS LAB LTD DR , NATESAN SELVAKUMAR , DAS JAGATTARAN , TAKHI MOHAMED , TREHAN SANJAY , IQBAL JAVED , MAGADI SITARAM KUMAR , KANDEPU SREENIVAS
Inventor: NATESAN SELVAKUMAR , DAS JAGATTARAN , TAKHI MOHAMED , TREHAN SANJAY , IQBAL JAVED , MAGADI SITARAM KUMAR , KANDEPU SREENIVAS
IPC: A61K31/395 , A61K31/495 , A61K31/55 , A61P31/00 , C07D401/14 , C07D403/10
CPC classification number: C07D401/14 , C07D403/10
Abstract: The present invention relates to novel triazole compounds of formula (I), their prodrugs, their pharmaceutically acceptable salts and their stereoisomers thereof. The present invention also relates to a process for the preparation of the novel compound of the formula (I).
Abstract translation: 本发明涉及式(I)的新型三唑化合物,其前药,其药学上可接受的盐及其立体异构体。 本发明还涉及制备式(I)的新型化合物的方法。
-
17.NEW ANTICANCER COMPOUNDS, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM 审中-公开
Title translation: 新型化合物及其制备方法及含有它们的药物组合物公开(公告)号:WO2004069145A2
公开(公告)日:2004-08-19
申请号:PCT/IB2004000299
申请日:2004-02-06
Applicant: REDDYS LAB LTD DR , VEDULA MANOHAR SHARMA , KATTUBOINA VENKATA ADISESHU , IQBAL JAVED , RAMANUJAM RAJAGOPALAN , RAJAGOPAL SRIRAM , MAMIDI NAGA VENKATA SRINIVASA , JOSYULA RAMANATHAM , GUTTA MADHUSUDHAN
Inventor: VEDULA MANOHAR SHARMA , KATTUBOINA VENKATA ADISESHU , IQBAL JAVED , RAMANUJAM RAJAGOPALAN , RAJAGOPAL SRIRAM , MAMIDI NAGA VENKATA SRINIVASA , JOSYULA RAMANATHAM , GUTTA MADHUSUDHAN
IPC: A61K20060101 , C07D215/00 , C07D215/44 , C07D215/54 , C07D239/72 , C07D239/94 , A61K
CPC classification number: C07D239/94 , C07D215/44 , C07D215/54
Abstract: The present invention relates to novel anticancer agents, their pharmaceutically acceptable salts, their geometrical isomers and their pharmaceutically acceptable compositions containing them. the present invention more particularly relates to novel quinazoline compounds, their pharmaceutically acceptable salts and their pharmaceutically acceptable compositions containing them. the novel quinazoline compounds have the general formula (I), where all symbols are as defined in the specification.
Abstract translation: 本发明涉及新型抗癌剂,其药学上可接受的盐,它们的几何异构体及其含有它们的药学上可接受的组合物。 本发明更具体地涉及新的喹唑啉化合物,其药学上可接受的盐及其含有它们的药学上可接受的组合物。 新的喹唑啉化合物具有通式(I),其中所有符号如说明书中所定义。
-
18.HETEROCYCLIC COMPOUNDS HAVING ANTIBACTERIAL ACTIVITY, PROCESS FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM 审中-公开
Title translation: 具有抗菌活性的杂环化合物,其制备方法和含有它们的药物组合物公开(公告)号:WO02051819A9
公开(公告)日:2003-08-07
申请号:PCT/IN0100227
申请日:2001-12-26
Applicant: REDDYS LAB LTD DR
Inventor: NATESAN SELVAKUMAR , DAS JAGATTARAN , IQBAL JAVED , MAGADI SITARAM KUMAR , MAMIDI NAGA VENKATA SRINIVASA , RAMANUJAM RAJAGOPALAN , SUNDARABABU BASKARAN , LOHRAY BRAJ BHUSHAN
IPC: A61K31/422 , A61K31/423 , A61P31/04 , C07D263/20 , C07D263/22 , C07D263/24 , C07D263/58 , C07D413/08 , C07D413/10 , C07D413/14 , C07D417/08 , C07D417/10 , A61K31/42 , C07D263/10 , C07D413/12 , C07D417/12
CPC classification number: C07D263/20 , C07D263/22 , C07D263/24 , C07D413/10 , C07D413/14 , C07D417/10
Abstract: The present invention relates to novel oxazolidinone compounds of the general formula (I) where R , R , R , Y , Y , Y , Y , and Z are as defined in the description; their derivatives, their analogs, their tautomeric forms, their stereoisomers, their polymorphs, their pharmaceutically acceptable salts, their pharmaceutically acceptable solvates and pharmaceutical compositions containing them.
Abstract translation: 本发明涉及通式(I)的新的恶唑烷酮化合物,其中R 1,R 2,R 3,Y 1,Y 1,Y 2,Y 3, ,Z如说明书所定义; 它们的衍生物,它们的类似物,它们的互变异构形式,它们的立体异构体,它们的多晶型物,其药学上可接受的盐,它们的药学上可接受的溶剂化物和含有它们的药物组合物。
-
19.NOVEL ANTIINFECTIVE COMPOUNDS AND THEIR PHARMACEUTICAL COMPOSITIONS 审中-公开
Title translation: 新型抗生素化合物及其药物组合物公开(公告)号:WO2004106329A2
公开(公告)日:2004-12-09
申请号:PCT/IB2004001811
申请日:2004-06-03
Applicant: REDDYS LAB LTD DR , MOHAMED TAKHI , DAS JAGATTARAN , NATESAN SELVAKUMAR , TREHAN SANJAY , IQBAL JAVED , MAGADI SITARAM KUMAR
Inventor: MOHAMED TAKHI , DAS JAGATTARAN , NATESAN SELVAKUMAR , TREHAN SANJAY , IQBAL JAVED , MAGADI SITARAM KUMAR
IPC: A61P31/04 , C07D405/10 , C07D405/14 , C07D409/10 , C07D409/14 , C07D405/00
CPC classification number: C07D405/10 , C07D405/14 , C07D409/10 , C07D409/14
Abstract: The present invention provides novel triazole compounds of formula (I), their pharmaceutically acceptable salts and their pharmaceutical compositions, where all symbols are as defined in the specification
Abstract translation: 本发明提供新的式(I)三唑化合物,其药学上可接受的盐及其药物组合物,其中所有符号如说明书中所定义
-
公开(公告)号:EP2702034A4
公开(公告)日:2015-03-25
申请号:EP12777520
申请日:2012-04-27
Applicant: REDDYS LAB LTD DR
Inventor: KATKAM SRINIVAS , SAGYAM RAJESWAR REDDY , MORTHALA RAGHAVENDAR RAO , IRENI BABU , VINIGARI KRISHNA , RAMDOSS SURESH KUMAR , RANGINENI SRINIVASULU , TUMMALA ARJUNKUMAR , IQBAL JAVED , ORUGANTI SRINIVAS , KANDAGATLA BHASKAR
IPC: C07C211/00 , C07C201/10 , C07C201/12 , C07C213/02 , C07D333/20
CPC classification number: C07C205/45 , C07C201/10 , C07C201/12 , C07C213/00 , C07C213/02 , C07C213/10 , C07C215/28 , C07C205/04
-
-
-
-
-
-
-
-
-