公开(公告)号：CA2666203A1

公开(公告)日：2008-04-17

申请号：CA2666203

申请日：2007-10-12

Applicant: BASF SE

Inventor： KEIL MICHAEL ,  LOEHR SANDRA ,  HAMPRECHT GERHARD ,  SAXELL HEIDI EMILIA ,  WOLF BERND ,  SIEVERNICH BERND ,  COX GERHARD ,  SCHMIDT THOMAS ,  MAYER GUIDO ,  SEITZ WERNER ,  GEBHARDT JOACHIM ,  MICHEL ALFRED ,  ERK PETER ,  WEVERS JAN HENDRIK ,  ZAGAR CYRILL ,  REINHARD ROBERT

IPC: C07D239/54 ,  A01N43/48

Abstract: The present invention relates to hydrates of 2-chloro-5-[3,6-dihydro-3-me thyl-2,6-dioxo-4-(trifluoromethyl)-1-(2H)-pyrimidinyl]-4-fluoro-N-[[methyl-( 1-methylethyl)amino]sulphonyl]benzamide. The invention also relates to a met hod for preparing these hydrates, and to formulations for crop protection wh ich comprise hydrates of the phenyluracil I.

公开(公告)号：AU2006310551A1

公开(公告)日：2007-05-10

申请号：AU2006310551

申请日：2006-10-26

Applicant: BASF SE

Inventor： KNELL MARCUS ,  BRINK MONIKA ,  WEVERS JAN HENDRIK

IPC: C07D213/81 ,  C07D213/79

Abstract: The invention relates to a process for the preparation of pyridylcarboxylic amides and esters I, Formula (I) wherein Hal, X and R1 have the meanings given in claim 1, which comprises the following steps: (a) heating a mixture consisting essentially of trichloromethylpyridine II, Formula (II), wherein Hal has the meaning given, and 1.0 to 1.5 equivalents of concentrated sulfuric acid, characterized in that the trichloromethylpyridine II in a liquid form is added to the concentrated sulfuric acid at a temperature from 110° C. to 160° C.; and (b) reacting the intermediate product obtained in step (a) with an amine or alcohol III, HXR1, wherein X and R1 have the meaning given, optionally in the presence of a solvent and/or a base.

公开(公告)号：BRPI0719214B1

公开(公告)日：2016-11-22

申请号：BRPI0719214

申请日：2007-10-12

Applicant: BASF SE

Inventor： MICHEL ALFRED ,  SIEVERNICH BERND ,  WOLF BERND ,  ZAGAR CYRILL ,  COX GERHARD ,  HAMPRECHT GERHARD ,  MAYER GUIDO ,  SAXELL HEIDI EMILIA ,  WEVERS JAN HENDRIK ,  GEBHARDT JOACHIM ,  KEIL MICHAEL ,  ERK PETER ,  REINHARD ROBERT ,  LÖHR SANDRA ,  SCHMIDT THOMAS ,  SEITZ WERNER

IPC: C07D239/54 ,  A01N43/48

公开(公告)号：CA2626465C

公开(公告)日：2016-07-12

申请号：CA2626465

申请日：2006-10-26

Applicant: BASF SE

Inventor： BRINK MONIKA ,  KNELL MARCUS ,  WEVERS JAN HENDRIK

IPC: C07D213/81 ,  C07D213/79

Abstract: The invention relates to a process for the preparation of pyridylcarboxylic amides and esters I, Formula (I) wherein Hal, X and R1 have the meanings given in claim 1, which comprises the following steps: (a) heating a mixture consisting essentially of trichloromethylpyridine II, Formula (II), wherein Hal has the meaning given, and 1.0 to 1.5 equivalents of concentrated sulfuric acid, characterized in that the trichloromethylpyridine II in a liquid form is added to the concentrated sulfuric acid at a temperature from 110~C to 160~C; and (b) reacting the intermediate product obtained in step (a) with an amine or alcohol III, HXR1, wherein X and R1 have the meaning given, optionally in the presence of a solvent and/or a base.

公开(公告)号：BRPI0609798B1

公开(公告)日：2015-01-27

申请号：BRPI0609798

申请日：2006-05-18

Applicant: BASF SE

Inventor： GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  SCHMIDT THOMAS ,  WEVERS JAN HENDRIK ,  ZECH HELMUT ,  HAEBERLE RUDOLF

IPC: C07D239/54

Abstract: The present invention relates to a process for preparing 1-alkyl-3-phenyluracils of the formula I where the variables R1 to R7 are as defined in the description by reacting 3-phenyluracils of the formula II and alkylating agents of the formula III R1-L1  III, with one another, wherein during the entire reaction the pH is kept in a range from 1 to 6 by adding base a little at a time.

