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公开(公告)号:WO2011022596A2
公开(公告)日:2011-02-24
申请号:PCT/US2010046091
申请日:2010-08-20
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR , BANDICHHOR RAKESHWAR , LEKKALA AMARNATH REDDY , HALDAR PRANAB , MYLAVARAPU RAVI KUMAR , GOLLA CHINA MALAKONDAIAH , VAGWALA RAGHUNATH , KARRI VIJAYA KUMAR , AKULA SWAPNA
Inventor: BANDICHHOR RAKESHWAR , LEKKALA AMARNATH REDDY , HALDAR PRANAB , MYLAVARAPU RAVI KUMAR , GOLLA CHINA MALAKONDAIAH , VAGWALA RAGHUNATH , KARRI VIJAYA KUMAR , AKULA SWAPNA
IPC: C07D403/12 , A61K31/404 , A61K31/55 , A61P5/30 , C07D403/10
CPC classification number: C07D403/12 , A61K31/404 , A61K31/55
Abstract: Processes for preparing bazedoxifene and its pharmaceutically acceptable salts, substantially free from process related impurities and process intermediates.
Abstract translation: 用于制备基本上不含过程相关杂质和过程中间体的巴多昔芬及其药学上可接受的盐的方法。
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2.
公开(公告)号:WO2012037187A3
公开(公告)日:2012-06-07
申请号:PCT/US2011051501
申请日:2011-09-14
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR , KANNIAH SUNDRA LAKSHMI , BOGE RAJESHAM , SUBBAREDDY PEDDIREDDY , KANWAR LALITA , RAMAKRISHNAN SRIVIDYA , KUMAR RAMYA , BANDICHHOR RAKESHWAR , LEKKALA AMARNATH REDDY , MYLAVARAPU RAVI KUMAR , RAGHUNATH VAGWALA
Inventor: KANNIAH SUNDRA LAKSHMI , BOGE RAJESHAM , SUBBAREDDY PEDDIREDDY , KANWAR LALITA , RAMAKRISHNAN SRIVIDYA , KUMAR RAMYA , BANDICHHOR RAKESHWAR , LEKKALA AMARNATH REDDY , MYLAVARAPU RAVI KUMAR , RAGHUNATH VAGWALA
IPC: C07D403/12 , A61K31/404 , A61K31/55 , C07C53/08 , C07C53/10 , C07D403/10
CPC classification number: C07D403/12 , C07D209/12
Abstract: Aspects of the present disclosure include crystalline bazedoxifene free base, crystalline bazedoxifene acetate Form D, and processes for their preparation. The drug compound having the adopted name "bazedoxifene acetate" has a chemical name 1-[4-(2-azepan-1-yl-ethoxy)benzyl]-2-(4-hydroxyphenyl)-3-methyl-1H-indol-5-ol acetic acid, and has the chemical structure shown below as Formula I.
Abstract translation: 本公开的方面包括结晶巴西多昔芬游离碱,结晶苯卓昔芬乙酸盐晶型D及其制备方法。 采用名称“醋酸巴泽多昔芬”的药物化合物具有化学名称1- [4-(2-氮杂环庚烷-1-基 - 乙氧基)苄基] -2-(4-羟基苯基)-3-甲基-1H-吲哚-1-基] 5-醇乙酸,并具有如下式I所示的化学结构。
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3.IMPROVED PROCESS FOR PREPARATION OF SAXAGLIPTIN AND ITS SALTS 审中-公开
Title translation: 改进萨伐他汀及其盐的制备方法公开(公告)号:WO2013175395A3
公开(公告)日:2014-01-30
申请号:PCT/IB2013054167
申请日:2013-05-21
Applicant: REDDYS LAB LTD DR
Inventor: VARANASI GANESH , MACHARLA PRABHAKAR , VEMPATI CHANDRASEKHAR , BANDICHHOR RAKESHWAR , DAHANUKAR VILAS HARESHWAR , IQBAL JAVED , ORUGANTI SRINIVAS , RAPOLU RAJESH KUMAR , NARIYAM MUNASWAMY SEKHAR , NETI SRINIVASAN
IPC: C07D209/02 , A61K31/403 , C07C13/615 , C07D209/52
CPC classification number: C07D209/52
Abstract: Improved processes for preparing saxagliptin or its salt and intermediates thereof are provided.
