公开(公告)号：DE60201089D1

公开(公告)日：2004-09-30

申请号：DE60201089

申请日：2002-04-06

Applicant: BASF AG

Inventor： TORMO I BLASCO JORDI ,  SAUTER HUBERT ,  MUELLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHAEFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N25/02 ,  A01N25/08 ,  A01N43/90 ,  C07D487/04

Abstract: 6-(2-Chloro-6-fluoro-phenyl)-triazolopyrimidines of formula (I), in which R 1 and R 2 independently denote hydrogen or alkyl, alkenyl, alkynyl, alkadienyl, or haloalkyl, cycloalkyl, bicycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R 1 and R 2 radicals may be unsubstituted or partially or fully halogenated or may be substituted as defined in the description. R 1 and R 2 together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; X is cyano, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi

公开(公告)号：HU0400210A2

公开(公告)日：2004-08-30

申请号：HU0400210

申请日：2002-03-13

Applicant: BASF AG

Inventor： AMMERMANN EBERHARD ,  GEWEHR MARKUS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  LORENZ GISELA ,  MUELLER BERND ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SAUTER HUBERT ,  SCHIEWECK FRANK ,  SCHAEFER PETER ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  TORMO I BLASCO JORDI

IPC: A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/64 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D239/42 ,  C07D401/14 ,  C07D403/04 ,  C07D471/04 ,  C07D473/06 ,  C07D487/04 ,  C07D521/00

Abstract: 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.

公开(公告)号：AU2003303097A1

公开(公告)日：2004-08-13

申请号：AU2003303097

申请日：2003-11-14

Applicant: BASF AG

Inventor： GROTE THOMAS ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH ,  BLASCO JORDI TORMO I

IPC: A01N43/90 ,  A01N55/10 ,  A01N47/38

Abstract: Disclosed are fungicidal mixtures containing A) a triazolopyrimidine derivative of formula (1), and B) an azole derivative or the salts or addition compound thereof selected among bromuconazole, difenoconazole, diniconazole, fenbuconazole, fluquinconazole, flusilazole, hexaconazole, prochloraz, tetraconazole, triflumizole, flutriafol, myclobutanil, penconazole, simeconazole, ipconazole, triticonazole, and prothioconazole as active components in a synergistically effective quantity, methods for controlling plant-pathogenic fungi by means of mixtures of compounds I and II-XVIII, substances containing said mixtures, and the use of compounds I and II-XVIII for producing such mixtures.

公开(公告)号：BR0211180A

公开(公告)日：2004-08-10

申请号：BR0211180

申请日：2002-07-08

Applicant: BASF AG

Inventor： BLASCO JORDI TORMO I ,  SAUTER HUBERT ,  LLER BERND M ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04

Abstract: Substituted 6-(2-tolyl)-triazolopyrimidines of formula (I) in which R and R independently denote hydrogen or alkyl, alkenyl, alkynyl, or alkadienyl, haloalkyl, haloalkenyl, cycloalkyl, phenyl, naphthyl, or 5- or 6-membered heterocyclyl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or 5- or 6-membered heteroaryl, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, or where R and R radicals may be unsubstituted or substituted as defined in the description, or R and R together with the interjacent nitrogen atom represent a 5- or 6-membered heterocyclic ring, containing one to four nitrogen atoms or one to three nitrogen atoms and one sulfur or oxygen atom, which may be substituted; R is halogen, cyano, alkyl, alkoxy, haloalkyl, or C(=O)A, wherein A is hydrogen, hydroxy, alkyl, amino, or mono- or dialkyl-amino; n is an integer from 1 to 4; and X is halogen, cyano, alkyl, alkoxy, haloalkoxy or alkenyloxy; processes for their preparation, compositions containing them and to their use for combating phytopathogenic fungi.

