PARA-SUBSTITUTED INDANYL AND TETRALINYL DERIVATIVES
    41.
    发明申请
    PARA-SUBSTITUTED INDANYL AND TETRALINYL DERIVATIVES 审中-公开
    对照衍生的吲哚和四氢吲哚衍生物

    公开(公告)号:WO2017012938A1

    公开(公告)日:2017-01-26

    申请号:PCT/EP2016/066603

    申请日:2016-07-13

    Applicant: BASF SE

    Abstract: Compounds of formula I, wherein the substituents R 1 , X, and the index k are as defined in the specification; a process for preparation of compounds of formula I, a process for preparation of its precursor compounds II, wherein the substituents R 1 , X, and the index k are as defined in the specification; intermediates for the production of compounds I, or II; use of compounds of formula I for the production of compounds of formula VI wherein the substituents R 1 , R 3 , and the index k are as defined in the specification; the use of compounds I, or II, for the production of active compounds.

    Abstract translation: 式I化合物,其中取代基R1,X和指数k如说明书中所定义; 制备式I化合物的方法,其前体化合物II的制备方法,其中取代基R1,X和指数k如说明书中所定义; 用于生产化合物I或II的中间体; 使用式I化合物来制备式VI化合物,其中取代基R 1,R 3和指数k如说明书中所定义; 使用化合物I或II来生产活性化合物。

    PROCESS FOR MANUFACTURING HALOACETAMIDES
    45.
    发明申请
    PROCESS FOR MANUFACTURING HALOACETAMIDES 审中-公开
    制备HALOACETAMIDES的方法

    公开(公告)号:WO2015003858A1

    公开(公告)日:2015-01-15

    申请号:PCT/EP2014/061591

    申请日:2014-06-04

    Applicant: BASF SE

    CPC classification number: C07C231/02 C07C51/58 C07C231/00 C07C233/05 C07C53/48

    Abstract: The present invention relates to a process for manufacturing haloacetamides of formula (I), comprising sub-step (a): reacting halones of formula (II) with oleum; followed by sub-step (b): reacting the reaction mixture obtained in sub-step(a) with an amine of formula (IV) optionally in the presence of a base; wherein the variables are defined according to the description.

    Abstract translation: 本发明涉及制备式(I)的卤代乙酰胺的方法,其包括以下步骤(a):使式(II)的卤酮与发烟硫酸反应; 然后是亚步骤(b):使在步骤(a)中获得的反应混合物与式(IV)的胺任选地在碱的存在下反应; 其中根据描述定义变量。

    ISOTHIAZOLINE COMPOUNDS FOR COMBATING INVERTEBRATE PESTS
    47.
    发明申请
    ISOTHIAZOLINE COMPOUNDS FOR COMBATING INVERTEBRATE PESTS 审中-公开
    用于组合反相胶束的异噻唑化合物

    公开(公告)号:WO2013092943A1

    公开(公告)日:2013-06-27

    申请号:PCT/EP2012/076539

    申请日:2012-12-21

    Applicant: BASF SE

    CPC classification number: C07D275/02 A01N43/80 C07D275/03 C07D417/04

    Abstract: The present invention relates to isothiazoline compounds of formula (I) wherein the variables are as defined in the claims or the description, which are useful for combating or controlling invertebrate pests, in particular arthropod pests and nematodes, and to a method for producing them. The invention also relates to a method for controlling invertebrate pests by using these compounds and to plant propagation material and to an agricultural and a veterinary composition comprising said compounds.

    Abstract translation: 本发明涉及式(I)的异噻唑啉化合物,其中变量如权利要求或描述中所定义,其可用于对抗或控制无脊椎动物害虫,特别是节肢动物害虫和线虫,以及其制备方法。 本发明还涉及通过使用这些化合物和植物繁殖材料以及包含所述化合物的农业和兽用组合物来控制无脊椎害虫的方法。

    PROCESS FOR PREPARING N-SUBSTITUTED 1H-PYRAZOLE-5-CARBOXYLATE COMPOUNDS AND DERIVATIVES THEREOF
    50.
    发明申请
    PROCESS FOR PREPARING N-SUBSTITUTED 1H-PYRAZOLE-5-CARBOXYLATE COMPOUNDS AND DERIVATIVES THEREOF 审中-公开
    制备N-取代的1H-吡唑-5-羧酸酯化合物及其衍生物的方法

    公开(公告)号:WO2013076092A1

    公开(公告)日:2013-05-30

    申请号:PCT/EP2012/073128

    申请日:2012-11-20

    Applicant: BASF SE

    CPC classification number: C07D401/04 C07D471/10

    Abstract: The present invention relates to a process for preparing an N-substituted 1 H-pyrazole- 5- carboxylate compound of the formula (l-A) comprising the steps of i) deprotonating a compound of the formula (II) in which the variables R 1 , R 2 and r are each as defined in the description and the claims, with a magnesium-organic base having a carbon bound magnesium; and ii) subjecting the product obtained in step (i) to a carbonylation by reacting it with a reagent selected from the group consisting carbon dioxide or a carbon dioxide equivalent, to obtain a compound of formula (l-A); and it relates to further conversions to yield a N-substituted 1H-pyrazole-5-carbonyl chloride compound of the formula (I).

    Abstract translation: 本发明涉及一种制备式(1A)的N-取代的1H-吡唑-5-羧酸酯化合物的方法,包括以下步骤:i)将式(II)的化合物去质子化,其中变量R1,R2 和r各自如说明书和权利要求中所定义,镁 - 有机碱具有碳结合的镁; 和ii)通过使步骤(i)中获得的产物与选自二氧化碳或二氧化碳当量的试剂反应来进行羰基化,得到式(I-A)化合物; 并且涉及进一步转化得到式(I)的N-取代的1H-吡唑-5-碳酰氯化合物。

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