Abstract translation: 提供了制备沙格列汀或其盐及其中间体的改进方法。
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公开(公告)号:WO2011025932A3
公开(公告)日:2011-07-21
申请号:PCT/US2010046938
申请日:2010-08-27
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR , BANDICHHOR RAKESHWAR , GUDIMALLA NAGARAJU , DWIVEDI NAMRATA , CHETLURU KIRAN KUMAR , GADE SRINIVAS REDDY , MUVVA VENKATESWARLU , SRIVASTAVA BINDU
Inventor: BANDICHHOR RAKESHWAR , GUDIMALLA NAGARAJU , DWIVEDI NAMRATA , CHETLURU KIRAN KUMAR , GADE SRINIVAS REDDY , MUVVA VENKATESWARLU , SRIVASTAVA BINDU
IPC: C07D487/04 , A61K31/4985 , A61P3/10
CPC classification number: C07D487/04 , A61K31/4985
Abstract: Processes for preparing sitagliptin and its pharmaceutically acceptable salts, and process intermediates.
Abstract translation: 制备西他列汀及其药学上可接受的盐和方法中间体的方法。
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公开(公告)号:WO2016009401A3
公开(公告)日:2016-03-17
申请号:PCT/IB2015055428
申请日:2015-07-17
Applicant: REDDYS LAB LTD DR
Inventor: SUD ABHISHEK , CHAUDHARI PRAMOD , BANDICHHOR RAKESHWAR , DAHANUKAR VILAS HARESHWAR , CHEEMALAPATI VENKATA ANNAPURNA SASI KALA , KAVITAPU DASAMESWARA RAO , LILAKAR JAYDEEPKUMAR DAHYABHAI
IPC: C07F9/6558
CPC classification number: C07F9/65583
Abstract: The present application relates to processes for the preparation of tedizolid phosphate.
Abstract translation: 本申请涉及制备磷酸泰替唑酯的方法。
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6.PHARMACEUTICAL COMPOSITIONS COMPRISING BORONIC ACID COMPOUNDS 审中-公开
Title translation: 包含硼酸化合物的药物组合物公开(公告)号:WO2013128419A3
公开(公告)日:2013-11-21
申请号:PCT/IB2013051644
申请日:2013-03-01
Applicant: REDDYS LAB LTD DR
Inventor: VAYA NAVIN , PRABHAKAR BHAGWATWAR HARSHAL , BANDICHHOR RAKESHWAR , KHATI NIRMAL , SHAIK RIYAZ AHMED , BHISE RAHUL , ASALLA YAKASWAMY , SHINDE RAJKUMAR BHIMRAO
IPC: A61K31/4985 , A61K9/08 , A61K38/05 , A61K47/12 , A61P35/00
CPC classification number: A61K47/18 , A61K31/133 , A61K31/194 , A61K31/497 , A61K31/69 , A61K47/12 , C07F5/025 , A61K2300/00
Abstract: A pharmaceutical composition and preparing processes thereof. The composition comprises bortezomib or pharmaceutically acceptable salt or solvate thereof, tromethamine and an organic carboxylic acid, and the pH of the composition is from about 3.0 to 6.0.