公开(公告)号：UA67778C2

公开(公告)日：2004-07-15

申请号：UA00126941

申请日：1999-04-23

Applicant: BASF AG

Inventor： SCHERER MARIA ,  SAUTER HUBERT ,  AMMERMANN EBERHARD ,  GROTE THOMAS ,  LORENZ GISELA

IPC: A01N47/24 ,  A01N37/50 ,  A01N47/12 ,  A01N47/18

Abstract: Винахідстосуєтьсяфунгіцидноїсуміші, щоміститьпринаймніоднусполукуз групи, щовключаєа1) карбаматиформулиІ, деТ означаєСНабо N, n дорівнює 0, 1 або 2 і R означаєгалоген, С1-С4алкілабоС1-С4галогеналкіл, причомузалишки R, якщо n дорівнює 2, можутьвідрізнятисяодинвідодного, a2) оксимовийефірскладногоефірукарбоновоїкислотиформули II абоа3) амідоксимовогоефірукарбоновоїкислотиформули III, іб) принаймніоднуактивнуречовинуформули IV, дезамісники R1-R3 маютьтакізначення: R1 означаєС1-С4алкіл, С2-С4алкеніл, С2-С4алкініл, С1-С4алкіл-С3-С7циклоалкіл, причомуцізалишкиможутьматизамісникиз групи, щовключаєгалоген, ціаной С1-С4алкокси, атакожозначаєС1-С4алкокси, R2 означаєС1-С4алкілабоС1-С4галогеналкіл, R3 означаєводень, галоген, С1-С4алкіл, С1-С4алкокси, С1-С4алкілтіо, N-С1-С4алкіламіно, С1-С4галогеналкілабоС1-С4галогеналкокси, Y означаєО, S, CHR4 або NR5, причому R4 і R5 можутьматизначення, наведенідля R2, n дорівнює 0, 1, 2 або 3, усинергічноефективнійкількості. , (I) , (II) , (III) (IV).

公开(公告)号：BR0210858A

公开(公告)日：2004-06-29

申请号：BR0210858

申请日：2002-07-03

Applicant: BASF AG

Inventor： MUELLER BERND ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  BLASCO JORDI TORMO I ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  RACK MICHAEL ,  LORENZ GISELA ,  STRATHMANN SIEGFRIED ,  AMMERMANN EBERHARD ,  STIERL REINHARD

IPC: A01N43/90 ,  C07D487/04 ,  A01N43/653

Abstract: 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines (I) are new. 5-(Alkyl, alkenyl or alkynyl)-7-(hydrocarbyl or heterocyclyl)-6-phenyl-1,2,4-triazolo[1,5-a]pyrimidines of formula (I) are new. [Image] n : 0-5; R : halo, CN, OH or OCN, or alkyl, alkenyl, alkynyl, T', haloalkenyl, OT, alkenyloxy, alkynyloxy, OT', cycloalkyl, cycloalkenyl, cycloalkoxy, alkoxycarbonyl, alkenyloxycarbonyl, alkynyloxycarbonyl, CONH 2, mono- or dialkylaminocarbonyl, alkoximinoalkyl, alkenyloximinocarbonyl, alkynyloximinoalkyl, alkylcarbonyl, alkenylcarbonyl, alkynylcarbonyl, cycloalkylcarbonyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); T : 1-6C alkyl; T' : 1-6C haloalkyl; Het : 5-10 membered, saturated, partially unsaturated or aromatic heterocycle containing 1-4 of O, N and/or S heteroatoms; R 11-10C alkyl, alkenyl, alkynyl, 3-12C cycloalkyl, 3-10C cycloalkenyl, phenyl, naphthyl or Het (all optionally partially or completely halogenated and optionally substituted by 1-4 R a); R ahalo, CN, NO 2, OH, T, T', COT, cycloalkyl, OT, OT', COOT, NHT, NT 2, 2-6C alkenyl, 2-6C alkenyloxy, 3-6C alkynyloxy, alkoximino, alkenyloximino, alkynyloximino, aralkoximino, alkynyl, alkynyloxycarbonyl, phenyl, naphthyl or Het (where all aliphatic, alicyclic or aromatic groups are optionally partially or completely halogenated and optionally substituted by 1-3 R aand/or 1-3 R c); R bhalo, CN, NO 2, OH, SH, NH 2, COOH, CONH 2, CSNH 2, T, T', 2-8C alkenyl, 2-8C alkenyloxy, 2-8C alkynyloxy, OT, OT', ST, NHT, NT 2, CHO, COT, SO 2T, SOT, COOT, OCOT, CONHT, CONT 2, CSNHT or CSNT 2; R ccycloalkyl, -O-cycloalkyl, heterocyclyl, -O-heterocyclyl, aryl, -O-aryl, -S-aryl, -O-T-aryl, -T-aryl, heteroaryl, -O-heteroaryl or -S-heteroaryl (where cycloalkyl or heterocyclyl rings are 3-10 membered, aryl rings are preferably 6-10 membered and heteroaryl rings are preferably 5-6 membered; and all rings are optionally partially or completely halogenated and optionally substituted by alkyl or haloalkyl); and R 21-4C alkyl, 2-4C alkynyl or 2-4C alkynyl (all optionally substituted by halo, CN, NO 2, OMe, OEt or 1-4C alkoxycarbonyl; Unless specified otherwise alkyl moieties have 1-8C, alkenyl or alkynyl moieties 2-10C and cycloalkyl or cycloalkenyl moieties 3-6C. Independent claims are also included for: (1) preparation of (I); and (2) dicarbonyl compound intermediates of formula (III), provided that n is not 0 and R 1and R 2are not both Me. [Image] ACTIVITY : Fungicide. 7-Cyclohexyl-5-methyl-6-(2-chloro-6-fluorophenyl)-1,2,4-triazolo[1,5-a]pyrimidine (Ia) at a concentration of 63 ppm gave at least 90 % protection of tomato plants against Alternaria solani. MECHANISM OF ACTION : None given.