公开(公告)号：AU2007306270B2

公开(公告)日：2013-09-26

申请号：AU2007306270

申请日：2007-10-12

Applicant: BASF SE

Inventor： HAMPRECHT GERHARD ,  LOHR SANDRA ,  SEITZ WERNER ,  KEIL MICHAEL ,  GEBHARDT JOACHIM ,  MICHEL ALFRED ,  COX GERHARD ,  SIEVERNICH BERND ,  SAXELL HEIDI EMILIA ,  MAYER GUIDO ,  ZAGAR CYRILL ,  SCHMIDT THOMAS ,  ERK PETER ,  WOLF BERND ,  REINHARD ROBERT ,  WEVERS JAN HENDRIK

IPC: C07D239/54 ,  A01N43/48

Abstract: The present invention relates to a crystalline form of 2-chloro-5-[3,6-dihydro-3-methyl-2,6-dioxo-4-(trifluoromethyl)-1-(2H)-pyrimidinyl]-4-fluoro-N-[[methyl-(1-methylethyl)amino]sulphonyl]benzamide. The invention also relates to a method for preparing this crystalline form and to formulations for crop protection which comprise this crystalline form of the phenyluracil.

公开(公告)号：UA98291C2

公开(公告)日：2012-04-25

申请号：UAA201101802

申请日：2006-11-23

Applicant: BASF SE

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  RACK MICHAEL ,  MAYER GUIDO ,  PLESCHKE AXEL

IPC: C07C303/40 ,  C07C201/00 ,  C07C205/00 ,  C07C311/00

Abstract: Способполучениясульфонамидовформулы I EMBED ISISServer I, гдезаместителиимеютзначение, приведенныев описании, реакциейхлоридовм-нитробензойнойкислотыформулы II саминосульфонамиформулы III, вприсутствииВ эквивалентовоснованияформулы IV, причемнастадииа) аминосульфоныформулы III реагируютс В1 эквивалентамиоснованияформулы IV, инастадии b) реакционнуюсмесь, полученнуюнастадииа), подвергаютвзаимодействиюс хлоридамим-нитробензойнойкислотыформулы II иВ2 эквивалентамиоснованияформулы IV, гдеВ, В1 иВ2 имеютзначение, приведенныев описании.

公开(公告)号：BRPI0619760A2

公开(公告)日：2012-02-22

申请号：BRPI0619760

申请日：2006-11-23

Applicant: BASF SE

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOEHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  RACK MICHAEL ,  MAYER GUIDO ,  PLESCHKE AXEL

IPC: C07C303/38 ,  C07C201/12 ,  C07C205/58 ,  C07C303/40 ,  C07C311/51

Abstract: A process for preparing sulfonamides I where the variables are each as defined in the description, by reacting m-nitrobenzoyl chlorides II with amino sulfones III, under the influence of B equivalents of base IV, wherein, in step a), the amino sulfone III is reacted with B1 equivalents of base IV, and, in step b), the reaction mixture resulting from step a) is reacted with m-nitrobenzoyl chlorides II and B2 equivalents of base IV; where B, B1 and B2 are each as defined in the description.

公开(公告)号：UA96281C2

公开(公告)日：2011-10-25

申请号：UAA200808447

申请日：2006-11-23

Applicant: BASF SE

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LOHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  RACK MICHAEL ,  MAYER GUIDO ,  PLESCHKE AXEL

IPC: C07C201/00 ,  C07C205/06 ,  C07C205/58 ,  C07C303/40

Abstract: Способполучениясульфонамидовформулы I EMBED ISISServer , (I) гдезаместителиимеютзначения, приведенныев описании, реакциейхлоридовм-нитробензойнойкислотыформулы II саминосульфонамиформулы III. Такжеописанспособполученияхлорангидридовм-нитробензойнойкислоты.

公开(公告)号：PL2081914T3

公开(公告)日：2011-07-29

申请号：PL07821246

申请日：2007-10-12

Applicant: BASF SE

Inventor： SCHMIDT THOMAS ,  GEBHARDT JOACHIM ,  LÖHR SANDRA ,  KEIL MICHAEL ,  WEVERS JAN HENDRIK ,  ERK PETER ,  SAXELL HEIDI EMILIA ,  HAMPRECHT GERHARD ,  SEITZ WERNER ,  MAYER GUIDO ,  WOLF BERND ,  COX GERHARD ,  MICHEL ALFRED ,  ZAGAR CYRILL ,  REINHARD ROBERT ,  SIEVERNICH BERND

IPC: A01N43/48 ,  C07D239/54