Abstract translation: 药物组合物及其制备方法。 组合物包含硼替佐米或其药学上可接受的盐或溶剂化物,氨丁三醇和有机羧酸,组合物的pH为约3.0至6.0。
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公开(公告)号:WO2008077035A3
公开(公告)日:2008-10-09
申请号:PCT/US2007087924
申请日:2007-12-18
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR , GADE SRINIVAS REDDY , MALLEPALLI SRINIVAS REDDY , MUVVA VENKATESHWARLU , AMIRISETTY RAVINDHRANATH TAGORE , HARIKEERTHI NARASIMHA MURTHY , RAMASAMY VIJAYA ANAND , BANDICHHOR RAKESHWAR , MYLAVARAPU RAVI KUMAR , KOPPARAPU RAMACHANDRA JANARDANA SARMA , MANUDHANE KUSHAL SURAJMAL , MADDULA SRINIVASULA REDDY
Inventor: GADE SRINIVAS REDDY , MALLEPALLI SRINIVAS REDDY , MUVVA VENKATESHWARLU , AMIRISETTY RAVINDHRANATH TAGORE , HARIKEERTHI NARASIMHA MURTHY , RAMASAMY VIJAYA ANAND , BANDICHHOR RAKESHWAR , MYLAVARAPU RAVI KUMAR , KOPPARAPU RAMACHANDRA JANARDANA SARMA , MANUDHANE KUSHAL SURAJMAL , MADDULA SRINIVASULA REDDY
IPC: C07D207/27
CPC classification number: C07D207/27
Abstract: A process for preparing levetiracetarn of the Formula (I) via a reaction between S-arnlnobutyramide or its salt: and 4-chlqrobutyrylchloride: which process comprses forming a reaction mixture that includes, the S-aminsbutyrarriide or its salt, the 4-chlorobutyrylchloride, and potassium hydroxide, wherein the potassium hydroxide is added to said reaction mixture in a lot-wise manner...
Abstract translation: 通过S-氨基异丁酰胺或其盐与4-氯丁酰氯的反应来制备式(I)的左乙拉西那嗪的方法:该方法包括形成包含S-氨基丁二酰亚胺或其盐的4-氯丁酰氯的反应混合物, 和氢氧化钾,其中将氢氧化钾以很多方式加入到所述反应混合物中...
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公开(公告)号:EP2470542A4
公开(公告)日:2013-04-24
申请号:EP10812650
申请日:2010-08-27
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR
Inventor: BANDICHHOR RAKESHWAR , GUDIMALLA NAGARAJU , DWIVEDI NAMRATA , CHETLURU KIRAN KUMAR , GADE SRINIVAS REDDY , MUVVA VENKATESWARLU , SRIVASTAVA BINDU
IPC: C07D487/04 , A61K31/4985 , A61P3/10
CPC classification number: C07D487/04 , A61K31/4985
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9.
公开(公告)号:EP2819673A4
公开(公告)日:2015-03-18
申请号:EP13755443
申请日:2013-03-01
Applicant: REDDYS LAB LTD DR
Inventor: VAYA NAVIN , PRABHAKAR BHAGWATWAR HARSHAL , BANDICHHOR RAKESHWAR , KHATI NIRMAL , SHAIK RIYAZ AHMED , BHISE RAHUL , ASALLA YAKASWAMY , SHINDE RAJKUMAR BHIMRAO
IPC: A61K38/05 , A61K9/08 , A61K31/133 , A61K31/194 , A61K31/497 , A61K31/69 , A61K47/12 , A61P35/00
CPC classification number: A61K47/18 , A61K31/133 , A61K31/194 , A61K31/497 , A61K31/69 , A61K47/12 , C07F5/025 , A61K2300/00
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公开(公告)号:EP2616463A4
公开(公告)日:2014-01-08
申请号:EP11825836
申请日:2011-09-14
Applicant: REDDYS LAB LTD DR , REDDYS LAB INC DR
Inventor: KANNIAH SUNDRA LAKSHMI , BOGE RAJESHAM , SUBBAREDDY PEDDIREDDY , KANWAR LALITA , RAMAKRISHNAN SRIVIDYA , KUMAR RAMYA , BANDICHHOR RAKESHWAR , LEKKALA AMARNATH REDDY , MYLAVARAPU RAVI KUMAR , RAGHUNATH VAGWALA
IPC: C07D403/12 , A61K31/404 , A61K31/55 , C07C53/08 , C07C53/10 , C07D403/10
CPC classification number: C07D403/12 , C07D209/12
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