公开(公告)号：BR0209835A

公开(公告)日：2004-06-15

申请号：BR0209835

申请日：2002-05-17

Applicant: BASF AG

Inventor： RHEINHEIMER JOACHIM ,  GYPSER ANDREAS ,  ROSE INGO ,  GROTE THOMAS ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  AMMERMANN EBERHARD ,  SPEAKMAN JOHN-BRYAN ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA

IPC: A01N43/86 ,  A01N43/90 ,  C07D265/24 ,  C07D498/04 ,  C07D513/04

Abstract: Oxazin(ethi)one compounds of the formula I: in which the variables Z, R 1 , R 2 , R 3 and n are as defined in claim 1 and A is a 5- or 6-membered carbocycle or a 5- or 6-membered heterocycle having 1, 2 or 3 heteroatoms selected from the group consisting of N, O and S, each of which cycles is attached via two carbon atoms to the oxazin(ethi)one ring, and the agriculturally useful salts of the oxazin(ethi)one compounds I are described. Moreover, the invention describes the use of compounds I and their salts for controlling phytopathogenic fungi, compositions which comprise the compounds I and/or their salts in a fungicidally effective amount and a method for controlling phytopathogenic fungi which comprises treating the fungi or the materials, plants, seeds or the soil threatened by fungal attack with a fungicidally effective amount of at least one compound of the formula I as claimed in claim 1 and/or a salt of I.

公开(公告)号：BR0207975A

公开(公告)日：2004-06-15

申请号：BR0207975

申请日：2002-03-13

Applicant: BASF AG

Inventor： GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  ROSE INGO ,  SCHOFER PETER ,  SCHIEWECK FRANK ,  SAUTER HUBERT ,  GEWEHR MARKUS ,  MUELLER BERND ,  BLASCO JORDI TORMO I ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED ,  LORENZ GISELA ,  STIERL REINHARD

IPC: A01N43/54 ,  A01N43/56 ,  A01N43/58 ,  A01N43/60 ,  A01N43/64 ,  A01N43/647 ,  A01N43/653 ,  A01N43/713 ,  A01N43/90 ,  C07D239/42 ,  C07D401/14 ,  C07D403/04 ,  C07D471/04 ,  C07D473/06 ,  C07D487/04 ,  C07D521/00 ,  C07D473/00

Abstract: 5-Phenylpyrimidines of the formula I, in which the substituents have the following meanings: R1 is a five- to ten-membered saturated, partially unsaturated or aromatic mono- or bicyclic heterocycle comprising one to four hetero atoms selected from the group consisting of O, N or S, which heterocycle can be substituted as defined in the description, R2 is hydrogen, halogen, cyano, alkyl, haloalkyl or alkoxy; R3, R4 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, R3 and R4 together with the nitrogen atom to which they are bonded may also form a five- or six-membered ring which can be interrupted by a hetero atom and have attached to it one or more substituents; R5, R6 are hydrogen, halogen, alkyl, haloalkyl or alkoxy; R7, R8 are hydrogen, halogen, alkyl or haloalkyl; R9 is hydrogen, halogen, alkyl, alkoxy, cycloalkoxy, haloalkoxy or alkoxycarbonyl, Processes and intermediates for the preparation of these compounds, and their use for controlling harmful fungi.

公开(公告)号：AU2003298117A1

公开(公告)日：2004-06-15

申请号：AU2003298117

申请日：2003-11-14

Applicant: BASF AG

Inventor： SCHOFL ULRICH ,  STIERL REINHARD ,  BLASCO JORDI TORMO I ,  BLETTNER CARSTEN ,  MULLER BERND ,  GEWEHR MARKUS ,  GRAMMENOS WASSILIOS ,  GROTE THOMAS ,  GYPSER ANDREAS ,  RHEINHEIMER JOACHIM ,  SCHAFER PETER ,  SCHIEWECK FRANK ,  SCHWOGLER ANJA ,  AMMERMANN EBERHARD ,  STRATHMANN SIEGFRIED

IPC: A01N43/90 ,  C07D487/04 ,  C07D249/00

Abstract: 2-Substituted triazolopyrimidines of the formula I, in which the substituents are as defined below: L are halogen, cyano, nitro, alkyl, alkenyl, alkynyl, haloalkyl, haloalkenyl, alkoxy, alkenyloxy, alkynyloxy, haloalkoxy, -C(-O)-A or S(-O) p A'; A and A' are as defined in the description; p is 0, 1 or 2; m is 0, 1, 2, 3, 4 or 5; X is cyano, alkyl, haloalkyl, alkoxy or haloalkoxy; R 1 ,R 2 are hydrogen, alkyl, haloalkyl, cycloalkyl, halocycloalkyl, alkenyl, alkadienyl, haloalkenyl, cycloalkenyl, alkynyl, haloalkynyl or cycloalkynyl, phenyl, naphthyl or a five- to ten-membered saturated, partially unsaturated or aromatic heterocycle which contains one to four heteroatoms from the group consisting of O, N and S, R 1 and R 2 together with the nitrogen atom to which they are attached may also form a five- or six-membered ring which may be interrupted by an atom from the group consisting of O, N and S, where R 1 and/or R 2 may be substituted as defined in the description; and R 3 is cyano, hydroxyl, alkoxy, alkenyloxy, haloalkoxy, haloalkenyloxy, NR 1 R 2 or S(O) n R 31 , where n and R 31 are as defined in the description; Processes and intermediates for preparing these compounds, compositions comprising them and their use for controlling phytopathogenic harmful fungi are described.

公开(公告)号：AU2003293690A1

公开(公告)日：2004-06-15

申请号：AU2003293690

申请日：2003-11-14

Applicant: BASF AG

Inventor： BLASCO JORDI TORMO I ,  GROTE THOMAS ,  AMMERMANN EBERHARD ,  STIERL REINHARD ,  STRATHMANN SIEGFRIED ,  SCHOFL ULRICH

IPC: A01N43/90 ,  A01N47/24

Abstract: Fungicidal mixtures comprising A) the triazolopyrimidine derivative of the formula I and B) carbamates of the formula II in which n is 1 or 2 and X is halogen, alkyl or haloalkyl, where the radicals X may be different if n is 2, in a synergistically effective amount, methods for controlling harmful fungi using mixtures of the compounds I and II, compositions comprising these compounds and the use of the compounds I and the compounds II for preparing such mixtures are described.